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458

抑制剂 & 化合物

52

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0547 FlutaMide Related CoMpound B

Others Others
FlutaMide Related CoMpound B 用作医药中间体。
T0535 Memantine Related Compound B

美金刚杂质B,3,5-Dimethyl-1-adamantanol

Others Others
Memantine Related Compound B (3,5-Dimethyl-1-adamantanol) 是Memantine 的杂质。
T21000 PiB

2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇,Pittsburgh Compound-B,6-OH-BTA-1

Others Others
PiB (Pittsburgh Compound-B) 是分析 11C-PiB 的标准品。 11C-PiB 是一种用于阿尔茨海默病诊断的 β-淀粉样蛋白 PET 成像示踪剂。
T20683 Letrozole related compound B

Letrozole specified impurity A

Letrozole related compound B is an impurity of aromatase inhibitor.
T125846 Clopidogrel Related Compound B

Clopidogrel Related Compound B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125846,CAS号为 144750-52-7。
T2028 NG 52

NG52,NG-52,Compound 52

CDK Cell Cycle/Checkpoint
NG 52 (NG-52) 是可逆和 ATP 相容性且具有口服活性的Cdc28p 和Pho85p 激酶抑制剂,IC50分别为 7 μM 和 2 μM。它还抑制磷酸甘油酸激酶 1 的活性,IC50值为 2.5 μM。
T124814 Barbaloin-related compound B

Barbaloin-related compound B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124814。
T29161 STOCK2S-26016

WNK IN B,WNK-IN-B,Compound B

WNK-IN-B is an inhibitor of Wnk signalling. WNK-IN-B is a cell-permeable diaminoacridine derivative that targets the CCT domain of SPAK and OSR1 via reversible binding. WNK-IN-B selectively suppress hypotonic shock-induced WNK signaling pathway activation
T71716 Nav1.1-IN-B

Nav1.1-IN-B is a selective NaV1.1 inhibitor which reduces visceral hypersensitivity.
T23732 Amoxicillin, L-

L-Amoxicillin,Amoxicillin trihydrate impurity B,Amoxicillin related compound B

Amoxicillin, L- is an antibiotic. It is also useful for the treatment of a number of bacterial infections.
T20564 Valsartan benzyl ester

Valsartan impurity B,Valsartan related compound C

Valsartan benzyl ester is a intermediate of Valsartan.
T70782 PF-05139962

PF-05139962 is a novel potent mTOR inhibitor with excellent mTOR biochemical inhibition, cellular potency, kinase selectivity and in vitro ADME properties. PF-05139962 has pS473 and pS6 cellular IC50 = 48 and 6 nM respectively. PF-05139962 has great selectivity against other receptors and kinases. No genotoxicity was observed on this compound and no more than 25% inhibiton was observed for major CYP enzymes (3A4, 1A2, 2C9, 2D6) at 3 uM. This compound has LE = 0.35 and LipE up to 6.8 which is in ...
T29476 6-OH-BTA-0

Pittsburgh Compound-B precursor,11C-PiB Precursor

6-OH-BTA-0 is the precursor for preparing 11C-PiB, which is a β-amyloid PET imaging tracer for Alzheimer's disease diagnosis.
T69381 Dechloro perphenazine

Dechloro perphenazine is the dechlorinated analogue of Perphenazine (P291100), an D2 dopamine receptor antagonist; α-adrenergic receptor antagonist and σ-receptor agonist.
T40284 B-Raf IN 2

Raf MAPK
B-Raf IN 2, compound Ia, is a highly effective and specific inhibitor of BRAF. It exhibits significant potential for cancer research.
T1832 Walrycin B

Antibacterial; Antibiotic Microbiology/Virology
Walrycin B 是一种能特异地靶向WalR 应答调节子的新型抗菌素。
T64021 GDC-6036-NH

Others Others
GDC-6036-NH 是化合物17a /b 的前体,化合物17a /b 是一种RAS 抑制剂,可用于癌症研究。
T63788 PCLX-001

Others Others
PCLX-001 is a small-molecule compound that acts as an orally active inhibitor of N-myristoyltransferase (NMT), specifically targeting NMT1 and NMT2 with IC50 values of 5 nM and 8 nM, respectively. This compound demonstrates anti-tumor effects and effectively inhibits the early signaling of B-cell receptor (BCR). Consequently, PCLX-001 is a valuable tool for researching B-cell malignancies [1] [2].
T35330 BTK inhibitor 1

BTK Angiogenesis; Tyrosine Kinase/Adaptors
BTK inhibitor 1 (Compound 27)是一种BTK 抑制剂(IC50:0.11nM),对hWB 中的B 细胞活化具有抑制作用,IC50为2nM。
T60932 MAO-B-IN-8

MAO Metabolism; Neuroscience
MAO-B-IN-8是一种高效且可逆的单胺氧化酶-B(MAO-B)抑制剂,同时也能抑制微胶质细胞产生的神经炎症介质。该化合物专为神经退行性疾病相关研究而设计[1]。
T125100 Pteroside B

