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Targets Recommended: Others

121

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TP1024 Rusalatide acetate (497221-38-2 free base)

Rusalatide acetate,TP508 amide acetate

Others Others
Rusalatide acetate (TP508 amide acetate) 是一种再生肽,可诱导干细胞再生修复,保护隐窝完整性,减缓辐照引起的胃肠道损伤。
T12107 MRS-3777 hemioxalate

Adenosine Receptor GPCR/G Protein; Neuroscience
MRS-3777 hemioxalate 是一种选择性腺苷 A3 受体拮抗剂,可逆转其相应激动剂的抗伤害感受作用,可用于研究炎症性疼痛。
T0374 Sunitinib Malate

苏尼替尼苹果酸盐,Sutent,SU 11248 (Malate),SU 11248,Sunitinib

Apoptosis; Mitophagy; VEGFR; FLT; IRE1; PDGFR; c-Kit; Autophagy Angiogenesis; Apoptosis; Autophagy; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors
Sunitinib Malate (Sunitinib) 是一种基于吲哚酮的酪氨酸激酶抑制剂,抑制 VEGFR2和 PDGFRβ的 IC50分别为80 nM 和 2 nM。它是 ATP 竞争性抑制剂,可通过抑制自身磷酸化和随后的 RNase 激活来有效抑制 Ire1α的磷酸化。
T13353 Xanomeline oxalate

LY246708 oxalate

AChR Neuroscience
Xanomeline oxalate (LY246708 oxalate)作为一种高效且选择性的胆碱能受体激动剂(SMRA),在体内有效促进磷脂酰肌醇水解。Xanomeline oxalate 对于阿尔茨海默病的研究具有重要价值。
T6120 Pralatrexate

Folotyn,10-炔丙基-10-去氮杂氨基蝶呤,10-Propargyl-10-deazaaminopterin,普拉曲沙

Apoptosis; DHFR; Antifolate; TAM Receptor Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Tyrosine Kinase/Adaptors
Pralatrexate (10-Propargyl-10-deazaaminopterin) 是一种抗叶酸剂,也是二氢叶酸还原酶抑制剂,Ki 值为 13.4 pM。它具有抗肿瘤活性,可研究复发/难治性 T 细胞淋巴瘤。它是叶酰聚谷氨酸合成酶的底物,具有改善的细胞摄取和保留能力。
T3355 Naloxegol oxalate

NKTR-118,NKTR-118 oxalate,AZ 13337019,AZ-13337019 oxalate

P450 Metabolism
Naloxegol oxalate (NKTR-118) 是一种外周选择性 opioid 样物质拮抗剂,用于治疗 opioid 样物质引起的便秘。
T68067L Etilefrine pivalate HCl

Etilefrine pivalate HCl(100696-30-8 Free base)

Etilefrine pivalate HCl 是一种具有口服活性的化合物,可用于治疗偏头痛。
T0601 Monobenzyl phthalate

邻苯二甲酸单苄酯,Phthalic Acid Monobenzyl Ester

Others; Endogenous Metabolite Metabolism; Others
Monobenzyl phthalate (Phthalic Acid Monobenzyl Ester) 是一种暴露于邻苯二甲酸盐(如,邻苯二甲酸二乙基己酯)后的尿代谢物 (urinary metabolite)。
T20168 Aurothiomalate sodium

金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate

Others; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Others
Aurothiomalate sodium (Miochrysin) 是一种选择性的致癌 PKCι信号传导抑制剂,可抑制肿瘤细胞增殖。它是一种硫氧还蛋白还原酶 (TrxR) 抑制剂,也是一种抗风湿剂。
T20802 Flumethasone pivalate

Locacorten,NSC-107680,特戊酸氟米松,Lorinden,NSC 107680,NSC107680,Locorten

Others Others
Flumethasone pivalate (Locorten) 具有止痒、抗炎和血管收缩的特性,可用于肾上腺皮质抑制、皮肤萎缩、血浆转皮质素结合和毛细血管扩张的研究。
T24588 Palatrigine

BW-A 256C,BW A256C

Adrenergic Receptor; Angiotensin-converting Enzyme (ACE) GPCR/G Protein; Metabolism; Neuroscience
Palatrigine (BW-A 256C) 是一种具有血管紧张素转换酶抑制和β肾上腺素受体阻断特性的化合物。
T1081 Naftidrofuryl oxalate

