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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T4981 Anisotropine Methylbromide

Prostaglandin Receptor; AChR GPCR/G Protein; Immunology/Inflammation; Neuroscience
Anisotropine Methylbromide 是一种抗胆碱能药物,已用于缓解胃肠道痉挛和抑制胃酸分泌。
T1575 Nizatidine

Axid,Acinon,尼扎替丁,Zanizal

AChE; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Nizatidine (Acinon) 是一种竞争性和可逆的组胺 H2 受体拮抗剂,具有抗酸活性,可用于胃溃疡的研究。
T1756L Ilaprazole

IY81149,艾普拉唑,IY 81149,IY-81149

Proton pump; TOPK MAPK; Membrane transporter/Ion channel
Ilaprazole (IY-81149) 是一种具有口服活性质子泵抑制剂,以剂量依赖性方式不可逆地抑制H+/K+-ATPase,在兔壁细胞制剂中的IC50为 6 μM。它也是一种有效的T 细胞起源蛋白激酶(TOPK)抑制剂,用于胃溃疡的研究。
T1756 Ilaprazole sodium

IY-81149 sodium,艾普拉唑钠

Proton pump; TOPK MAPK; Membrane transporter/Ion channel
Ilaprazole sodium (IY-81149 sodium) 是一种具有口服活性质子泵抑制剂,以剂量依赖性方式不可逆地抑制 H+/K+-ATPase,在兔壁细胞制剂中的 IC50为 6 μM。它也是一种有效的 T 细胞起源蛋白激酶(TOPK)抑制剂,用于胃溃疡的研究。
T14975 CJ-42794

CJ-042794

Others Others
CJ-42794 (CJ-042794)是前列腺素受体 EP4的选择性拮抗剂, 抑制[3H]-PGE2与 EP4受体结合的平均 pKi 为8.5, 对 EP4选择性比 EP1, EP2和 EP3高200多倍。
T15687 Thioflosulide

L-745337

COX Immunology/Inflammation; Neuroscience
Thioflosulide (L-745337) 是一种具有选择性和高效性的 COX2 抑制剂(IC50:2.3 nM),具有抗炎活性,可用于研究胃溃疡。
T28136 NC-1300-B

NC1300B,NC 1300 B

ATPase Membrane transporter/Ion channel
NC-1300-B 抑制 H(+)-K(+)-ATP 酶,可用于研究胃溃疡。
T14546 Bermoprofen

AD-1590,AJ-1590

Others Others
Bermoprofen (AD-1590) 是一种口服活性非甾体抗炎化合物, 具有抗炎镇痛活性,可用于研究胃溃疡。
T19826 Rabeprazole

LY307640

Potassium Channel; STAT JAK/STAT signaling; Membrane transporter/Ion channel; Stem Cells
Rabeprazole (LY307640) 是一种 H+/K+-ATPase 抑制剂,通过靶向 STAT3 介导的糖酵解来抑制胃上皮细胞中的细胞增殖,可用于研究胃溃疡。
T7099 Gefarnate

Others Others
Gefarnate 是一种胃炎和胃溃疡的研究药物,目前也用于研究干眼症。
T13145 Thiazolidinone-Derivatives-1

Others Others
Thiazolidinone-Derivatives-1 抑制胃酸分泌,可用于研究胃和十二指肠溃疡的治疗。
T3610 Ranitidine

雷尼替丁,HSDB 3925,Ranitidin

P450; Antibacterial; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Ranitidine (HSDB 3925) 是一种选择性的,具有口服活性的组胺 H2 受体拮抗剂,IC50为 3.3 μM。它还一种是CYP2C19和CYP2C9的弱抑制剂,可抑制胃液分泌。
T22267 Cetalkonium chloride

Benzylcetyldimethylammonium chloride hydrate

Antibacterial Microbiology/Virology
Cetalkonium chloride(Benzylcetyldimethylammonium chloride hydrate) 是一种铵盐防腐剂,具有抗炎活性,可用于研究口疮性溃疡。
T1639 Amlexanox

