57
19
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15033 |
Cyproconazole
|
Antibacterial | Microbiology/Virology |
Cyproconazole 是一种三唑类杀菌剂,在农业上用于保护作物免受多种真菌病原体的侵害。 | |||
T4553 |
Procaine penicillin G
普鲁卡因青霉素,Duphapen,Hydracillin,Hostacillin |
Antibiotic | Microbiology/Virology |
Procaine penicillin G (Duphapen) 是一种抗生素,可用于治疗多种细菌感染。具体来说,它用于梅毒、炭疽、口腔感染、肺炎、白喉、蜂窝组织炎和动物咬伤。 | |||
T0018 |
Procainamide hydrochloride
Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺 |
DNA Methyltransferase; Sodium Channel; AChR; Autophagy | Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Neuroscience |
Procainamide hydrochloride (Procapan) 是一种用于研究心律失常的抗心律失常制剂。 | |||
T20625 |
Prochloraz
咪鲜胺,Sporgon,Prelude |
Estrogen Receptor/ERR; AhR; Androgen Receptor; Antifungal | Endocrinology/Hormones; Immunology/Inflammation; Metabolism; Microbiology/Virology |
Prochloraz (Prelude) 是咪唑类抗真菌剂。Prochloraz 抑制羊毛甾醇的细胞色素 P450 依赖性 14α-脱甲基作用,由此抑制麦角固醇的生物合成,从而导致真菌细胞膜破裂和细胞死亡。它也是雌激素受体和 雄激素受体的拮抗剂,IC50分别为25 μM 和4 μM, 并激活芳烃受体,EC50为1μM。 | |||
T0249 |
N-Acetylprocainamide
NAPA,Acecainide,乙酰普卡胺,N-乙酰普鲁卡因胺 |
Potassium Channel; Sodium Channel; Drug Metabolite | Membrane transporter/Ion channel; Metabolism |
N-Acetylprocainamide (NAPA) 是K+通道抑制剂,是第三代抗心律失常剂。 | |||
T0378 |
Oxybuprocaine hydrochloride
Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐 |
Sodium Channel | Membrane transporter/Ion channel |
Oxybuprocaine hydrochloride (Oxybuprocaine HCl) 是可逆的钠通道阻断剂,可防止角膜,结膜和巩膜中疼痛神经的冲动传播。Oxybuprocaine hydrochloride 专用于眼科与耳鼻喉科。 | |||
T7817 |
Aprocitentan
ACT-132577,N-[5-(4-溴苯基)-6-[2-[(5-溴-2-嘧啶基)氧基]乙氧基]-4-嘧啶基]氨基磺酰胺 |
Endothelin Receptor | GPCR/G Protein |
Aprocitentan (ACT-132577) 是一种 Macitentan 的主要活性代谢物。它是 ETA/ETB 的双重拮抗剂,其 pA2值分别为 6.7 和 5.5,IC50分别为 3.4 nM 和 987 nM。 | |||
T6443 |
Chloroprocaine hydrochloride
盐酸氯普鲁卡因,Chloroprocaine HCl |
ATPase; Others | Membrane transporter/Ion channel; Others |
Chloroprocaine hydrochloride (Chloroprocaine HCl) 是一种 Na/K-ATPase 活性抑制剂,IC50为 13 mM,可阻断外周神经。 | |||
T0288 |
Procodazole
2-Benzimidazolepropionic acid,Propazol,丙考达唑 |
Antibacterial | Microbiology/Virology |
Procodazole (2-Benzimidazolepropionic acid) 是一种针对病毒和细菌感染的非特异性活性免疫保护剂。 | |||
T0385 |
Prochlorperazine Maleate
Prochlorperazin,Capazine,Prochlorperazine dimaleate salt,Stemetil,Compazine,丙氯拉嗪 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Prochlorperazine Maleate (Capazine) 是一种吩噻嗪类抗精神病药,主要用于治疗恶心、呕吐和眩晕。它比氯丙嗪更容易引起锥体外系疾病。 | |||
T7636 |
Phenprocoumon
乙苄香豆,苯丙羟基香豆素 |
||
Phenprocoumon 是一种长效口服抗凝剂和维生素 K 的拮抗剂,是香豆素衍生物。 | |||
T0802 |
Procaine hydrochloride
Novocaine HCl,Procaine HCl,盐酸普鲁卡因 |