萘呋胺酯 草酸盐,Nafronyl oxalate,Nafronyl oxalate salt

5-HT Receptor GPCR/G Protein; Neuroscience
Naftidrofuryl oxalate (Nafronyl oxalate) 是一种用于治疗外周和脑血管疾病的药物,可增加细胞氧化能力,也是一种 5-HT2 受体拮抗剂。
T3608 Carbasalate calcium

Rheomin,Omegin,Alcacyl,Iromin,卡巴匹林钙,Solupsan,Carbasalate Calcium

Platelet aggregation Others
Carbasalate calcium (Rheomin) 是抗炎和解热剂,可用于研究疼痛的缓解。
T0225 Pizotifen Malate

Pizotyline (malate),BC-105 (malate),BC-105,苯噻啶苹果酸盐

5-HT Receptor GPCR/G Protein; Neuroscience
Pizotifen Malate (BC-105 malate) 是5-HT2受体的拮抗剂,对5-HT1C 有高亲和力。
T7420 Valifenalate

霜霉灭,Valiphenal,IR5885

Antibacterial Microbiology/Virology
Valifenalate (IR5885) 是一种抗真菌剂,对各种类型的霉菌都有效,可用于葡萄,西红柿和其他蔬菜等高价值作物防护。
T16007 MALAT1-IN-1

Others Others
MALAT1-IN-1 是Malat1(转移相关的肺腺癌转录本 1) 的特异性抑制剂。它能够以剂量依赖性方式调节Malat1下游基因,但对Neat1(富核丰富转录本 1) 的表达无影响。
T20322 Diisopropyl phthalate

NSC15315,NSC 15315,NSC-15315

Others Others
Diisopropyl phthalate 广泛用作化学工业中塑料和消费品的添加剂。
T1797 Cabozantinib S-malate

苹果酸卡博替尼,Cabozantinib,卡博替尼苹果酸盐,XL184,Cabozantinib Malate

Apoptosis; VEGFR; c-Met/HGFR; TAM Receptor; c-Kit Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Cabozantinib S-malate (XL184) 是一种多受体酪氨酸激酶抑制剂, 抑制VEGFR2,c-Met,Kit,Axl 和Flt3的IC50分别为0.035,1.3,4.6,7 和 11.3 nM。
T0498 Salsalate

Disalicylic acid,Salicylsalicylic acid,Sasapyrine,NSC-49171,双水杨酸酯

Reactive Oxygen Species; COX Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Salsalate (Sasapyrine) 是一种有效的抗风湿药物,是一种非乙酰化水杨酸盐,可以绕过胃的吸收,也可以避免环氧合酶的抑制。它具有抗炎活性,降低血糖水平、胰岛素抵抗和细胞因子表达,可用于研究 2 型糖尿病。
TD0099 Malachite green oxalate

Apoptosis; Others; IκB/IKK; NF-κB Apoptosis; NF-κB; Others
Malachite green oxalate 是一种三苯基甲烷染料,可用于检测酶促反应中磷酸盐的释放。它也是一种选择性IKBKE 抑制剂,在体内外均表现出抗肿瘤活性。
T0071 Homosalate

Homomenthyl salicylate,原膜散酯,胡莫柳酯

Others Others
Homosalate (Homomenthyl salicylate) 是一种有机防晒剂,能够过滤紫外线,保护皮肤免受阳光损伤。
T0640 Benzyl butyl phthalate

BBP,邻苯二甲酸丁苄酯,1,2-benzenedicarboxylic acid,butyl phenylmethyl ester,Butyl benzyl phthalate

Others; Aryl Hydrocarbon Receptor Immunology/Inflammation; Others
Benzyl butyl phthalate (1,2-benzenedicarboxylic acid) 是邻苯二甲酸酯的一员,可激活乳腺癌细胞中的芳香烃受体,刺激 SPHK1/S1P/S1PR3 信号传导,促进转移性乳腺癌干细胞的形成。它通过上调 Zeb1 的表达,可引起血管瘤细胞的迁移和侵袭。
T39211 PD 144418 oxalate

