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68

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T15500 HPi1

Others; Antibacterial Microbiology/Virology; Others
HPi1 是一种有口服活性的,针对幽门螺杆菌的选择性抗菌剂,IC50为 0.24 μM,MIC 为 0.08-0.16 μg/mL。
T38612 Linaprazan glurate

Others Others
Linaprazan glurate 抑制外源性或内源性刺激的胃酸分泌。 Linaprazan glurate 可用于胃肠道炎症性疾病和消化性溃疡疾病的研究。
T5051 Isopropamide Iodide

AChR Neuroscience
Isopropamide iodide 是长效季铵盐抗胆碱能药物。它用于研究消化性溃疡和其他胃肠道疾病,尤其是胃酸过多和运动过度。
T6710 Troxipide

曲昔派特,曲昔匹特,Aplace

Others Others
Troxipide (Aplace) 是非分泌型胃保护剂,是口服具有活力的胃炎和胃溃疡的防御因子的增强剂,具有抗溃疡、抗炎和粘液分泌作用。
T0044 Oxethazaine

奥昔卡因,Oxetacaine

HBV; Sodium Channel Membrane transporter/Ion channel; Microbiology/Virology
Oxethazaine (Oxetacaine) 是一种具有耐酸性和口服活性试剂,是芬特明的酸性前体,有潜力缓解消化性溃疡疾病或食管炎引起的疼痛。
T1562 Rebamipide

Proamipide,OPC12759,瑞巴派特

Free radical scavengers; COX; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience; oxidation-reduction
Rebamipide (OPC12759) 是一种粘膜保护剂,可诱导COX-2表达,增加PGE2水平,并以 COX-2 依赖性方式增强胃粘膜防御。
T0157 Roxatidine Acetate hydrochloride

HOE 760,盐酸罗沙替丁醋酸酯,Roxatidine Acetate HCl

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Roxatidine Acetate hydrochloride (HOE 760) 是一种特异性和竞争性的组胺 H2 受体拮抗剂,能抑制胃酸分泌,可用于胃溃疡和十二指肠溃疡的研究。
TP1035 Cyclic somatostatin

SRIF-14,合成生长抑素,环状生长激素抑制素,Somatostatin-14

Others Others
Cyclic somatostatin (SRIF-14) 是生长激素释放抑制因子,可用于研究胃十二指肠溃疡出血。
T6928 Pantoprazole

SKF96022,泮托拉唑,BY1023

Apoptosis; Proton pump; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel
Pantoprazole (BY1023) 是一种质子泵抑制剂,用于短期治疗由胃食管反流病引起的食管糜烂和溃疡。它联合阿霉素可显著增加肿瘤生长延迟。它是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。
T21254 Vonoprazan Fumarate

TAK-438,TAK 438,Vonoprazan Fumurate,TAK438,富马酸沃诺拉赞

Proton pump Membrane transporter/Ion channel
Vonoprazan Fumarate (TAK438) 是质子泵的有效抑制剂,是口服有效的高效钾竞争性酸阻断剂,具有抗分泌活性。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50为 19 nM。它被开发用于研究酸相关疾病,如消化性溃疡和胃食管反流病。
T8388 Vonoprazan

TAK-438 (free base),沃诺拉赞

Proton pump Membrane transporter/Ion channel
Vonoprazan (TAK-438 (free base)) 是一种质子泵抑制剂,是口服活性钾竞争性酸阻断剂,有抗分泌作用。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50值为 19 nM。它可用于研究胃酸相关疾病。
T19763 Cetraxate hydrochloride

DV-1006,DV 1006,Cetraxate HCl,盐酸西曲酸酯,DV1006

Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism
Cetraxate hydrochloride (DV10062) 是一种有效的顶体蛋白酶 (acrosomal proteinase acrosin) 抑制剂,Ki 和 IC50分别为 0.94 μM 和 3.3 μM。它是一种口服有活性的抗溃疡试剂 (anti-ulcer),具有粘膜保护作用,可用于研究胃溃疡。
T0161 Pantoprazole Sodium Hydrate

SKF96022 sodium hydrate,泮托拉唑钠水合物,BY1023 (sodium hydrate),SKF96022 (sodium hydrate)