Histone Demethylase; 5-HT Receptor; DNA/RNA Synthesis; Sodium Channel; NMDAR; AChR | Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Procaine hydrochloride (Novocaine HCl) 是DNA 脱甲基剂,是一种苯甲酸衍生物,具有局部麻醉和抗心律失常特性。 | |||
T1488 |
Procarbazine hydrochloride
NSC-77213 HCl,盐酸甲基苄肼,Procarbazine HCl |
DNA Alkylator/Crosslinker; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Procarbazine hydrochloride (NSC-77213 HCl) 是一种烷化剂,是甲基肼衍生物的盐酸盐,具有抗肿瘤和诱变活性。 | |||
T60322 |
Procainamide
Biocoryl,Novocainamide |
DNA Methyltransferase | Chromatin/Epigenetic |
Procainamide (Novocainamide) 是 DNA 甲基转移酶 1 (DNMT1) 的特异性强效抑制剂。Procainamide 是一种 1A 类抗心律失常药物。Procainamide 具有研究癌症和心律失常的潜力。 | |||
T31659 |
Eprociclovir
AV10,AV-10,A-5021,A 5021,A5021,AV 10 |
Antifection | Microbiology/Virology |
Eprociclovir (A-5021) 是一种新型阿昔洛韦类似物,是 EHV1 复制的强效抑制剂,可能用于治疗和/或预防该病毒感染。Eprociclovir 对大多数人类疱疹病毒都有很强的抗疱疹活性。 | |||
T21746 |
Terameprocol
tetramethyl Nordihydroguaiaretic Acid,EM-1421 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Terameprocol (EM-1421) 是 Nordihydroguaiaretic acid 的合成衍生物,是非选择性脂氧合酶抑制剂。 | |||
TP1868 |
Proctolin
直肠肽 |
Others | Others |
Proctolin 是内源性五肽,也是兴奋性神经调节剂。 | |||
T4548 |
Procaterol hydrochloride
|
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Procaterol hydrochloride 用于治疗哮喘的短效β2-肾上腺素受体激动剂。 | |||
T69013 |
Alaproclate
|
NMDAR | Neuroscience |
Alaproclate 是一种非竞争性 NMDA 受体拮抗剂,也是一种新的选择性5-HT摄取抑制剂,可用于研究抑郁症和老年痴呆。 | |||
T23702 |
Alaproclate, (S)-
(-)-Alaproclate,S-(-)-Alaproclate |
||
Alaproclate, (S)- is a selective inhibitor of serotonin reuptake. | |||
T4979 |
Procyclidine hydrochloride
(±)-Procyclidine hydrochlorid,丙环定盐酸盐 |
NMDAR; iGluR | Membrane transporter/Ion channel; Neuroscience |
Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) 是具有NMDA 拮抗剂特性的抗胆碱能试剂。 | |||
T70027 |
Eprociclovir potassium
|
||
Eprociclovir potassium is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica... | |||
T25988 |
Proclonol
R 8284,R-8284,Kilacar,R8284 |
||
Proclonol is used as a pesticide. | |||
T19049 |
Procion Blue HB
蓝色染料,Reactive Blue 2 |
Others | Others |
Procion Blue HB is an antagonist of purinergic. | |||
T124398 |
Procerine
|
||
Procerine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124398。 | |||
T69817 |
Eprociclovir Na
|
||
Eprociclovir Na is the salt form of Eprociclovir, also known as A-5021, a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applie... | |||
T0029 |
Procaine
Duracaine,Spinocaine,普鲁卡因,Novocaine,Vitamin H3,奴夫卡因 |
Histone Demethylase; DNA/RNA Synthesis; Sodium Channel | Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Membrane transporter/Ion channel |
