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71

抑制剂 & 化合物

14

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Cat. No. Product Name Target Signaling Pathways
T38361 GSK717

IL Receptor; NOD Immunology/Inflammation; NF-κB
GSK717 是 NOD2(核苷酸结合寡聚结构域 2) 的选择性抑制剂。它抑制壁酰二肽 (MDP) 诱导的 NOD2 介导的信号转导,抑制 MDP 刺激的 HEK293/hNOD2 细胞分泌 IL-8 (IC50为 400 nM)。
T7123 AMG-47a

VEGFR; p38 MAPK; JAK; Src Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; MAPK; Stem Cells; Tyrosine Kinase/Adaptors
AMG-47a 是具有口服活性的 Lck 抑制剂,IC50值为 0.2 nM。它具有抗炎作用,对 VEGF2、p38α、p38α、Jak3、MLR 和 IL-2的 IC50值分别为 1、3、72、30 和 21 nM。
T4686 Simeprevir

TMC435,西咪匹韦,TMC-435350,Olysio

HCV Protease; SARS-CoV Microbiology/Virology; Proteases/Proteasome
Simeprevir (TMC435) 是一种有效的 HCV NS3/4A 蛋白酶抑制剂,抑制 HCV 复制,EC50 为 7.8 nM。它也是 SARS-CoV-2 3CLpro 抑制剂。
T77761 BMS-502

Others Others
BMS-502 是一种二酰基甘油激酶 (DGK) α 和 ζ 的强效双重抑制剂, 诱导人和小鼠T细胞的免疫反应,阻断 T 细胞中细胞内检查点信号传导。BMS-502 以剂量依赖的方式刺激免疫反应,可用于研究与免疫相关的疾病。
T21608L β-Interleukin I (163-171), human Acetate

β-Interleukin I (163-171), human Acetate(106021-96-9 Free base)

Others Others
β-Interleukin I (163-171), human Acetate 是一种参与调节免疫反应、炎症反应和造血的肽。
T76699 Sabatolimab

MBG453,NVP-MBG453

Others Others
Sabatolimab (MBG453) 是一种靶向 TIM-3的人源化 IgG4 (S228P) 抗体,是一种有效的调节适应性和先天免疫反应的抑制性受体。Sabatolimab 具有潜在的免疫抑制活性,可选择性与免疫细胞和骨髓细胞上的 TIM-3 结合。
T14513 BBIQ

TLR Immunology/Inflammation
BBIQ 是一种有效且选择性的 toll 样受体 7 (TLR7) 激动剂,对人 TLR7 的 EC50 为 59.1 nM。BBIQ 还是一种功能强大的疫苗佐剂,可增强机体的先天免疫应答。
T50068 2-[(2S,5S)-5-(carbamoylmethyl)-3,6-dioxopiperazin-2-yl]acetamide

Others Others
2-[(2S,5S)-5-(carbamoylmethyl)-3,6-dioxopiperazin-2-yl]acetamide 是一种用作分子结构单元的化合物,为环状二肽。它可以诱导细胞凋亡、抑制细胞增殖和调节免疫反应,具有广泛的生物活性,包括抗肿瘤、抗真菌、抗细菌、抗病毒和免疫条件活性等。
T6964 Resiquimod

R848,雷西莫特,S28463

HCV Protease; TLR Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Resiquimod (R848) 是一种 Toll 样受体7/8的激动剂,可诱导细胞因子上调。
T3614 Inosine pranobex

Groprinosin,Isoprinosine,异丙肌苷,Immunovir,Delimmun

IL Receptor; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Inosine pranobex (Delimmun) 是一种免疫增强剂,它是一种广谱抗病毒剂,用于 HIV 感染。
T78362 Transglutaminase

TG

Transglutaminase (TG) 是一种硫醇酶,促使蛋白质分子间交联,通过催化谷氨酰胺残基的γ-羧酰胺基团与其他化合物的一级ε-胺基团形成异肽键。该酶在包括凝血、抗菌免疫反应和光合作用在内的多种生理过程中发挥作用。
T10865 Cot inhibitor-1

