103
6
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T17030 |
Tegoprazan
|
ATPase; Proton pump | Membrane transporter/Ion channel |
Tegoprazan 是一种口服有效的、高选择性胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,能够控制胃酸分泌和运动,在体外检测的对猪、犬、人的 H+/K+-ATP 酶的 IC50为0.29-0.52 μM。 | |||
T38612 |
Linaprazan glurate
|
Others | Others |
Linaprazan glurate 抑制外源性或内源性刺激的胃酸分泌。 Linaprazan glurate 可用于胃肠道炎症性疾病和消化性溃疡疾病的研究。 | |||
T22724 |
Dimaprit dihydrochloride
|
NOS; NO Synthase; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Dimaprit dihydrochloride 是组胺H2受体的一种选择性激动剂,可刺激胃酸的分泌。它还抑制nNOS,IC50值为 49 μM。 | |||
T4579 |
Pentagastrin
五肽胃泌素,ICI-50123 |
Others; cholecystokinin | GPCR/G Protein; Others |
Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂,IC50=11 nM。它能够增强胃粘膜对酸的防御机制,并保护胃粘膜免受损伤。 | |||
T4981 |
Anisotropine Methylbromide
|
Prostaglandin Receptor; AChR | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Anisotropine Methylbromide 是一种抗胆碱能药物,已用于缓解胃肠道痉挛和抑制胃酸分泌。 | |||
T0498 |
Salsalate
Disalicylic acid,Salicylsalicylic acid,Sasapyrine,NSC-49171,双水杨酸酯 |
Reactive Oxygen Species; COX | Immunology/Inflammation; Metabolism; Neuroscience; NF-κB |
Salsalate (Sasapyrine) 是一种有效的抗风湿药物,是一种非乙酰化水杨酸盐,可以绕过胃的吸收,也可以避免环氧合酶的抑制。它具有抗炎活性,降低血糖水平、胰岛素抵抗和细胞因子表达,可用于研究 2 型糖尿病。 | |||
T8599 |
Betazole dihydrochloride
盐酸倍他唑,Betazole hydrochloride |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Betazole dihydrochloride (Betazole hydrochloride) 是吡唑类组胺,是一种口服活性 H2受体激动剂,能诱导胃酸分泌,导致胆总管压力立即显著升高。它作为一种诊断剂,用于研究胃酸分泌能力。 | |||
T1756L |
Ilaprazole
IY81149,艾普拉唑,IY 81149,IY-81149 |
Proton pump; TOPK | MAPK; Membrane transporter/Ion channel |
Ilaprazole (IY-81149) 是一种具有口服活性质子泵抑制剂,以剂量依赖性方式不可逆地抑制H+/K+-ATPase,在兔壁细胞制剂中的IC50为 6 μM。它也是一种有效的T 细胞起源蛋白激酶(TOPK)抑制剂,用于胃溃疡的研究。 | |||
T0686 |
Orlistat
Ro-18-0647,奥利司他,Tetrahydrolipstatin |
Apoptosis; Others; Fatty Acid Synthase | Apoptosis; Metabolism; Others |
Orlistat (Tetrahydrolipstatin) 是一种不可逆的胰腺和胃脂肪酶抑制剂,也是一种脂肪酸合成酶抑制剂,可研究肥胖症,具有抗动脉粥样硬化作用。 | |||
T6700 |
Tenatoprazole
泰妥拉唑,TU-199 |
Proton pump | Membrane transporter/Ion channel |
Tenatoprazole (TU-199) 是一种口服有效的,基于咪唑吡啶的质子泵抑制剂。它抑制猪胃H+/K+-ATP 酶活性,IC50为6.2 μM。它阻断泛素与 ESCRT-1 因子 Tsg101 的相互作用,抑制几种包膜病毒的产生,包括 EBV。 | |||
T1756 |
Ilaprazole sodium
IY-81149 sodium,艾普拉唑钠 |
Proton pump; TOPK | MAPK; Membrane transporter/Ion channel |
Ilaprazole sodium (IY-81149 sodium) 是一种具有口服活性质子泵抑制剂,以剂量依赖性方式不可逆地抑制 H+/K+-ATPase,在兔壁细胞制剂中的 IC50为 6 μM。它也是一种有效的 T 细胞起源蛋白激酶(TOPK)抑制剂,用于胃溃疡的研究。 | |||
T8388 |
Vonoprazan
TAK-438 (free base),沃诺拉赞 |
Proton pump | Membrane transporter/Ion channel |
Vonoprazan (TAK-438 (free base)) 是一种质子泵抑制剂,是口服活性钾竞争性酸阻断剂,有抗分泌作用。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50值为 19 nM。它可用于研究胃酸相关疾病。 | |||
T0674 |
Lansoprazole
兰索拉唑,A-65006,AG-1749 |
Proton pump; Phospholipase; Antibacterial | Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Lansoprazole (A-65006) 是一种可抑制胃酸生成的质子泵抑制剂。它是中性鞘磷脂酶的外泌体抑制剂。 | |||
T21254 |
Vonoprazan Fumarate
TAK-438,TAK 438,Vonoprazan Fumurate,TAK438,富马酸沃诺拉赞 |
Proton pump | Membrane transporter/Ion channel |
