458
52
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0547 |
FlutaMide Related CoMpound B
|
Others | Others |
FlutaMide Related CoMpound B 用作医药中间体。 | |||
T0535 |
Memantine Related Compound B
美金刚杂质B,3,5-Dimethyl-1-adamantanol |
Others | Others |
Memantine Related Compound B (3,5-Dimethyl-1-adamantanol) 是Memantine 的杂质。 | |||
T21000 |
PiB
2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇,Pittsburgh Compound-B,6-OH-BTA-1 |
Others | Others |
PiB (Pittsburgh Compound-B) 是分析 11C-PiB 的标准品。 11C-PiB 是一种用于阿尔茨海默病诊断的 β-淀粉样蛋白 PET 成像示踪剂。 | |||
T20683 |
Letrozole related compound B
Letrozole specified impurity A |
||
Letrozole related compound B is an impurity of aromatase inhibitor. | |||
T125846 |
Clopidogrel Related Compound B
|
||
Clopidogrel Related Compound B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125846,CAS号为 144750-52-7。 | |||
T2028 |
NG 52
NG52,NG-52,Compound 52 |
CDK | Cell Cycle/Checkpoint |
NG 52 (NG-52) 是可逆和 ATP 相容性且具有口服活性的Cdc28p 和Pho85p 激酶抑制剂,IC50分别为 7 μM 和 2 μM。它还抑制磷酸甘油酸激酶 1 的活性,IC50值为 2.5 μM。 | |||
T124814 |
Barbaloin-related compound B
|
||
Barbaloin-related compound B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124814。 | |||
T29161 |
STOCK2S-26016
WNK IN B,WNK-IN-B,Compound B |
||
WNK-IN-B is an inhibitor of Wnk signalling. WNK-IN-B is a cell-permeable diaminoacridine derivative that targets the CCT domain of SPAK and OSR1 via reversible binding. WNK-IN-B selectively suppress hypotonic shock-induced WNK signaling pathway activation | |||
T71716 |
Nav1.1-IN-B
|
||
Nav1.1-IN-B is a selective NaV1.1 inhibitor which reduces visceral hypersensitivity. | |||
T23732 |
Amoxicillin, L-
L-Amoxicillin,Amoxicillin trihydrate impurity B,Amoxicillin related compound B |
||
Amoxicillin, L- is an antibiotic. It is also useful for the treatment of a number of bacterial infections. | |||
T20564 |
Valsartan benzyl ester
Valsartan impurity B,Valsartan related compound C |
||
Valsartan benzyl ester is a intermediate of Valsartan. | |||
T70782 |
PF-05139962
|
||
PF-05139962 is a novel potent mTOR inhibitor with excellent mTOR biochemical inhibition, cellular potency, kinase selectivity and in vitro ADME properties. PF-05139962 has pS473 and pS6 cellular IC50 = 48 and 6 nM respectively. PF-05139962 has great selectivity against other receptors and kinases. No genotoxicity was observed on this compound and no more than 25% inhibiton was observed for major CYP enzymes (3A4, 1A2, 2C9, 2D6) at 3 uM. This compound has LE = 0.35 and LipE up to 6.8 which is in ... | |||
T29476 |
6-OH-BTA-0