Sigma receptor GPCR/G Protein
PD 144418 oxalate is a highly potent and selective sigma 1 (σ1) receptor ligand, displaying a Ki value of 0.08 nM for σ1 and 1377 nM for σ2. It exhibits negligible affinity for other receptors, ion channels, and enzymes. Additionally, PD 144418 oxalate demonstrates potential antipsychotic activity.
T0027 Octisalate

水杨酸辛酯,2-Ethylhexyl salicylate,Octyl salicylate

Others Others
Octisalate (Octyl salicylate) 能够吸收 UVB 射线,可用于防晒剂和化妆品。
T19282 Diisohexyl phthalate

Others Others
Diisohexyl phthalate 是一种可用作增塑剂的邻苯二甲酸二烷基酯。
T6353 (-)-p-Bromotetramisole Oxalate

(-)-对溴四咪唑草酸盐,L-p-Bromotetramisole oxalate,6-Bromolevamisole oxalate,(-)-p-Bromolevamisole oxalate

Phosphatase; Phosphorylase Metabolism
(-)-p-Bromotetramisole Oxalate (6-Bromolevamisole oxalate) 是一种强效的、非特异性碱性磷酸酶抑制剂。
T31932 GJ071 oxalate

GJ 071,GJ-071,GJ071

Others Others
GJ071 oxalate 是一种无义抑制剂。无义抑制剂(NonSups)诱导“读出”,即在提前终止密码子处选择近同源tRNA,并将相应的氨基酸插入新生多肽中。
T7569 Clebopride malate

苹果酸氯波必利,氯波必利

Dopamine Receptor GPCR/G Protein; Neuroscience
Clebopride malate 是多巴胺拮抗剂,可用于功能性胃肠功能紊乱的研究。
T2317 Almotriptan Malate

LAS 31416,PNU180638,马来酸阿莫曲坦

5-HT Receptor GPCR/G Protein; Neuroscience
Almotriptan Malate (PNU180638) 是一种选择性 5-HT1B/1D 受体激动剂,用于治疗成人偏头痛发作。
T6493 Escitalopram Oxalate

草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate

Others; 5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience; Others
Escitalopram Oxalate ((S)-(+)Citalopram oxalate) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。
T22514 4F 4PP oxalate

5-HT Receptor GPCR/G Protein; Neuroscience
4F 4PP oxalate 是一种选择性5-HT2A 拮抗剂。
T67063 4-Amino-4-methyl-2-pentanone oxalate

4-Amino-4-methyl-2-pentanone oxalate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67063,CAS号为 625-03-6。
T27771 L-703606 Oxalate

L 703606,L703,606,L-703,606,L703606,L 703,606,L-703606

L-703,606 is a potent, selective human NK1 receptor antagonist.
T25981 Pralatrexate, (S)-

Pralatrexate, (S)- is a folate analog dihydrofolate reductase (DHFR) inhibitor exhibiting high affinity for reduced folate carrier-1 (RFC-1) with antineoplastic and immunosuppressive activities. Pralatrexate selectively enters cells expressing RFC-1; intr
T124567 Alatolin

Alatolin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124567,CAS号为 60389-86-8。
T20274 Dibenzyl phthalate

AI300364,AI3-00364

Dibenzyl phthalate is an endocrine-disrupting chemical. It also interferes with different cell signaling pathways involved in weight and glucose homeostasis.
T12738 Rivanicline hemioxalate

RJR-2403 hemioxalate,(E)-Metanicotine hemioxalate

Others Others
Rivanicline hemioxalate (RJR-2403 hemioxalate; (E)-Metanicotine hemioxalate) 是一种神经元烟碱受体 (neuronal nicotinic receptor) 激动剂,对 α4β2 亚型有高度选择性(Ki= 26 nM),比对于 α7 受体的选择性高1000倍(Ki=3.6 μM)。
T37012 (±)-PPCC oxalate

(±)-PPCC (oxalate) 是 sigma-1 激动剂,能与 sigma-1 受体相互作用(Ki=1.5 nM)。(±)-PPCC (oxalate) 在有认知障碍的大鼠中具有抗遗忘作用,可以改善大鼠的认知能力。
T40060 Nicotinamide riboside malate

Nicotinamide riboside malate is an orally active NAD+ precursor that elevates NAD+ levels and stimulates the activity of SIRT1 and SIRT3. Functioning as a vitamin B3 (niacin) source, it augments oxidative metabolism and provides protection against metabolic abnormalities induced by a high-fat diet. Additionally, Nicotinamide riboside malate mitigates cognitive decline in a genetically modified mouse model of Alzheimer's disease.
T65547 4-(Chlorosulfonyl)phenyl pivalate