Apoptosis; Potassium Channel; Proton pump; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel
Pantoprazole Sodium Hydrate (BY1023 (sodium hydrate)) 是一种具有口服活性的质子泵抑制剂。它是取代的苯并咪唑,是H+/K+-ATPase 抑制剂。它可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T6929 Pantoprazole sodium

Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc

Apoptosis; Others; Proton pump; HIF; Autophagy Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Others
Pantoprazole sodium (Pantecta) 是一种具有口服活性的质子泵抑制剂,是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,IC50为 6.8 μM。它可以改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T10124 Antiulcer Agent 1

Others Others
Antiulcer Agent 1 是一种用于口服给药的 2-(3,4-二甲氧基苯基)乙胺衍生物。
T76577 Antiulcer Agent 2

Antiulcer Agent 2 是一种四肽,组成包括天冬氨酸、丙氨酸、组氨酸和赖氨酸,存在于人白蛋白N端,并在溃疡及活性氧生成中显示出潜在应用。
T28665 Saviprazole

Hoe731,Hoe 731,Hoe-731

Proton pump Membrane transporter/Ion channel
Saviprazole (Hoe-731) 是一种质子泵抑制剂,可用于治疗胃溃疡。
T5008 Teprenone

Tetraprenylacetone,Geranylgeranylacetone,替普瑞酮

HSP Cytoskeletal Signaling; Metabolism
Teprenone (Geranylgeranylacetone) 是一种热休克蛋白诱导剂,有抗溃疡作用。
T12215 Nexopamil racemate

(Rac)-Nexopamil

Calcium Channel; 5-HT Receptor GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Nexopamil racemate((Rac)-Nexopamil) 是 Nexopamil 的外消旋体。Nexopamil racemate 具有潜在的抗哮喘和抗溃疡活性。
T31195 Dalcotidine

KU 1257,KU-1257

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Dalcotidine (KU 1257) 是一种新型组胺H2受体拮抗剂,具有组胺H9受体拮抗活性和抗分泌作用,与豚鼠大脑皮层结合的Ki 值为0.040 对分离性豚鼠右心房组胺诱导的正变时反应的拮抗作用的KB 值为0.041。Dalcotidine 提高了溃疡愈合的质量,可能有助于降低溃疡的复发率和复发率。
T29015 Trithiozine

Tresanil,Sulmetozine,Tritiozinum,舒美吗啉,Tritiozine,Tritiozina

Others Others
Trithiozine (Tritiozinum) 具有抗分泌和抗溃疡能力。 Trithiozine 可用于治疗消化性溃疡病和高分泌障碍的研究。
T6548 Irsogladine

Dicloguamine,伊索拉定

PDE; AChR Metabolism; Neuroscience
Irsogladine (Dicloguamine) 是抗胃溃疡剂,通过 M1 毒蕈碱乙酰胆碱受体结合促进间隙连接细胞间通讯。
T4510 Polaprezinc

Zinc L-carnosine,聚普瑞锌,L-肌肽锌

Others Others
Polaprezinc是一种含有锌和L-carnosine的生物可用螯合物,以其胃肠保护性能、抗溃疡、抗氧化和抗炎效果而闻名。
T6349 Sitafloxacin Hydrate

西他沙星水合物,DU-6859a,DU6859a hydrate

Antibacterial; Antibiotic Microbiology/Virology
Sitafloxacin Hydrate (DU-6859a) 是一种口服有效的氟喹诺酮类抗生素,在体外可对抗广泛的革兰氏阳性和阴性细菌有活性。Sitafloxacin 可研究呼吸道感染和尿路感染。
T77618 COX-2-IN-34

COX Immunology/Inflammation; Neuroscience
COX-2-IN-34 是一种选择性的、口服有效的 COX-2 抑制剂,在小鼠实验过程中显示出抗炎活性且无胃溃疡毒性。
T1639 Amlexanox

氨来呫诺,CHX3673,Amoxanox,氨来诺,AA673

IL Receptor; FGFR; Others; IκB/IKK Angiogenesis; Immunology/Inflammation; NF-κB; Others; Tyrosine Kinase/Adaptors
Amlexanox (AA673) 是一种特异性的 IKKε和 TBK1抑制剂,其 IC50=1-2 μM。
T62396 KB-5492 free base

KB-5492 free base 是一种有效的和选择性的sigma 受体抑制剂,抑制 [3H]1,3-di(2-tolyl)guanidine (DTG) 与sigma 受体结合,IC50值为 3.15 μM。KB-5492 free base 是一种抗溃疡剂。
T16865 SCH28080