Vonoprazan Fumarate (TAK438) 是质子泵的有效抑制剂,是口服有效的高效钾竞争性酸阻断剂,具有抗分泌活性。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50为 19 nM。它被开发用于研究酸相关疾病,如消化性溃疡和胃食管反流病。 | |||
T7615 |
Xenopsin
爪蟾肽,Xenopsin(2TFA) |
Others | Others |
Xenopsin (Xenopsin(2TFA)) 是一种神经降压素样八肽,来自于非洲爪蟾皮肤,能够抑制胃泌素刺激的胃酸分泌。 | |||
T15005 |
CP-66948
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
CP-66948 是一种有效的 histamine H2 受体拮抗剂,对胃酸分泌有抑制作用,可用于保护胃黏膜和肠粘膜。 | |||
T13145 |
Thiazolidinone-Derivatives-1
|
Others | Others |
Thiazolidinone-Derivatives-1 抑制胃酸分泌,可用于研究胃和十二指肠溃疡的治疗。 | |||
T1627 |
Famotidine
MK-208,法莫替丁 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Famotidine (MK-208) 是一种具有抗酸活性的丙脒和组胺 H2 受体拮抗剂。 | |||
TP1309 |
Gastric mucin
|
Antibacterial; Antibiotic | Microbiology/Virology |
Gastric mucin 是一种能保护胃肠道免受酸、蛋白酶、致病微生物和机械创伤影响的糖蛋白。 | |||
T0081 |
Lafutidine
拉呋替丁,FRG-8813 |
5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Lafutidine (FRG-8813) 是一种组胺受体 H2RA 拮抗剂,可抑制胃酸分泌,具有胃粘膜保护作用,可用于研究胃食管反流疾病。 | |||
T10221 |
Abeprazan hydrochloride
DWP14012 hydrochloride,Fexuprazan hydrochloride |
Proton pump | Membrane transporter/Ion channel |
Abeprazan hydrochloride (Fexuprazan hydrochloride) 是一种有效的、可逆的、具有口服活性的potassium-competitive acid 阻滞剂,通过竞争性的与钾离子结合抑制 H+,K+- ATPase,而无需酸激活。Abeprazan hydrochloride 是一种质子泵抑制剂(PPI),通过减少胃酸的产生而起作用,可用于治疗胃酸相关疾病,如胃食管反流病(GERD)和消化性溃疡。 | |||
T20561L |
BPC 157 acetate(137525-51-0 free base)
BPC157 acetate,BPC-157 acetate,Bpc 15 acetate,Bpc15 acetate,Bpc-15 acetate |
Others | Others |
BPC 157 acetate(137525-51-0 free base) 是一种具有保肝作用的胃肽 (BPC) 的 15 个氨基酸片段。 | |||
TP2030L1 |
Gastrin I (human) acetate
Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐 |
cholecystokinin | GPCR/G Protein |
Gastrin I (human) acetate (Gastrin-17 acetate) 是在胃中产生的内源性肽,通过胆囊收缩素 2 (CCK2) 受体增加胃酸分泌。 | |||
T0157 |
Roxatidine Acetate hydrochloride
HOE 760,盐酸罗沙替丁醋酸酯,Roxatidine Acetate HCl |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Roxatidine Acetate hydrochloride (HOE 760) 是一种特异性和竞争性的组胺 H2 受体拮抗剂,能抑制胃酸分泌,可用于胃溃疡和十二指肠溃疡的研究。 | |||
T0797 |
Cimetidine
西米替汀,SKF-92334,西咪替丁 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Cimetidine (SKF-92334) 是一种可口服的可逆组胺H2受体拮抗剂,Ki 为 0.6 μM。它抑制胃酸分泌,以及胃蛋白酶和胃泌素的输出,具有抗癌和抗炎活性。 | |||
TP1705 |
Gastrin I (1-14), human
|
Others | Others |
Gastrin I (1-14), human 是人胃泌素 I 肽的 1-14 片段。其中Gastrin I 是内源性胃肠肽激素。Gastrin 是胃酸分泌的主要激素调节剂。 | |||
T37588L |
GIP (1-30) amide, porcine acetate
|
IGF-1R | Tyrosine Kinase/Adaptors |
GIP (1-30) amide, porcine acetate 是完全葡萄糖依赖性促胰岛素多肽 (GIP) 受体的激动剂。它可弱抑制胃酸分泌,强烈刺激胰岛素。 | |||
T6929 |
Pantoprazole sodium
Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc |
Apoptosis; Others; Proton pump; HIF; Autophagy | Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Others |
Pantoprazole sodium (Pantecta) 是一种具有口服活性的质子泵抑制剂,是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,IC50为 6.8 μM。它可以改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。 | |||
T68016 |
Spiroglumide
CR-2194 |
cholecystokinin | GPCR/G Protein |
Spiroglumide 是一种CCKB-胃泌素拮抗剂,能够抑制剂量依赖性五肽胃泌素诱导的酸分泌过多,其ID50为20.1(8.67-46.4)mg / kg,可用于探索胃泌素在调节人类胃酸分泌中的生理作用。 | |||
TP2018L |
GIP (human) acetate