氨来呫诺,CHX3673,Amoxanox,氨来诺,AA673

IL Receptor; FGFR; Others; IκB/IKK Angiogenesis; Immunology/Inflammation; NF-κB; Others; Tyrosine Kinase/Adaptors
Amlexanox (AA673) 是一种特异性的 IKKε和 TBK1抑制剂,其 IC50=1-2 μM。
T25737 Linetastine

TMK 688,TMK-688,TMK688

Lipoxygenase; LTR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Linetastine (TMK-688) 是一种 5-脂氧合酶抑制剂(5-LOX),能抑制白三烯的产生,并能拮抗组胺的作用。Linetastine可用于研究哮喘、动脉粥样硬化和消化性溃疡。
T23667 AGN-201904

AGN201904,AGN 201904

ATPase Membrane transporter/Ion channel
AGN-201904 是质子泵抑制剂,是一种奥美拉唑前药,可延缓衰老,可用于预防和治疗消化性溃疡。
T0674 Lansoprazole

兰索拉唑,A-65006,AG-1749

Proton pump; Phospholipase; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Lansoprazole (A-65006) 是一种可抑制胃酸生成的质子泵抑制剂。它是中性鞘磷脂酶的外泌体抑制剂。
T3442 UK-371804

UK371804

PAI-1; Serine Protease Metabolism; Proteases/Proteasome
UK-371804 是一种尿嘧啶型纤溶酶原激活物的抑制剂,Ki=10 nM。
T33584 Namirotene

CBS 211A,Cbs 211 A

Others Others
Namirotene (CBS 211A) 是一种蛋白质生物合成抑制剂,是一种人工合成的维甲酸类似物,可用于研究角膜疾病、角膜溃疡和干眼综合征。
T1651 Rabeprazole sodium

Dexrabeprazole Sodium,LY307640 sodium,Habeprazole Sodium,雷贝拉唑钠,Rebeprazole sodium,Aciphex Sodium

Apoptosis; Proton pump Apoptosis; Membrane transporter/Ion channel
Rabeprazole sodium (Habeprazole Sodium) 是一种质子泵抑制剂,不可逆地抑制胃 H+/K+-ATPase,可研究胃溃疡和胃食管反流。它诱导细胞凋亡,也抑制尿苷核苷核糖水解酶 ,IC50为 0.3 μM。
T68122 Oxmetidine

SKF 92994,Oxmetidina,Oxmetidinum

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Oxmetidine (SKF 92994) 是一种新型 H2 受体拮抗剂,具有细胞毒性。 Oxmetidine 抑制心脏和血管组织中跨膜钙通量,可用于治疗活动性十二指肠溃疡。
T68100 Mifentidine

DA 4577

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mifentidine (DA 4577) 是一种可口服的 H2 受体拮抗剂,可用于研究胃排空和实验性胃和十二指肠溃疡。
T1052 Proglumide

二丙谷酰胺

cholecystokinin GPCR/G Protein
Proglumide (Binoside) 是一种非肽的、口服具有活性的胆囊收缩素(CCK)-A/B 受体拮抗剂。它能够选择性阻断 CCK 在中枢神经系统中的作用。它能够抑制胃分泌,具有保护胃十二指肠粘膜的能力,并表现出抗癫痫和抗氧化活性。
T33846 Oxyphenonium bromide

Spasmophen,Oxifenon,奥芬溴铵,Oxyfenon,Atrenyl,Oxyphenon

Others Others
Oxyphenonium bromide (Oxyfenon) 具有抗胆碱能活性,可用于治疗胃和十二指肠溃疡以及缓解内脏痉挛的研究。
T8679 Epidermal Growth Factor

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Epidermal Growth Factor 与表皮生长因子受体 (EGFR) 结合并刺激细胞生长和增殖。它被批准用于治疗糖尿病足溃疡。
T0992 Carbenoxolone disodium

Biogastrone,Duogastrone,甘珀酸钠,Bioral

Gap Junction Protein Cytoskeletal Signaling
Carbenoxolone disodium (Duogastrone) 是甘草酸的活性代谢物和人11β-HSD 和细菌3α, 20β-HSD 的抑制剂。它是一种缝隙连接的解耦剂,可抑制牛痘病毒生长,用于消化性、食道和口腔溃疡和炎症的相关研究。
T5051 Isopropamide Iodide