Procaine (Vitamin H3) 是DNA 脱甲基剂,是一种酯类局部麻醉剂。它起效缓慢,作用持续时间短,主要用于浸润麻醉、周围神经阻滞和脊髓阻滞。 | |||
TMIH-0453 |
Procaterol-d7
(Rac)-Procaterol-d7 |
||
Procaterol-d7 是 Procaterol 的氘代化合物。Procaterol 的 CAS 号为 81262-93-3。Procaterol hydrochloride用于治疗哮喘的短效β2-肾上腺素受体激动剂。 | |||
T10351 |
Aprocitentan D4
ACT-132577 D4 |
Others | Others |
Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM; pA2s: 6.7 and 5.5). | |||
T16466 |
Penicillin G Procaine
PGP |
Others | Others |
Penicillin G Procaine is a β-lactam antibiotic and is a crystalline complex produced by chemically combining penicillin G with procaine. | |||
T1488L |
Procarbazine free base
CB 400-497,NSC-77213,Ro 4-6467/1,Ro 4-6467,Procarbazine |
||
Procarbazine is an antineoplastic chemotherapy drug for the treatment of Hodgkin's lymphoma and certain brain cancers. The drug is metabolized and activated in the liver. It also inhibits MAO thus increasing the effects of sympathomimetics, TCAs, and tyra | |||
T125167 |
Proctorione C
|
||
Proctorione C 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125167,CAS号为 263250-03-9。 | |||
T36521 |
Alaproclate (hydrochloride)
|
||
Alaproclate is a selective serotonin reuptake inhibitor (SSRI).1,2 It inhibits depletion of serotonin (5-HT) induced by 4-methyl-α-ethyl-m-tyramine in rat cerebral cortex, hippocampus, hypothalamus, and striatum (EC50s = 18, 4, 8, and 12 mg/kg, respectively).1 Alaproclate inhibits NMDA-evoked currents and depolarization-induced voltage-dependent potassium currents in rat hippocampal neurons (IC50s = 1.1 and 6.9 μM, respectively) and does not inhibit GABA-evoked currents when used at concentratio... | |||
T60578 |
Procyclidine
|
||
Procyclidine (Tricyclamol; (±)-Procyclidine) 是一种抗胆碱能剂。它是一种毒蕈碱受体 (muscarinic receptor) 拮抗剂,也是 N-甲基-D-天冬氨酸 (NMDA) 拮抗剂。Procyclidine 可用于帕金森症和相关精神疾病的研究,如Soman 诱发的癫痫。 | |||
T60469 |
Chloroprocaine
|
||
Chloroprocaine (2-Chloroprocaine) 是一种有效的Na,K-ATPase 酶活性抑制剂(IC50 = 13 mM)。Chloroprocaine 是一种阻滞外周神经的局部麻醉剂。 | |||
T20621 |
Isoprocarb
异丙威,Etrofolan,Mipcine,Hytox,Mipcin,Mipsin |
||
Isoprocarb is a metabolite of the pesticide. | |||
T34075 |
Piprocurarium iodide
Brevicurarine,LD2480,LD 2480,LD-2480 |
||
Piprocurarium iodide is a bioactive chemical. | |||
T78518 |
Prochloraz manganese
|
||
Prochloraz manganese为用于农业工业的抗真菌剂。 | |||
T126112 |
Epiprocurcumenol
|
||
Epiprocurcumenol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126112。 | |||
TMIH-0454 |
Prochlorperazine-d8
|
||
Prochlorperazine-d8 是 Prochlorperazine 的氘代化合物。Prochlorperazine 的 CAS 号为 58-38-8。Prochlorperazine 是一种抗精神病药phenothiazine衍生物。 | |||
T34074 |
Piproctanyl bromide