Pittsburgh Compound-B precursor,11C-PiB Precursor |
||
6-OH-BTA-0 is the precursor for preparing 11C-PiB, which is a β-amyloid PET imaging tracer for Alzheimer's disease diagnosis. | |||
T69381 | Dechloro perphenazine | ||
Dechloro perphenazine is the dechlorinated analogue of Perphenazine (P291100), an D2 dopamine receptor antagonist; α-adrenergic receptor antagonist and σ-receptor agonist. | |||
T40284 |
B-Raf IN 2
|
Raf | MAPK |
B-Raf IN 2, compound Ia, is a highly effective and specific inhibitor of BRAF. It exhibits significant potential for cancer research. | |||
T1832 |
Walrycin B
|
Antibacterial; Antibiotic | Microbiology/Virology |
Walrycin B 是一种能特异地靶向WalR 应答调节子的新型抗菌素。 | |||
T64021 |
GDC-6036-NH
|
Others | Others |
GDC-6036-NH 是化合物17a /b 的前体,化合物17a /b 是一种RAS 抑制剂,可用于癌症研究。 | |||
T63788 |
PCLX-001
|
Others | Others |
PCLX-001 is a small-molecule compound that acts as an orally active inhibitor of N-myristoyltransferase (NMT), specifically targeting NMT1 and NMT2 with IC50 values of 5 nM and 8 nM, respectively. This compound demonstrates anti-tumor effects and effectively inhibits the early signaling of B-cell receptor (BCR). Consequently, PCLX-001 is a valuable tool for researching B-cell malignancies [1] [2]. | |||
T35330 |
BTK inhibitor 1
|
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
BTK inhibitor 1 (Compound 27)是一种BTK 抑制剂(IC50:0.11nM),对hWB 中的B 细胞活化具有抑制作用,IC50为2nM。 | |||
T60932 |
MAO-B-IN-8
|
MAO | Metabolism; Neuroscience |
MAO-B-IN-8是一种高效且可逆的单胺氧化酶-B(MAO-B)抑制剂,同时也能抑制微胶质细胞产生的神经炎症介质。该化合物专为神经退行性疾病相关研究而设计[1]。 | |||
T125100 |
Pteroside B
|
||
Pteroside B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125100。 | |||
T14299 |
AP20187
B/B Homodimerizer |
Others | Others |
AP20187 (B/B Homodimerizer) 是一种细胞渗透性配体,用于二聚化 FK506 结合蛋白 (FKBP) 融合蛋白。它启动生物信号级联和基因表达或破坏蛋白质-蛋白质相互作用。 | |||
T10337 |
Antimicrobial Compound 1
|
Antibacterial | Microbiology/Virology |
Antimicrobial Compound 1 是一种烷基吡啶鎓化合物,尾部为 12C,头部为 4-羧基。 Antimicrobial Compound 1 对枯草芽孢杆菌和大肠杆菌具有抗菌活性。 | |||
T67879 |
hMAO-B-IN-5
|
MAO; Monoamine Oxidase | Metabolism; Neuroscience |
hMAO-B-IN-5 是有一种有效的、可逆的、具有选择性的人类单胺氧化酶 hMAO-B 抑制剂( IC50 :0.12 μM)。 hMAO-B-IN-5 可以透过血脑屏障,可用于对帕金森疾病的研究,是中枢神经系统疾病的治疗和诊断中都是有潜力的化合物。 | |||
T126461 |
Aloenin B
|
||
Aloenin B 是一种从芦荟的叶和根中分离得到的化合物,对谷氨酸诱导的HT22细胞神经元死亡具有神经保护活性。 | |||
T39043 |
Tenofovir amibufenamide
HS-10234 |
HBV | Microbiology/Virology |
Tenofovir amibufenamide (HS-10234) (HS-10234) 是一种 Tenofovir 前药,是一种具有口服活性的抗病毒化合物。Tenofovir amibufenamide 对乙型肝炎病毒 (HBV)具有抑制作用,可用于慢性乙型肝炎 (CHB) 研究。 | |||
T20641 |
Propagermanium