Pteroside B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125100。
T14299 AP20187

B/B Homodimerizer

Others Others
AP20187 (B/B Homodimerizer) 是一种细胞渗透性配体,用于二聚化 FK506 结合蛋白 (FKBP) 融合蛋白。它启动生物信号级联和基因表达或破坏蛋白质-蛋白质相互作用。
T10337 Antimicrobial Compound 1

Antibacterial Microbiology/Virology
Antimicrobial Compound 1 是一种烷基吡啶鎓化合物,尾部为 12C,头部为 4-羧基。 Antimicrobial Compound 1 对枯草芽孢杆菌和大肠杆菌具有抗菌活性。
T67879 hMAO-B-IN-5

MAO; Monoamine Oxidase Metabolism; Neuroscience
hMAO-B-IN-5 是有一种有效的、可逆的、具有选择性的人类单胺氧化酶 hMAO-B 抑制剂( IC50 :0.12 μM)。 hMAO-B-IN-5 可以透过血脑屏障,可用于对帕金森疾病的研究,是中枢神经系统疾病的治疗和诊断中都是有潜力的化合物。
T126461 Aloenin B

Aloenin B 是一种从芦荟的叶和根中分离得到的化合物,对谷氨酸诱导的HT22细胞神经元死亡具有神经保护活性。
T39043 Tenofovir amibufenamide

HS-10234

HBV Microbiology/Virology
Tenofovir amibufenamide (HS-10234) (HS-10234) 是一种 Tenofovir 前药,是一种具有口服活性的抗病毒化合物。Tenofovir amibufenamide 对乙型肝炎病毒 (HBV)具有抑制作用,可用于慢性乙型肝炎 (CHB) 研究。
T20641 Propagermanium

Dipropanoic acid germanium sequioxide,SK-818,Ge 132,二羧乙基三氧化二锗,Ge132,SK 818,Ge-132

Others Others
Propagermanium (Ge132) 是一种锗的有机金属化合物,在日本已被用作治疗慢性乙型肝炎的药物。
T67764 hMAO-B-IN-4

MAO Metabolism; Neuroscience
hMAO-B-IN-4 (compound B10) 是一种选择性的、可逆的、血脑屏障通透性 (BBB) 的人单胺氧化-B (hMAO-B) 抑制剂 (IC50= 0.067, Ki= 0.03 μM)。hMAO-B-IN-4 抑制 hMAO-A 的活性较低, IC50 值为 33.82 μM。
T62404 SHMT-IN-2

Others Others
SHMT-IN-2 (compound 2) 是一种特异性人 SHMT1/2 小分子抑制剂,能够作用于 SHMT1 (IC50: 13 nM) 和 SHMT2 (IC50: 66 nM)。SHMT-IN-2 对许多人类癌细胞的生长具有抑制作用,对 B 细胞淋巴瘤具有敏感性。
T67748 ROCK-IN-5

ROCK; ERK Cell Cycle/Checkpoint; Cytoskeletal Signaling; MAPK; Stem Cells
ROCK-IN-5(化合物I-B-37)是一种有效的蛋白激酶抑制剂,包括ROCK、ERK、GSK 和AGC。ROCK-IN-5在心脏病、增殖性疾病和神经退行性疾病研究方面具有潜力。
T77656 LW3

Antifungal Microbiology/Virology
LW3 是一种有效的广谱抗真菌化合物。 LW3 具有抗真菌活性,对 B. cinerea、R. solani、S. sclerotiorum 和 F. graminearum 具有抑制作用, EC50 值分别为 0.54、0.09、1.52 和 2.65 mg/L。
T50009L sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate

Others Others
sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate 是一种有机硫化合物。它已被用作研究含硫化合物对酶活性和代谢途径的影响的模型化合物,也被用于研究含硫化合物对细菌生长和基因表达调控的影响。
T6075 Epothilone B

帕妥匹隆,Patupilone,EPO 906

Apoptosis; Microtubule Associated; Antibiotic; Antifungal Apoptosis; Cytoskeletal Signaling; Microbiology/Virology
Epothilone B (EPO 906) 是微管稳定剂,Ki 为0.71 μM。 它与αβ-微管蛋白异二聚体亚基结合,使αβ-微管蛋白解离减少。
T6998 Tedizolid Phosphate

TR-701FA,Torezolid phosphate,磷酸特地唑胺

Antibacterial; Antibiotic Microbiology/Virology
Tedizolid Phosphate (TR-701FA) 是 MAO-A 和 MAO-B 抑制剂,具有抗革兰氏阳性菌的活性。
T15704 Lagociclovir

MIV-210

HBV Microbiology/Virology
Lagociclovir (MIV-210) 是一种核苷类似物,是一种可用治疗 HBV82的抗病毒化合物,可抑制野生型乙型肝炎病毒 (HBV) 在永久表达 HBV 的人肝癌细胞系中的复制。
T67789 Bazinaprine