4-(Chlorosulfonyl)phenyl pivalate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65547,CAS号为 150374-99-5。
T74010 (Rac)-Mono(3,5,5-trimethylhexyl) phthalate

(Rac)-Mono(3,5,5-trimethylhexyl) phthalate 为常见邻苯二甲酸酯增塑剂的关键代谢物,具备免疫抑制功能。
TP2394 Nifalatide

Nifalatide is a analog of enkephalin.
T35713 N-desethyl Brinzolamide (oxalate)

N-desethyl Brinzolamide is an active metabolite of the carbonic anhydrase (CA) inhibitor brinzolamide .1It inhibits CAII and CAIV activities (IC50s = 1.28 and 128 nM, respectively). 1.Kim, C.-Y., Whittington, D.A., Chang, J.S., et al.Structural aspects of isozyme selectivity in the binding of inhibitors to carbonic anhydrases II and IVJ. Med. Chem.45(4)888-893(2002)
T37013 (+/-)-PPCC oxalate

Selective sigma (σ) receptor ligand. Displays high affinity for σ1; also binds at σ2 sites (Ki = 1.5 nM and 50.8 nM respectively). Selective over a range of receptor types including dopaminergic and muscarinic receptors, DAT and SERT. Prezzavento et al (2007) Novel sigma receptor ligands: synthesis and biological profile. J.Med.Chem. 50 951 PMID:17328523 |Prezzavento et al (2008) A new sigma ligand, (±)-PPCC, antagonizes kappa opioid receptor-mediated antinociceptive effect. Life Sci. 82 549 PMI...
T71600 Benazoline oxalate salt

Benazoline oxalate salt is a pharmacological active compound that inhibits casein kinase Iε (CKIε) or CKIδ phosphorylation of the PER2 protein.
T28154 Nemonoxacin Malate

TG-873870,TG873870,TG 873870

Nemonoxacin is a non-fluorinated quinolone antibiotic.
T20349 Diethyl terephthalate

NSC-68816,NSC68816,NSC 68816

Diethyl terephthalate is an agent that is used in the production of polyesters.
T10835L Cletoquine oxalate

Desethylhydroxychloroquine oxalate

Others Others
Cletoquine oxalate (Desethylhydroxychloroquine oxalate) is a major active metabolite of Hydroxychloroquine. Cletoquine has the ability to against the chikungunya virus (CHIKV). Cletoquine has antimalarial effects and has the potential for autoimmune disea
T12739 Rivanicline oxalate

RJR-2403 oxalate,(E)-Metanicotine oxalate

Others Others
Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).
T13007 ST1936 oxalate

5-HT Receptor GPCR/G Protein; Neuroscience
ST1936 oxalate 是一种 5-HT6 受体的选择性纳摩尔亲和激动剂,对人5-HT6、5-HT7和 5-HT2B 受体的 Ki 值分别为 13、168 和 245 nM。