ATPase; Proton pump Membrane transporter/Ion channel
SCH28080 是一种可逆且具有 K+ 竞争性的胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,IC50 值为 20 nM (家兔微粒体膜)。SCH28080 在体内是有效的酸分泌抑制剂,具有抗溃疡活性、抗分泌和细胞保护活性。
T1756L Ilaprazole

IY81149,艾普拉唑,IY 81149,IY-81149

Proton pump; TOPK MAPK; Membrane transporter/Ion channel
Ilaprazole (IY-81149) 是一种具有口服活性质子泵抑制剂,以剂量依赖性方式不可逆地抑制H+/K+-ATPase,在兔壁细胞制剂中的IC50为 6 μM。它也是一种有效的T 细胞起源蛋白激酶(TOPK)抑制剂,用于胃溃疡的研究。
T10872L CP 96021

5-HT Receptor GPCR/G Protein; Neuroscience
CP 96021是一组5-HT1受体和5-HT2受体拮抗剂,具有抗炎特性,是治疗胃肠道和呼吸道哮喘的非自身抗溃疡化合物。
T77617 MMP-9-IN-6

MMP Proteases/Proteasome
MMP-9-IN-6 是一种 MMP-9 抑制剂,其 IC50 值为50 μM, 具有较好的抗溃疡功效。MMP-9-IN-6 具有潜在的抗肿瘤活性,可用于研究组织重塑、伤口修复和动脉粥样硬化。
T21385 Cinitapride

西尼必利,Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove

5-HT Receptor GPCR/G Protein; Neuroscience
Cinitapride (Blaston) 是一种促胃药。它减缓肌肉的活动,以减轻诸如胃酸反流、胃排空延迟和溃疡性消化不良等病症的症状。 Cinitapride 作为 5-HT2 受体的拮抗剂和 5-HT1 和 5-HT4 受体的激动剂。
T0786 Clidinium bromide

克利溴铵,Ro 2-3773

AChR Neuroscience
Clidinium bromide (Ro 2-3773) 是季胺抗毒蕈碱剂,可通过减少胃酸和减慢肠道速度,缓解痉挛和腹部疼痛的症状。
T24728 Rosaprostol

C 83

Rosaprostol is an agent of the anti-ulcer drug.
T33710 Nocloprost

Nocloprost is a prostaglandin E2 analog with local gastroprotective and ulcer-healing activity.
T32599 Lauroylglycyrrhetinic acid

BX 24,BX24,BX-24

Lauroylglycyrrhetinic acid, an analog of carbenoxolone, can be used in the treatment of stomach ulcer.
T23725 Amicoumacin A

Amicoumacin A has antibacterial activity. It also strongly suppresses inflammatory and ulcer activity.
T10008 BTM-1086

Others Others
BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.
T34087 Plaunotol

Kelnac,Plaunotolum

Plaunotol is a gastric protective agent that increases prostaglandins in the gastric mucosa and accelerates ulcer healing.
T34936 Tridihexethyl chloride

Propethonum,Pathilon,Tridihexethyl

Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.
T68200 Roxatidine hydrochloride

Roxatidine hydrochloride is an anti-ulcer agent and histamine antagonist that suppresses gastric acid secretion. It effectively heals duodenal and gastric ulcers and reduces ulcer pain. Roxatidine acetate has an improved safety profile compared to other similar drugs, in part because lower doses of roxatidine acetate are therapeutically effective.
T69801 AU-461

AU-461 is a gastric H(+)/K(+) ATPase inhibitor which acts as an anti-ulcer agent.
T31743 Famotine hydrochloride

Famotine HCl,UK-2054

Famotine Hydrochloride is a histamine H2 receptor antagonist that suppresses acid production in the stomach and commonly treats peptic ulcer disease and gastroesophageal reflux disease.
T69805 AU-006

AU-006 is an anti-ulcer drug which is effective in the treatment of gastric ulcers by inhibiting gastric acid secretion.
T28613 RP73870

RP 73870,RP-73870

RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.
T24254 KB-5492 anhydrous

KB-5492,KB5492,KB 5492

KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.
T19929 Ranitidine-S-oxide