GIP (human) acetate(100040-31-1 Free base) |
IGF-1R | Tyrosine Kinase/Adaptors |
GIP (human) acetate 是葡萄糖依赖性胰岛素分泌的刺激剂和胃酸分泌的弱抑制剂。 GIP (human) acetate 在脂质代谢和肥胖的发展中起着至关重要的作用。 | |||
T1467 |
Acemetacin
阿西美辛,K-708,TVX 1322 |
COX | Immunology/Inflammation; Neuroscience |
Acemetacin (TVX 1322) 是一种非甾体抗炎类的化合物。 | |||
T22391 |
Omeprazole Sodium
|
P450; Proton pump; Antibacterial; Autophagy | Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Omeprazole 是有效的质子泵抑制剂,在胃肠道疾病的研究中具有价值。它竞争性抑制CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阴性菌和革兰氏阳性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。 | |||
T16865 |
SCH28080
|
ATPase; Proton pump | Membrane transporter/Ion channel |
SCH28080 是一种可逆且具有 K+ 竞争性的胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,IC50 值为 20 nM (家兔微粒体膜)。SCH28080 在体内是有效的酸分泌抑制剂,具有抗溃疡活性、抗分泌和细胞保护活性。 | |||
T2686 |
Esomeprazole Magnesium
(S)-Omeprazole magnesium,NEXIUM,埃索美拉唑镁,(-)-Omeprazole magnesium |
ATPase; Proton pump | Membrane transporter/Ion channel |
Esomeprazole Magnesium (NEXIUM) 是一种口服有效的 H+, K+-ATPase 抑制剂,在上消化道疾病和胃食管反流疾病中具有研究价值。Esomeprazole magnesium 是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。 | |||
T21385 |
Cinitapride
西尼必利,Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Cinitapride (Blaston) 是一种促胃药。它减缓肌肉的活动,以减轻诸如胃酸反流、胃排空延迟和溃疡性消化不良等病症的症状。 Cinitapride 作为 5-HT2 受体的拮抗剂和 5-HT1 和 5-HT4 受体的激动剂。 | |||
TP1325L |
Gastrin-Releasing Peptide, human(TFA)
|
Others | Others |
Gastrin-Releasing Peptide, human(TFA) (93755-85-2 free base) 是一种调节性人类肽,可引发胃泌素释放并调节胃酸分泌和肠道运动功能。支配胃G 细胞的迷走神经节后纤维释放GRP,刺激G 细胞释放胃泌素。 | |||
T77599 |
Methyl retinoate
Retinoic acid, methyl ester |
Others | Others |
Methyl retinoate (Retinoic acid, methyl ester) 在体内实验中会诱导给部位发生无菌炎症,会使血液中白细胞数量增加,而红细胞和Hb含量减少。Methyl retinoate 可促进自发性白血病的产生。Methyl retinoate 可用于治疗因维生素A缺乏而产生的胃肥大和溃疡。 | |||
T1083L |
Theophylline monohydrate
Quibron,茶碱一水合物 |
HDAC; PDE; Adenosine Receptor | Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience |
Theophylline monohydrate (Quibron) 似乎抑制磷酸二酯酶和前列腺素的产生,调节钙通量和细胞内钙分布,并拮抗腺苷。茶碱是黄嘌呤的天然生物碱衍生物,从植物山茶花和小粒咖啡中分离出来。在生理上,该药剂可放松支气管平滑肌,产生血管舒张(脑血管除外),刺激中枢神经系统,刺激心肌,利尿,增加胃酸分泌;它还可以抑制炎症并改善横膈膜的收缩性。 | |||
T31958 |
Glycine-pentagastrin
Glycine pentagastrin,Boc-gly-trp-met-asp-phe-NH2,Tbgtmap |
||
Glycine-pentagastrin can enhance gastric mucosal defence mechanisms against acid and protect the gastric mucosa from experimental injury. | |||
T27669 |
JNJ-26070109
JNJ26070109 |
||
JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat. | |||
T27092 |
CS-526
R-105266,R 105266,R105266 |
||
CS-526 is a proton pump inhibitor. The inhibitory mechanism of CS-526 on H+,K+-ATPase was a competitive antagonism to the K+ binding site of H+,K+-ATPase, and it was also a reversible inhibition. CS-526 has a potent antisecretory effect on gastric acid se | |||
T69805 | AU-006 | ||
AU-006 is an anti-ulcer drug which is effective in the treatment of gastric ulcers by inhibiting gastric acid secretion. | |||
T69164 | Dibenamine | ||
Dibenamine is an alpha adrenergic antagonist that blocks basal and histamine-stimulated gastric acid secretion. | |||
T20660 |