Dipropanoic acid germanium sequioxide,SK-818,Ge 132,二羧乙基三氧化二锗,Ge132,SK 818,Ge-132 |
Others | Others |
Propagermanium (Ge132) 是一种锗的有机金属化合物,在日本已被用作治疗慢性乙型肝炎的药物。 | |||
T67764 |
hMAO-B-IN-4
|
MAO | Metabolism; Neuroscience |
hMAO-B-IN-4 (compound B10) 是一种选择性的、可逆的、血脑屏障通透性 (BBB) 的人单胺氧化-B (hMAO-B) 抑制剂 (IC50= 0.067, Ki= 0.03 μM)。hMAO-B-IN-4 抑制 hMAO-A 的活性较低, IC50 值为 33.82 μM。 | |||
T62404 |
SHMT-IN-2
|
Others | Others |
SHMT-IN-2 (compound 2) 是一种特异性人 SHMT1/2 小分子抑制剂,能够作用于 SHMT1 (IC50: 13 nM) 和 SHMT2 (IC50: 66 nM)。SHMT-IN-2 对许多人类癌细胞的生长具有抑制作用,对 B 细胞淋巴瘤具有敏感性。 | |||
T67748 |
ROCK-IN-5
|
ROCK; ERK | Cell Cycle/Checkpoint; Cytoskeletal Signaling; MAPK; Stem Cells |
ROCK-IN-5(化合物I-B-37)是一种有效的蛋白激酶抑制剂,包括ROCK、ERK、GSK 和AGC。ROCK-IN-5在心脏病、增殖性疾病和神经退行性疾病研究方面具有潜力。 | |||
T77656 |
LW3
|
Antifungal | Microbiology/Virology |
LW3 是一种有效的广谱抗真菌化合物。 LW3 具有抗真菌活性,对 B. cinerea、R. solani、S. sclerotiorum 和 F. graminearum 具有抑制作用, EC50 值分别为 0.54、0.09、1.52 和 2.65 mg/L。 | |||
T50009L |
sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate
|
Others | Others |
sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate 是一种有机硫化合物。它已被用作研究含硫化合物对酶活性和代谢途径的影响的模型化合物,也被用于研究含硫化合物对细菌生长和基因表达调控的影响。 | |||
T6075 |
Epothilone B
帕妥匹隆,Patupilone,EPO 906 |
Apoptosis; Microtubule Associated; Antibiotic; Antifungal | Apoptosis; Cytoskeletal Signaling; Microbiology/Virology |
Epothilone B (EPO 906) 是微管稳定剂,Ki 为0.71 μM。 它与αβ-微管蛋白异二聚体亚基结合,使αβ-微管蛋白解离减少。 | |||
T6998 |
Tedizolid Phosphate
TR-701FA,Torezolid phosphate,磷酸特地唑胺 |
Antibacterial; Antibiotic | Microbiology/Virology |
Tedizolid Phosphate (TR-701FA) 是 MAO-A 和 MAO-B 抑制剂,具有抗革兰氏阳性菌的活性。 | |||
T15704 |
Lagociclovir
MIV-210 |
HBV | Microbiology/Virology |
Lagociclovir (MIV-210) 是一种核苷类似物,是一种可用治疗 HBV82的抗病毒化合物,可抑制野生型乙型肝炎病毒 (HBV) 在永久表达 HBV 的人肝癌细胞系中的复制。 | |||
T67789 |
Bazinaprine
|
MAO | Metabolism; Neuroscience |
Bazinaprine 是一种选择性的、可逆的单胺氧化酶抑制剂(MAOI),是治疗抑郁症的候选化合物。Bazinaprine 对A 型单胺氧化酶显示出较强的抑制作用,对b 型单胺氧化酶只显示出较弱的抑制作用。Bazinaprine 在体内可逆,但在体外不可逆。 | |||
T9518 |
Inarigivir ammonium
ORI-9020 ammonium,SB-9200 ammonium,Inarigivir铵 |
HBV | Microbiology/Virology |
Inarigivir ammonium (SB-9200 ammonium) 是一种二核苷酸抗病毒化合物,可显着降低表达乙型肝炎病毒的转基因小鼠的 HBV DNA。它是一种激活细胞内先天免疫的视黄酸诱导基因-I 激动剂。 | |||
T77632 |
Antiviral agent 34
|
Antiviral; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation |
Antiviral agent 34 是一种可口服且作用效果较强的抗病毒化合物,抑制甲型和乙型流感病毒。Antiviral agent 34 通过调节 RNA 聚合酶来抑制流感病毒的增殖。Antiviral agent 34 可用于研究病毒感染。 | |||
T4019 |
Cambinol
SIRT1/2 Inhibitor IV,NSC 112546 |
Apoptosis; Phospholipase; Sirtuin | Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism |
Cambinol (SIRT1/2 Inhibitor IV) 是一种SIRT1和SIRT2的抑制剂,IC50值分别为 56 μM 和 59 μM。它是中性鞘磷脂酶的外泌体抑制剂。 | |||
T61131 |
MAO-B-IN-11
|
||
MAO-B-IN-11, also known as Compound 8c, is a highly potent inhibitor of monoamine oxidase B (MAO-B), with an IC50 value of 1.3 μM. Additionally, MAO-B-IN-11 exhibits neuroprotective properties [1]. | |||
T60660 |
MAO-B-IN-14
|
||
MAO-B-IN-14 (Compound 9) 是选择性的单胺氧化酶-B (MAO-B)抑制剂。MAO-B-IN-14 对人 MAO-B 的 IC50值为 0.95 μM,Ki 值为 0.55 μM。 | |||
T79895 |
Cbl-b-IN-8
|
E1/E2/E3 Enzyme | Ubiquitination |
Cbl-b-IN-8 (Compound 293),一种casitas B系淋巴瘤(Cbl-b)及c-Cbl的抑制剂,其IC50值分别为5.5 nM和7.8 nM。 | |||
T79894 |
Cbl-b-IN-7
|
E1/E2/E3 Enzyme | Ubiquitination |
Cbl-b-IN-7 (Compound 248)作为针对casitas B系淋巴瘤(Cbl-b)和c-Cbl的抑制剂,其IC50值分别为6.7 nM与5.2 nM。 | |||
T79896 |
Cbl-b-IN-9
|
E1/E2/E3 Enzyme | Ubiquitination |
Cbl-b-IN-9(Compound 300)为针对casitas B系淋巴瘤(Cbl-b)及c-Cbl的抑制剂,其IC50值分别为5.6 nM与4.7 nM。 | |||
T61321 |
MAO-B-IN-12
|
||
MAO-B-IN-12 (Compound 16c) is a highly effective inhibitor of monoamine oxidase B (MAO-B), displaying significant potency with an IC50 value of 1.3 μM. Additionally, MAO-B-IN-12 exhibits notable neuroprotective activity [1]. | |||
T79897 |
Cbl-b-IN-10
|
E1/E2/E3 Enzyme | Ubiquitination |
Cbl-b-IN-10(Compound 463)为针对casitas B系淋巴瘤(Cbl-b)和c-Cbl的抑制剂,其IC50值分别为6.0 nM和3.5 nM。 | |||
T79893 |
Cbl-b-IN-6
|
E1/E2/E3 Enzyme | Ubiquitination |
Cbl-b-IN-6 (Compound 246),作为casitas B系淋巴瘤(Cbl-b)和c-Cbl的抑制剂,其IC50值分别为5.8 nM和4.4 nM。 | |||
T10310 |
Amphotericin B methyl ester
|
Others | Others |
Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses significant antifungal activity. It disrupts HIV-1 particle production and potently inhibits HIV | |||
T61830 | MAO-B-IN-10 | ||
MAO-B-IN-10 (compound 4f) is a highly potent and selective inhibitor of MAO-B (monoamine oxidase-B). It effectively penetrates the blood-brain barrier and exhibits an IC50 of 5.3 μM. This compound demonstrates the ability to inhibit self-mediated Aβ (amyloid β) aggregation by 58.2% and disaggregate it by 43.3%. Thus, MAO-B-IN-10 holds promise for Alzheimer's disease research [1]. | |||
T79898 |
Cbl-b-IN-11
|
E1/E2/E3 Enzyme | Ubiquitination |
Cbl-b-IN-11 (Compound 466)作为casitas B系淋巴瘤 (Cbl-b) 及c-Cbl的抑制剂,显示出对Cbl-b和c-Cbl的高度选择性,其IC50值分别为6.4 nM 和6.1 nM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0948L |
Corticosterone
皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants) |
Glucocorticoid Receptor; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Corticosterone (Kendall's compound B) 是一种肾上腺皮质类固醇,有盐皮质激素和糖皮质激素的活性,具有口服活性。Corticosterone 参与体内能量、免疫反应和应激反应的调节。 | |||
T2S0062 |
Pulchinenoside B