AChR Neuroscience
Isopropamide iodide 是长效季铵盐抗胆碱能药物。它用于研究消化性溃疡和其他胃肠道疾病,尤其是胃酸过多和运动过度。
T1338 Sucralfate

硫糖铝,Sucrose octasulfate–aluminum complex

FGFR; Others; Antibacterial; Prostaglandin Receptor Angiogenesis; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Others; Tyrosine Kinase/Adaptors
Sucralfate (Sucrose octasulfate–aluminum complex) 是一种口服活性胃保护剂。它抑制消化性活性,并与黏膜损伤时暴露的带负电荷的上皮下蛋白结合,形成一层粘性层,保护血管床和增殖区。它可用于预防和治疗胃肠道疾病。
T4195 Betahistine

PT 9 base,倍他司汀,Vasomotal,Serc base

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Betahistine (Vasomotal) 是可口服的组胺 H1 受体激动剂和 H3 受体的拮抗剂,可用作血管扩张剂,用于类风湿性关节炎的研究。
T10221 Abeprazan hydrochloride

DWP14012 hydrochloride,Fexuprazan hydrochloride

Proton pump Membrane transporter/Ion channel
Abeprazan hydrochloride (Fexuprazan hydrochloride) 是一种有效的、可逆的、具有口服活性的potassium-competitive acid 阻滞剂,通过竞争性的与钾离子结合抑制 H+,K+- ATPase,而无需酸激活。Abeprazan hydrochloride 是一种质子泵抑制剂(PPI),通过减少胃酸的产生而起作用,可用于治疗胃酸相关疾病,如胃食管反流病(GERD)和消化性溃疡。
T77599 Methyl retinoate

Retinoic acid, methyl ester

Others Others
Methyl retinoate (Retinoic acid, methyl ester) 在体内实验中会诱导给部位发生无菌炎症,会使血液中白细胞数量增加,而红细胞和Hb含量减少。Methyl retinoate 可促进自发性白血病的产生。Methyl retinoate 可用于治疗因维生素A缺乏而产生的胃肥大和溃疡。
T69805 AU-006

AU-006 is an anti-ulcer drug which is effective in the treatment of gastric ulcers by inhibiting gastric acid secretion.
T25805 Metoquizine

Ly-42406,Ly 42406,Ly42406,Lilly 42406

Metoquizine 是一种抗胆碱能化合物。它是一种蕈毒碱型乙酰胆碱受体拮抗剂,曾用于治疗溃疡。
T12914 Siltenzepine

Others Others
Siltenzepine is an agent of anti-acid agent,and used in the treatment of peptic ulcers.
T2138L Oxyphencyclimine

Oxiphencycliminum,Antulcus,Zamanil,Manir,Caridan,Naridan

Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.
T26090 Rioprostil

TR 4698,TR4698,Rioprostilum,TR-4698

Rioprostil is a methyl prostaglandin E1 analog that decreases gastric acid secretion and enhances the gastric mucus-bicarbonate barrier. It is effective in the treatment of gastric ulcers and gives significant protection against NSAID-induced gastric muco
T27640 Itriglumide

CR-2945,CR2945,CR 2945

Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, and gastroesophageal reflux disease (GERD).
T12047 Misoprostol acid

Others Others
Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.
T70135 Nepaprazole sodium dihydrate

Nepaprazole sodium dihydrate is a proton pump inhibitor potentially for treatment of gastric ulcers.
T24254 KB-5492 anhydrous

KB-5492,KB5492,KB 5492

KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.
T16152 Betamethasone 17-benzoate

Kinesin Cytoskeletal Signaling
Betamethasone 17-benzoate is a representative steroid. It also can be used in the treatment of recurrent aphothous ulcers (RAU).
T32224 Isopropamide

Priazimide,Dipramide,Piaccamide,Chloroisopropamide,Dipramid

Isopropamide (R5) is a long-acting anticholinergic drug. It is used to treat peptic ulcers and other gastrointestinal disorders involving excess gastric acid (gastrointestinal acidosis) and hyperactivity.
T37470 Bismuth subcarbonate