化合物

Rusalatide acetate (497221-38-2 free base)
Cat.No: TP1024
Synonym: Rusalatide acetate,TP508 amide acetate
Target: Others
MRS-3777 hemioxalate
Cat.No: T12107
Synonym:
Target: Adenosine Receptor
Sunitinib Malate
Cat.No: T0374
Synonym: 苏尼替尼苹果酸盐,Sutent,SU 11248 (Malate),SU 11248,Sunitinib
Target: Apoptosis, Mitophagy, VEGFR, FLT, IRE1, PDGFR, c-Kit, Autophagy
Xanomeline oxalate
Cat.No: T13353
Synonym: LY246708 oxalate
Target: AChR
Pralatrexate
Cat.No: T6120
Synonym: Folotyn,10-炔丙基-10-去氮杂氨基蝶呤,10-Propargyl-10-deazaaminopterin,普拉曲沙
Target: Apoptosis, DHFR, Antifolate, TAM Receptor
Naloxegol oxalate
Cat.No: T3355
Synonym: NKTR-118,NKTR-118 oxalate,AZ 13337019,AZ-13337019 oxalate
Target: P450
Etilefrine pivalate HCl
Cat.No: T68067L
Synonym: Etilefrine pivalate HCl(100696-30-8 Free base)
Target:
Monobenzyl phthalate
Cat.No: T0601
Synonym: 邻苯二甲酸单苄酯,Phthalic Acid Monobenzyl Ester
Target: Others, Endogenous Metabolite
Aurothiomalate sodium
Cat.No: T20168
Synonym: 金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate
Target: Others, PKC
Flumethasone pivalate
Cat.No: T20802
Synonym: Locacorten,NSC-107680,特戊酸氟米松,Lorinden,NSC 107680,NSC107680,Locorten
Target: Others
Palatrigine
Cat.No: T24588
Synonym: BW-A 256C,BW A256C
Target: Adrenergic Receptor, Angiotensin-converting Enzyme (ACE)
Naftidrofuryl oxalate
Cat.No: T1081
Synonym: 萘呋胺酯 草酸盐,Nafronyl oxalate,Nafronyl oxalate salt
Target: 5-HT Receptor
Carbasalate calcium
Cat.No: T3608
Synonym: Rheomin,Omegin,Alcacyl,Iromin,卡巴匹林钙,Solupsan,Carbasalate Calcium
Target: Platelet aggregation
Pizotifen Malate
Cat.No: T0225
Synonym: Pizotyline (malate),BC-105 (malate),BC-105,苯噻啶苹果酸盐
Target: 5-HT Receptor
Valifenalate
Cat.No: T7420
Synonym: 霜霉灭,Valiphenal,IR5885
Target: Antibacterial
MALAT1-IN-1
Cat.No: T16007
Synonym:
Target: Others
Diisopropyl phthalate
Cat.No: T20322
Synonym: NSC15315,NSC 15315,NSC-15315
Target: Others
Cabozantinib S-malate
Cat.No: T1797
Synonym: 苹果酸卡博替尼,Cabozantinib,卡博替尼苹果酸盐,XL184,Cabozantinib Malate
Target: Apoptosis, VEGFR, c-Met/HGFR, TAM Receptor, c-Kit
Salsalate
Cat.No: T0498
Synonym: Disalicylic acid,Salicylsalicylic acid,Sasapyrine,NSC-49171,双水杨酸酯
Target: Reactive Oxygen Species, COX
Malachite green oxalate
Cat.No: TD0099
Synonym:
Target: Apoptosis, Others, IκB/IKK, NF-κB
Homosalate
Cat.No: T0071
Synonym: Homomenthyl salicylate,原膜散酯,胡莫柳酯
Target: Others
Benzyl butyl phthalate
Cat.No: T0640
Synonym: BBP,邻苯二甲酸丁苄酯,1,2-benzenedicarboxylic acid,butyl phenylmethyl ester,Butyl benzyl phthalate
Target: Others, Aryl Hydrocarbon Receptor
PD 144418 oxalate
Cat.No: T39211
Synonym:
Target: Sigma receptor
Octisalate
Cat.No: T0027
Synonym: 水杨酸辛酯,2-Ethylhexyl salicylate,Octyl salicylate
Target: Others
Diisohexyl phthalate
Cat.No: T19282
Synonym:
Target: Others
(-)-p-Bromotetramisole Oxalate
Cat.No: T6353
Synonym: (-)-对溴四咪唑草酸盐,L-p-Bromotetramisole oxalate,6-Bromolevamisole oxalate,(-)-p-Bromolevamisole oxalate
Target: Phosphatase, Phosphorylase
GJ071 oxalate
Cat.No: T31932
Synonym: GJ 071,GJ-071,GJ071
Target: Others
Clebopride malate
Cat.No: T7569
Synonym: 苹果酸氯波必利,氯波必利
Target: Dopamine Receptor
Almotriptan Malate
Cat.No: T2317
Synonym: LAS 31416,PNU180638,马来酸阿莫曲坦
Target: 5-HT Receptor
Escitalopram Oxalate
Cat.No: T6493
Synonym: 草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate
Target: Others, 5-HT Receptor, Serotonin Transporter
4F 4PP oxalate
Cat.No: T22514
Synonym:
Target: 5-HT Receptor
4-Amino-4-methyl-2-pentanone oxalate
Cat.No: T67063
Synonym:
Target:
L-703606 Oxalate
Cat.No: T27771
Synonym: L 703606,L703,606,L-703,606,L703606,L 703,606,L-703606
Target:
Pralatrexate, (S)-
Cat.No: T25981
Synonym:
Target:
Alatolin
Cat.No: T124567
Synonym:
Target:
Dibenzyl phthalate
Cat.No: T20274
Synonym: AI300364,AI3-00364
Target:
Rivanicline hemioxalate
Cat.No: T12738
Synonym: RJR-2403 hemioxalate,(E)-Metanicotine hemioxalate
Target: Others
(±)-PPCC oxalate
Cat.No: T37012
Synonym:
Target:
Nicotinamide riboside malate
Cat.No: T40060
Synonym:
Target:
4-(Chlorosulfonyl)phenyl pivalate
Cat.No: T65547
Synonym:
Target:
(Rac)-Mono(3,5,5-trimethylhexyl) phthalate
Cat.No: T74010
Synonym:
Target:
Nifalatide
Cat.No: TP2394
Synonym:
Target:
N-desethyl Brinzolamide (oxalate)
Cat.No: T35713
Synonym:
Target:
(+/-)-PPCC oxalate
Cat.No: T37013
Synonym:
Target:
Benazoline oxalate salt
Cat.No: T71600
Synonym:
Target:
Nemonoxacin Malate
Cat.No: T28154
Synonym: TG-873870,TG873870,TG 873870
Target:
Diethyl terephthalate
Cat.No: T20349
Synonym: NSC-68816,NSC68816,NSC 68816
Target:
Cletoquine oxalate
Cat.No: T10835L
Synonym: Desethylhydroxychloroquine oxalate
Target: Others
Rivanicline oxalate
Cat.No: T12739
Synonym: RJR-2403 oxalate,(E)-Metanicotine oxalate
Target: Others
ST1936 oxalate
Cat.No: T13007
Synonym:
Target: 5-HT Receptor
Cat. No. Product Name Target Signaling Pathways
T8319 Butyl isobutyl phthalate