白头翁皂苷B |
||
Compound T2S0062 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T2S0062,CAS号为 135247-95-9。 | |||
T4961 |
9''-Methyl salvianolate B
9'-Methyl lithospermate B,9’-丹酚酸B单甲酯,9''-丹酚酸B单甲酯 |
Others | Others |
9'-Methyl lithospermate B 是一种酚类化合物,提取自 RadixSalvia miltiorrhizae。 | |||
TN2359 |
Iristectorigenin B
Iristectrigenin B |
Liver X Receptor | Metabolism |
Iristectorigenin B (Iristectrigenin B) 是一种有效的肝脏 X 受体 (LXR) 调节剂,是从 Belamcanda chinensis 中分离的小分子化合物。Iristectrigenin B 可促进巨噬细胞 RAW 1.1 细胞中 ABCA264 和 ABCG7 的表达。 | |||
T22286 |
Cyanosafracin B
Cyanoquinonamine,氰基番红菌素 B,CBR28-1 |
Others | Others |
Cyanosafracin B (Cyanoquinonamine) 是一种合成 Phthalascidin Pt-650 及 Ecteinascidin ET-743 的起始原料。 | |||
TN2043 |
Pasakbumin B
13-alpha-(21)-Epoxyeurycomanone,13ALPHA(21)-环氧宽缨酮 |
Others | Others |
Pasakbumin B (13-alpha-(21)-Epoxyeurycomanone) 是一种从 Eurycoma longifoliaJack 中获得的具有生物活性的化合物,显示出抗溃疡作用。 | |||
T1922 |
Pseudolaric Acid B
土槿乙酸B,土荆皮乙酸 |
Apoptosis; p38 MAPK; Ferroptosis; HBV; Autophagy; Antifungal | Apoptosis; Autophagy; MAPK; Microbiology/Virology |
Pseudolaric Acid B 是一种从Pseudolarix kaempferiGorden (pinaceae) 根部分离的二萜酸,具有抗癌、抗真菌、抗受精和免疫抑制活性。它还诱导细胞自噬。 | |||
TN3628 |
Chamaejasmenin B
|
Others | Others |
Chamaejasmenin B 是一种从 Stellera chamaejasme L 中分离得到的化合物。Chamaejasmenin B 具有抗癌和抗肿瘤活性,可抑制癌细胞迁移和侵袭,抑制肿瘤转移。Chamaejasmenin B 可用于研究如乳腺癌类的癌症。 | |||
T3408 |
Syringin
Lilacin,Syringoside,eleutheroside-b,Methoxyconiferine,紫丁香苷 |
NOS; Autophagy | Autophagy; Immunology/Inflammation |
Syringin (eleutheroside-b) 是欧丁香中的一种苯丙素类天然产物,通过抑制自噬来防止压力超载引起的心肌肥厚,具有抗肿瘤、抗增殖、抗骨质疏松、免疫调节和血小板聚集抑制作用。 | |||
T3519 |
Formosanin C
Polyphyllin B,重楼皂苷 B,重楼皂苷B |
Apoptosis; Caspase | Apoptosis; Proteases/Proteasome |
Formosanin C (Polyphyllin B) 是从滇重楼中分离的一种薯蓣皂苷,可诱导细胞凋亡。它是一种免疫调节剂,具有抗肿瘤活性。 | |||
TN5254 |
Wighteone
Erythrinin B,6-Isopentenylgenistein |
Antifungal | Microbiology/Virology |
Wighteone (Erythrinin B) 是一种从 Genista ephedroides 中提取出来的小分子化合物,具有潜在的抗真菌和抗癌活性,对 EGFR L858R/T790M 突变非小细胞肺癌具有抗肿瘤作用。。 | |||
TN1880 |
Lucidenic acid B
Lucidenicacid B |
Apoptosis; Caspase | Apoptosis; Proteases/Proteasome |
Lucidenic acid B (Lucidenicacid B) 是从灵芝中提取得到的天然化合物,可诱导caspase-9 和 caspase-3 的活化和 PARP 的裂解,可通过线粒体介导诱导人白血病细胞凋亡 。 Lucidenic acid B通过灭活MAPK / ERK信号转导途径和降低NF-kappaB和AP-1的结合活性来抑制PMA诱导的人肝癌细胞侵袭。。Lucidenic acid B 对细胞周期和坏死细胞没有影响。 | |||
T8002 |
3-Hydroxycoumarin
|
Lipoxygenase | Metabolism |
3-hydroxycoumarin 是一种 15-LOX-1的有效氧化还原抑制剂,近期被证明能保护海胆生殖细胞免受紫外线 B 的损伤。 | |||
T4S0350 |
Licochalcone B
甘草查尔酮 B,甘草查尔酮B |
Beta Amyloid; Others | Neuroscience; Others |
