购物车

搜索结果

Search Results for " har "
Targets Recommended: Others

45

抑制剂 & 化合物

83

天然产物

4

化合物库

12

重组蛋白

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name
L1010 FDA上市及药典收录分子库

3158 compounds
3158 个上市及药典分子集合,可用于高通量筛选和高内涵筛选;
L6800 中国药典收录天然产物库

2051 compounds
2051 种中国药典收录的天然产物,是药物开发、药理研究等领域的有力工具;
L7830 高溶解性片段药效团化合物库

985 compounds
高溶解性片段药效团库包含985 个片段小分子。
L6140 糖类及苷类化合物库

362 compounds
362 种糖类或苷类的化合物,可用于高通量筛选和高内涵筛选;

化合物库

FDA上市及药典收录分子库
Cat.No: L1010
Compounds: 3158
中国药典收录天然产物库
Cat.No: L6800
Compounds: 2051
高溶解性片段药效团化合物库
Cat.No: L7830
Compounds: 985
糖类及苷类化合物库
Cat.No: L6140
Compounds: 362
Cat. No. Product Name Target Signaling Pathways
T5020 Eptifibatide

Eptifibatide Acetate,Mpr-Har-Gly-Asp-Trp-Pro-Cys-NH2,依替巴肽

Others Others
Eptifibatide (Eptifibatide Acetate) 是一种糖蛋白 IIb/IIIa 抑制剂类的抗血小板药物,是一种由 6 个氨基酸和一个巯基丙酰基残基构成的环状七肽。
T79600 Zharp2-1

RIP kinase Apoptosis; NF-κB
Zharp2-1是一种 RIPK2 抑制剂,抑制了 MDP 诱导或单核细胞增生李斯特菌感染诱导的炎症细胞因子的转录,缓解MDP诱导的小鼠腹膜炎症状,可用于研究炎症性肠病 (IBD)。
T0582 Fructooligosaccharides

Others Others
Fructooligosaccharides 是一种左旋单糖,是葡萄糖的异构体。
T0889 Saccharin

O-Sulfobenzimide,O-Benzoic sulfimide,Saccharimide,Benzoic sulfimide,糖精

Others; Antibacterial Microbiology/Virology; Others
Saccharin (O-Sulfobenzimide) 是一种口服有效的人造甜味剂,具有抑菌和微生物调节特性。
T10789 Chitosan oligosaccharide

COS,壳聚糖低聚乳酸酯

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Chitosan oligosaccharide (COS) 是 β-(1→4)-连接的 D-氨基葡萄糖的寡聚体,Chitosan oligosaccharide可激活 AMPK ,抑制NF-κB 和 MAPK在内的炎症信号通路。
T6974 Saccharin 1-methylimidazole

糖精-1-甲基咪唑盐,SMI,Saccharin 1-methylimidazole (SMI)

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Saccharin 1-methylimidazole (SMI) 是一种用于 DNA 和 RNA 合成的通用激活剂。
T3158L Harman hydrochloride

哈尔满盐酸盐,Harmane hydrochloride(486-84-0 Free base)

P450 Metabolism
Harman hydrochloride 可以以 AhR 依赖性方式直接诱导 CYP1A1 基因表达,可能代表了harman 促进致突变性、共致突变性和致癌性的新机制。
T7871 Calcium D-saccharate tetrahydrate

D-Glucaric acid calcium salt,葡萄糖二酸鈣,Calcium D-saccharate tetrahydrate,D-Saccharic acid calcium salt

Others Others
Calcium D-saccharate tetrahydrate (Calcium D-saccharate tetrahydrate) 是一种氧化的非环状己糖。它可以抑制癌细胞的癌变和增殖。
T8673 FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR

Fmoc-Tpi-OH,FMOC-L-1,2,3,4-四氢-Β-咔啉-3-羧酸

Others Others
FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR (Fmoc-Tpi-OH) 是THN 的衍生物。
T4983 Isoetharine mesylate salt

Isoetarine mesilate,异丙肾上腺素甲磺酸盐

Others; Adrenergic Receptor GPCR/G Protein; Neuroscience; Others
Isoetharine mesylate salt (Isoetarine mesilate) 是一种 β-肾上腺素能受体激动剂。它还是能够上调 CYP450 表达的孕烷 X 受体(PXR) 激活剂。
T41319 D-Saccharic acid 1,4-lactone hydrate

Others Others
D-Saccharic acid 1,4-lactone hydrate 是β-葡萄糖醛酸酶的有效抑制剂(IC50=48.4 μM),可用作标准药物。D-Saccharic acid 1,4-lactone hydrate 显示出抗癌、解毒和抗氧化的活性性。
T124661 Cepharadione B

Cepharadione B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124661。
T10786 Charantin

GSK-3 PI3K/Akt/mTOR signaling; Stem Cells
Charantin is a steroidal saponin isolated from Momordica charantia. It increases the release of insulin and slowing down gluconeogenesis. Charantin can inhibit GSK-3.
T35744 Ivermectin B1a monosaccharide

Ivermectin B1a monosaccharide is produced by selective hydrolysis of the terminal saccharide unit of ivermectin. It can inhibit nematode larval development, but does not cause paralytic activity. This compound has been used as a probe to detect some types of ivermectin resistance.
T19977 Saccharin sodium

CCRIS 706,Saccharin, sodium

Saccharin sodium is a type of artificial or nonnutritive sweetener. Saccharin sodium is used in the production of various foods and pharmaceutical products.
T77217 Saccharopine hydrochloride

Saccharopine hydrochloride(L-Saccharopine hydrochloride)是赖氨酸降解的中间体,兼具线粒体毒性。该化合物由赖氨酸-酮戊二酸还原酶催化赖氨酸与α-酮戊二酸生成。继而,糖精脱氢酶作用于Saccharopine hydrochloride,生成α-氨基己酸酯半醛和谷氨酸。其通过干扰线粒体的稳态平衡,对生物体的发育造成损害。
T72319 Lewis y tetrasaccharide