ButylIsobutylPhthalate,邻苯二甲酸-1-丁酯-2-异丁酯

Glucosidase Metabolism
Butyl isobutyl phthalate (ButylIsobutylPhthalate) 是一种非竞争性 α-葡萄糖苷酶抑制剂,IC50=38 μM,可以从海带的根状茎中分离得到。它具有降血糖作用,可用于糖尿病相关的研究。
T5112 DI-N-OCTYL PHTHALATE

Others Others
DI-N-OCTYL PHTHALATE 用作增塑剂和添加剂。用于毒理学研究以及通过邻苯二甲酸盐从食品接触材料 (FCM) 迁移到食品中而发生的食品污染风险评估研究。
TN6745 PALATINOSE

TNP-470,帕拉金糖水合物,Isomaltulose

Others Others
PALATINOSE (TNP-470) 是一种天然存在的二糖,由α-1,6-连接的葡萄糖和果糖组成。PALATINOSE 对肝脏代谢功能具有有益的影响,因此可能是蔗糖甜味剂的良好替代品。
TN1162 Dibutyl phthalate

1,2-Benzenedicarboxylic acid

Antifection Microbiology/Virology
Dibutyl phthalate (1,2-Benzenedicarboxylic acid) 是一种增塑剂,广泛用于工业制造。Dibutyl phthalate可调节 MSH6 巴豆酰化,可诱导诱导氧化损伤和遗传毒性,可破坏果蝇和人体细胞中保守的昼夜节律。
T0606 Monobutyl Phthalate

邻苯二甲酸单丁酯,Mono-n-butyl phthalate,Butyl hydrogen phthalate

Others Others
Monobutyl Phthalate (Butyl hydrogen phthalateButyl hydrogen phthalate) 是邻苯二甲酸二丁酯的主要代谢物,是一种胚胎毒物,具有抗雄激素作用。
T4914 Mesoxalate sodium (monohydrate)

Sodium mesoxalate monohydrate,丙酮二酸钠

Others; Endogenous Metabolite Metabolism; Others
Mesoxalate sodium (monohydrate) 是内源性代谢产物的一种。
TN6982 Diethyl phthalate