Ranitidine-S-oxide is a metabolite of Ranitidine. It is commonly used in the treatment of peptic ulcer disease, Zollinger–Ellison syndrome,and gastroesophageal reflux disease.
T70127 Famotine

Famotine is a histamine H2 receptor antagonist that inhibits stomach acid production. It is commonly used in the treatment of peptic ulcer disease and gastroesophageal reflux disease.
T70090 Nizatidine amide

Nizatidine amide is a histamine H2 receptor antagonist that inhibits stomach acid production. It is commonly used in the treatment of peptic ulcer disease and gastroesophageal reflux disease.
T71049 Famotidine disulfide

Famotidine disulfide is a histamine H2-receptor antagonist that inhibits stomach acid production. It is commonly used in the treatment of peptic ulcer disease and gastroesophageal reflux disease.

化合物

HPi1
Cat.No: T15500
Synonym:
Target: Others, Antibacterial
Linaprazan glurate
Cat.No: T38612
Synonym:
Target: Others
Isopropamide Iodide
Cat.No: T5051
Synonym:
Target: AChR
Troxipide
Cat.No: T6710
Synonym: 曲昔派特,曲昔匹特,Aplace
Target: Others
Oxethazaine
Cat.No: T0044
Synonym: 奥昔卡因,Oxetacaine
Target: HBV, Sodium Channel
Rebamipide
Cat.No: T1562
Synonym: Proamipide,OPC12759,瑞巴派特
Target: Free radical scavengers, COX, Prostaglandin Receptor
Roxatidine Acetate hydrochloride
Cat.No: T0157
Synonym: HOE 760,盐酸罗沙替丁醋酸酯,Roxatidine Acetate HCl
Target: Histamine Receptor
Cyclic somatostatin
Cat.No: TP1035
Synonym: SRIF-14,合成生长抑素,环状生长激素抑制素,Somatostatin-14
Target: Others
Pantoprazole
Cat.No: T6928
Synonym: SKF96022,泮托拉唑,BY1023
Target: Apoptosis, Proton pump, Autophagy
Vonoprazan Fumarate
Cat.No: T21254
Synonym: TAK-438,TAK 438,Vonoprazan Fumurate,TAK438,富马酸沃诺拉赞
Target: Proton pump
Vonoprazan
Cat.No: T8388
Synonym: TAK-438 (free base),沃诺拉赞
Target: Proton pump
Cetraxate hydrochloride
Cat.No: T19763
Synonym: DV-1006,DV 1006,Cetraxate HCl,盐酸西曲酸酯,DV1006
Target: Serine/threonin kinase
Pantoprazole Sodium Hydrate
Cat.No: T0161
Synonym: SKF96022 sodium hydrate,泮托拉唑钠水合物,BY1023 (sodium hydrate),SKF96022 (sodium hydrate)
Target: Apoptosis, Potassium Channel, Proton pump, Autophagy
Pantoprazole sodium
Cat.No: T6929
Synonym: Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc
Target: Apoptosis, Others, Proton pump, HIF, Autophagy
Antiulcer Agent 1
Cat.No: T10124
Synonym:
Target: Others
Antiulcer Agent 2
Cat.No: T76577
Synonym:
Target:
Saviprazole
Cat.No: T28665
Synonym: Hoe731,Hoe 731,Hoe-731
Target: Proton pump
Teprenone
Cat.No: T5008
Synonym: Tetraprenylacetone,Geranylgeranylacetone,替普瑞酮
Target: HSP
Nexopamil racemate
Cat.No: T12215
Synonym: (Rac)-Nexopamil
Target: Calcium Channel, 5-HT Receptor
Dalcotidine
Cat.No: T31195
Synonym: KU 1257,KU-1257
Target: Histamine Receptor
Trithiozine
Cat.No: T29015
Synonym: Tresanil,Sulmetozine,Tritiozinum,舒美吗啉,Tritiozine,Tritiozina
Target: Others
Irsogladine
Cat.No: T6548
Synonym: Dicloguamine,伊索拉定
Target: PDE, AChR
Polaprezinc
Cat.No: T4510
Synonym: Zinc L-carnosine,聚普瑞锌,L-肌肽锌
Target: Others
Sitafloxacin Hydrate
Cat.No: T6349
Synonym: 西他沙星水合物,DU-6859a,DU6859a hydrate
Target: Antibacterial, Antibiotic
COX-2-IN-34
Cat.No: T77618
Synonym:
Target: COX
Amlexanox
Cat.No: T1639
Synonym: 氨来呫诺,CHX3673,Amoxanox,氨来诺,AA673
Target: IL Receptor, FGFR, Others, IκB/IKK
KB-5492 free base
Cat.No: T62396
Synonym:
Target:
SCH28080
Cat.No: T16865
Synonym:
Target: ATPase, Proton pump
Ilaprazole
Cat.No: T1756L
Synonym: IY81149,艾普拉唑,IY 81149,IY-81149
Target: Proton pump, TOPK
CP 96021
Cat.No: T10872L
Synonym:
Target: 5-HT Receptor
MMP-9-IN-6
Cat.No: T77617
Synonym:
Target: MMP
Cinitapride
Cat.No: T21385
Synonym: 西尼必利,Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove
Target: 5-HT Receptor
Clidinium bromide
Cat.No: T0786
Synonym: 克利溴铵,Ro 2-3773
Target: AChR
Rosaprostol
Cat.No: T24728
Synonym: C 83
Target:
Nocloprost
Cat.No: T33710
Synonym:
Target:
Lauroylglycyrrhetinic acid
Cat.No: T32599
Synonym: BX 24,BX24,BX-24
Target:
Amicoumacin A
Cat.No: T23725
Synonym:
Target:
BTM-1086
Cat.No: T10008
Synonym:
Target: Others
Plaunotol
Cat.No: T34087
Synonym: Kelnac,Plaunotolum
Target:
Tridihexethyl chloride
Cat.No: T34936
Synonym: Propethonum,Pathilon,Tridihexethyl
Target:
Roxatidine hydrochloride
Cat.No: T68200
Synonym:
Target:
AU-461
Cat.No: T69801
Synonym:
Target:
Famotine hydrochloride
Cat.No: T31743
Synonym: Famotine HCl,UK-2054
Target:
AU-006
Cat.No: T69805
Synonym:
Target:
RP73870
Cat.No: T28613
Synonym: RP 73870,RP-73870
Target:
KB-5492 anhydrous
Cat.No: T24254
Synonym: KB-5492,KB5492,KB 5492
Target:
Ranitidine-S-oxide
Cat.No: T19929
Synonym:
Target:
Famotine
Cat.No: T70127
Synonym:
Target:
Nizatidine amide
Cat.No: T70090
Synonym:
Target:
Famotidine disulfide
Cat.No: T71049
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3605 Gastrodenol

