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97

抑制剂 & 化合物

12

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP2137L pp60 c-src (521-533) (phosphorylated) acetate

Others Others
pp60 c-src (521-533) (phosphorylated) acetate 是粘着斑形成和细胞扩散的调节剂。它还调节细胞运动,是由促运动透明质酸受体 RHAMM 触发的信号通路中的关键成分。
T39185 pp60 (v-SRC) Autophosphorylation Site, Phosphorylated

pp60 (v-SRC) Autophosphorylation Site, Phosphorylated

pp60 (v-SRC) Autophosphorylation Site, Phosphorylated is a phosphorylated peptide derived from an EGFR substrate. It serves as a valuable tool for quantifying phosphorylated substrates in screening EGFR Kinase inhibitors.
TP1590 MARCKS Peptide(151-175), Phosphorylated

Myristoylated Alanine-Rich C Kinase Substrate peptide (151-175) is a high affinity Protein Kinase C substrate.
TP2137 pp60 c-src (521-533) (phosphorylated)

Peptide corresponding to the pp60c-src carboxy terminal regulatory domain; phosphorylated at Tyr527. Binds to pp60c-src and pp60v-src at the SH2 domain, suppressing their tyrosine kinase activity and transforming potential.
T81578 p60c-src substrate II, phosphorylated

p60c-src substrate II, phosphorylated 是磷酸化的五肽,为 p60c-src substrate II 的磷酸化形式。其代表了蛋白质翻译后修饰的一种,对生物调控具有重要作用。
T7704 KY-226

Phosphatase Metabolism
KY-226 是选择性的,口服活性的和变构蛋白酪氨酸磷酸酶 1B 抑制剂,IC50=0.25 μM,且不激活 PPARγ 。它可以保护神经元免受脑缺血损伤。它通过增强胰岛素和瘦素信号传导发挥抗糖尿病和抗肥胖作用。
T3071 Olverembatinib

GZD 824

Bcr-Abl Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Olverembatinib (GZD 824) 是一种高效的、口服具有活性的pan-Bcr-Abl 抑制剂,具有抗肿瘤活性。它能广泛而有效地抑制突变型 Bcr-Abl。它对天然的 Bcr-Abl 和 Bcr-AblT315I 作用的IC50值分别为 0.34 nM 和 0.68 nM。
T2429 Olverembatinib dimesylate

GZD824 Dimesylate,HQP1351

Bcr-Abl Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Olverembatinib dimesylate (GZD824 Dimesylate) 是一种高效的、口服具有活性的pan-Bcr-Abl 抑制剂,具有抗肿瘤活性。它能广泛而有效地抑制突变型 Bcr-Abl。它对天然的 Bcr-Abl 和 Bcr-AblT315I 作用的IC50值分别为 0.34 nM 和 0.68 nM。
T31929 Giripladib

PLA 695,PLA-695,PLA695

Phospholipase Metabolism
Giripladib (PLA695)(PLX-695)是一种cPLA2特异性抑制剂,可抑制辐射诱导的内皮细胞磷酸化ERK 和磷酸化Akt 的增加。
T26193 SKLB-163

SKLB163

MAPK; Akt; Caspase; Rho; JNK Apoptosis; Cell Cycle/Checkpoint; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling; Proteases/Proteasome
SKLB-163 通过下调 RhoGDI、激活 JNK-1 信号通路和 caspase-3 以及减少磷酸化 Akt 和 p44/42 MAPK 发挥作用。
TP1789L Malantide acetate(86555-35-3 free base)

PKA; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Malantide acetate(86555-35-3 free base) 是一种由环 AMP 依赖性蛋白激酶 (PKA) 磷酸化的十二肽,可增加 PKA 活性。 Malantide 是一种由 PKA 磷酸化的合成肽,用于在体外测量 PKA 活性。
T67772 Phos-tag Acrylamide AAL-107

Phos-tag Acrylamide AAL-107 是一种丙烯酰胺悬垂物,可用作可视化磷酸化蛋白质的工具。
T3438 S107

Others Others
S107 是一种 RyR 选择性 1, 4-苯并硫氮杂卓衍生物,通过增强 calstabin2 与突变和/或 PKA 磷酸化通道的结合亲和力来稳定 RyR2 通道。
T26078 Rhodblock 6