MAO Metabolism; Neuroscience
Bazinaprine 是一种选择性的、可逆的单胺氧化酶抑制剂(MAOI),是治疗抑郁症的候选化合物。Bazinaprine 对A 型单胺氧化酶显示出较强的抑制作用,对b 型单胺氧化酶只显示出较弱的抑制作用。Bazinaprine 在体内可逆,但在体外不可逆。
T9518 Inarigivir ammonium

ORI-9020 ammonium,SB-9200 ammonium,Inarigivir铵

HBV Microbiology/Virology
Inarigivir ammonium (SB-9200 ammonium) 是一种二核苷酸抗病毒化合物,可显着降低表达乙型肝炎病毒的转基因小鼠的 HBV DNA。它是一种激活细胞内先天免疫的视黄酸诱导基因-I 激动剂。
T77632 Antiviral agent 34

Antiviral; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation
Antiviral agent 34 是一种可口服且作用效果较强的抗病毒化合物,抑制甲型和乙型流感病毒。Antiviral agent 34 通过调节 RNA 聚合酶来抑制流感病毒的增殖。Antiviral agent 34 可用于研究病毒感染。
T4019 Cambinol

SIRT1/2 Inhibitor IV,NSC 112546

Apoptosis; Phospholipase; Sirtuin Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Cambinol (SIRT1/2 Inhibitor IV) 是一种SIRT1和SIRT2的抑制剂,IC50值分别为 56 μM 和 59 μM。它是中性鞘磷脂酶的外泌体抑制剂。
T61131 MAO-B-IN-11

MAO-B-IN-11, also known as Compound 8c, is a highly potent inhibitor of monoamine oxidase B (MAO-B), with an IC50 value of 1.3 μM. Additionally, MAO-B-IN-11 exhibits neuroprotective properties [1].
T60660 MAO-B-IN-14

MAO-B-IN-14 (Compound 9) 是选择性的单胺氧化酶-B (MAO-B)抑制剂。MAO-B-IN-14 对人 MAO-B 的 IC50值为 0.95 μM,Ki 值为 0.55 μM。
T79895 Cbl-b-IN-8

E1/E2/E3 Enzyme Ubiquitination
Cbl-b-IN-8 (Compound 293),一种casitas B系淋巴瘤(Cbl-b)及c-Cbl的抑制剂,其IC50值分别为5.5 nM和7.8 nM。
T79894 Cbl-b-IN-7

E1/E2/E3 Enzyme Ubiquitination
Cbl-b-IN-7 (Compound 248)作为针对casitas B系淋巴瘤(Cbl-b)和c-Cbl的抑制剂,其IC50值分别为6.7 nM与5.2 nM。
T79896 Cbl-b-IN-9

E1/E2/E3 Enzyme Ubiquitination
Cbl-b-IN-9(Compound 300)为针对casitas B系淋巴瘤(Cbl-b)及c-Cbl的抑制剂,其IC50值分别为5.6 nM与4.7 nM。
T61321 MAO-B-IN-12

MAO-B-IN-12 (Compound 16c) is a highly effective inhibitor of monoamine oxidase B (MAO-B), displaying significant potency with an IC50 value of 1.3 μM. Additionally, MAO-B-IN-12 exhibits notable neuroprotective activity [1].
T79897 Cbl-b-IN-10

E1/E2/E3 Enzyme Ubiquitination
Cbl-b-IN-10(Compound 463)为针对casitas B系淋巴瘤(Cbl-b)和c-Cbl的抑制剂,其IC50值分别为6.0 nM和3.5 nM。
T79893 Cbl-b-IN-6

E1/E2/E3 Enzyme Ubiquitination
Cbl-b-IN-6 (Compound 246),作为casitas B系淋巴瘤(Cbl-b)和c-Cbl的抑制剂,其IC50值分别为5.8 nM和4.4 nM。
T10310 Amphotericin B methyl ester

Others Others
Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses significant antifungal activity. It disrupts HIV-1 particle production and potently inhibits HIV
T61830 MAO-B-IN-10

MAO-B-IN-10 (compound 4f) is a highly potent and selective inhibitor of MAO-B (monoamine oxidase-B). It effectively penetrates the blood-brain barrier and exhibits an IC50 of 5.3 μM. This compound demonstrates the ability to inhibit self-mediated Aβ (amyloid β) aggregation by 58.2% and disaggregate it by 43.3%. Thus, MAO-B-IN-10 holds promise for Alzheimer's disease research [1].
T79898 Cbl-b-IN-11

E1/E2/E3 Enzyme Ubiquitination
Cbl-b-IN-11 (Compound 466)作为casitas B系淋巴瘤 (Cbl-b) 及c-Cbl的抑制剂,显示出对Cbl-b和c-Cbl的高度选择性,其IC50值分别为6.4 nM 和6.1 nM。