Piproctanylium bromide,Stemtrol;Piproctanyl bromide,Stemtrol,Piproctanyl bromide,Piproctanyliumbromid,Alden |
||
Piproctanyl bromide is an agricultural growth regulator. | |||
T23701 |
Alaproclate hydrochloride, (S)-
|
||
Alaproclate hydrochloride, (S)- is a selective inhibitor of serotonin reuptake. | |||
T69533 |
Procinolol
|
||
Procinolol is a beta adrenergic receptor antagonist. | |||
T68957 |
Eprociclovir dihydrate
|
||
Eprociclovir dihydrate is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica... | |||
T0378L |
Oxybuprocaine
Butoxyprocaine,BNX,Benoxinate,Novescine,Novesin |
||
Oxybuprocaine is an ester-type local anesthetic that is used especially in ophthalmology and otolaryngology. Oxybuprocaine binds to sodium channels and reversibly stabilizes the neuronal membrane which decreases its permeability to sodium ions. | |||
T60970 |
Caprochlorone
|
||
Caprochlorone 对正痘病毒具有抗病毒活性,可以降低被感染的小鼠肺部中流感病毒的滴度。Caprochlorone 可以抑制病毒穿透细胞,并且延迟新形成的病毒从细胞释放。 | |||
T69379 |
Iproclozide
|
||
Iproclozide is a potent monamine oxydase inhibitor (MAOI). | |||
T69027 |
Procaine merethoxylline
|
||
Procaine merethoxylline is a noted sodium channel blocker with a variety of inhibitory effects. | |||
T20811 |
Procymidone
Dicyclidine,S-7131,S 7131,SP 751011,SP-751011,S7131 |
||
Procymidone, a dicarboximide fungicide, is mainly used for vineyard protection but also for different crops. | |||
T36380 |
GLP-1 (1-36) amide (human, rat) (trifluoroacetate salt)
|
||
GLP-1 amide is a peptide hormone cleaved from proglucagon in the pancreas.1,2 Mice lacking the glucagon receptor (Gcgr-/-) have approximately nine-fold higher levels of total GLP-1 amide, including GLP-1 (1-36) amide and truncated GLP-1 (7-36) amide , in pancreatic tissue compared to wild-type mice.2References1. Schjoldager, B.T., Mortensen, P.E., Christiansen, J., et al. GLP-1 (glucagon-like peptide 1) and truncated GLP-1, fragments of human proglucagon, inhibit gastric acid secretion in humans... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0205 |
Procyanidin B1
原花青素B1,原花青素 B1 |
TLR | Immunology/Inflammation |
Procyanidin B1 是水果中常见的多酚类黄酮,能够与TLR4/MD-2复合体结合,具有抗炎活性。 | |||
TN1136 |
Procyanidin A1
原花青素 A1,Proanthocyanidin A1,原花色素A1 |
LDL; Calcium Channel; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism |
Procyanidin A1 (Proanthocyanidin A1) 是一种原花青素二聚体,具有抗过敏作用,可抑制蛋白激酶 C 激活下游脱粒或 RBL-213 细胞内部储存的 Ca2+流入。 | |||
TN6904 |
Procurcumadiol
5-Hydroxyprocurcumenol |
Others | Others |
Procurcumadiol (5-Hydroxyprocurcumenol) 是来自姜黄的天然产物。 | |||
TN2103 |
PROCYANIDIN C1
原花青素 C1,原花青素C1 |
Apoptosis | Apoptosis |