Rhodblock6,Rhodblock-6

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
Rhodblock 6 是一种 Rho 激酶 (ROCK) 抑制剂,可抑制磷酸化 MRLC(肌球蛋白调节轻链)定位,通过特异性抑制 Rho 激酶的活性发挥作用。
T6762 AS1842856

Autophagy; FOXO1 Apoptosis; Autophagy
AS1842856 是一种特异性的Foxo1抑制剂,IC50为 30 nM。它抑制自噬,直接与 FoxO1 结合而降低 FoxO1 的活性。
T17205 UNC2541

Others; FLT; TAM Receptor Angiogenesis; Others; Tyrosine Kinase/Adaptors
UNC2541 是 Mer 酪氨酸激酶特异性抑制剂,与 MerTK ATP 结合口袋结合的IC50值为 4.4 nM,对其选择性远高于 Axl,Tyro3 和 Flt3。它能够抑制磷酸化的 MerTK (pMerTK;EC50,510 nM)。
T14569 BI8626

E1/E2/E3 Enzyme Ubiquitination
BI8626 是一种泛素连接酶 HUWE1 抑制剂,对 NOD/ShiLtj 小鼠自发性干燥综合征具有保护作用。BI8626 抑制细胞内胆固醇并降低磷酸化 ZAP-70、CD25 和其他激活标志物的表达,抑制 CD4 T 细胞的增殖。
T1790 Fosaprepitant dimeglumine

福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt

Neurokinin receptor GPCR/G Protein; Neuroscience
Fosaprepitant dimeglumine (MK-0517) 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。
T7280 CAY10594

Phospholipase Metabolism
CAY10594 是磷脂酶 D2 抑制剂 (体外IC50=140 nM,细胞IC50=110 nM)。它在体外显著阻碍乳腺癌细胞的侵袭性迁移,并调节磷酸化 GSK-3β/JNK 轴改善扑热息痛诱导的急性肝损伤。
T27242 EF24

EF 24,EF-24,3,5-Bis[(2-fluorophenyl)Methylene]-4-piperidinone

ERK; MEK; Caspase Apoptosis; MAPK; Proteases/Proteasome
EF24 (3,5-Bis[(2-fluorophenyl)Methylene]-4-piperidinone) 是姜黄素类似物,口服生物利用度高,抗肿瘤作用强。它可增强活化的 Caspase3 及 Caspase9 的水平,并抑制 MEK1 及 ERK 的磷酸化形式的表达。它可以抑制口腔鳞状细胞癌细胞的 MAPK/ERK 信号通路,从而发挥抗肿瘤作用。
T16961 Supinoxin

RX-5902

Apoptosis; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Supinoxin (RX-5902) 是磷酸化 p68 RNA 解旋酶的强效口服活性抑制剂,是一种抗肿瘤试剂。它与 Y593 磷酸化的 p68 相互作用并减弱 β-catenin 的核穿梭性。它诱导细胞凋亡并抑制 TNBC 癌细胞系的生长,IC50的范围为 10 nM 至 20 nM。
T15378L Gemcitabine elaidate hydrochloride

CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride

Others Others
Gemcitabine elaidate (CP-4126) hydrochloride 是 Gemcitabine 的亲脂性前药。Gemcitabine elaidate hydrochloride 通过酯酶转化为 Gemcitabine 以被磷酸化。Gemcitabine elaidate hydrochloride 可以口服给药,具有抗肿瘤活性。
T1643 Penciclovir

喷昔洛韦,BRL 39123,VSA 671

HCV Protease; Antifection; HSV Microbiology/Virology; Proteases/Proteasome
Penciclovir (BRL 39123) 是一种疱疹病毒核苷类似物 DNA 聚合酶抑制剂。它作用于HSV1 和 2,IC50分别为 0.04-1.8 μg/mL 和 0.06-4.4 μg/mL。
T9636 Dalpiciclib