Lewis y

Lewis Y tetrasaccharide (Lewis Y, LeY) 是Lewis X trisaccharide 的四糖衍生物。Lewis Y tetrasaccharide 是一种与恶性卵巢癌转移和预后不良相关的抗原。
T75594 Harpactira Baviana Venom

Harpactira Baviana Venom (Baboon Tarantula Venom) 是一种蜘蛛毒液,能够从皇帝巴布蜘蛛蜘蛛中获得。Harpactira Baviana Venom 可以调节 NaV1.8和诱导痛觉过敏。
T60502 Isoetharine hydrochloride

Isoetharine (hydrochloride) (compound I) 是一种选择性和口服活性的短效β-肾上腺能受体激动剂,广泛用作吸入治疗研究中的支气管扩张剂。
T30217 Avadharidine

Avadharidine is a biochemical.
T125719 Harzianic acid

Harzianic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125719。
T126414 Harmalidine

Harmalidine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126414。
T64850 Chinese Pharmacopoeia Compound Library

Chinese Pharmacopoeia Compound Library 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64850。
T4983L Isoetharine

Isoetarine,Bronkosol,Bronkometer,Etyprenalinum

Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.
T125160 Harmalacidine

Harmalacidine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125160。
T68721 Cantharidin imide

Cantharidin imide is a PP1/2A inhibitor found in Canarthis vesicatoria. It inhibits proliferation of colorectal cancer cells, increases MCP-1, IL-6, and IL-β levels, and inhibits differentiation and resorptive activity of osteoclasts. This compound can produce severe skin inflammation, and is extremely toxic if ingested orally.
T126029 8-cis-Cinnamoylharpagide

8-cis-Cinnamoylharpagide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126029,CAS号为 133645-36-0。
T37730 Saccharocarcin A

Saccharocarcin A is an antibiotic originally isolated from S. aerocolonigenes subsp. antibiotica. It is active against M. luteus, S. aureus, E. coli, P. aeruginosa, and C. albicans in a disc assay. Saccharocarcin A inhibits C. trachomatis infection by 88% without inducing cytotoxicity in McCoy cells when used at a concentration of 0.5 μg/ml.
T81424 Polysaccharidase

Tremella polysaccharide

Polysaccharidase (Tremella polysaccharide) 是一种提升免疫功能的真菌多糖。该化合物展现出治疗化疗和放疗导致的白细胞减少症的研究潜力。
T123890 Catharantin; Catharanthine

Catharantin; Catharanthine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T123890,CAS号为 94444-28-7。
T19979 Saccharin sodium hydrate

O-benzoic sulfimide sodium salt,糖精钠,Saccharin, sodium salt hydrate

Saccharin, sodium salt hydrate is used in the food industry and for sweetening diabetes diet. It is also used as a synthetic sweet ignorance agent. Saccharin, sodium salt hydrate is the first generation′ synthetic sugar alternative that has been studied f
T35756 Avermectin B1a monosaccharide

Avermectin B1a monosaccharide is a macrolide anthelmintic and monosaccharide form of avermectin B1a . It is lethal to C. elegans with a minimum active concentration (MAC) value of 0.1 μM. Avermectin B1a monosaccharide also stimulates conductance in isolated shore crab muscle.
T37509 Saccharocarcin B

Saccharocarcin B 是从放线菌 Saccharothrix aerocolongenes subsp.antibiotica SCC1886 的发酵液中分离出来的。
T30265 Navafenterol saccharinate

AZD8871 saccharinate,LAS-191351 saccharinate,LAS191351 saccharinate,AZD-8871 saccharinate

AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).
T68494 Octenidine saccharin

Octenidine saccharin is a Dental Plaque Inhibitor
T126028 8-O-4-Hydroxycinnamoylharpagide

8-O-4-Hydroxycinnamoylharpagide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126028,CAS号为 133645-37-1。
T75728 Charybdotoxin TFA

Charybdotoxin TFA 是一种含 37 个氨基酸的肽,是一个K+通道阻滞剂。
TP2059 Charybdotoxin

Specific inhibitor of the big conductance Ca2+-activated K+ channel.
T124022 8-p-Coumaroylharpagide

T26790 Bharangin

Bharangin is a inhibitor of penicillinase enzyme in E coli.
T35734 Doramectin monosaccharide

Doramectin monosaccharide is an acid degradation product of doramectin , a disaccharide-containing anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in nematodes. Doramectin undergoes acid-catalyzed hydrolysis to form doramectin monosaccharide.
T82583 Deoxyharringtonine

Deoxyharringtonine为从Cephalotaxus属植物中分离的生物碱,具备显著的抗白血病活性。
T32900 Saccharopine

L-Saccharopine,accharopin

L-Saccharopine is a product of the breakdown of essential amino acid Lysine.
T30870 Chartreusin sodium

X465A sodium salt

Chartreusin sodium is a biochemical.
T12323 ORM-15341

Androgen Receptor Endocrinology/Hormones
ORM-15341 是雄激素受体拮抗剂,作用于 AR-HEK293细胞(IC50:38 nM)。