Procyanidin C1 是一种天然多酚,可造成 DNA 损伤,细胞周期停滞,诱导凋亡。它降低癌细胞中 Bcl-2 的蛋白水平,增强 BAX,caspase 3 和 9 的表达。 | |||
TN1132 |
Procyanidin A2
原花青素 A2,原花青素A2 |
IL Receptor; TNF; transporter; Antibacterial | Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology |
Procyanidin A2 是一种具有抗癌、抗氧化、抗菌和抗炎活性的黄酮类天然产物,存在于蔓越莓和越橘中。 | |||
T6S1367 |
Procyanidin B2
原花青素 B2,Proanthocyanidin B2 |
Reactive Oxygen Species; NOD | Immunology/Inflammation; Metabolism; NF-κB |
Procyanidin B2 (Proanthocyanidin B2) 是天然黄酮类物质,具有抗肿瘤,抗氧化等活性。 | |||
TN1150 |
Procyanidin B3
原花青素B3,原花青素 B3 |
Histone Acetyltransferase | Chromatin/Epigenetic |
Procyanidin B3 是从葡萄中提取的一种黄酮类天然产物,是组蛋白乙酰转移酶特异性抑制剂,可与 p300的其他位点而非活性位点结合,选择性抑制 p300 介导的 androgen 受体乙酰化。 | |||
TN2102 | Procurcumenol | Others; TNF | Apoptosis; Others |
Procurcumenol is an inhibitor of Nitric Oxide. Procurcumenol and epicurcumenol have inhibitory effects on release of tumor necrosis factor-a (TNF-a). | |||
TN5497 |
Procyanidin B2 3,3'-di-O-gallate
Procyanidin B-2 3,3'-di-O-gallate,原花青素B2-3,3'-二-O-没食子酸酯 |
||
Procyanidin B2 3,3'-di-O-gallate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5497,CAS号为 79907-44-1。 | |||
TN5492 |
Procyanidin B2 3''-O-gallate
Epicatechin-(4β→8)-epicatechin 3''-O-gallate,原花青素B2-3"-O-没食子酸 |
||
Procyanidin B2 3''-O-gallate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5492,CAS号为 73086-04-1。 | |||
T81398 |
Procyanidin A5'
|
||
Procyanidin A5是一种属于A型二聚体的原花青素,具有两个(flavan-3-ol)单元通过碳-碳键连接的结构,通常存在于各种植物中,例如苹果和葡萄皮。 | |||
TN4831 |
Procumbide
|
||
Procumbide has anti-inflammatory activity. | |||
TN1151 |
Procyanidol B4
原花青素B4,Procyanidin B4 |
Nrf2 | Immunology/Inflammation |
Procyanidin B4 reveals significant antioxidant activity | |||
T81397 |
Procyanidin C2
Procyanidine C2 |
||
Procyanidin C2,源自Fagopyrum dibotrys (D. Don) Hara,为酚苷类化合物。 | |||
TN5493 |
Procyanidin B5
原花青素B5,Procyanidin B-5,Epicatechin-(4β→6)-epicatechin |
||
Procyanidin B5 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5493,CAS号为 12798-57-1。 | |||
T60692 |
Masoprocol
|
||
Masoprocol (meso-Nordihydroguaiaretic acid) 是口服有效的脂氧合酶 (lipoxygenase) 抑制剂。Masoprocol 具有出抗高血糖活性,可用于 II 型糖尿病的研究。 Masoprocol 可降低体内肝甘油三酯和葡萄糖浓度。 | |||
TN4641 |
Neoprocurcumenol
|
Others | Others |
Neoprocurcumenol exerts significant toxicity on mosquito larvae. | |||
TN5489 |
Procyanidin B-5 3,3'-di-O-gallate
原花青素B5-3,3'-二-O-没食子酸酯,Procyanidin B5 3,3'-di-O-gallate |
||
Procyanidin B-5 3,3'-di-O-gallate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5489,CAS号为 106533-60-2。 | |||
TN4320 |
Isoprocurcumenol
|
Others | Others |
Isoprocurcumenol is an inhibitor of Nitric Oxide. |