SHR-6390

CDK Cell Cycle/Checkpoint
Dalpiciclib (SHR-6390) 是一种高选择性、口服生物利用度和相当效力的 CDK4 和 CKD6 抑制剂,IC50 分别为 12.4 nM 和 9.9 nM。它通过抑制磷酸化 Rb 蛋白和诱导 G1 细胞周期阻滞在食管鳞状细胞癌中发挥有效的抗肿瘤活性。
T37207L Cdk5 Substrate acetate

CDK Cell Cycle/Checkpoint
Cdk5 Substrate acetate 是一种丝氨酸/苏氨酸激酶,主要在神经元组织中具有活性。与 p25 或 p35 一起,Cdk5 磷酸化一系列蛋白质,包括组蛋白 H1 和 tau。 它是一种合成肽 (PKTPKKAKKL),对应于组蛋白 H1 的序列。它被 Cdk5 磷酸化,Km 值为 5 µM。
T6501 Fludarabine Phosphate

NSC 312887 Phosphate,fludara Phosphate,F-ara-A (NSC 312887) Phosphate,F-ara-AMP,磷酸氟达拉滨

Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Fludarabine Phosphate (NSC 312887 Phosphate) 是一种腺苷和脱氧腺苷类似物,与 dATP 竞争,并入到 DNA,可以抑制 DNA 聚合酶 α、核糖核苷酸还原酶和 DNA 引发酶,从而中断 DNA 合成并抑制肿瘤细胞生长。
T6446 Clevudine

L-FMAU,克拉夫定,Levovir

HBV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Clevudine (Levovir) 是一种非自然 L-构型的核苷类似物,是一种与聚合酶结合的非竞争性抑制剂,具有较强的抗 HBV 活性,半衰期长,毒性低的特点。
T27709 K67

K 67,K-67

K67 is a specific inhibitor against the interaction between KEAP1 DC domain and S349-phosphorylated KIR of p62/SQSTM1.
TP1789 Malantide

Malantide is a dodecapeptide phosphorylated by cyclic AMP-dependent protein kinase (PKA), and increases PKA activity.Malantide is a synthetic peptide that is phosphorylated by PKA and is used to measure PKA activity in vitro.
T40829 D-Erythritol 4-phosphate

D-erythritol 4-phosphate is a phosphorylated component isolated from the hydrolysate.
T29731 Agrocinopine

Agrocinopine A

Agrocinopine is an Opine phosphorylated sugar synthesized by crown gall tumors.
T27655 JG-48

JG-48 is an inhibitor of Hsp70. JG-48 suppresses phosphorylated and total Tau in cells, endogenous Tau in neuroblastoma cells.
T36944 Ara-G

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Ara-G 是一种脱氧鸟苷 (GdR) 类似物和核苷类似物,可被 T 淋巴谱系细胞迅速转化为其相应的阿拉伯糖基鸟嘌呤核苷酸三磷酸 (araGTP),从而抑制 DNA 合成和对 T 淋巴母细胞的选择性体外毒性细胞系以及来自 T 细胞急性淋巴细胞白血病 (ALL) 患者的新鲜分离的白血病细胞。
T73179 HDAC-IN-50

HDAC-IN-50是一种口服活性的有效FGFR和HDAC双重抑制剂,其IC50值针对FGFR1、FGFR2、FGFR3、FGFR4、HDAC1、HDAC2、HDAC6、HDAC8分别为0.18、1.2、0.46、1.4、1.3、1.6、2.6、13 nM。该化合物能诱导(Apoptosis)及使细胞周期在G0/G1期停滞,降低pFGFR1、pERK、pSTAT3的表达,展现出抗肿瘤活性。
T83052 Anti-inflammatory agent 60

NF-κB NF-κB
Anti-inflammatory agent 60 (compound 21) 的 IC50 值针对一氧化氮生成为 12.95 μM。此化合物通过浓度依赖性方式降低 iNOS、phosphorylated p65 以及 β-catenin 的表达。
TP1602 [pThr3]-CDK5 Substrate

[pThr3]-CDK5 Substrate is an effective Phospho-Thr3CDK5 Substrate.[pThr3]-CDK5 Substrate is phosphorylated by CDK5 with a Km value of 6 µM[1].
TP1660 [pThr3]-CDK5 Substrate (TFA)