Revaprazan
SB-641257,SB 641257,SB641257 |
||
Revaprazan is a novel, selective potassium-competitive acid blocker, to be specific, it reversibly inhibits gastric H(+)/K(+)-ATPase and shows effective acid suppression comparable to PPIs. | |||
T32224 |
Isopropamide
Priazimide,Dipramide,Piaccamide,Chloroisopropamide,Dipramid |
||
Isopropamide (R5) is a long-acting anticholinergic drug. It is used to treat peptic ulcers and other gastrointestinal disorders involving excess gastric acid (gastrointestinal acidosis) and hyperactivity. | |||
T26090 |
Rioprostil
TR 4698,TR4698,Rioprostilum,TR-4698 |
||
Rioprostil is a methyl prostaglandin E1 analog that decreases gastric acid secretion and enhances the gastric mucus-bicarbonate barrier. It is effective in the treatment of gastric ulcers and gives significant protection against NSAID-induced gastric muco | |||
T30250 |
AZD0865
AZD-0865,AZD 0865 |
||
AZD0865 is an effective drug that inhibits gastric H(+), K(+) -ATPase activity and acid formation in vitro, with rapid onset. | |||
T13261 |
CCK-B Receptor Antagonist 1
|
Others | Others |
CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid. | |||
T68200 |
Roxatidine hydrochloride
|
||
Roxatidine hydrochloride is an anti-ulcer agent and histamine antagonist that suppresses gastric acid secretion. It effectively heals duodenal and gastric ulcers and reduces ulcer pain. Roxatidine acetate has an improved safety profile compared to other similar drugs, in part because lower doses of roxatidine acetate are therapeutically effective. | |||
T15722 |
Lavoltidine
Loxtidine,AH-234844 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hypergastrinemia. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3727 |
Methyl syringate
Syringic Acid Methyl Ester,丁香酸甲酯 |
TRP/TRPV Channel | Membrane transporter/Ion channel |
Methyl syringate (Syringic Acid Methyl Ester) 是水仙花蜜的化学标记物,是有效的细菌和真菌漆酶酚介质。它也是TRPA1激动剂。 | |||
T20604L |
Litorin acetate(55749-97-8 Free base)
|
Bombesin Receptor | GPCR/G Protein |
Litorin acetate 是一种两栖类铃蟾肽衍生物,是一种铃蟾肽受体激动剂。它刺激平滑肌收缩,刺激胃泌素、胃酸和胰腺分泌,抑制体内营养。 | |||
TN2601 |
12-O-Methylcarnosic acid
|
Reductase | Endocrinology/Hormones; Metabolism |
12-O-Methylcarnosic acid 是分离自小叶丹参的丙酮提取物的一种二萜肉桂酸,可抑制 5α-还原酶 (5α-reductase) 活性,IC50为 61.7 μM。它抑制 LNCaP 细胞的增殖。它具有抗微生物活性、抗氧化和抗癌活性。 | |||
T2A2532 |
L-Histidine
Glyoxaline-5-alanine,L-(-)-Histidine,L-组氨酸,histidine,组氨酸,L-Hisidine |
Mitochondrial Metabolism; Endogenous Metabolite | Metabolism |
L-Histidine (L-(-)-Histidine) 是人类生长和组织修复所需的一种半必需氨基酸(儿童应从食物中获得)。 L-Histidine 是线粒体谷氨酰胺转运的抑制剂。 | |||
T20604 |
Litorin
|
||
Litorin, an amphibian bombesin peptide derivative, is found to suppress the nutriment, to stimulate the contraction of smooth muscle, to stimulate gastrin, gastric acid, and pancreatic secretion. | |||
TN3740 |
Cyclocommunol
|
PAFR | GPCR/G Protein |
Cyclocommunol exhibits cytotoxicity against hepatocellular carcinoma (SMMC-7721) and gastric carcinoma (BGC-823 and SGC-7901) cell lines. It also shows strong inhibition of arachidonic acid (AA)- and collagen-induced platelet aggregation. |