化合物

Eptifibatide
Cat.No: T5020
Synonym: Eptifibatide Acetate,Mpr-Har-Gly-Asp-Trp-Pro-Cys-NH2,依替巴肽
Target: Others
Zharp2-1
Cat.No: T79600
Synonym:
Target: RIP kinase
Fructooligosaccharides
Cat.No: T0582
Synonym:
Target: Others
Saccharin
Cat.No: T0889
Synonym: O-Sulfobenzimide,O-Benzoic sulfimide,Saccharimide,Benzoic sulfimide,糖精
Target: Others, Antibacterial
Chitosan oligosaccharide
Cat.No: T10789
Synonym: COS,壳聚糖低聚乳酸酯
Target: AMPK
Saccharin 1-methylimidazole
Cat.No: T6974
Synonym: 糖精-1-甲基咪唑盐,SMI,Saccharin 1-methylimidazole (SMI)
Target: DNA/RNA Synthesis
Harman hydrochloride
Cat.No: T3158L
Synonym: 哈尔满盐酸盐,Harmane hydrochloride(486-84-0 Free base)
Target: P450
Calcium D-saccharate tetrahydrate
Cat.No: T7871
Synonym: D-Glucaric acid calcium salt,葡萄糖二酸鈣,Calcium D-saccharate tetrahydrate,D-Saccharic acid calcium salt
Target: Others
FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR
Cat.No: T8673
Synonym: Fmoc-Tpi-OH,FMOC-L-1,2,3,4-四氢-Β-咔啉-3-羧酸
Target: Others
Isoetharine mesylate salt
Cat.No: T4983
Synonym: Isoetarine mesilate,异丙肾上腺素甲磺酸盐
Target: Others, Adrenergic Receptor
D-Saccharic acid 1,4-lactone hydrate
Cat.No: T41319
Synonym:
Target: Others
Cepharadione B
Cat.No: T124661
Synonym:
Target:
Charantin
Cat.No: T10786
Synonym:
Target: GSK-3
Ivermectin B1a monosaccharide
Cat.No: T35744
Synonym:
Target:
Saccharin sodium
Cat.No: T19977
Synonym: CCRIS 706,Saccharin, sodium
Target:
Saccharopine hydrochloride
Cat.No: T77217
Synonym:
Target:
Lewis y tetrasaccharide
Cat.No: T72319
Synonym: Lewis y
Target:
Harpactira Baviana Venom
Cat.No: T75594
Synonym:
Target:
Isoetharine hydrochloride
Cat.No: T60502
Synonym:
Target:
Avadharidine
Cat.No: T30217
Synonym:
Target:
Harzianic acid
Cat.No: T125719
Synonym:
Target:
Harmalidine
Cat.No: T126414
Synonym:
Target:
Chinese Pharmacopoeia Compound Library
Cat.No: T64850
Synonym:
Target:
Isoetharine
Cat.No: T4983L
Synonym: Isoetarine,Bronkosol,Bronkometer,Etyprenalinum
Target:
Harmalacidine
Cat.No: T125160
Synonym:
Target:
Cantharidin imide
Cat.No: T68721
Synonym:
Target:
8-cis-Cinnamoylharpagide
Cat.No: T126029
Synonym:
Target:
Saccharocarcin A
Cat.No: T37730
Synonym:
Target:
Polysaccharidase
Cat.No: T81424
Synonym: Tremella polysaccharide
Target:
Catharantin; Catharanthine
Cat.No: T123890
Synonym:
Target:
Saccharin sodium hydrate
Cat.No: T19979
Synonym: O-benzoic sulfimide sodium salt,糖精钠,Saccharin, sodium salt hydrate
Target:
Avermectin B1a monosaccharide
Cat.No: T35756
Synonym:
Target:
Saccharocarcin B
Cat.No: T37509
Synonym:
Target:
Navafenterol saccharinate
Cat.No: T30265
Synonym: AZD8871 saccharinate,LAS-191351 saccharinate,LAS191351 saccharinate,AZD-8871 saccharinate
Target:
Octenidine saccharin
Cat.No: T68494
Synonym:
Target:
8-O-4-Hydroxycinnamoylharpagide
Cat.No: T126028
Synonym:
Target:
Charybdotoxin TFA
Cat.No: T75728
Synonym:
Target:
Charybdotoxin
Cat.No: TP2059
Synonym:
Target:
8-p-Coumaroylharpagide
Cat.No: T124022
Synonym:
Target:
Bharangin
Cat.No: T26790
Synonym:
Target:
Doramectin monosaccharide
Cat.No: T35734
Synonym:
Target:
Deoxyharringtonine
Cat.No: T82583
Synonym:
Target:
Saccharopine
Cat.No: T32900
Synonym: L-Saccharopine,accharopin
Target:
Chartreusin sodium
Cat.No: T30870
Synonym: X465A sodium salt
Target:
ORM-15341
Cat.No: T12323
Synonym:
Target: Androgen Receptor
Cat. No. Product Name Target Signaling Pathways
TN7211 Tetrahydroharmine

Leptaflorine

MAO Metabolism; Neuroscience
Tetrahydroharmine (Leptaflorine) 是一种天然产物,存在于植物Banisteriopsis caapi cultivar Da Vine 的茎和枝中。四氢骆驼蓬碱是一种Monoamine oxidase A 抑制剂。
T2782 Catharanthine

(+)-3, 4-Didehydrocoronaridine,长春质碱,(+)-3,4-Didehydrocoronaridine

Calcium Channel; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience
Catharanthine ((+)-3,4-Didehydrocoronaridine) 是长春花中的一种生物碱,可抑制电压门控 L 型钙离子通道,具有抗肿瘤和降血压活性。
T3158 Harmane

Loturine,Harman,Aribine,哈尔满碱

Adrenergic Receptor; Monoamine Oxidase; Imidazoline Receptor GPCR/G Protein; Neuroscience
Harmane (Loturine) 是一种在咖啡和烟草烟雾中发现的 β-咔啉生物碱,是有效的神经毒素,可引起严重的动作震颤和精神病学表现。它还是选择性的单胺氧化酶抑制剂,具有致突变作用,对 MAO A/B 的 IC50值分别为 0.5 和 5 μM。
T1711 Harmine