[pThr3]-CDK5 Substrate TFA is an effective Phospho-Thr3CDK5 Substrate. [pThr3]-CDK5 Substrate is phosphorylated by CDK5 with a Km value of 6 µM.
T40447 T-705RMP

T-705RMP, the phosphorylated metabolite derived from T-705, demonstrates a limited inhibitory impact on the host cells' IMP dehydrogenase (IMPDH) activities, with an IC 50 value of 601 μM.
T35652 2'-Deoxyguanosine 5'-monophosphate (sodium salt hydrate)

2'-Deoxyguanosine 5'-monophosphate (dGMP) is used as a substrate of guanylate kinases to generate dGDP, which in turn is phosphorylated to dGTP, a nucleotide precursor used in DNA synthesis. In addition, dGMP can be efficiently phosphorylated by the type I thymidylate kinase of the malarial agent P. falciparum. In humans, deficiency of mitochondrial deoxyguanosine kinase, which synthesizes dGMP from ATP and deoxyguanosine, contributes to mitochondrial DNA depletion syndrome.
T37602 GSK 143

Spleen tyrosine kinase (Syk) inhibitor (pIC50 = 7.5). Also inhibits phosphorylated Erk (pIC50 = 7.1). Decreases cell number and viability in chronic lymphocytic leukemia (CCL) cell lines. Liddle et al (2011) Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor. Bioorg.Med.Chem.Lett. 21 6188 PMID:21903390 |Varghese et al (2018) Highly selective SYK inhibitor, GSK143, abrogates survival signals in chronic lymphocytic leukaemia. Br.J.Haematol 182 9...
T10407 Gartisertib

ATR inhibitor 2

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
ATR inhibitor 2 is an orally active, ATP-competitive, and selective ATR inhibitor (Ki <150 pM) with antitumor activity. ATR inhibitor 2 potently inhibits ATR-driven phosphorylated checkpoint kinase-1 (Chk1) phosphorylation (IC50: 8 nM).
T22421 S107 hydrochloride

Others Others
S107 hydrochloride, a RyR-selective 1,4-benzothiazepine derivative, could stabilize RyR2 channels via enhancing the binding affinity of calstabin2 to mutant and/or PKA-phosphorylated channels.
T73303 BTK-IN-17

BTK-IN-17是一种选择性且具有BTK 抑制剂,IC50值为 13.7 nM。BTK-IN-17 降低 p-BTKY223和 p-PLCγ2Y1217的表达。BTK-IN-17 具有抗炎作用。
T76475 Casein Kinase II Substrate

Casein KinaseII Substrate 是一种酪蛋白激酶 II (CK2) 肽底物,可被CK2选择性磷酸化。
T39586 Cantrixil

TRX-E-002-1

Cantrixil (TRX-E-002-1) is a second-generation super-benzopyran (SBP) compound, derived from TRX-E-002. It elicits an increase in phosphorylated c-Jun levels, leading to caspase-mediated apoptosis in ovarian cancer cells. Cantrixil exhibits potent pan anti-cancer activity against various cancer phenotypes.
TP1716 Calmodulin-Dependent Protein Kinase II (281-309)

Calmodulin-Dependent Protein Kinase II 281-309

Calmodulin-Dependent Protein Kinase II (281-309) is a synthetic peptide that can be phosphorylated at Thr286 by PKC and inhibits CaM kinase II (IC50 = 80 nM).
T78131 Emtricitabine triphosphate tetrasodium salt

(-)-Emtricitabine triphosphate tetrasodium salt

Reverse Transcriptase Microbiology/Virology
Emtricitabinetriphosphatetetrasodium salt 为 Emtricitabinetriphosphate 的四钠盐。 Emtricitabinetriphosphate 本身为 Emtricitabine 的磷酸化代谢物,后者作为核苷类逆转录酶抑制剂对抗 HIV 与 HBV。
TP1641 [pSer2, pSer5, pSer7]-CTD TFA