Bismuth subcarbonate, also known as bismuth carbonate oxide, is a versatile semiconductor compound based on bismuth, commonly utilized for its antibacterial properties, as well as in various applications such as sensors, super capacitors, and photocatalysts. Additionally, bismuth subcarbonate serves as a protective agent against gastric acid erosion, particularly in the treatment of gastric ulcers[1][2].
T25104 Aprofene

aprophen,Aprofenum

Aprofene (Aprophen) is an antagonist of muscarinic and nicotinic acetylcholine receptors. It may be used in the therapy of peptic ulcers, endarteritis (inflammation of the inner shell of the artery), cholecystitis (inflammation of the gallbladder), and sp
T78237 Urease-IN-6

Urease-IN-6为一种高效Urease抑制剂,IC50值为14.2 μM,适用于消化性溃疡和胃溃疡研究。
T20937 Dodecenylsuccinic anhydride

2-十二烯基-丁二酸酐,Rikacid DDSA,Dodecenylsuccinic acid anhydride,DDSA

Others Others
Dodecenylsuccinic anhydride (DDSA) 可与胶原水凝胶接枝,作为疏水性伤口敷料掺入辛伐他汀后,在治疗溃疡和预防伤口感染方面具有潜在应用。
T6415 Bismuth Subcitrate Potassium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Bismuth subcitrate potassium 是针对 12 种幽门螺杆菌菌株的抗生素,MIC50为 8 μg/ml。它用于幽门螺杆菌感染的上胃肠道疾病的研究。
T25375 Enprostil

RS-84135,RS 84135,Gardrin,RS84135

Enprostil is a synthetic PGE2 analog that has an inhibitory effect on gastric acid secretion, a mucoprotective effect, and a postprandial lowering effect on gastrin. It has efficient and safe in the therapy of gastroduodenal ulcers.
T68206 Arbortristoside A

Arbortristoside A is an anti-inflammatory and antinociceptive. This activity may be due to the inhibiting effect of prostaglandin, histamine and serotonin. Arbortristoside A has also been shown to act on ulcerations and may facilitate healing of peptic ulcers.
T33314 Methantheline Bromide

Frenogastrico,Dixamone bromide,Banthine,Asabaine,Methanthelinium bromide

Methantheline Bromide is a synthetic spasmolytic used to relieve cramps or spasms of the stomach, bowel, and bladder. It is also useful for intestinal or gastric ulcers (peptic ulcer disease), intestinal problems, pancreatitis, gastritis, biliary dysmotil