Telepathine,去氢骆驼蓬碱

MAO; 5-HT Receptor; DYRK Cell Cycle/Checkpoint; GPCR/G Protein; Metabolism; Neuroscience; Tyrosine Kinase/Adaptors
Harmine (Telepathine) 是一种从山茱萸种子中分离出来的生物碱,具有抗癌和抗炎活性。它是双特异性酪氨酸磷酸化调节激酶抑制剂,对5-HT2A 血清素受体具有高亲和力,Ki 值为 397 nM。
T5791 Fructo-​oligosaccharide DP7/GF6

Fructoheptasaccharide,蔗果七糖

Others Others
Fructo-​oligosaccharide DP7/GF6 (Fructoheptasaccharide) 属于一种聚果糖,聚合度 (DP=7)。其中 Fructo-oligosaccharides (FOS) 由 6 个果糖单元通过 (2→1)-β-糖苷键连接,并在非还原性末端具有 1 个 D-葡萄糖单元。
T3023 Catharanthine sulfate

AChR Neuroscience
Catharanthine sulfate 抑制烟碱样受体介导的隔膜收缩。
T3013 Catharanthine tartrate

Catharanthine hemitartrate,酒石酸长春质碱

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Catharanthine tartrate (Catharanthine hemitartrate) 是长春花中的一种生物碱,可抑制电压门控 L 型钙离子通道,具有抗肿瘤和降血压活性。
TN2376 Fructo-oligosaccharide DP8/GF7

蔗果八糖,Fructo-oligosaccharide DP8 / GF7

Others Others
Fructo-oligosaccharide DP8/GF7 (Fructo-oligosaccharide DP8 / GF7) 是一种聚果糖,聚合度(DP=8)。Fructo-oligosaccharides 由 7 个果糖单元通过 (2→1)-β-糖苷键连接,并在非还原性末端具有 1 个 D-葡萄糖单元。
T11855 Lipopolysaccharides

脂多糖,LPS

Others Others
Lipopolysaccharides (LPS) 是革兰氏阴性细菌细胞壁的一种特有成分,由脂质A、寡糖核心和 O -特异性多糖 (O-antigen) 3个区域组成。Lipopolysaccharides 有利于维持细胞外膜的完整性,保护细菌免受胆汁盐和脂类抗生素的破坏。Lipopolysaccharides 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
T0131 Cepharanthine

NSC-623442,千金藤碱,千金藤素

Apoptosis; TNF; HIV Protease; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Cepharanthine (NSC-623442) 是从Stephania cepharanthaHayata 中提取的一种生物碱,具有抗炎、抗氧化作用。它可抑制肿瘤坏死因子 (TNF)-α 介导的 NFκB 刺激、质膜脂质过氧化和血小板聚集,并抑制细胞因子的产生。
TN6640 1,2,3,4-Tetrahydronorharman-1-one

1,2,3,4-四羟基去甲哈尔满-1-酮,L-Oxonoreleagnine

Parasite; Antifection Microbiology/Virology
1,2,3,4-Tetrahydronorharman-1-one (L-Oxonoreleagnine) 是从印度尼西亚海海绵 Acanthostrongylophora ingens 中分离得到的。
T8770 Harmalol

骆驼蓬酚,Harmidol

AChR Neuroscience
Harmalol (Harmidol) 是一种具有生物活性的 β-咔啉,是 harmalal 生物碱的成员
T41078 Lipopolysaccharides, Escherichiacoli

Lipopolysaccharide, E. coli O111:B4

Others Others
Lipopolysaccharides, Escherichiacoli (E. coli O111:B4) 是革兰氏阴性细菌细胞壁的一种特有成分,由脂质A、寡糖核心和 O -特异性多糖 (O-antigen) 3个区域组成。Lipopolysaccharides, Escherichiacoli 有利于维持细胞外膜的完整性,保护细菌免受胆汁盐和脂类抗生素的破坏。Lipopolysaccharides, Escherichiacoli 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
T8286 Harringtonine

三尖杉酯碱,三尖杉脂碱

Others; Influenza Virus Microbiology/Virology; Others
Harringtonine 是一种天然的 Cephalotaxus 生物碱,可抑制蛋白质合成,有抗基孔肯雅病毒活性,EC50为 0.24 μM。
T2782L Catharanthine Tartrate(2468-21-5(free base))

Calcium Channel Membrane transporter/Ion channel; Metabolism
Catharanthine Tartrate(2468-21-5(free base)) 是从马达加斯加长春花中分离得到的天然产物,Catharanthine Tartrate 抑制电压操作的L 型Ca2+通道,具有抗癌和降血压活性。
T2894 Norcantharidin

Norcantharadine,去甲斑蝥素,Endothall anhydride

EGFR; c-Met/HGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Norcantharidin (Norcantharadine) 是一种合成的抗癌化合物,是人类结肠癌中 c-Met 和 EGFR 的双重抑制剂。
T3380 Homoharringtonine

Myelostat,Ceflatonin,高三尖杉酯碱,HHT,Omacetaxine mepesuccinate

STAT JAK/STAT signaling; Stem Cells
Homoharringtonine (HHT) 属于生物碱类天然产物,可以抑制蛋白质的翻译,具有细胞毒性。Homoharringtonine 作用于肿瘤细胞的核糖体,抑制蛋白质翻译的延伸步骤,从而抑制蛋白质合成,具有抗肿瘤活性。
T2736 Sodium Demethylcantharidate

Sodium norcantharidin,去甲斑蝥酸钠

Others; Endogenous Metabolite Metabolism; Others
Sodium Demethylcantharidate (Sodium norcantharidin) 是内源性代谢产物的一种。
T3152 Harmol