化合物

FlutaMide Related CoMpound B
Cat.No: T0547
Synonym:
Target: Others
Memantine Related Compound B
Cat.No: T0535
Synonym: 美金刚杂质B,3,5-Dimethyl-1-adamantanol
Target: Others
PiB
Cat.No: T21000
Synonym: 2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇,Pittsburgh Compound-B,6-OH-BTA-1
Target: Others
Letrozole related compound B
Cat.No: T20683
Synonym: Letrozole specified impurity A
Target:
Clopidogrel Related Compound B
Cat.No: T125846
Synonym:
Target:
NG 52
Cat.No: T2028
Synonym: NG52,NG-52,Compound 52
Target: CDK
Barbaloin-related compound B
Cat.No: T124814
Synonym:
Target:
STOCK2S-26016
Cat.No: T29161
Synonym: WNK IN B,WNK-IN-B,Compound B
Target:
Nav1.1-IN-B
Cat.No: T71716
Synonym:
Target:
Amoxicillin, L-
Cat.No: T23732
Synonym: L-Amoxicillin,Amoxicillin trihydrate impurity B,Amoxicillin related compound B
Target:
Valsartan benzyl ester
Cat.No: T20564
Synonym: Valsartan impurity B,Valsartan related compound C
Target:
PF-05139962
Cat.No: T70782
Synonym:
Target:
6-OH-BTA-0
Cat.No: T29476
Synonym: Pittsburgh Compound-B precursor,11C-PiB Precursor
Target:
Dechloro perphenazine
Cat.No: T69381
Synonym:
Target:
B-Raf IN 2
Cat.No: T40284
Synonym:
Target: Raf
Walrycin B
Cat.No: T1832
Synonym:
Target: Antibacterial, Antibiotic
GDC-6036-NH
Cat.No: T64021
Synonym:
Target: Others
PCLX-001
Cat.No: T63788
Synonym:
Target: Others
BTK inhibitor 1
Cat.No: T35330
Synonym:
Target: BTK
MAO-B-IN-8
Cat.No: T60932
Synonym:
Target: MAO
Pteroside B
Cat.No: T125100
Synonym:
Target:
AP20187
Cat.No: T14299
Synonym: B/B Homodimerizer
Target: Others
Antimicrobial Compound 1
Cat.No: T10337
Synonym:
Target: Antibacterial
hMAO-B-IN-5
Cat.No: T67879
Synonym:
Target: MAO, Monoamine Oxidase
Aloenin B
Cat.No: T126461
Synonym:
Target:
Tenofovir amibufenamide
Cat.No: T39043
Synonym: HS-10234
Target: HBV
Propagermanium
Cat.No: T20641
Synonym: Dipropanoic acid germanium sequioxide,SK-818,Ge 132,二羧乙基三氧化二锗,Ge132,SK 818,Ge-132
Target: Others
hMAO-B-IN-4
Cat.No: T67764
Synonym:
Target: MAO
SHMT-IN-2
Cat.No: T62404
Synonym:
Target: Others
ROCK-IN-5
Cat.No: T67748
Synonym:
Target: ROCK, ERK
LW3
Cat.No: T77656
Synonym:
Target: Antifungal
sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate
Cat.No: T50009L
Synonym:
Target: Others
Epothilone B
Cat.No: T6075
Synonym: 帕妥匹隆,Patupilone,EPO 906
Target: Apoptosis, Microtubule Associated, Antibiotic, Antifungal
Tedizolid Phosphate
Cat.No: T6998
Synonym: TR-701FA,Torezolid phosphate,磷酸特地唑胺
Target: Antibacterial, Antibiotic
Lagociclovir
Cat.No: T15704
Synonym: MIV-210
Target: HBV
Bazinaprine
Cat.No: T67789
Synonym:
Target: MAO
Inarigivir ammonium
Cat.No: T9518
Synonym: ORI-9020 ammonium,SB-9200 ammonium,Inarigivir铵
Target: HBV
Antiviral agent 34
Cat.No: T77632
Synonym:
Target: Antiviral, DNA/RNA Synthesis
Cambinol
Cat.No: T4019
Synonym: SIRT1/2 Inhibitor IV,NSC 112546
Target: Apoptosis, Phospholipase, Sirtuin
MAO-B-IN-11
Cat.No: T61131
Synonym:
Target:
MAO-B-IN-14
Cat.No: T60660
Synonym:
Target:
Cbl-b-IN-8
Cat.No: T79895
Synonym:
Target: E1/E2/E3 Enzyme
Cbl-b-IN-7
Cat.No: T79894
Synonym:
Target: E1/E2/E3 Enzyme
Cbl-b-IN-9
Cat.No: T79896
Synonym:
Target: E1/E2/E3 Enzyme
MAO-B-IN-12
Cat.No: T61321
Synonym:
Target:
Cbl-b-IN-10
Cat.No: T79897
Synonym:
Target: E1/E2/E3 Enzyme
Cbl-b-IN-6
Cat.No: T79893
Synonym:
Target: E1/E2/E3 Enzyme
Amphotericin B methyl ester
Cat.No: T10310
Synonym:
Target: Others
MAO-B-IN-10
Cat.No: T61830
Synonym:
Target:
Cbl-b-IN-11
Cat.No: T79898
Synonym:
Target: E1/E2/E3 Enzyme
Cat. No. Product Name Target Signaling Pathways
T0948L Corticosterone

皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Corticosterone (Kendall's compound B) 是一种肾上腺皮质类固醇,有盐皮质激素和糖皮质激素的活性,具有口服活性。Corticosterone 参与体内能量、免疫反应和应激反应的调节。
T2S0062 Pulchinenoside B

白头翁皂苷B

Compound T2S0062 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T2S0062,CAS号为 135247-95-9。
T4961 9''-Methyl salvianolate B

9'-Methyl lithospermate B,9’-丹酚酸B单甲酯,9''-丹酚酸B单甲酯

Others Others
9'-Methyl lithospermate B 是一种酚类化合物,提取自 RadixSalvia miltiorrhizae。
TN2359 Iristectorigenin B

Iristectrigenin B

Liver X Receptor Metabolism
Iristectorigenin B (Iristectrigenin B) 是一种有效的肝脏 X 受体 (LXR) 调节剂,是从 Belamcanda chinensis 中分离的小分子化合物。Iristectrigenin B 可促进巨噬细胞 RAW 1.1 细胞中 ABCA264 和 ABCG7 的表达。
T22286 Cyanosafracin B

Cyanoquinonamine,氰基番红菌素 B,CBR28-1

Others Others
Cyanosafracin B (Cyanoquinonamine) 是一种合成 Phthalascidin Pt-650 及 Ecteinascidin ET-743 的起始原料。
TN2043 Pasakbumin B

13-alpha-(21)-Epoxyeurycomanone,13ALPHA(21)-环氧宽缨酮

Others Others
Pasakbumin B (13-alpha-(21)-Epoxyeurycomanone) 是一种从 Eurycoma longifoliaJack 中获得的具有生物活性的化合物,显示出抗溃疡作用。
T1922 Pseudolaric Acid B

土槿乙酸B,土荆皮乙酸

Apoptosis; p38 MAPK; Ferroptosis; HBV; Autophagy; Antifungal Apoptosis; Autophagy; MAPK; Microbiology/Virology
Pseudolaric Acid B 是一种从Pseudolarix kaempferiGorden (pinaceae) 根部分离的二萜酸,具有抗癌、抗真菌、抗受精和免疫抑制活性。它还诱导细胞自噬。
TN3628 Chamaejasmenin B

Others Others
Chamaejasmenin B 是一种从 Stellera chamaejasme L 中分离得到的化合物。Chamaejasmenin B 具有抗癌和抗肿瘤活性,可抑制癌细胞迁移和侵袭,抑制肿瘤转移。Chamaejasmenin B 可用于研究如乳腺癌类的癌症。
T3408 Syringin

Lilacin,Syringoside,eleutheroside-b,Methoxyconiferine,紫丁香苷

NOS; Autophagy Autophagy; Immunology/Inflammation
Syringin (eleutheroside-b) 是欧丁香中的一种苯丙素类天然产物,通过抑制自噬来防止压力超载引起的心肌肥厚,具有抗肿瘤、抗增殖、抗骨质疏松、免疫调节和血小板聚集抑制作用。
T3519 Formosanin C

Polyphyllin B,重楼皂苷 B,重楼皂苷B

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Formosanin C (Polyphyllin B) 是从滇重楼中分离的一种薯蓣皂苷,可诱导细胞凋亡。它是一种免疫调节剂,具有抗肿瘤活性。
TN5254 Wighteone

Erythrinin B,6-Isopentenylgenistein

Antifungal Microbiology/Virology
Wighteone (Erythrinin B) 是一种从 Genista ephedroides 中提取出来的小分子化合物,具有潜在的抗真菌和抗癌活性,对 EGFR L858R/T790M 突变非小细胞肺癌具有抗肿瘤作用。。
TN1880 Lucidenic acid B

Lucidenicacid B

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Lucidenic acid B (Lucidenicacid B) 是从灵芝中提取得到的天然化合物,可诱导caspase-9 和 caspase-3 的活化和 PARP 的裂解,可通过线粒体介导诱导人白血病细胞凋亡 。 Lucidenic acid B通过灭活MAPK / ERK信号转导途径和降低NF-kappaB和AP-1的结合活性来抑制PMA诱导的人肝癌细胞侵袭。。Lucidenic acid B 对细胞周期和坏死细胞没有影响。
T8002 3-Hydroxycoumarin

Lipoxygenase Metabolism
3-hydroxycoumarin 是一种 15-LOX-1的有效氧化还原抑制剂,近期被证明能保护海胆生殖细胞免受紫外线 B 的损伤。
T4S0350 Licochalcone B

甘草查尔酮 B,甘草查尔酮B

Beta Amyloid; Others Neuroscience; Others
Licochalcone B 是从Glycyrrhiza inflate 根中提取的。它能够抑制淀粉样蛋白 β 自聚集作用 (IC50=2.16 μM) ,分解预先形成的 Aβ42原纤维,并通过螯合金属离子抑制金属诱导的 Aβ42聚集。
T1040 Vitamin B12