TNF; MAPK Apoptosis; MAPK
Cot inhibitor-1 是一种选择性的 Cot 蛋白激酶(也被称为 Tpl2或 MAP3K8)抑制剂(IC50 为 28 nM)。Cot inhibitor-1 抑制人全血中 TNF-alpha 的产生,其 IC50 为 5.7 nM。Cot 参与多种细胞信号通路,特别是与炎症和免疫反应有关的信号通路。Cot inhibitor-1抑制 Cot 活性,可能对类风湿关节炎、炎症性肠病和某些类型的癌症具有潜在的治疗效果。
T28708 Sch 24937

Sch 24937 is a potent immunosuppressant on B lymphocyte mediated immune responses.
T61110 UC-1V150

UC-1V150 is a distinct TLR7 agonist, which activates cellular immune responses and exhibits anti-tumor effects. It also serves as a precursor for the synthesis of ISAC molecules, known as immune-stimulating antibody conjugates [1] [2].
T25319 Diacetylsplenopentin HCl

Diacetylsplenopentin hydrochloride

Diacetylsplenopentin HCl is used as a synthetic immunomodulator that affects the proliferation and differentiation of bone marrow stem cells without stimulating pathological immune responses beyond the balance of the immune system. This effect is specific
T27099 CU-3

CU 3,CU3

CU-3 is a potent and selective inhibitor of diacylglycerol kinase alpha (DGKalpha). CU-3 attenuates cancer cell proliferation and simultaneously enhances immune responses including anti-cancer immunity.
T34026 Phevamine A

PHVA

Others Others
Phevamine A (PHVA) 是植物免疫反应的抑制剂。
T38614 TLR7 agonist 3

TLR7 agonist 3 (Compound 2), a potent activator of toll-like receptor 7 (TLR7), plays a critical role in initiating immune responses, positioning it as a promising target for immunomodulator development.
T40452 N-Acetylpsychosine

N-Acetylpsychosine,C2 Galactosylceramide (d18:1/2:0)

N-Acetylpsychosine, also known as α-galactosylated C2-ceramide (d18:1/2:0), exhibits immunostimulatory properties. This compound, N-Acetylpsychosine, holds potential as a valuable tool for studying the mechanisms of apoptosis and immune responses activated by dendritic cells (DCs).
T73990 Lipid M

Lipid M (pKa: 6.75) 可用于递送 mRNA 疫苗,引发强大的免疫反应并提高耐受性。
T74872 ODN 105870

ODN 105870 是一种 G 修饰的抑制性寡核苷酸 (INH-ODN),是一种选择性 TLR7抑制剂。ODN 105870 可用于炎症免疫反应研究。
T80131 C5a Anaphylatoxin (human)

Complement System Immunology/Inflammation
C5a Anaphylatoxin (human)为促炎多肽及白细胞化学引诱剂,主要应用于炎症与免疫领域研究,例如过敏性哮喘。
T39292 NS2 (114-121), Influenza

NS2 (114-121), Influenza

NS2 (114-121), Influenza, is a fragment derived from the nonstructural protein 2 (NS2) of the influenza virus. This compound serves as an epitope for influenza research and can be utilized to study the CD8+ cytotoxic T lymphocyte (CTL) in antiviral immune responses.
T14035 3M-011

TLR Immunology/Inflammation
3M-011, a potent dual toll-like receptor TLR7/8 agonist and cytokine inducer, serves as a powerful adjuvant to radiotherapy, eliciting significant local and systemic immune responses. Additionally, it effectively inhibits H3N2 influenza viral replication in the nasal cavity and exhibits strong antitumor activity[1][2][3].
T40216 PTPN22-IN-1