哈尔酚(骆驼蓬醇),Methylpyridoindolol

Others Others
Harmol (Methylpyridoindolol) 一种 β-carboline 生物碱,是单胺氧化酶抑制剂,可用作分析参考标准品。
T2811 Harmine hydrochloride

telepathine hydrochloride,盐酸哈尔明碱

5-HT Receptor; DYRK; GluR Cell Cycle/Checkpoint; GPCR/G Protein; Neuroscience; Tyrosine Kinase/Adaptors
Harmine hydrochloride (telepathine hydrochloride) 是一种 DYRK 抑制剂,具有抗癌和抗炎活性。它对5-HT2A 血清素受体具有高亲和力,Ki 值为 397 nM。
T2797 Harmaline

Others Others
Harmaline 是一种来自harmala 生物碱和β-咔啉的荧光精神活性吲哚生物碱。它是harmine 的还原氢化形式。
T5086 Pharmatose DCL 14

D-乳糖一水合物,D-Lactose monohydrate

Others; Endogenous Metabolite Metabolism; Others
Pharmatose DCL 14 (D-Lactose monohydrate) 是内源性代谢产物的一种。
TN1724 Harmalol hydrochloride

Harmidol hydrochloride

P450; Antioxidant Metabolism; oxidation-reduction
Harmalol hydrochloride (Harmidol hydrochloride) 是一种可从Peganum harmala L.的种子中提取出来的β-咔啉生物碱。Harmalol hydrochloride 是Harmaline 的主要代谢产物,在转录和翻译后水平上显著抑制二恶英介导的 CYP1A1 诱导。Harmalol hydrochloride 在去氧肾上腺素或KCl 预先收缩的分离大鼠胸主动脉制剂中显示出血管松弛活性。 Harmalol hydrochloride 具有抗氧化活性.
T6S2025 8-​O-​Acetylharpagide

8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide

Antibacterial Microbiology/Virology
8-O-Acetylharpagide 是从 Ajuga reptans 中分离得到的一种环烯醚萜,有抗肿瘤、抗病毒、抗菌和抗炎作用。它对豚鼠的离体平滑肌有生物活性。
T6S2024 Harpagide

Antibacterial; Parasite Microbiology/Virology
Harpagide 是从Scrophularia cryptophila 中分离出来的一种鸢尾糖苷,具有抗炎和抗寄生虫活性,对T.b. rhodesiense 具有体外锥虫杀虫活性,IC50为 21 μg/mL,它对L. donovani 的IC50值为 2.0 μg/mL。
T5656 (±)-Norcantharidin

Endothall anhydride,去甲斑蝥素,Norcantharidin

EGFR; c-Met/HGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
(±)-Norcantharidin (Endothall anhydride) 是一种人类结肠癌中 c-Met 和 EGFR 的双重抑制剂,可研究抗癌,具有抗血管生成活性。
T6S2023 Harpagoside

Others; COX; NO Synthase Immunology/Inflammation; Neuroscience; Others
Harpagoside 是从爪钩草中分离出来的一种天然产物,可抑制COX-1和COX-2活性,并抑制 NO 的产生。
T8769 Harmaline hydrochloride

Harmidine hydrochloride

Others Others
Harmaline hydrochloride (Harmidine hydrochloride) 是一种荧光吲哚生物碱,来自 harmala 生物碱和 β-咔啉。它是 harmine 的部分氢化形式。 Harmaline 通过诱导下橄榄神经元的节律性放电在正常大鼠中产生全身性震颤。
T8154 Fructo-oligosaccharide DP9/GF8

Fructo-oligosaccharide DP9 / GF8,蔗果九糖

Others Others
Fructo-oligosaccharide DP9/GF8 (Fructo-oligosaccharide DP9 / GF8) 是一种低聚果糖(FOS),其聚合度DP=9。低聚果糖(FOS)由 8 个果糖单元通过 (2→1)-β-糖苷键连接,并在非还原性末端具有 1 个 D-葡萄糖单元。
T2S0837 Astragalus Polysacharin

2-(Chloromethyl)-4-(4-nitrophenyl)thiazole,黄芪多糖,89250-26-0

TAM Receptor Tyrosine Kinase/Adaptors
2-(Chloromethyl)-4-(4-nitrophenyl)thiazole 是一种从黄芪 (Astragalus propinquus) 中提取得到的天然产物。2-(Chloromethyl)-4-(4-nitrophenyl)thiazole 具有抗癌活性,通过抑制肿瘤相关巨噬细胞 (TAM) 的 M2 极化在肝细胞癌 (HCC) 中显示除抗肿瘤活性。
TN3355 Agatharesinol acetonide

Antifection Microbiology/Virology
Agatharesinol acetonide shows anticancer activity towards the A549 non-small-cell lung-cancer cell line (IC50 = 27.1 microM).
TN6014 Norcepharadione B

鱼腥草

Norcepharadione B shows good inhibitory activity against the replication of HSV-1, it also shows antimalarial activity with EC50 values of 7.5mug/ml. Norcepharadione B exhibits significant cytotoxicity against five human tumor cell lines (A-549, SK-OV-3,
TN4622 N9-Methylharman

Others Others
N9-Methylharman 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4622,CAS号为 16498-64-9。
TN1483 Charantadiol A

苦瓜二醇A

Others Others
Charantadiol A is a natural product from Momordica charantia.
TN4526 Methyl 2alpha-hydroxyhardwickiate

Others Others
Methyl 2alpha-hydroxyhardwickiate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4526,CAS号为 50428-93-8。
TN6283 Stepharine

Stepharine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6283,CAS号为 2810-21-1。
TN3611 Catharticin

Others Others
Catharticin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3611,CAS号为 39723-40-5。
T81937 Lewis a trisaccharide

Lewis a

Lewis a trisaccharide 是精子聚糖结构和 HL-60 细胞表面聚糖结构的主要组分。
T75637 Demethylcantharidate disodium