Bismuth tripotassium dicitrate,枸橼酸铋钾,Bismuth subcitrate

Others Others
Gastrodenol (Bismuth tripotassium dicitrate) 是一种对溃疡和胃不适具有潜在的应用价值的药物。
T2833 Dehydrocostus Lactone

Epiligulyl oxide,去氢木香内酯,(-)-Dehydrocostus lactone,去氢木香烃内酯

IκB/IKK NF-κB
Dehydrocostus Lactone ((-)-Dehydrocostus lactone) 是一种倍半萜内酯,从云木香中分离得到。
TN6577 Bletilloside A

3-Methoxyshancigusin I

Others Others
Bletilloside A(3-Methoxyshancigusin I) 是从条纹苜蓿的块茎中分离出一种新型葡萄糖苷,具有抗胃溃疡活性。
TN1568 Deoxyartemisinin

2-deoxyartemisinin

Deoxyartemisinin (2-deoxyartemisinin) 是一种口服有效的抗炎和抗溃疡化合物,可从青蒿素青蒿中分离得到。
T21651 Lansoprazole sodium

兰索拉唑钠,Lansoprazole (sodium), AG-1749 sodium

Proton pump; Phospholipase; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Lansoprazole sodium (Lansoprazole (sodium)) 是一种质子泵抑制剂,是中性鞘磷脂酶的外泌体抑制剂,能抑制胃酸生成。
TN2233 Spathulenol

Antioxidant; Antifungal Microbiology/Virology; oxidation-reduction
Spathulenol 是一种来自 Aristolochia yunnanensis 的天然成分,具有抗炎、抗氧化、抗增殖、抗溃疡和抗分枝杆菌活性。 Spathulenol 在 DPPH 系统中显示出显著的抗氧化活性,IC50 为 85.60 μg/mL。
T12681 (±)​-​Vasicine