Licochalcone B 是从Glycyrrhiza inflate 根中提取的。它能够抑制淀粉样蛋白 β 自聚集作用 (IC50=2.16 μM) ,分解预先形成的 Aβ42原纤维,并通过螯合金属离子抑制金属诱导的 Aβ42聚集。 | |||
T1040 |
Vitamin B12
Cyanocobalamin,Cobalamin,维生素B12 |
Endogenous Metabolite | Metabolism |
Vitamin B12 (Cobalamin) 是一种维生素,在维持血流形成和脑、神经系统正常功能等方面发挥关键作用。 | |||
T83545 |
(E)-(-)-Aspongopusamide B
|
||
(E)-(-)-Aspongopusamide B (Compound 9) 是从昆虫Aspongopus chinensis 分离得到的一种天然产物。 | |||
T83271 |
6-Aldehydoisoophiopogonone B
|
||
6-Aldehydoisoophiopogonone B (Compound 24) 是从Ophiopogon japonicus 提取的同型异黄酮化合物。 | |||
T81298 |
Renchangianin B
|
||
Renchanginin B(compound 2)是从Kadsura renchangiana茎中分离得到的一种二苯并环辛烯型木酚素。 | |||
T82554 |
Dihydroisocucurbitacin B
|
||
Dihydroisocucurbitacin B为一种源自Wilbrandia ebracteata根部的活性化合物。 | |||
T38481 |
Camellianin B
|
||
Camellianin B, a flavonoid compound and metabolite of Camellianin A, exhibits antioxidant properties and acts as an angiotensin converting enzyme (ACE) inhibitor. | |||
T83155 |
Agonodepside B
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Agonodepside B, 分离自非孢子丝状真菌F7524,是一种化合物。 | |||
T8174 |
Saikosaponin F
柴胡皂苷F,柴胡皂苷 F |
Others | Others |
Saikosaponin F 是一种柴胡中的天然成分。 | |||
T38837 |
Microcolin B
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Microcolin B, an acylpeptide immunosuppressant, is a highly potent and biologically unique compound containing proline. It is derived from the blue-green alga Lyngbya majuscule. | |||
T81742 |
Mulberrofuran B
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Mulberrofuran B,一种从Morus alba乙醇提取物中分离得到的化合物,展现了抗氧化活性。 | |||
T80702 |
α-Thevetin B
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α-Thevetin B(Compound 24), 一种从Thevetia peruviana分离得到的心脏苷,用于肺癌、胃癌和胰腺癌的研究。 | |||
T40383 |
Monensin B
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Monensin B is a polyketide compound derived from the bacterium Streptomyces cinnamonensis. Its production involves the fermentation of Streptomyces cinnamonensis, resulting in a mixture of Monensin A and Monensin B. The ratio of these two compounds depends on the concentrations of ethylmalonyl-CoA and methylmalonyl-CoA. | |||
T80000 |
Multiflorin B
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NO Synthase | Immunology/Inflammation |
Multiflorin B为一种山奈酚苷,源自蕨类植物Neocheiropteris palmatopedata的根部提取。在20 μg/ml的浓度下,Multiflorin B能够抑制一氧化氮的生成,其抑制率达到52%。 | |||
T82396 |
Fissitungfine B
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Fissitungfine B,一种从热带药用植物Fissistigma tungfangense提取的化合物,展示出显著的抗癌活性。 | |||
T82302 |
Glucodichotomine B