PTPN22-IN-1

PTPN22-IN-1 is a potent PTPN22 inhibitor ( IC 50 =1.4 μM; K i =0.50 μM). PTPN22-IN-1 exhibits >7-10 fold selectivity for PTPN22 over similar phosphatases. PTPN22-IN-1 augments antitumor immune responses. From WO2021007491A1 compound L-1.
T13667 Dusquetide TFA (931395-42-5 free base)

SGX942 TFA,Dusquetide TFA

Others Others
Dusquetide TFA is a kind of innate defense regulator (IDR).Dusquetide TFA has been shown to be active in reducing inflammation and increasing clearance of bacterial infections.Dusquetide TFA regulates innate immune responses to PAMPs and DAMPs in combinat
T82142 Hymenistatin I

Hymenistatin I,一种环八肽[c-(-Pro-Pro-Tyr-Val-Pro-Leu-Ile-ile-Ile-)],具有免疫抑制活性,影响体液和细胞免疫应答。
T69834 Tivumecirnon

FLX475

Tivumecirnon (FLX475) 是一种有效的 CCR4拮抗剂,可以阻断干扰有效抗肿瘤免疫反应的调节性 T 细胞,具有抗肿瘤活性。
T77775 TP-1454

TP-1454是一种针对PKM2的激活剂,其生化测定的AC50为10 Nm。它可通过作用于T调节细胞来调控肿瘤的免疫反应。
T76748 Foralumab

Foralumab(NI-0401)为口服有效的人源化单克隆抗体,针对CD3进行靶向。其能够调控NSG小鼠体内,由人类造血干细胞重建的人类细胞的免疫反应。
T79927 Pectate Lyase

Pectate Lyase为植物病原菌分泌的关键酶,主要功能包括在果胶降解和真菌毒力形成中发挥作用。此外,Pectate Lyase还能诱导植物的免疫反应并参与其毒力过程。
T74873 ODN 105871

ODN 105871,一种G修饰的抑制性寡核苷酸(INH-ODN),作为选择性TLR7抑制剂,适用于炎症免疫反应的研究。
T74584 5-Methylcytidine 5′-triphosphate

5-Methylcytidine 5′-triphosphate (5-Methyl-CTP) 为修饰核苷三磷酸,用以替代未修饰 mRNA,以增强翻译性能与稳定性,显著降低人类及其他哺乳动物细胞的先天免疫反应。
T81022 Tegoprubart

Tegoprubart为针对CD40配体(CD40L)的单克隆抗体,该配体为共刺激介质的核心。通过抑制CD40L,可减弱细胞与抗体介导的免疫反应,促进免疫环境趋向耐受性。在移植动物模型中,Tegoprubart已展现出体内活性。
T27638 Israpafant

Y-24180,Y 24180,Y24180

Israpafant is a selective antagonist for the platelet-activating factor receptor ( IC50 = 0.84nM). Israpafant inhibits PAF-induced human platelet aggregation. Israpafant inhibits the activation of eosinophil cells and consequently delays the development o
T82858 Bleselumab

ASKP 1240,Anti-Human CD40 Recombinant Antibody

Bleselumab (ASKP 1240)为人源化抗-CD40单克隆抗体,通过高亲和力(Kd: 0.24 nM)与CD40结合,阻断CD40与CD40L配体的相互作用,从而抑制免疫反应,用于预防器官移植排斥。
T73659 HLF1-11

HLF1-11,一种人乳铁蛋白衍生肽,是一种广谱抗菌剂。HLF1-11 抑制MPO(human) 的活性。HLF1-11 还使GM-CSF 驱动的单核细胞向巨噬细胞分化,并增强其免疫反应。
T76241 Trichomide A

Trichomide A 是一种有效的 SHP2激活剂。Trichomide A 是一种天然的环缩肽。Trichomide A 在 Con A 激活的 T 细胞中对激活的 T 淋巴细胞介导的免疫反应具有免疫抑制活性。Trichomide A 具有研究免疫相关皮肤病的潜力。
T74268 STING agonist-13