[pSer2, pSer5, pSer7]-CTD (TFA) is a substrate for CDK7(cyclin-dependent protein kinase), a phosphorylated polypeptide at ser2, ser5, and ser7 of RNA polymerase II carboxyl terminus (CTD).
T62519 SW02

SW02 是一种有效的 Hsp70 的 ATPase 活性激活剂 (EC50: 150 μM)。SW02 能够积累总 tau 和磷酸化 tau (pTau)。
T35928 NVS-PAK1-C

NVS-PAK1-C

NVS-PAK1-C 是一种有效的、ATP 竞争的特异性变构 PAK1抑制剂探针。NVS-PAK1-C 可抑制去磷酸化的 PAK1(IC50= 5 nM) 和磷酸化的 PAK1(IC50= 6 nM)。NVS-PAK1-C 也可以抑制去磷酸化的 PAK2 (IC50=270 nM) 和磷酸化的 PAK2 (IC50=720 nM)。

化合物

pp60 c-src (521-533) (phosphorylated) acetate
Cat.No: TP2137L
Synonym:
Target: Others
pp60 (v-SRC) Autophosphorylation Site, Phosphorylated
Cat.No: T39185
Synonym: pp60 (v-SRC) Autophosphorylation Site, Phosphorylated
Target:
MARCKS Peptide(151-175), Phosphorylated
Cat.No: TP1590
Synonym:
Target:
pp60 c-src (521-533) (phosphorylated)
Cat.No: TP2137
Synonym:
Target:
p60c-src substrate II, phosphorylated
Cat.No: T81578
Synonym:
Target:
KY-226
Cat.No: T7704
Synonym:
Target: Phosphatase
Olverembatinib
Cat.No: T3071
Synonym: GZD 824
Target: Bcr-Abl
Olverembatinib dimesylate
Cat.No: T2429
Synonym: GZD824 Dimesylate,HQP1351
Target: Bcr-Abl
Giripladib
Cat.No: T31929
Synonym: PLA 695,PLA-695,PLA695
Target: Phospholipase
SKLB-163
Cat.No: T26193
Synonym: SKLB163
Target: MAPK, Akt, Caspase, Rho, JNK
Malantide acetate(86555-35-3 free base)
Cat.No: TP1789L
Synonym:
Target: PKA, PKC
Phos-tag Acrylamide AAL-107
Cat.No: T67772
Synonym:
Target:
S107
Cat.No: T3438
Synonym:
Target: Others
Rhodblock 6
Cat.No: T26078
Synonym: Rhodblock6,Rhodblock-6
Target: ROCK
AS1842856
Cat.No: T6762
Synonym:
Target: Autophagy, FOXO1
UNC2541
Cat.No: T17205
Synonym:
Target: Others, FLT, TAM Receptor
BI8626
Cat.No: T14569
Synonym:
Target: E1/E2/E3 Enzyme
Fosaprepitant dimeglumine
Cat.No: T1790
Synonym: 福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt
Target: Neurokinin receptor
CAY10594
Cat.No: T7280
Synonym:
Target: Phospholipase
EF24
Cat.No: T27242
Synonym: EF 24,EF-24,3,5-Bis[(2-fluorophenyl)Methylene]-4-piperidinone
Target: ERK, MEK, Caspase
Supinoxin
Cat.No: T16961
Synonym: RX-5902
Target: Apoptosis, DNA/RNA Synthesis
Gemcitabine elaidate hydrochloride
Cat.No: T15378L
Synonym: CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride
Target: Others
Penciclovir
Cat.No: T1643
Synonym: 喷昔洛韦,BRL 39123,VSA 671
Target: HCV Protease, Antifection, HSV
Dalpiciclib
Cat.No: T9636
Synonym: SHR-6390
Target: CDK
Cdk5 Substrate acetate
Cat.No: T37207L
Synonym:
Target: CDK
Fludarabine Phosphate
Cat.No: T6501
Synonym: NSC 312887 Phosphate,fludara Phosphate,F-ara-A (NSC 312887) Phosphate,F-ara-AMP,磷酸氟达拉滨
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Clevudine
Cat.No: T6446
Synonym: L-FMAU,克拉夫定,Levovir
Target: HBV, DNA/RNA Synthesis
K67
Cat.No: T27709
Synonym: K 67,K-67
Target:
Malantide
Cat.No: TP1789
Synonym:
Target:
D-Erythritol 4-phosphate
Cat.No: T40829
Synonym:
Target:
Agrocinopine
Cat.No: T29731
Synonym: Agrocinopine A
Target:
JG-48
Cat.No: T27655
Synonym:
Target:
Ara-G
Cat.No: T36944
Synonym:
Target: Nucleoside Antimetabolite/Analog
HDAC-IN-50
Cat.No: T73179
Synonym:
Target:
Anti-inflammatory agent 60
Cat.No: T83052
Synonym:
Target: NF-κB
[pThr3]-CDK5 Substrate
Cat.No: TP1602
Synonym:
Target:
[pThr3]-CDK5 Substrate (TFA)
Cat.No: TP1660
Synonym:
Target:
T-705RMP
Cat.No: T40447
Synonym:
Target:
2'-Deoxyguanosine 5'-monophosphate (sodium salt hydrate)
Cat.No: T35652
Synonym:
Target:
GSK 143
Cat.No: T37602
Synonym:
Target:
Gartisertib
Cat.No: T10407
Synonym: ATR inhibitor 2
Target: ATM/ATR
S107 hydrochloride
Cat.No: T22421
Synonym:
Target: Others
BTK-IN-17
Cat.No: T73303
Synonym:
Target:
Casein Kinase II Substrate
Cat.No: T76475
Synonym:
Target:
Cantrixil
Cat.No: T39586
Synonym: TRX-E-002-1
Target:
Calmodulin-Dependent Protein Kinase II (281-309)
Cat.No: TP1716
Synonym: Calmodulin-Dependent Protein Kinase II 281-309
Target:
Emtricitabine triphosphate tetrasodium salt
Cat.No: T78131
Synonym: (-)-Emtricitabine triphosphate tetrasodium salt
Target: Reverse Transcriptase
[pSer2, pSer5, pSer7]-CTD TFA
Cat.No: TP1641
Synonym:
Target:
SW02
Cat.No: T62519
Synonym:
Target:
NVS-PAK1-C
Cat.No: T35928
Synonym: NVS-PAK1-C
Target:
Cat. No. Product Name Target Signaling Pathways
T5113 L-GLUCOSE

