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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T8239 Cromoglicic acid

Others Others
Cromoglicic acid 可防止肥大细胞释放炎性化学物质,例如组胺。
T0211 Azelastine

Azelastina,Astelin,Azelastinum,氮卓斯汀

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine (Azelastinum) 是一种选择性组胺 1 拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T3979 Emedastine

LY188695,依美斯汀,Emadine

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Emedastine (LY188695) 是一种可口服的,选择性和高亲和力的组胺 H1受体拮抗剂,Ki 值为 1.3 nM。它是苯并咪唑衍生物,可用于过敏性鼻炎、过敏性皮肤疾病和过敏性结膜炎的研究。
T0118 Mizolastine

SL 850324,咪唑司汀,咪唑斯汀

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mizolastine (SL 850324) 是组胺 H1 受体拮抗剂,IC50为 47 nM。它用于治疗过敏反应,如花粉热和荨麻疹等。
T21404 Fluticasone furoate

Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate

Glucocorticoid Receptor Endocrinology/Hormones
Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇,衍生自氟替卡松,Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。
T6242 Rupatadine Fumarate

富马酸卢帕他定,Rinialer,Rupafin,Alergoliber

PAFR; Autophagy; Histamine Receptor Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Rupatadine Fumarate (Rinialer) 是一种可口服的长效PAF/H1受体的双抑制剂,Ki 值分别为 0.55 μM 和 0.1 μM。它可研究过敏性鼻炎和荨麻疹。
T0059 Diphenylpyraline hydrochloride

盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂,抑制多巴胺的吸收。它是可口服的抗组胺试剂,具有抗胆碱和抗过敏作用,可用于缓解过敏性疾病,如鼻炎、花粉热和瘙痒性皮肤疾病等。
T3185 R112

(E)-Elafibranor

Syk Angiogenesis; Tyrosine Kinase/Adaptors
R112 ((E)-Elafibranor) 是ATP 竞争性的 Syk 激酶抑制剂,它能够抑制Syk 激酶活性,Ki=6 nM,IC50=226 nM。
T0211L Azelastine hydrochloride

Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine hydrochloride (Astelin) 是一种选择性组胺 1拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T1030 Triprolidine hydrochloride monohydrate

盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Triprolidine hydrochloride monohydrate 是一种组胺 H1 拮抗剂,用于过敏性鼻炎、哮喘。
T1269 Tripelennamine hydrochloride

Pyribenzamine hydrochloride,去敏灵,Tripelennamine HCl,Pyribenzamine HCl,盐酸曲吡那敏

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) 是一种组胺 H1 拮抗剂,具有低镇静作用,但经常刺激胃肠道。
T2335 Ebastine

Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ebastine (Kestine) 是一种可口服的组胺 H1 受体拮抗剂,用于过敏性鼻炎的症状和慢性特发性荨麻疹的研究。
T0205 Brompheniramine maleate

Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Brompheniramine maleate (Dimotane) 是一种可口服的丙胺类抗组胺剂,具有抗胆碱能和抗抑郁作用,可用于过敏性鼻炎和缓解疼痛的研究。它是一种选择性组胺 H1 受体拮抗剂,Kd 为 6.06 nM。
T0188 Fluticasone (propionate)

丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate

Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Microbiology/Virology
Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,亲和力KD 为 0.5 nM。具有抗病毒活性。
T0089 Cetirizine dihydrochloride

盐酸西替利嗪,P071,UCB P071,Cetirizine DiHCl

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Cetirizine dihydrochloride (UCB P071) 是羟嗪的羧化代谢物,是特异性口服有效的 H1 受体长效拮抗剂。它标记抗过敏特性,抑制过敏反应期间嗜酸性粒细胞趋化,可有效治疗过敏性鼻炎、确诊荨麻疹和花粉诱发的哮喘。
T1553 Chlorpheniramine maleate

马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Chlorpheniramine maleate (NCI-C55265) 是一种组胺 H1 拮抗剂,IC50为12 nM,用于过敏反应、花粉热、鼻炎、荨麻疹和哮喘。
T6660 SB-705498

TRP/TRPV Channel Membrane transporter/Ion channel
SB705498 是一种口服有效的 TRPV1选择性拮抗剂,pIC50值为 7.1。
T1531 Mometasone furoate

糠酸莫美他松,糠酸莫米松,Sch32088

Glucocorticoid Receptor Endocrinology/Hormones
Mometasone furoate (Sch32088) 是糖皮质激素受体激动剂,具有抗炎和抗过敏作用。它是皮质固醇类试剂,动物模型中,可局部应用于气道炎症、慢性皮肤湿疹、哮喘。
T1278 Astemizole

Laridal,Histaminos,Paralergin,阿司咪唑

Potassium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Astemizole (Laridal) 是一种长效、非镇静抗组胺药,用于治疗季节性过敏性鼻炎、哮喘、过敏性结膜炎和慢性特发性荨麻疹。它是组胺 H1 受体的拮抗剂,IC50值为 4 nM,还阻断 hERG K+通道,IC50值为 0.9 nM,具有抗胆碱能和止痒作用。
T2270 Trans-Tranilast

Tranilast trans-,反式-曲尼司特,反-曲尼司特

RAAS Endocrinology/Hormones
Trans-Tranilast 是抗过敏剂,可用于过敏性鼻炎、支气管哮喘和特应性皮炎的研究。
T77426 Pascolizumab