STINGagonist-13 是一种STING 激动剂,通过STING 介导的免疫激活进行癌症免疫。STINGagonist-13 可刺激STING 下游信号传导并促进 I 型干扰素免疫反应。STINGagonist-13 能显著降低肿瘤体积并具有免疫记忆衍生的癌症抑制活性。
T79320 Antitumor agent-114

STING Immunology/Inflammation
Antitumor agent-114为一种强效STING激动剂,具有激活免疫功能并在乳腺癌小鼠模型中缩减肿瘤体积的作用,适用于免疫与癌症疾病研究之用。
T74706 Vidutolimod

Vidutolimod 是一种CpG-A 类寡核苷酸,是TLR9的激动剂。Vidutolimod 激活浆细胞样树突状细胞(pDCs)并触发IFNα的释放,导致抗肿瘤免疫作用。
T68383 BIIB028

BIIB028 is a small-molecule inhibitor of heat shock protein (Hsp) 90 with potential antineoplastic activity. Hsp90 inhibitor BIIB028 blocks the binding of oncogenic client proteins to Hsp90, which may result in the proteasomal degradation of these proteins and so the inhibition of tumor cell proliferation. Hsp90 is a molecular chaperone that plays a key role in the conformational maturation of oncogenic signaling proteins, such as Her2/Erbb2, Akt, Raf1, Bcr-Abl, and mutated p53, in addition to o...
T79488 RNase L-IN-1

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
RNase L-IN-1(compound 17a)为RNase L的特异性抑制剂,能有效地防止该酶降解RNA,从而抑制病毒复制,并对先天性免疫反应及炎症过程具调控作用。
T74585 5-Methylcytidine 5′-triphosphate trisodium

5-Methylcytidine 5′-triphosphate (5-Methyl-CTP) trisodium 为一种修饰核苷三磷酸,可用以替换原生mRNA,进而提升翻译效率与稳定性,同时在人类及其他哺乳动物细胞中显著降低先天免疫反应。
T82793 Caerin 1.1 TFA

Apoptosis Apoptosis
Caerin 1.1 TFA 是澳大利亚树蛙Litoria腺体分泌物中分离出的宿主防御肽,具有抑制 HeLa 细胞增殖及介导细胞凋亡 (apoptosis) 的能力,并可能促进适应性 T 细胞免疫反应。
T76786 Cabiralizumab

Cabiralizumab (FPA 008) 是一种抗 CSF1R 单克隆抗体 (MAb)。Cabiralizumab 可增强 T 细胞浸润和抗肿瘤 T 细胞免疫反应。Cabiralizumab 抑制破骨细胞的活化并阻止骨质破坏,可用于类风湿性关节炎 (RA) 的研究。Cabiralizumab 可与 Nivolumab 结合用于肺癌研究。
T74910 ODN 24888

ODN 24888 是一种鸟嘌呤修饰的抑制性寡核苷酸 (INH-ODN),对TLR7/TLR9介导的信号通路表现出强烈的抑制作用。ODN 24888 损害 IFN-α 水平和NF-κB 激活,抑制IL-6的释放。ODN 24888 参与免疫和炎症应答,可作为疫苗佐剂使用。
T74905 ODN 2007

ODN 2007是一种B类CpG ODN(寡脱氧核苷酸),兼具Toll样受体(TLR)配体功能。作为免疫调节剂和疫苗佐剂,它能够增强哺乳动物、鱼类及人类的免疫反应。其序列为5'-TCGTCGTTGTCGTTTTGTCGTT-3'。
T80761 XQ2B

XQ2B为cGAS抑制剂,针对蛋白质-DNA相互作用及其相分离。该化合物可阻止单纯疱疹病毒1(HSV-1)触发的抗病毒免疫响应,在体外与体内都能增强HSV-1的感染效果。
T74693 CDN-A

CDN-A为一种环二核苷酸,主要用于抗体-活性分子偶联物(ADC)的合成。作为先天免疫及适应性免疫反应的关键激活剂,环状二核苷酸能由内源性外来DNA或侵入性细菌病原体生成,在人体内通过促进干扰素基因表达激活先天免疫系统。