邻苯二甲酸二乙酯,1,2-diethyl benzene-1,2-dicarboxylate

Apoptosis Apoptosis
Diethyl phthalate (1,2-diethyl benzene-1,2-dicarboxylate) 是一种内分泌干扰物,影响 PC12 细胞凋亡系统。Diethyl phthalate 广泛用于许多塑料和个人护理产品。
T3S1873 Talatisamine

塔拉乌头胺,塔拉萨敏

Potassium Channel Membrane transporter/Ion channel
Talatisamine 是一种乌头生物碱,对K+通道有特异性阻滞作用。它能减弱 beta- 淀粉样低聚物对培养的皮层神经元的毒性。
T8084 Dimethyl 4-hydroxyisophthalate

二甲基 4-羟基异邻苯二甲酸酯,Dimetghyl 4-Hydroxyisophthalate

Others Others
Dimethyl 4-hydroxyisophthalate (Dimetghyl 4-Hydroxyisophthalate) 是水杨酸甲酯类似物。
T5119 Dicyclo hexyl Phthalate

Others Others
Dicyclo hexyl Phthalate 是一种固体增塑剂。
T4875 Palatinose hydrate

6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物

Others; Endogenous Metabolite Metabolism; Others
Palatinose hydrate (6-O-α-D-Glucopyranosyl-D-fructose, Isoma) 是内源性代谢产物的一种。
T3746 Dimethyl phthalate

邻苯二甲酸二甲酯,Solvanom,Avolin,Fermine,避蚊酯

Others Others
Dimethyl phthalate (Fermine) 是一种邻苯二甲酸酯 (PAEs),是一种已知的内分泌干扰物,也是一种普遍存在的污染物。它常作为增塑剂,赋予硬质聚氯乙烯 (PVC) 树脂以柔韧性。
T20200 Citrulline malate

L-Citrulline DL-malate,Stimol

Citrulline malate is a cpd of anti-fatigue.
T39836 Monoethyl phthalate

Monoethyl phthalate is a metabolite of diethyl phthalate, serving as a urinary biomarker for phthalate exposure, and indicating potential risks of thyroid cancer and benign nodules.
T20273 Diamyl phthalate

NSC 4720,NSC-4720,NSC4720

Diamyl phthalate is an agent of endocrine disruptor.
T31429 Dibutyl terephthalate

Dibutyl terephthalate is a biochemical.
T20473 Bis(2-ethylhexyl) terephthalate

Bis(2-ethylhexyl) terephthalate is an agent of biochemical.
TN4826 Prerubialatin

Others Others
Prerubialatin is a precursor of rubialatins A and B.
TN5631 Alaternin

2-羟基大黄素,2-Hydroxyemodin

Alaternin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5631,CAS号为 641-90-7。
T31536 Ditridecyl phthalate

DTDP,Phthalic acid, ditridecyl ester,Nuoplaz,BRN 2023076,Polycizer 962BPA

Ditridecyl phthalate is a kind of phthalate ester. Phthalate esters are esters of phthalic acid and are mainly used as plasticizers to soften polyvinyl chloride. They can be found in many different kind if products, including glues, building materials, pe
T20241 Diphenyl phthalate

NSC-4052,NSC 4052,NSC4052

Diphenyl phthalate is an agent of biochemical.