Cyanocobalamin,Cobalamin,维生素B12

Endogenous Metabolite Metabolism
Vitamin B12 (Cobalamin) 是一种维生素,在维持血流形成和脑、神经系统正常功能等方面发挥关键作用。
T83545 (E)-(-)-Aspongopusamide B

(E)-(-)-Aspongopusamide B (Compound 9) 是从昆虫Aspongopus chinensis 分离得到的一种天然产物。
T83271 6-Aldehydoisoophiopogonone B

6-Aldehydoisoophiopogonone B (Compound 24) 是从Ophiopogon japonicus 提取的同型异黄酮化合物。
T81298 Renchangianin B

Renchanginin Bcompound 2)是从Kadsura renchangiana茎中分离得到的一种二苯并环辛烯型木酚素。
T82554 Dihydroisocucurbitacin B

Dihydroisocucurbitacin B为一种源自Wilbrandia ebracteata根部的活性化合物。
T38481 Camellianin B

Camellianin B, a flavonoid compound and metabolite of Camellianin A, exhibits antioxidant properties and acts as an angiotensin converting enzyme (ACE) inhibitor.
T83155 Agonodepside B

Agonodepside B, 分离自非孢子丝状真菌F7524,是一种化合物。
T8174 Saikosaponin F

柴胡皂苷F,柴胡皂苷 F

Others Others
Saikosaponin F 是一种柴胡中的天然成分。
T38837 Microcolin B

Microcolin B, an acylpeptide immunosuppressant, is a highly potent and biologically unique compound containing proline. It is derived from the blue-green alga Lyngbya majuscule.
T81742 Mulberrofuran B

Mulberrofuran B,一种从Morus alba乙醇提取物中分离得到的化合物,展现了抗氧化活性。
T80702 α-Thevetin B

α-Thevetin BCompound 24), 一种从Thevetia peruviana分离得到的心脏苷,用于肺癌、胃癌和胰腺癌的研究。
T40383 Monensin B

Monensin B is a polyketide compound derived from the bacterium Streptomyces cinnamonensis. Its production involves the fermentation of Streptomyces cinnamonensis, resulting in a mixture of Monensin A and Monensin B. The ratio of these two compounds depends on the concentrations of ethylmalonyl-CoA and methylmalonyl-CoA.
T80000 Multiflorin B

NO Synthase Immunology/Inflammation
Multiflorin B为一种山奈酚苷,源自蕨类植物Neocheiropteris palmatopedata的根部提取。在20 μg/ml的浓度下,Multiflorin B能够抑制一氧化氮的生成,其抑制率达到52%。
T82396 Fissitungfine B

Fissitungfine B,一种从热带药用植物Fissistigma tungfangense提取的化合物,展示出显著的抗癌活性。
T82302 Glucodichotomine B

Glucodichotomine B (Compound 13) 是一种从中药植物 Stellaria dichotoma L. var. lanceolata 根中分离得到的天然产物,具有抗癌活性。
T83459 11α-O-Tigloyl-12β-O-acetyltenacigenin B

Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic
11α-O-Tigloyl-12β-O-acetyltenacigenin B 是Tenacigenin B 的酯类衍生物,源自藤黄藤 (MTC)。该化合物具有调节Aurora-A活性,对淋巴瘤显示出潜在的抗肿瘤效果。
TN2408 Evofolin B

Cannabinoid Receptor GPCR/G Protein
Evofolin B 是从Zanthoxylum ailanthoides 的茎皮中分离出来的天然化合物。Evofolin B 对人类中性粒细胞对甲酰-L-蛋氨酸-L-亮氨酸-L-苯丙氨酸/cytochalasin B(fMLP/CB)产生的超氧阴离子有抑制作用。
T80860 Vitisin B

(-)-Vitisin B,E-Vitisin B

Vitisin B,从Vitis thunbergii var. taiwaniana分离提取,对脂多糖(LPS)诱导的关节炎表现出抗炎活性。
T38609 Mycalolide B

Mycalolide-B is a marine sponge-derived compound that functions as a selective inhibitor of actomyosin ATPase. It effectively hinders ATP-induced contraction and Mg2+-ATPase activity in the absence of Ca2+.
T74196 Inophyllum B

Inophyllum B ((+)-Inophyllum B) 是一种有效的HIV 逆转录酶 (Reverse Transcriptase) 抑制剂,IC50为 38 nM。Inophyllum B 在体外细胞培养中抑制HIV-1(IC50=1.4 μM)。Inophyllum B 可从非洲大蜗牛Achatina fulica 的丙酮提取物中分离得到。
T81169 Shishijimicin B

Shishijimicin B为活性的烯二炔类化合物,具有强烈的细胞毒性,IC50值介于2.0 - 3.3 nM。此化合物表现出抗肿瘤活性,常用于癌症研究中。作为点击化学试剂,Shishijimicin B内含Alkyne基团,能通过含Azide基团的分子在铜催化下发生(CuAAc)反应。
T82445 Erinacine P