化合物

GSK717
Cat.No: T38361
Synonym:
Target: IL Receptor, NOD
AMG-47a
Cat.No: T7123
Synonym:
Target: VEGFR, p38 MAPK, JAK, Src
Simeprevir
Cat.No: T4686
Synonym: TMC435,西咪匹韦,TMC-435350,Olysio
Target: HCV Protease, SARS-CoV
BMS-502
Cat.No: T77761
Synonym:
Target: Others
β-Interleukin I (163-171), human Acetate
Cat.No: T21608L
Synonym: β-Interleukin I (163-171), human Acetate(106021-96-9 Free base)
Target: Others
Sabatolimab
Cat.No: T76699
Synonym: MBG453,NVP-MBG453
Target: Others
BBIQ
Cat.No: T14513
Synonym:
Target: TLR
2-[(2S,5S)-5-(carbamoylmethyl)-3,6-dioxopiperazin-2-yl]acetamide
Cat.No: T50068
Synonym:
Target: Others
Resiquimod
Cat.No: T6964
Synonym: R848,雷西莫特,S28463
Target: HCV Protease, TLR
Inosine pranobex
Cat.No: T3614
Synonym: Groprinosin,Isoprinosine,异丙肌苷,Immunovir,Delimmun
Target: IL Receptor, HIV Protease
Transglutaminase
Cat.No: T78362
Synonym: TG
Target:
Cot inhibitor-1
Cat.No: T10865
Synonym:
Target: TNF, MAPK
Sch 24937
Cat.No: T28708
Synonym:
Target:
UC-1V150
Cat.No: T61110
Synonym:
Target:
Diacetylsplenopentin HCl
Cat.No: T25319
Synonym: Diacetylsplenopentin hydrochloride
Target:
CU-3
Cat.No: T27099
Synonym: CU 3,CU3
Target:
Phevamine A
Cat.No: T34026
Synonym: PHVA
Target: Others
TLR7 agonist 3
Cat.No: T38614
Synonym:
Target:
N-Acetylpsychosine
Cat.No: T40452
Synonym: N-Acetylpsychosine,C2 Galactosylceramide (d18:1/2:0)
Target:
Lipid M
Cat.No: T73990
Synonym:
Target:
ODN 105870
Cat.No: T74872
Synonym:
Target:
C5a Anaphylatoxin (human)
Cat.No: T80131
Synonym:
Target: Complement System
NS2 (114-121), Influenza
Cat.No: T39292
Synonym: NS2 (114-121), Influenza
Target:
3M-011
Cat.No: T14035
Synonym:
Target: TLR
PTPN22-IN-1
Cat.No: T40216
Synonym: PTPN22-IN-1
Target:
Dusquetide TFA (931395-42-5 free base)
Cat.No: T13667
Synonym: SGX942 TFA,Dusquetide TFA
Target: Others
Hymenistatin I
Cat.No: T82142
Synonym:
Target:
Tivumecirnon
Cat.No: T69834
Synonym: FLX475
Target:
TP-1454
Cat.No: T77775
Synonym:
Target:
Foralumab
Cat.No: T76748
Synonym:
Target:
Pectate Lyase
Cat.No: T79927
Synonym:
Target:
ODN 105871
Cat.No: T74873
Synonym:
Target:
5-Methylcytidine 5′-triphosphate
Cat.No: T74584
Synonym:
Target:
Tegoprubart
Cat.No: T81022
Synonym:
Target:
Israpafant
Cat.No: T27638
Synonym: Y-24180,Y 24180,Y24180
Target:
Bleselumab
Cat.No: T82858
Synonym: ASKP 1240,Anti-Human CD40 Recombinant Antibody
Target:
HLF1-11
Cat.No: T73659
Synonym:
Target:
Trichomide A
Cat.No: T76241
Synonym:
Target:
STING agonist-13
Cat.No: T74268
Synonym:
Target:
Antitumor agent-114
Cat.No: T79320
Synonym:
Target: STING
Vidutolimod
Cat.No: T74706
Synonym:
Target:
BIIB028
Cat.No: T68383
Synonym:
Target:
RNase L-IN-1
Cat.No: T79488
Synonym:
Target: DNA/RNA Synthesis
5-Methylcytidine 5′-triphosphate trisodium
Cat.No: T74585
Synonym:
Target:
Caerin 1.1 TFA
Cat.No: T82793
Synonym:
Target: Apoptosis
Cabiralizumab
Cat.No: T76786
Synonym:
Target:
ODN 24888
Cat.No: T74910
Synonym:
Target:
ODN 2007
Cat.No: T74905
Synonym:
Target:
XQ2B
Cat.No: T80761
Synonym:
Target:
CDN-A
Cat.No: T74693
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T13502 3-Oxo-5β-cholanoic acid