Demethylcantharidate disodium 是一种内源性代谢产物,能通过诱导内质网应激来促进肝癌细胞的凋亡,并且对多种类型的癌症展现出良好的抗癌活性。
T79978 6,6′-Dihydroxythiobinupharidine

6,6′-Dihydroxythiobinupharidine 作为一种抑制剂,主要针对半胱氨酸蛋白酶(cysteine proteases)。研究表明,该化合物能显著促进人拓扑异构酶IIα(topoisomeraseIIα)和IIβ(topoisomeraseIIβ)介导的DNA裂解,分别提高了8倍和3倍的效率。
TN1321 6'-​O-​Cinnamoyl harpagide

6'-O-Cinnamoylharpagide,(1S,4AS,5R,7S,7AR)-1,4A,5,6,7,7A-六氢-4A,5,7-三羟基-7-甲基环戊二烯并[C]吡喃-1-基 BETA-D-吡喃葡萄糖苷 6-[(2E)-3-苯基-2-丙烯酸酯],6'-O-肉桂酰基哈巴苷,6'-O-肉桂酰哈巴苷

Others Others
6'-O-Cinnamoylharpagide has anti-inflammatory activity.
T19328 Fructo-oligosaccharide DP11/GF10

Others Others
Fructo-oligosaccharide DP11/GF10 is a fructooligosaccharide (FOS) compound with a degree of polymerization (DP) equal to 11. FOS consists of 10 fructose units connected by (2→1)-β-glycosidic bonds, with a single D-glucosyl unit present at the non-reducing end.
TN2629 15,16-Dihydro-15-methoxy-16-oxohardwickiic acid

Others Others
15,16-Dihydro-15-methoxy-16-oxohardwickiic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2629,CAS号为 115783-35-2。
TN4184 Harmol hydrochloride monohydrate

Others Others
Harmol hydrochloride monohydrate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4184,CAS号为 40580-83-4。
T82369 Fructo-oligosaccharide DP14

Fructo-oligosaccharide DP14为从Atractylodes lancea中提取的寡糖。
TN2057 Perisesaccharide C

Others Others
Perisesaccharide C is a natural product
T83300 5′-Des-O-methylharringtonine

5′-Des-O-methylharringtonine为Cephalotaxus harringtonia植物中提取的天然化合物。
T82277 GM1a Ganglioside oligosaccharide

GM1a Ganglioside oligosaccharide为ganglioside GM1的半合成形式,后者作为霍乱毒素的天然受体,在生长调节及激素诱导反应的耦合中具有关键功能。
T4024 Norharmane

2-Azacarbazole,2,9-Diazafluorene,β-Carboline,去甲哈尔满

DNA; Endogenous Metabolite; Monoamine Oxidase DNA Damage/DNA Repair; Metabolism; Neuroscience
Norharmane (β-Carboline) 是一种有效的选择性单胺氧化酶 A (MAO-A) 抑制剂,Ki=3.34 μM。
TN3162 6-Epi-8-O-acetylharpagide

Others Others
6-Epi-8-O-acetylharpagide是一种天然产物,属于玄参科玄参属,其产品编号为 TN3162,CAS号为 97169-44-3。6-Epi-8-O-acetylharpagide可用作对照参考。
------------------------ 更多 ------------------------