化合物

Anisotropine Methylbromide
Cat.No: T4981
Synonym:
Target: Prostaglandin Receptor, AChR
Nizatidine
Cat.No: T1575
Synonym: Axid,Acinon,尼扎替丁,Zanizal
Target: AChE, Histamine Receptor
Ilaprazole
Cat.No: T1756L
Synonym: IY81149,艾普拉唑,IY 81149,IY-81149
Target: Proton pump, TOPK
Ilaprazole sodium
Cat.No: T1756
Synonym: IY-81149 sodium,艾普拉唑钠
Target: Proton pump, TOPK
CJ-42794
Cat.No: T14975
Synonym: CJ-042794
Target: Others
Thioflosulide
Cat.No: T15687
Synonym: L-745337
Target: COX
NC-1300-B
Cat.No: T28136
Synonym: NC1300B,NC 1300 B
Target: ATPase
Bermoprofen
Cat.No: T14546
Synonym: AD-1590,AJ-1590
Target: Others
Rabeprazole
Cat.No: T19826
Synonym: LY307640
Target: Potassium Channel, STAT
Gefarnate
Cat.No: T7099
Synonym:
Target: Others
Thiazolidinone-Derivatives-1
Cat.No: T13145
Synonym:
Target: Others
Ranitidine
Cat.No: T3610
Synonym: 雷尼替丁,HSDB 3925,Ranitidin
Target: P450, Antibacterial, Histamine Receptor
Cetalkonium chloride
Cat.No: T22267
Synonym: Benzylcetyldimethylammonium chloride hydrate
Target: Antibacterial
Amlexanox
Cat.No: T1639
Synonym: 氨来呫诺,CHX3673,Amoxanox,氨来诺,AA673
Target: IL Receptor, FGFR, Others, IκB/IKK
Linetastine
Cat.No: T25737
Synonym: TMK 688,TMK-688,TMK688
Target: Lipoxygenase, LTR, Histamine Receptor
AGN-201904
Cat.No: T23667
Synonym: AGN201904,AGN 201904
Target: ATPase
Lansoprazole
Cat.No: T0674
Synonym: 兰索拉唑,A-65006,AG-1749
Target: Proton pump, Phospholipase, Antibacterial
UK-371804
Cat.No: T3442
Synonym: UK371804
Target: PAI-1, Serine Protease
Namirotene
Cat.No: T33584
Synonym: CBS 211A,Cbs 211 A
Target: Others
Rabeprazole sodium
Cat.No: T1651
Synonym: Dexrabeprazole Sodium,LY307640 sodium,Habeprazole Sodium,雷贝拉唑钠,Rebeprazole sodium,Aciphex Sodium
Target: Apoptosis, Proton pump
Oxmetidine
Cat.No: T68122
Synonym: SKF 92994,Oxmetidina,Oxmetidinum
Target: Histamine Receptor
Mifentidine
Cat.No: T68100
Synonym: DA 4577
Target: Histamine Receptor
Proglumide
Cat.No: T1052
Synonym: 二丙谷酰胺
Target: cholecystokinin
Oxyphenonium bromide
Cat.No: T33846
Synonym: Spasmophen,Oxifenon,奥芬溴铵,Oxyfenon,Atrenyl,Oxyphenon
Target: Others
Epidermal Growth Factor
Cat.No: T8679
Synonym:
Target: EGFR
Carbenoxolone disodium
Cat.No: T0992
Synonym: Biogastrone,Duogastrone,甘珀酸钠,Bioral
Target: Gap Junction Protein
Isopropamide Iodide
Cat.No: T5051
Synonym:
Target: AChR
Sucralfate
Cat.No: T1338
Synonym: 硫糖铝,Sucrose octasulfate–aluminum complex
Target: FGFR, Others, Antibacterial, Prostaglandin Receptor
Betahistine
Cat.No: T4195
Synonym: PT 9 base,倍他司汀,Vasomotal,Serc base
Target: Histamine Receptor
Abeprazan hydrochloride
Cat.No: T10221
Synonym: DWP14012 hydrochloride,Fexuprazan hydrochloride
Target: Proton pump
Methyl retinoate
Cat.No: T77599
Synonym: Retinoic acid, methyl ester
Target: Others
AU-006
Cat.No: T69805
Synonym:
Target:
Metoquizine
Cat.No: T25805
Synonym: Ly-42406,Ly 42406,Ly42406,Lilly 42406
Target:
Siltenzepine
Cat.No: T12914
Synonym:
Target: Others
Oxyphencyclimine
Cat.No: T2138L
Synonym: Oxiphencycliminum,Antulcus,Zamanil,Manir,Caridan,Naridan
Target:
Rioprostil
Cat.No: T26090
Synonym: TR 4698,TR4698,Rioprostilum,TR-4698
Target:
Itriglumide
Cat.No: T27640
Synonym: CR-2945,CR2945,CR 2945
Target:
Misoprostol acid
Cat.No: T12047
Synonym:
Target: Others
Nepaprazole sodium dihydrate
Cat.No: T70135
Synonym:
Target:
KB-5492 anhydrous
Cat.No: T24254
Synonym: KB-5492,KB5492,KB 5492
Target:
Betamethasone 17-benzoate
Cat.No: T16152
Synonym:
Target: Kinesin
Isopropamide
Cat.No: T32224
Synonym: Priazimide,Dipramide,Piaccamide,Chloroisopropamide,Dipramid
Target:
Bismuth subcarbonate
Cat.No: T37470
Synonym:
Target:
Aprofene
Cat.No: T25104
Synonym: aprophen,Aprofenum
Target:
Urease-IN-6
Cat.No: T78237
Synonym:
Target:
Dodecenylsuccinic anhydride
Cat.No: T20937
Synonym: 2-十二烯基-丁二酸酐,Rikacid DDSA,Dodecenylsuccinic acid anhydride,DDSA
Target: Others
Bismuth Subcitrate Potassium
Cat.No: T6415
Synonym:
Target: Others, Antibacterial, Antibiotic
Enprostil
Cat.No: T25375
Synonym: RS-84135,RS 84135,Gardrin,RS84135
Target:
Arbortristoside A
Cat.No: T68206
Synonym:
Target:
Methantheline Bromide
Cat.No: T33314
Synonym: Frenogastrico,Dixamone bromide,Banthine,Asabaine,Methanthelinium bromide
Target:
Cat. No. Product Name Target Signaling Pathways
T0070 Pentoxifylline