3-氧代-5β-胆烷酸,Dehydrolithocholic acid

ROR Metabolism
3-Oxo-5β-cholanoic acid (Dehydrolithocholic acid) 是胆汁酸的一种代谢产物。3-Oxo-5β-cholanoic acid 直接与关键转录因子RORγt(Kd=1.13 μM) 结合抑制TH17细胞分化。
TN2088 Platycodin D2

桔梗皂苷D2

IL Receptor; HBV Immunology/Inflammation; Microbiology/Virology
Platycodin D2 是分离自桔梗的皂苷类物质,显示除抗癌活性。
T0948L Corticosterone

皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Corticosterone (Kendall's compound B) 是一种肾上腺皮质类固醇,有盐皮质激素和糖皮质激素的活性,具有口服活性。Corticosterone 参与体内能量、免疫反应和应激反应的调节。
T5S0993 Kurarinone

苦参酮,苦参黄素

BCL; Others; IκB/IKK; TNF; NF-κB; JAK; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; NF-κB; Others; Stem Cells
Kurarinone 是从灌木苦参中提取的黄酮类化合物,具有抗肿瘤、雌激素和抗炎活性,对免疫反应也有很强的抑制作用。
T67710 3-Indoleacrylic acid

Endogenous Metabolite Metabolism
3-Indoleacrylic acid 是由链球菌属产生的色氨酸的代谢产物。3-Indoleacrylic acid 对肠上皮屏障功能有有益作用,并减轻免疫细胞的炎症反应。
T5731 1-Kestose

蔗果三糖,1-蔗果三糖

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
1-Kestose 是低聚果糖成分,有效刺激了 Faecalibacterium prausnitzii 和 Bifidobacteria。它有抗羟基自由基的潜力。它可促进肠道内乳酸菌数量,影响微生物以及肠道和全身免疫反应。
TN1879 Lucideric acid A

Lucidenic acid A,赤芝酸A

MMP; p38 MAPK; JNK MAPK; Proteases/Proteasome
Lucideric acid A (Lucidenic acid A) 是分离自灵芝的天然产物,可抑制 PMA 诱导的MMP-9活性,具有抵抗肝癌细胞侵袭的作用。
T1614 Hydrocortisone

氢化可的松,Cortisol

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Hydrocortisone (Cortisol) 是一种糖皮质激素,由肾上腺素皮质分泌。Hydrocortisone 激动糖皮质激素受体,可促进蛋白质分解代谢、糖异生、毛细血管壁稳定性、肾脏钙排泄,并抑制免疫和炎症反应。
T5S1895 Norisoboldine

Laurelliptine,去甲异波尔定,(+)-Laurelliptine

MAPK; Adenosine Receptor GPCR/G Protein; MAPK; Neuroscience
Norisoboldine ((+)-Laurelliptine) 是一种可口服的芳基烃受体激动剂,是乌药中主要的异喹啉类生物碱,可用于类风湿性关节炎和溃疡性结肠炎的研究。
T4928 L-Kynurenine