L-葡萄糖,L-(-)-Glucose

Others Others
L-Glucose (L-(-)-Glucose) 是一种 D-glucose 的对映体,可促进食物的摄取。
T3262 Phosphocreatine disodium

Disodium phosphocreatine,Phosphocreatine disodium salt,Creatine phosphate disodium salt,磷酸肌酸钠

Others; Endogenous Metabolite Metabolism; Others
Phosphocreatine disodium (Phosphocreatine disodium salt) 是一种磷酸化的肌酸分子,在肌肉、骨骼和大脑中作为一种可快速动员的高能磷酸盐储备。
T0894 Thiamine hydrochloride

盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride

Apoptosis; HBV; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology
Thiamine hydrochloride (Vitamin B1) 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。
T4726 D-Glucose 6-phosphate sodium

G6P sodium salt,D-Glucose 6-phosphate sodium salt,D-葡萄糖-6-磷酸钠盐,Sodium Glucose-6-Phosphate

Others; Endogenous Metabolite Metabolism; Others
D-Glucose 6-phosphate sodium (G6P sodium salt) 是内源性代谢产物的一种。
T5057 DL-O-Phosphoserine

DL-O-磷酸丝氨酸,DL-2-Amino-3-hydroxypropanoic acid 3-phosphate,O-PHOSPHO-L-SERINE,DL-SOP

Others; Endogenous Metabolite Metabolism; Others
DL-O-Phosphoserine (DL-SOP) 是丝氨酸和磷酸的酯,是人类生物流体中的正常代谢物。
T78473 Sphingosine (d17:1)

C17 Sphingosine

Sphingosine (d17:1) (C17 Sphingosine)是一种存在于人类皮肤中的17碳鞘脂,可被鞘氨醇激酶的磷酸化。Sphingosine C-17作为内标可用于进行鞘脂类化合物的光谱分析。
T7989 Trimethyl phosphate