Erinacine P(化合物1)为担子菌猴头菇YB4-6237菌丝体分离得到的木犀草素亲代代谢产物。其在温和条件下可化学转化为猴头素B,继而可转化为猴头素A。
TN4605 Myriceric acid B

HIV Protease Microbiology/Virology; Proteases/Proteasome
Myriceric acid B is a potent HIV-1 entry inhibitor targeting gp41 and can serve as a lead compound for developing novel anti-HIV-1 drug. Myriceric acid B scavenges DPPH free radicals with IC50 value of 21.8 uM, it inhibits aromatase activity with IC50 val
T75692 Hypoglaunine D

Hypoglaunine D 是 Triptonine B 的类似物,是一种抗HIV 的化合物,Hypoglaunine D 抑制 H9 淋巴细胞中HIV 病毒复制的EC50值为 22 μg/ml。
T82983 Aplyronine B

Aplyronine B是一种具有抗肿瘤活性的活性化合物,对HeLa-S3细胞表现出细胞毒性,IC50值为2.9 nM,适用于癌症研究。
T81321 Quercetin-3-O-b-D-galactopyranosyl-(1→6)-b-D-glucopyranoside

Quercetin-3-O-b-D-galactopyranosyl-(1→6)-b-D-glucopyranoside (化合物 1),为自白仙茅 (M. delavayi) 叶中分离的黄酮甙类化合物。
T81095 Stenophyllol B

Stenophyllol B (compound 4) 是一种具有双环及桥联三环骨架的三聚芪类化合物。该化合物最初在龙脑香科植物中被鉴定,随后在Hopea、Neobalanocarpus、Shorea、Stemonoporus以及Vateri等属的多种物种中发现。
T72916 Justicidin B

爵床脂素B

Justicidin B是一种高效的抗癌木脂素及促凋亡剂,同时具备显著的骨吸收抑制作用,并展现出强大的抗病毒、杀真菌和抗原虫能力。此外,Justicidin B能显着抑制血小板聚集。
T75468 Asperglaucin B

Asperglaucin B 是一种来自真菌Aspergillus chevalieriSQ-8 的烷基化水杨醛衍生物,具有抗菌活性。Asperglaucin B 对两种植物病原体Pseudomonas syringae pv actinidae(Psa)和Bacillus cereus 显示出有效的抗菌活性,MIC 值为 6.25 μM。
T79949 Foenumoside B

PPAR DNA Damage/DNA Repair; Metabolism
Foenumoside B为从Lysimachia foenum-graecum中提取的三萜皂苷。该化合物通过激活AMPK信号传导和抑制PPARγ诱导的脂肪生成,调节脂质代谢向脂肪分解方向转变。因其调控作用,Foenumoside B常用于研究肥胖及相关代谢疾病。
T81856 Marsdenoside B

Marsdenoside B(化合物8), 一种海芋属植物中的提取物,显示对MGC-803和HT-29肿瘤细胞系具有抑制作用,其IC50s 分别为25.6 μg/mL 和32.4 μg/mL。
T79970 Taxamairin B

Taxamairin B是有效的抗炎化合物,能显著抑制LPS诱导的RAW264.7细胞中促炎因子(TNF-α, IL-1β和IL-6)表达及NO、ROS生成,并对LPS引起的急性肺损伤模型小鼠具有保护效果。
T83903 Polymyxin B2 sulfate

Polymyxin B2是一种抗生素,并且是从B. polymyxa分离出的阳离子脂肽抗生素polymyxin B的主要成分。该化合物对P. aeruginosa、A. baumannii、K. pneumoniae和E. cloacae菌株具有活性(MICs分别为1-2、0.5-1、0.25-0.5和0.25-1 µg/ml)。在体内实验中,以4 mg/kg剂量的Polymyxin B2能显著降低P. aeruginosa血液感染小鼠模型中的血液集落形成单位(CFUs)数量。
T31471 Dihydroisoalantolactone

Dihydroisoalantolactone is found in herbs and spices. Dihydroisoalantolactone is isolated from roots of Inula helenium (elecampane). This compound Aliphatic heteropolycyclic, belongs to the class of organic compounds known as eudesmanolides, secoeudesmano
T79976 Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside

HBV Microbiology/Virology
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside 作为一种抗HBV剂,在Hep G2.2.15细胞系上能够抑制HBsAg和HBeAg的分泌,其IC50值分别约为1.67 mM和>2.15 mM。
T81201 Sartorypyrone B

Sartorypyrone B为Chevalone C的2β-乙酰氧基衍生物,由海绵源真菌Neosartorya tsunodae(KUFC 9213)的培养物中乙酸乙酯提取得到。该化合物对MCF-7、NCI-H460和A375-C5细胞系展示出较强的生长抑制活性,GI50s值分别为17.8、20.5和25.0 μM,显示其在乳腺癌、非小细胞肺癌和黑色素瘤研究中的应用潜力。
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天然产物