L-犬尿氨酸,(S)-Kynurenine

AhR; Aryl Hydrocarbon Receptor; Endogenous Metabolite Immunology/Inflammation; Metabolism
L-Kynurenine ((S)-Kynurenine) 是L-色氨酸的代谢物,是芳香烃受体激动剂,可抑制同种异体 T 细胞增殖并增加恶性 U87 神经胶质瘤细胞侵入胶原基质。
T3386 Kaempferitrin

Lespedin,Kaempferol,Lespenephryl,Lespenefril,Kaempferol 3,7-dirhamnoside,山奈苷

cell cycle arrest; Glucokinase; IGF-1R Cell Cycle/Checkpoint; Metabolism; Tyrosine Kinase/Adaptors
Kaempferitrin (Lespenephryl) 是天然黄酮苷类化合物,具有缓解疼痛、抗糖尿病、消炎、抗肿瘤和化疗作用,可激活胰岛素信号传导。
TN4804 Platycoside A

Antifection Microbiology/Virology
Platycoside A has hemolytic activity and adjuvant potential on the immune responses to Newcastle disease virus-based recombinant avian influenza vaccine. It induces the IgG and IgG1 antibody responses in the immunized mice.
TN2181 Sarmentosin

Others Others
Sarmentosin significantly lowers the SGPT level of patients suffering from chronic viral hepatitis, and shows a suppressive effect on cell-mediated immune responses in mice. It shows a good effect in lowering serum glutamate-pyruvate transaminase.
T38838 QS-21

Stimulon,QS-21

QS-21, an immunostimulatory saponin, is a powerful vaccine adjuvant that stimulates both Th2 humoral and Th1 cell-mediated immune responses by interacting with antigen presenting cells (APCs) and T cells. Additionally, QS-21 activates the NLRP3 inflammasome, leading to the release of cytokines IL-1β and IL-18, which are dependent on caspase-1.

天然产物

3-Oxo-5β-cholanoic acid
Cat.No: T13502
Synonym: 3-氧代-5β-胆烷酸,Dehydrolithocholic acid
Target: ROR
Platycodin D2
Cat.No: TN2088
Synonym: 桔梗皂苷D2
Target: IL Receptor, HBV
Corticosterone
Cat.No: T0948L
Synonym: 皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)
Target: Glucocorticoid Receptor, Endogenous Metabolite
Kurarinone
Cat.No: T5S0993
Synonym: 苦参酮,苦参黄素
Target: BCL, Others, IκB/IKK, TNF, NF-κB, JAK, STAT
3-Indoleacrylic acid
Cat.No: T67710
Synonym:
Target: Endogenous Metabolite
1-Kestose
Cat.No: T5731
Synonym: 蔗果三糖,1-蔗果三糖
Target: Others, Endogenous Metabolite, Antibacterial
Lucideric acid A
Cat.No: TN1879
Synonym: Lucidenic acid A,赤芝酸A
Target: MMP, p38 MAPK, JNK
Hydrocortisone
Cat.No: T1614
Synonym: 氢化可的松,Cortisol
Target: Glucocorticoid Receptor, Endogenous Metabolite
Norisoboldine
Cat.No: T5S1895
Synonym: Laurelliptine,去甲异波尔定,(+)-Laurelliptine
Target: MAPK, Adenosine Receptor
L-Kynurenine
Cat.No: T4928
Synonym: L-犬尿氨酸,(S)-Kynurenine
Target: AhR, Aryl Hydrocarbon Receptor, Endogenous Metabolite
Kaempferitrin
Cat.No: T3386
Synonym: Lespedin,Kaempferol,Lespenephryl,Lespenefril,Kaempferol 3,7-dirhamnoside,山奈苷
Target: cell cycle arrest, Glucokinase, IGF-1R
Platycoside A
Cat.No: TN4804
Synonym:
Target: Antifection
Sarmentosin
Cat.No: TN2181
Synonym:
Target: Others
QS-21
Cat.No: T38838
Synonym: Stimulon,QS-21
Target:
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