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Glucodichotomine B (Compound 13) 是一种从中药植物 Stellaria dichotoma L. var. lanceolata 根中分离得到的天然产物,具有抗癌活性。 | |||
T83459 |
11α-O-Tigloyl-12β-O-acetyltenacigenin B
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Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic |
11α-O-Tigloyl-12β-O-acetyltenacigenin B 是Tenacigenin B 的酯类衍生物,源自藤黄藤 (MTC)。该化合物具有调节Aurora-A活性,对淋巴瘤显示出潜在的抗肿瘤效果。 | |||
TN2408 |
Evofolin B
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Cannabinoid Receptor | GPCR/G Protein |
Evofolin B 是从Zanthoxylum ailanthoides 的茎皮中分离出来的天然化合物。Evofolin B 对人类中性粒细胞对甲酰-L-蛋氨酸-L-亮氨酸-L-苯丙氨酸/cytochalasin B(fMLP/CB)产生的超氧阴离子有抑制作用。 | |||
T80860 |
Vitisin B
(-)-Vitisin B,E-Vitisin B |
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Vitisin B,从Vitis thunbergii var. taiwaniana分离提取,对脂多糖(LPS)诱导的关节炎表现出抗炎活性。 | |||
T38609 |
Mycalolide B
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Mycalolide-B is a marine sponge-derived compound that functions as a selective inhibitor of actomyosin ATPase. It effectively hinders ATP-induced contraction and Mg2+-ATPase activity in the absence of Ca2+. | |||
T74196 |
Inophyllum B
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Inophyllum B ((+)-Inophyllum B) 是一种有效的HIV 逆转录酶 (Reverse Transcriptase) 抑制剂,IC50为 38 nM。Inophyllum B 在体外细胞培养中抑制HIV-1(IC50=1.4 μM)。Inophyllum B 可从非洲大蜗牛Achatina fulica 的丙酮提取物中分离得到。 | |||
T81169 |
Shishijimicin B
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Shishijimicin B为活性的烯二炔类化合物,具有强烈的细胞毒性,IC50值介于2.0 - 3.3 nM。此化合物表现出抗肿瘤活性,常用于癌症研究中。作为点击化学试剂,Shishijimicin B内含Alkyne基团,能通过含Azide基团的分子在铜催化下发生(CuAAc)反应。 | |||
T82445 |
Erinacine P
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Erinacine P(化合物1)为担子菌猴头菇YB4-6237菌丝体分离得到的木犀草素亲代代谢产物。其在温和条件下可化学转化为猴头素B,继而可转化为猴头素A。 | |||
TN4605 | Myriceric acid B | HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Myriceric acid B is a potent HIV-1 entry inhibitor targeting gp41 and can serve as a lead compound for developing novel anti-HIV-1 drug. Myriceric acid B scavenges DPPH free radicals with IC50 value of 21.8 uM, it inhibits aromatase activity with IC50 val | |||
T75692 | Hypoglaunine D | ||
Hypoglaunine D 是 Triptonine B 的类似物,是一种抗HIV 的化合物,Hypoglaunine D 抑制 H9 淋巴细胞中HIV 病毒复制的EC50值为 22 μg/ml。 | |||
T82983 |
Aplyronine B
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Aplyronine B是一种具有抗肿瘤活性的活性化合物,对HeLa-S3细胞表现出细胞毒性,IC50值为2.9 nM,适用于癌症研究。 | |||
T81321 |
Quercetin-3-O-b-D-galactopyranosyl-(1→6)-b-D-glucopyranoside
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Quercetin-3-O-b-D-galactopyranosyl-(1→6)-b-D-glucopyranoside (化合物 1),为自白仙茅 (M. delavayi) 叶中分离的黄酮甙类化合物。 | |||