Corticosterone
Cat.No: T0948L
Synonym: 皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)
Target: Glucocorticoid Receptor, Endogenous Metabolite
Pulchinenoside B
Cat.No: T2S0062
Synonym: 白头翁皂苷B
Target:
9''-Methyl salvianolate B
Cat.No: T4961
Synonym: 9'-Methyl lithospermate B,9’-丹酚酸B单甲酯,9''-丹酚酸B单甲酯
Target: Others
Iristectorigenin B
Cat.No: TN2359
Synonym: Iristectrigenin B
Target: Liver X Receptor
Cyanosafracin B
Cat.No: T22286
Synonym: Cyanoquinonamine,氰基番红菌素 B,CBR28-1
Target: Others
Pasakbumin B
Cat.No: TN2043
Synonym: 13-alpha-(21)-Epoxyeurycomanone,13ALPHA(21)-环氧宽缨酮
Target: Others
Pseudolaric Acid B
Cat.No: T1922
Synonym: 土槿乙酸B,土荆皮乙酸
Target: Apoptosis, p38 MAPK, Ferroptosis, HBV, Autophagy, Antifungal
Chamaejasmenin B
Cat.No: TN3628
Synonym:
Target: Others
Syringin
Cat.No: T3408
Synonym: Lilacin,Syringoside,eleutheroside-b,Methoxyconiferine,紫丁香苷
Target: NOS, Autophagy
Formosanin C
Cat.No: T3519
Synonym: Polyphyllin B,重楼皂苷 B,重楼皂苷B
Target: Apoptosis, Caspase
Wighteone
Cat.No: TN5254
Synonym: Erythrinin B,6-Isopentenylgenistein
Target: Antifungal
Lucidenic acid B
Cat.No: TN1880
Synonym: Lucidenicacid B
Target: Apoptosis, Caspase
3-Hydroxycoumarin
Cat.No: T8002
Synonym:
Target: Lipoxygenase
Licochalcone B
Cat.No: T4S0350
Synonym: 甘草查尔酮 B,甘草查尔酮B
Target: Beta Amyloid, Others
Vitamin B12
Cat.No: T1040
Synonym: Cyanocobalamin,Cobalamin,维生素B12
Target: Endogenous Metabolite
(E)-(-)-Aspongopusamide B
Cat.No: T83545
Synonym:
Target:
6-Aldehydoisoophiopogonone B
Cat.No: T83271
Synonym:
Target:
Renchangianin B
Cat.No: T81298
Synonym:
Target:
Dihydroisocucurbitacin B
Cat.No: T82554
Synonym:
Target:
Camellianin B
Cat.No: T38481
Synonym:
Target:
Agonodepside B
Cat.No: T83155
Synonym:
Target:
Saikosaponin F
Cat.No: T8174
Synonym: 柴胡皂苷F,柴胡皂苷 F
Target: Others
Microcolin B
Cat.No: T38837
Synonym:
Target:
Mulberrofuran B
Cat.No: T81742
Synonym:
Target:
α-Thevetin B
Cat.No: T80702
Synonym:
Target:
Monensin B
Cat.No: T40383
Synonym:
Target:
Multiflorin B
Cat.No: T80000
Synonym:
Target: NO Synthase
Fissitungfine B
Cat.No: T82396
Synonym:
Target:
Glucodichotomine B
Cat.No: T82302
Synonym:
Target:
11α-O-Tigloyl-12β-O-acetyltenacigenin B
Cat.No: T83459
Synonym:
Target: Aurora Kinase
Evofolin B
Cat.No: TN2408
Synonym:
Target: Cannabinoid Receptor
Vitisin B
Cat.No: T80860
Synonym: (-)-Vitisin B,E-Vitisin B
Target:
Mycalolide B
Cat.No: T38609
Synonym:
Target:
Inophyllum B
Cat.No: T74196
Synonym:
Target:
Shishijimicin B
Cat.No: T81169
Synonym:
Target:
Erinacine P
Cat.No: T82445
Synonym:
Target:
Myriceric acid B
Cat.No: TN4605
Synonym:
Target: HIV Protease
Hypoglaunine D
Cat.No: T75692
Synonym:
Target:
Aplyronine B
Cat.No: T82983
Synonym:
Target:
Quercetin-3-O-b-D-galactopyranosyl-(1→6)-b-D-glucopyranoside
Cat.No: T81321
Synonym:
Target:
Stenophyllol B
Cat.No: T81095
Synonym:
Target:
Justicidin B
Cat.No: T72916
Synonym: 爵床脂素B
Target:
Asperglaucin B
Cat.No: T75468
Synonym:
Target:
Foenumoside B
Cat.No: T79949
Synonym:
Target: PPAR
Marsdenoside B
Cat.No: T81856
Synonym:
Target:
Taxamairin B
Cat.No: T79970
Synonym:
Target:
Polymyxin B2 sulfate
Cat.No: T83903
Synonym:
Target:
Dihydroisoalantolactone
Cat.No: T31471
Synonym:
Target:
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside
Cat.No: T79976
Synonym:
Target: HBV
Sartorypyrone B
Cat.No: T81201
Synonym:
Target:
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