天然产物

Butyl isobutyl phthalate
Cat.No: T8319
Synonym: ButylIsobutylPhthalate,邻苯二甲酸-1-丁酯-2-异丁酯
Target: Glucosidase
DI-N-OCTYL PHTHALATE
Cat.No: T5112
Synonym:
Target: Others
PALATINOSE
Cat.No: TN6745
Synonym: TNP-470,帕拉金糖水合物,Isomaltulose
Target: Others
Dibutyl phthalate
Cat.No: TN1162
Synonym: 1,2-Benzenedicarboxylic acid
Target: Antifection
Monobutyl Phthalate
Cat.No: T0606
Synonym: 邻苯二甲酸单丁酯,Mono-n-butyl phthalate,Butyl hydrogen phthalate
Target: Others
Mesoxalate sodium (monohydrate)
Cat.No: T4914
Synonym: Sodium mesoxalate monohydrate,丙酮二酸钠
Target: Others, Endogenous Metabolite
Diethyl phthalate
Cat.No: TN6982
Synonym: 邻苯二甲酸二乙酯,1,2-diethyl benzene-1,2-dicarboxylate
Target: Apoptosis
Talatisamine
Cat.No: T3S1873
Synonym: 塔拉乌头胺,塔拉萨敏
Target: Potassium Channel
Dimethyl 4-hydroxyisophthalate
Cat.No: T8084
Synonym: 二甲基 4-羟基异邻苯二甲酸酯,Dimetghyl 4-Hydroxyisophthalate
Target: Others
Dicyclo hexyl Phthalate
Cat.No: T5119
Synonym:
Target: Others
Palatinose hydrate
Cat.No: T4875
Synonym: 6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物
Target: Others, Endogenous Metabolite
Dimethyl phthalate
Cat.No: T3746
Synonym: 邻苯二甲酸二甲酯,Solvanom,Avolin,Fermine,避蚊酯
Target: Others
Citrulline malate
Cat.No: T20200
Synonym: L-Citrulline DL-malate,Stimol
Target:
Monoethyl phthalate
Cat.No: T39836
Synonym:
Target:
Diamyl phthalate
Cat.No: T20273
Synonym: NSC 4720,NSC-4720,NSC4720
Target:
Dibutyl terephthalate
Cat.No: T31429
Synonym:
Target:
Bis(2-ethylhexyl) terephthalate
Cat.No: T20473
Synonym:
Target:
Prerubialatin
Cat.No: TN4826
Synonym:
Target: Others
Alaternin
Cat.No: TN5631
Synonym: 2-羟基大黄素,2-Hydroxyemodin
Target:
Ditridecyl phthalate
Cat.No: T31536
Synonym: DTDP,Phthalic acid, ditridecyl ester,Nuoplaz,BRN 2023076,Polycizer 962BPA
Target:
Diphenyl phthalate
Cat.No: T20241
Synonym: NSC-4052,NSC 4052,NSC4052
Target:
Cat. No. Product Name Species Expression System
TMPY-01099 GPT Protein, Rat, Recombinant (His)

Gpt1,ALAT,glutamic-pyruvate transaminase (alanine a...

Rat Baculovirus Insect Cells
Alanine aminotransferase (ALT), also known as glutamate pyruvate transaminase (GPT), is a pyridoxal enzyme that belongs to the class-I pyridoxal-phosphate-dependent aminotransferase family, Alanine aminotransferase subfamily. Gpt / Gpt1 / ALT catalyzes the reversible interconversion of L-alanine and 2-oxoglutalate to pyruvate and L-glutamate and plays a key role in the intermediary metabolism of glucose and amino acids. Gpt / Gpt1 / ALT is expressed in the liver, kidney, heart, and skeletal musc...
TMPH-00824 Oxalate oxidase 1 Protein, Hordeum vulgare, Recombinant (His & Myc)

Hordeum vulgare E. coli
Releases hydrogen peroxide in the apoplast which may be important for cross-linking reactions in the cell wall biochemistry. May play an important role in several aspects of plant growth and defense mechanisms. Oxalate oxidase 1 Protein, Hordeum vulgare, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 28.2 kDa and the accession number is P45850.
TMPH-00312 Malate dehydrogenase Protein, Brucella abortus, Recombinant (His & Myc & SUMO)

Brucella abortus E. coli
Catalyzes the reversible oxidation of malate to oxaloacetate. Malate dehydrogenase Protein, Brucella abortus, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 53.7 kDa and the accession number is B2S881.
TMPH-03060 NaD1 Protein, Nicotiana alata, Recombinant (His & SUMO)

Nicotiana alata E. coli
Plant defense peptide with antifungal activity against F.oxysporum and B.cinerea. Retards the growth of the Lepidopteran insect pests H.armigera and H.punctigera.

重组蛋白

GPT Protein, Rat, Recombinant (His)
Cat.No: TMPY-01099
Species: Rat
Expression System: Baculovirus Insect Cells
Oxalate oxidase 1 Protein, Hordeum vulgare, Recombinant (His & Myc)
Cat.No: TMPH-00824
Species: Hordeum vulgare
Expression System: E. coli
Malate dehydrogenase Protein, Brucella abortus, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00312
Species: Brucella abortus
Expression System: E. coli
NaD1 Protein, Nicotiana alata, Recombinant (His & SUMO)
Cat.No: TMPH-03060
Species: Nicotiana alata
Expression System: E. coli
TargetMol Loading
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