T81095 |
Stenophyllol B
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Stenophyllol B (compound 4) 是一种具有双环及桥联三环骨架的三聚芪类化合物。该化合物最初在龙脑香科植物中被鉴定,随后在Hopea、Neobalanocarpus、Shorea、Stemonoporus以及Vateri等属的多种物种中发现。 | |||
T72916 |
Justicidin B
爵床脂素B |
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Justicidin B是一种高效的抗癌木脂素及促凋亡剂,同时具备显著的骨吸收抑制作用,并展现出强大的抗病毒、杀真菌和抗原虫能力。此外,Justicidin B能显着抑制血小板聚集。 | |||
T75468 | Asperglaucin B | ||
Asperglaucin B 是一种来自真菌Aspergillus chevalieriSQ-8 的烷基化水杨醛衍生物,具有抗菌活性。Asperglaucin B 对两种植物病原体Pseudomonas syringae pv actinidae(Psa)和Bacillus cereus 显示出有效的抗菌活性,MIC 值为 6.25 μM。 | |||
T79949 |
Foenumoside B
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PPAR | DNA Damage/DNA Repair; Metabolism |
Foenumoside B为从Lysimachia foenum-graecum中提取的三萜皂苷。该化合物通过激活AMPK信号传导和抑制PPARγ诱导的脂肪生成,调节脂质代谢向脂肪分解方向转变。因其调控作用,Foenumoside B常用于研究肥胖及相关代谢疾病。 | |||
T81856 |
Marsdenoside B
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Marsdenoside B(化合物8), 一种海芋属植物中的提取物,显示对MGC-803和HT-29肿瘤细胞系具有抑制作用,其IC50s 分别为25.6 μg/mL 和32.4 μg/mL。 | |||
T79970 |
Taxamairin B
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Taxamairin B是有效的抗炎化合物,能显著抑制LPS诱导的RAW264.7细胞中促炎因子(TNF-α, IL-1β和IL-6)表达及NO、ROS生成,并对LPS引起的急性肺损伤模型小鼠具有保护效果。 | |||
T83903 |
Polymyxin B2 sulfate
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Polymyxin B2是一种抗生素,并且是从B. polymyxa分离出的阳离子脂肽抗生素polymyxin B的主要成分。该化合物对P. aeruginosa、A. baumannii、K. pneumoniae和E. cloacae菌株具有活性(MICs分别为1-2、0.5-1、0.25-0.5和0.25-1 µg/ml)。在体内实验中,以4 mg/kg剂量的Polymyxin B2能显著降低P. aeruginosa血液感染小鼠模型中的血液集落形成单位(CFUs)数量。 | |||
T31471 |
Dihydroisoalantolactone
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Dihydroisoalantolactone is found in herbs and spices. Dihydroisoalantolactone is isolated from roots of Inula helenium (elecampane). This compound Aliphatic heteropolycyclic, belongs to the class of organic compounds known as eudesmanolides, secoeudesmano | |||
T79976 |
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside
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HBV | Microbiology/Virology |
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside 作为一种抗HBV剂,在Hep G2.2.15细胞系上能够抑制HBsAg和HBeAg的分泌,其IC50值分别约为1.67 mM和>2.15 mM。 | |||
T81201 |
Sartorypyrone B
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Sartorypyrone B为Chevalone C的2β-乙酰氧基衍生物,由海绵源真菌Neosartorya tsunodae(KUFC 9213)的培养物中乙酸乙酯提取得到。该化合物对MCF-7、NCI-H460和A375-C5细胞系展示出较强的生长抑制活性,GI50s值分别为17.8、20.5和25.0 μM,显示其在乳腺癌、非小细胞肺癌和黑色素瘤研究中的应用潜力。 | |||
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