天然产物

Tetrahydroharmine
Cat.No: TN7211
Synonym: Leptaflorine
Target: MAO
Catharanthine
Cat.No: T2782
Synonym: (+)-3, 4-Didehydrocoronaridine,长春质碱,(+)-3,4-Didehydrocoronaridine
Target: Calcium Channel, AChR
Harmane
Cat.No: T3158
Synonym: Loturine,Harman,Aribine,哈尔满碱
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
Harmine
Cat.No: T1711
Synonym: Telepathine,去氢骆驼蓬碱
Target: MAO, 5-HT Receptor, DYRK
Fructo-​oligosaccharide DP7/GF6
Cat.No: T5791
Synonym: Fructoheptasaccharide,蔗果七糖
Target: Others
Catharanthine sulfate
Cat.No: T3023
Synonym:
Target: AChR
Catharanthine tartrate
Cat.No: T3013
Synonym: Catharanthine hemitartrate,酒石酸长春质碱
Target: Others, Calcium Channel
Fructo-oligosaccharide DP8/GF7
Cat.No: TN2376
Synonym: 蔗果八糖,Fructo-oligosaccharide DP8 / GF7
Target: Others
Lipopolysaccharides
Cat.No: T11855
Synonym: 脂多糖,LPS
Target: Others
Cepharanthine
Cat.No: T0131
Synonym: NSC-623442,千金藤碱,千金藤素
Target: Apoptosis, TNF, HIV Protease, Autophagy
1,2,3,4-Tetrahydronorharman-1-one
Cat.No: TN6640
Synonym: 1,2,3,4-四羟基去甲哈尔满-1-酮,L-Oxonoreleagnine
Target: Parasite, Antifection
Harmalol
Cat.No: T8770
Synonym: 骆驼蓬酚,Harmidol
Target: AChR
Lipopolysaccharides, Escherichiacoli
Cat.No: T41078
Synonym: Lipopolysaccharide, E. coli O111:B4
Target: Others
Harringtonine
Cat.No: T8286
Synonym: 三尖杉酯碱,三尖杉脂碱
Target: Others, Influenza Virus
Catharanthine Tartrate(2468-21-5(free base))
Cat.No: T2782L
Synonym:
Target: Calcium Channel
Norcantharidin
Cat.No: T2894
Synonym: Norcantharadine,去甲斑蝥素,Endothall anhydride
Target: EGFR, c-Met/HGFR
Homoharringtonine
Cat.No: T3380
Synonym: Myelostat,Ceflatonin,高三尖杉酯碱,HHT,Omacetaxine mepesuccinate
Target: STAT
Sodium Demethylcantharidate
Cat.No: T2736
Synonym: Sodium norcantharidin,去甲斑蝥酸钠
Target: Others, Endogenous Metabolite
Harmol
Cat.No: T3152
Synonym: 哈尔酚(骆驼蓬醇),Methylpyridoindolol
Target: Others
Harmine hydrochloride
Cat.No: T2811
Synonym: telepathine hydrochloride,盐酸哈尔明碱
Target: 5-HT Receptor, DYRK, GluR
Harmaline
Cat.No: T2797
Synonym:
Target: Others
Pharmatose DCL 14
Cat.No: T5086
Synonym: D-乳糖一水合物,D-Lactose monohydrate
Target: Others, Endogenous Metabolite
Harmalol hydrochloride
Cat.No: TN1724
Synonym: Harmidol hydrochloride
Target: P450, Antioxidant
8-​O-​Acetylharpagide
Cat.No: T6S2025
Synonym: 8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide
Target: Antibacterial
Harpagide
Cat.No: T6S2024
Synonym:
Target: Antibacterial, Parasite
(±)-Norcantharidin
Cat.No: T5656
Synonym: Endothall anhydride,去甲斑蝥素,Norcantharidin
Target: EGFR, c-Met/HGFR
Harpagoside
Cat.No: T6S2023
Synonym:
Target: Others, COX, NO Synthase
Harmaline hydrochloride
Cat.No: T8769
Synonym: Harmidine hydrochloride
Target: Others
Fructo-oligosaccharide DP9/GF8
Cat.No: T8154
Synonym: Fructo-oligosaccharide DP9 / GF8,蔗果九糖
Target: Others
Astragalus Polysacharin
Cat.No: T2S0837
Synonym: 2-(Chloromethyl)-4-(4-nitrophenyl)thiazole,黄芪多糖,89250-26-0
Target: TAM Receptor
Agatharesinol acetonide
Cat.No: TN3355
Synonym:
Target: Antifection
Norcepharadione B
Cat.No: TN6014
Synonym: 鱼腥草
Target:
N9-Methylharman
Cat.No: TN4622
Synonym:
Target: Others
Charantadiol A
Cat.No: TN1483
Synonym: 苦瓜二醇A
Target: Others
Methyl 2alpha-hydroxyhardwickiate
Cat.No: TN4526
Synonym:
Target: Others
Stepharine
Cat.No: TN6283
Synonym:
Target:
Catharticin
Cat.No: TN3611
Synonym:
Target: Others
Lewis a trisaccharide
Cat.No: T81937
Synonym: Lewis a
Target:
Demethylcantharidate disodium
Cat.No: T75637
Synonym:
Target:
6,6′-Dihydroxythiobinupharidine
Cat.No: T79978
Synonym:
Target:
6'-​O-​Cinnamoyl harpagide
Cat.No: TN1321
Synonym: 6'-O-Cinnamoylharpagide,(1S,4AS,5R,7S,7AR)-1,4A,5,6,7,7A-六氢-4A,5,7-三羟基-7-甲基环戊二烯并[C]吡喃-1-基 BETA-D-吡喃葡萄糖苷 6-[(2E)-3-苯基-2-丙烯酸酯],6'-O-肉桂酰基哈巴苷,6'-O-肉桂酰哈巴苷
Target: Others
Fructo-oligosaccharide DP11/GF10
Cat.No: T19328
Synonym:
Target: Others
15,16-Dihydro-15-methoxy-16-oxohardwickiic acid
Cat.No: TN2629
Synonym:
Target: Others
Harmol hydrochloride monohydrate
Cat.No: TN4184
Synonym:
Target: Others
Fructo-oligosaccharide DP14
Cat.No: T82369
Synonym:
Target:
Perisesaccharide C
Cat.No: TN2057
Synonym:
Target: Others
5′-Des-O-methylharringtonine
Cat.No: T83300
Synonym:
Target:
GM1a Ganglioside oligosaccharide
Cat.No: T82277
Synonym:
Target:
Norharmane
Cat.No: T4024
Synonym: 2-Azacarbazole,2,9-Diazafluorene,β-Carboline,去甲哈尔满
Target: DNA, Endogenous Metabolite, Monoamine Oxidase
6-Epi-8-O-acetylharpagide
Cat.No: TN3162
Synonym:
Target: Others
--------- 更多 ---------
Cat. No. Product Name Species Expression System
TMPJ-00533 LYVE1 Protein, Human, Recombinant (His)

XLKD1,Cell Surface Retention Sequence-Binding Protein 1,Extr...

Human HEK293 Cells
Lymphatic Vessel Endothelial Hyaluronic Acid Receptor 1 is a single-pass type I membrane protein. LYVE-1 is a CD44 homolog found primarily on lymphatic endothelial cells 1. LYVE-1 mainly expressed in endothelial cells lining lymphatic vessels. While LYVE-1 functions is a Ligand-specific transporter trafficking between intracellular organelles (TGN) and the plasma membrane. LYVE-1 plays a role in autocrine regulation of cell growth mediated by growth regulators containing cell surface retention s...
TMPY-04932 SUC2 Protein, Saccharomyces cerevisiae, Recombinant (His)

Saccharomyces cerevisiae P. pastoris (Yeast)
SUC2 Protein, Saccharomyces cerevisiae, Recombinant (His) is expressed in yeast with His tag. The predicted molecular weight is 60 kDa and the accession number is P00724-1.
TMPH-02466 Ribonuclease MC Protein, Momordica charantia, Recombinant (His & Myc)

Momordica charantia E. coli
Ribonuclease MC Protein, Momordica charantia, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 28.7 kDa and the accession number is P23540.
TMPH-00363 Cyanovirin-N homolog Protein, Ceratopteris richardii, Recombinant (His)