(±)​-Peganine

Others Others
(±)-Vasicine is the racemate of Vasicine. Vasicine isolated from Peganum harmala seeds, with anti-ulcer activity.
TN1893 Luteolin-3',7-di-O-glucoside

Others Others
Luteolin-3',7-di-O-glucoside has anti-ulcer and antioxidant activities.
TN3852 Dihydrolicoisoflavone

Antifection Microbiology/Virology
Dihydrolicoisoflavone A possesses weaker anti-H. pylori activity, it may be useful chemopreventive agents for peptic ulcer or gastric cancer in H. pylori-infected individuals.
TN1302 6,8-Diprenylorobol

6,8-二异戊烯基香豌豆苷元

Others; HIV Protease; Antifection Microbiology/Virology; Others; Proteases/Proteasome
6,8-Diprenylorobol possesses weaker anti-H. pylori activity, it may be a useful chemopreventive agent for peptic ulcer or gastric cancer in H. pylori-infected individuals.
TN3926 Eicosanyl caffeate

Others Others
Eicosanyl caffeate has anti-ulcer and moderate antioxidant properties, it exhibits potent elastase inhibitory activity, with the IC(50) value of 0.99 microg/mL.
TN1913 Marmin

Calcium Channel; Antifection; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and secondarily due to the prevention of the effects of endogenous acetylcholine and histamine.
T73653 Pexiganan

Pexiganan(MSI 78 free base),maganin 2 的合成类似物,是一种具有口服活性的广谱强效抗菌肽,主要用于研究糖尿病足溃疡等相关感染。
TN4322 Isopulegol

ATPase; Potassium Channel; GABA Receptor Membrane transporter/Ion channel; Neuroscience
Isopulegol presents depressant- and anxiolytic-like effects, it also has anticonvulsant and bioprotective effects against PTZ-induced convulsions are possibly related to positive modulation of benzodiazepine-sensitive GABAA receptors and to antioxidant properties.Isopulegol presents significant gastroprotective effects in both ethanol- and indomethacin-induced ulcer models, which appear to be mediated, at least in part, by endogenous prostaglandins, K(ATP) channel opening, and antioxidant proper...
TN4223 Homopterocarpin

Antifection Microbiology/Virology
Homopterocarpin and Pterocarpus extract offer gastroprotection against indomethacin- induced ulcer by antioxidative mechanism and the modulation of gastric homeostasis, homopterocarpin may be responsible for, or contribute to the antiulcerogenic property

天然产物

Gastrodenol
Cat.No: T3605
Synonym: Bismuth tripotassium dicitrate,枸橼酸铋钾,Bismuth subcitrate
Target: Others
Dehydrocostus Lactone
Cat.No: T2833
Synonym: Epiligulyl oxide,去氢木香内酯,(-)-Dehydrocostus lactone,去氢木香烃内酯
Target: IκB/IKK
Bletilloside A
Cat.No: TN6577
Synonym: 3-Methoxyshancigusin I
Target: Others
Deoxyartemisinin
Cat.No: TN1568
Synonym: 2-deoxyartemisinin
Target:
Lansoprazole sodium
Cat.No: T21651
Synonym: 兰索拉唑钠,Lansoprazole (sodium), AG-1749 sodium
Target: Proton pump, Phospholipase, Antibacterial
Spathulenol
Cat.No: TN2233
Synonym:
Target: Antioxidant, Antifungal
(±)​-​Vasicine
Cat.No: T12681
Synonym: (±)​-Peganine
Target: Others
Luteolin-3',7-di-O-glucoside
Cat.No: TN1893
Synonym:
Target: Others
Dihydrolicoisoflavone
Cat.No: TN3852
Synonym:
Target: Antifection
6,8-Diprenylorobol
Cat.No: TN1302
Synonym: 6,8-二异戊烯基香豌豆苷元
Target: Others, HIV Protease, Antifection
Eicosanyl caffeate
Cat.No: TN3926
Synonym:
Target: Others
Marmin
Cat.No: TN1913
Synonym:
Target: Calcium Channel, Antifection, Histamine Receptor
Pexiganan
Cat.No: T73653
Synonym:
Target:
Isopulegol
Cat.No: TN4322
Synonym:
Target: ATPase, Potassium Channel, GABA Receptor
Homopterocarpin
Cat.No: TN4223
Synonym:
Target: Antifection
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