Oxpentifylline,PTX,己酮可可碱,BL-191

HIV Protease; PDE; Adenosine Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Pentoxifylline (PTX) 是一种具有口服活性的磷酸二酯酶非选择性抑制剂,具有免疫调节、抗炎、抗纤溶、抗增殖和血液流变学改善作用。它可研究周围血管疾病、脑血管疾病和其他一些涉及局部微循环缺陷的疾病。
TN2078 Pinocembrin chalcone

2',4',6'-Trihydroxychalcone,Pinocembrinchalcone

Calcium Channel; Tyrosinase; Antibacterial; Antifection Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Proteases/Proteasome
Pinocembrin chalcone 是一种具有抗诱变作用的酪氨酸酶抑制剂。 Pinocembrin 查尔酮可用于预防胃溃疡的研究。
T7908 DL-Methionine Methylsulfonium Chloride

DL-蛋氨酸甲基氯化锍,维生素U

Others Others
DL-methionine methylsulfonium chloride 是天然的蛋氨酸衍生物。它能够有效保护胃粘膜,避免其受到乙醇诱导的损伤。
TN4465 Luvangetin

COX; Prostaglandin Receptor; Antifection GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Luvangetin may have anti-inflammatory activity, it can inhibit NO and PGE2 production in LPS-stimulated BV2 cells. Luvangetin shows significant protection against pylorus-ligated and aspirin-induced gastric ulcers in rats and cold restraint stress-induced
T83258 7(18)-Dehydroschisandro A

7(18)-Dehydroschisandro A (化合物2) 是从Schizandra chinensis Baill分离得到的木脂素,对激性胃溃疡显示出抑制效果。
T83257 7(8)-Dehydroschisandrol A

7(8)-Dehydroschisandrol A (Compound 4a)为从Schizandra chinensis Baill分离的木脂素,对激性胃溃疡表现出较弱抑制效果。
TN4659 Nimbin

COX Immunology/Inflammation; Neuroscience
Nimbin is an anti-pyretic, can be used to treat arthritis, hypoglycaemia, peptic ulcers, anti-secretory activity, and it can also be used as an antibiotic. Nimbin requires to elicit a 50% inhibition of this steroid hydroxylase activity in the three insect
T75507 1-Methyl-2-(8E)-8-tridecenyl-4(1H)-quinolinone

1-Methyl-2-(8E)-8-tridecenyl-4(1H)-quinolinone 对幽门螺杆菌菌株 51 表现出有效的抗菌活性,MIC50 值和 MIC90 值分别为 22 µM 和 50 µM。该化合物展现了在研究胃及十二指肠溃疡方面的潜力。

天然产物

Pentoxifylline
Cat.No: T0070
Synonym: Oxpentifylline,PTX,己酮可可碱,BL-191
Target: HIV Protease, PDE, Adenosine Receptor, Autophagy
Pinocembrin chalcone
Cat.No: TN2078
Synonym: 2',4',6'-Trihydroxychalcone,Pinocembrinchalcone
Target: Calcium Channel, Tyrosinase, Antibacterial, Antifection
DL-Methionine Methylsulfonium Chloride
Cat.No: T7908
Synonym: DL-蛋氨酸甲基氯化锍,维生素U
Target: Others
Luvangetin
Cat.No: TN4465
Synonym:
Target: COX, Prostaglandin Receptor, Antifection
7(18)-Dehydroschisandro A
Cat.No: T83258
Synonym:
Target:
7(8)-Dehydroschisandrol A
Cat.No: T83257
Synonym:
Target:
Nimbin
Cat.No: TN4659
Synonym:
Target: COX
1-Methyl-2-(8E)-8-tridecenyl-4(1H)-quinolinone
Cat.No: T75507
Synonym:
Target:
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