CV-N homolog,Cyanovirin-N homolog

Ceratopteris richardii P. pastoris (Yeast)
Mannose-binding lectin. Cyanovirin-N homolog Protein, Ceratopteris richardii, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 14.4 kDa and the accession number is P86326.
TMPH-00395 Autolysin Protein, Chlamydomonas reinhardtii, Recombinant (His & SUMO)

Autolysin,GLE,Gametolysin,Gamete lytic enzyme

Chlamydomonas reinhardtii E. coli
Mediates digestion of the cell walls of the 2 mating type gametes during mating as a necessary prelude to cell fusion. This enzyme acts specifically on the framework proteins (inner wall) of the cell wall, cleaving several model peptides at specific sites. Autolysin Protein, Chlamydomonas reinhardtii, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 65.6 kDa and the accession number is P31178.
TMPY-05413 HARS/HisRS Protein, Human, Recombinant (His)

histidyl-tRNA synthetase,USH3B,HRS

Human Baculovirus Insect Cells
HARS/HisRS Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.6 kDa and the accession number is P12081-1.
TMPH-00130 Mannosyl-oligosaccharide alpha-1,2-mannosidase 1B Protein, Aspergillus phoenicis, Recombinant (His & Myc)

Aspergillus phoenicis E. coli
Involved in the maturation of Asn-linked oligosaccharides. Progressively trims alpha-1,2-linked mannose residues from Man(9)GlcNAc(2) to produce Man(5)GlcNAc(2). Mannosyl-oligosaccharide alpha-1,2-mannosidase 1B Protein, Aspergillus phoenicis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 61.3 kDa and the accession number is Q12563.
TMPY-02176 Harmonin/USH1C Protein, Human, Recombinant (His)

PDZD7C,PDZ-73,PDZ73,DFNB18A,PDZ-73/NY-CO-38,DFNB18,NY-CO-37,...

Human E. coli
Harmonin, also known as Antigen NY-CO-38 / NY-CO-37, Autoimmune enteropathy-related antigen AIE-75, Protein PDZ-73, Renal carcinoma antigen NY-REN-3, Usher syndrome type-1C protein and USH1C, is a protein that is expressed in small intestine, colon, kidney, eye and weakly in pancreas. USH1C is expressed also in vestibule of the inner ear. USH1C contains 3 PDZ (DHR) domains. USH1C may be involved in protein-protein interaction. Defects in USH1C are the cause of Usher syndrome type 1C (USH1C), als...
TMPH-03372 Sharpin Protein, Rat, Recombinant (His & Myc)

Rat E. coli
Sharpin Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 47.7 kDa and the accession number is Q9EQL9.
TMPH-03485 L-saccharopine oxidase Protein, S. pombe, Recombinant (His & Myc)

Fission yeast E. coli
L-saccharopine oxidase Protein, S. pombe, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 52.2 kDa and the accession number is Q9UTM9.
TMPH-02983 Mumps virus (strain Miyahara vaccine) Hemagglutinin-neuraminidase Protein (His)

MuV E. coli
Attaches the virus to sialic acid-containing cell receptors and thereby initiating infection. Binding of HN protein to the receptor induces a conformational change that allows the F protein to trigger virion/cell membranes fusion.; Neuraminidase activity ensures the efficient spread of the virus by dissociating the mature virions from the neuraminic acid containing glycoproteins. Mumps virus (strain Miyahara vaccine) Hemagglutinin-neuraminidase Protein (His) is expressed in E. coli expression sy...
TMPH-01193 Human cytomegalovirus (HCMV) (strain AD169) Uncharacterized protein UL128 (His)

HHV-5 E. coli
Human cytomegalovirus (HCMV) (strain AD169) Uncharacterized protein UL128 (His) is expressed in E. coli.

重组蛋白

LYVE1 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00533
Species: Human
Expression System: HEK293 Cells
SUC2 Protein, Saccharomyces cerevisiae, Recombinant (His)
Cat.No: TMPY-04932
Species: Saccharomyces cerevisiae
Expression System: P. pastoris (Yeast)
Ribonuclease MC Protein, Momordica charantia, Recombinant (His & Myc)
Cat.No: TMPH-02466
Species: Momordica charantia
Expression System: E. coli
Cyanovirin-N homolog Protein, Ceratopteris richardii, Recombinant (His)
Cat.No: TMPH-00363
Species: Ceratopteris richardii
Expression System: P. pastoris (Yeast)
Autolysin Protein, Chlamydomonas reinhardtii, Recombinant (His & SUMO)
Cat.No: TMPH-00395
Species: Chlamydomonas reinhardtii
Expression System: E. coli
HARS/HisRS Protein, Human, Recombinant (His)
Cat.No: TMPY-05413
Species: Human
Expression System: Baculovirus Insect Cells
Mannosyl-oligosaccharide alpha-1,2-mannosidase 1B Protein, Aspergillus phoenicis, Recombinant (His & Myc)
Cat.No: TMPH-00130
Species: Aspergillus phoenicis
Expression System: E. coli
Harmonin/USH1C Protein, Human, Recombinant (His)
Cat.No: TMPY-02176
Species: Human
Expression System: E. coli
Sharpin Protein, Rat, Recombinant (His & Myc)
Cat.No: TMPH-03372
Species: Rat
Expression System: E. coli
L-saccharopine oxidase Protein, S. pombe, Recombinant (His & Myc)
Cat.No: TMPH-03485
Species: Fission yeast
Expression System: E. coli
Mumps virus (strain Miyahara vaccine) Hemagglutinin-neuraminidase Protein (His)
Cat.No: TMPH-02983
Species: MuV
Expression System: E. coli
Human cytomegalovirus (HCMV) (strain AD169) Uncharacterized protein UL128 (His)
Cat.No: TMPH-01193
Species: HHV-5
Expression System: E. coli
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