Others Others
Trimethyl phosphate 是一种有机磷化合物,是催化磷酸化化合物水解的酶的抑制剂,已被用作合成肽和其他蛋白质的反应物,用作合成有机和无机化合物的催化剂,以及用作合成药物的试剂。
T5069 D-Glucose 6-phosphate potassium salt

Others Others
在细胞中,当葡萄糖被己糖激酶或葡萄糖激酶磷酸化或在糖原分解过程中通过磷酸葡萄糖变位酶转化葡萄糖 1-磷酸时,会产生D-glucose 6-phosphate (G6P)。 G6P 位于糖酵解和戊糖磷酸途径的起点。当血糖水平高时,它也可以作为糖原储存。
T5079 Adenosine 5'-diphosphate sodium salt

腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt

Others; Endogenous Metabolite Metabolism; Others
Adenosine 5'-diphosphate sodium salt (ADP sodium salt) 是一种核苷二磷酸,是一种 ATP 酶对 ATP 去磷酸化的产物。它通过在 P2T-嘌呤受体上的作用诱导人血小板聚集并抑制刺激的腺苷酸环化酶。
TL0008 Gigantol

Wnt/beta-catenin; Glucosidase Cytoskeletal Signaling; Metabolism; Stem Cells
Gigantol 是一种联苄基化合物,从几种药用兰花中获得,是一种Wnt/β-catenin 通路抑制剂,具有抗肿瘤活性。
T19263 D-Glucose 6-phosphate

Others Others
D-glucose 6-phosphate is glucose that is phosphorylated on the carbon 6 hydroxyl group.
T35415 α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)

α-D-Glucose-1,6-bisphosphate is abis-phosphorylated derivative of α-D-glucose that has roles in carbohydrate metabolism.1It is the product of the reaction of glucose-1- or 6-phosphate with glucose-1,6-bisphosphate synthase (PGM2LI) in the conversion of 1,3-bisphosphoglycerate to 3-phosphoglycerate.2It is also a cofactor for the bacterial enzyme phosphopentomutase.3,4α-D-Glucose-1,6-bisphosphate has been used in the study of carbohydrate metabolism. 1.Beitner, R.Regulation of carbohydrate metabol...

天然产物

L-GLUCOSE
Cat.No: T5113
Synonym: L-葡萄糖,L-(-)-Glucose
Target: Others
Phosphocreatine disodium
Cat.No: T3262
Synonym: Disodium phosphocreatine,Phosphocreatine disodium salt,Creatine phosphate disodium salt,磷酸肌酸钠
Target: Others, Endogenous Metabolite
Thiamine hydrochloride
Cat.No: T0894
Synonym: 盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride
Target: Apoptosis, HBV, Endogenous Metabolite
D-Glucose 6-phosphate sodium
Cat.No: T4726
Synonym: G6P sodium salt,D-Glucose 6-phosphate sodium salt,D-葡萄糖-6-磷酸钠盐,Sodium Glucose-6-Phosphate
Target: Others, Endogenous Metabolite
DL-O-Phosphoserine
Cat.No: T5057
Synonym: DL-O-磷酸丝氨酸,DL-2-Amino-3-hydroxypropanoic acid 3-phosphate,O-PHOSPHO-L-SERINE,DL-SOP
Target: Others, Endogenous Metabolite
Sphingosine (d17:1)
Cat.No: T78473
Synonym: C17 Sphingosine
Target:
Trimethyl phosphate
Cat.No: T7989
Synonym:
Target: Others
D-Glucose 6-phosphate potassium salt
Cat.No: T5069
Synonym:
Target: Others
Adenosine 5'-diphosphate sodium salt
Cat.No: T5079
Synonym: 腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt
Target: Others, Endogenous Metabolite
Gigantol
Cat.No: TL0008
Synonym:
Target: Wnt/beta-catenin, Glucosidase
D-Glucose 6-phosphate
Cat.No: T19263
Synonym:
Target: Others
α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)
Cat.No: T35415
Synonym:
Target:
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