SB-240683

IL Receptor Immunology/Inflammation
Pascolizumab (SB-240683) 是一种人源化抗 IL-4 单克隆抗体。Pascolizumab 具有哮喘作用,可用于研究过敏性鼻炎。
T1470 Fexofenadine hydrochloride

Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,盐酸非索非那定,Telfast,Fexofenadine HCl,Allegra,MDL 16455A

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) 是一种抗组胺药,用于治疗过敏性鼻炎、血管性水肿和慢性荨麻疹。
T61213 PF-03654764

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
PF-03654764 是一种具有口服活性、高效性和选择性的组胺 H3 受体拮抗剂,对人 H3 和大鼠 H3 具有抑制作用, Ki 值分别为 1.2 nM 和 7.9 nM。PF-03654764 常与 Fexofenadine 一起联合用药来治疗过敏性鼻炎。
T2396 Ramatroban

BAY u3405,雷马曲班

GPR; Prostaglandin Receptor; PPAR DNA Damage/DNA Repair; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism
Ramatroban (BAY u3405) 是一种血栓素 A(2) (TxA(2)) 拮抗剂,IC50为 14 nM。它还通过抑制PGD2结合从而拮抗CRTH2,IC50为113 nM。它用于治疗过敏性鼻炎,可用于治疗哮喘的研究。
T22354 Levocetirizine Dihydrochloride

Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydrochloride is the R-enantiomer of Cetirizine, which gives it a higher affinity for the H1-receptor than the S-enantiomer. Due to this enhanced affinity, Levocetirizine Dihydrochloride is effective in treating allergic rhinitis and chronic idiopathic urticaria.
T1097 Loratadine

氯雷他定,SCH 29851,Loratidine

Influenza Virus; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Loratadine (SCH 29851) 是一种组胺 H1受体反向激动剂,IC50>32 μM。它抑制炎症介质的免疫释放,具有抗登革热病毒的活性。
T2392 Nafamostat mesylate

甲磺酸萘莫司他,FUT-175

Apoptosis; Serine/threonin kinase; SARS-CoV; Serine Protease Apoptosis; Cell Cycle/Checkpoint; Metabolism; Microbiology/Virology; Proteases/Proteasome
Nafamostat mesylate (FUT-175) 是一种广谱丝氨酸蛋白酶抑制剂,血管舒缓素抑制剂,能抑制血液凝固。它通过降低颗粒酶活性和 CTL 细胞溶解抑制T 细胞自身反应活性,可抑制SARS-CoV-2 的激活。它还是潜在的补体抑制剂。
T4563 Thonzylamine

neohetramine,松齐拉敏

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Thonzylamine (neohetramine) 是可口服的H1组胺受体拮抗剂,具有抗组胺和抗过敏特性,可用于鼻充血、过敏性结膜炎和其他过敏性疾病的研究。
T21112 Triprolidine hydrochloride

295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil

Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.
T10437 AZD8848

TLR Immunology/Inflammation
AZD8848 is a selective antedrug agonist of toll-like receptor 7 (TLR7). It is developed for the research of asthma and allergic rhinitis.
T69737 SCH-79687

SCH-79687 is a histamine antagonist selective for the H3 subtype. This H3 antagonist may play a role in allergic rhinitis.
T29951 Ambicromil

Ambicromil is used for allergic rhinitis.
T0785L Dexchlorpheniramine free base

Polaramine,Dexchlorpheniramine Maleate,Mylaramine

Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.
T27556 HSR-609

HSR609,FY609,FY-609,FY 609

HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.
T37386 Dihydro Montelukast

Dihydro montelukast is a potential impurity found in commercial montelukast preparations. Montelukast (sodium salt) is a potent and selective cysteinyl leukotriene 1 (CysLT1) receptor antagonist. Formulations containing montelukast are used for the treatment of asthma as well as for the symptoms associated with allergic rhinitis.
T27445 GSK-1004723

GSK 1004723

GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.
T74646 PM-81I

PM-81I为一种高效STAT6抑制剂(针对SH2结构域),可显著减少STAT6的磷酸化水平。适用于研究过敏性肺病、过敏性鼻炎、慢性阻塞性肺病或癌症。
T21247 Carbinoxamine

Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine

Carbinoxamine, an anticholinergic and antihistamine agent, is used for hay fever, angioedema, vasomotor rhinitis, mild urticaria, dermatographism and allergic conjunctivitis. It is a histamine antagonist, specifically an H1-antagonist.
T68280 Adriforant

Adriforant, also known as ZPL-3893787, PF-3893787 and ZPL-389, is a novel histamine H4 receptor antagonist. Adriforant shows an excellent in vitro profile that warrants their further investigation in relevant models of human disease. Histamine H4 receptor (H4R) has become a promising target for immuno-inflammatory diseases, such as allergic rhinitis, asthma or dermal allergies.
T26770 Bencycloquidium Bromide

BCQB

Bencycloquidium Bromide is a muscarinic M3 antagonist. Bencycloquidium bromide inhibits nasal hypersecretion in a rat model of allergic rhinitis. Bencycloquidium Bromide showed high affinity toward the M(3) receptor in Chinese hamster ovary (CHO) cells (M
T16476 PF-03654746

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。
T73972 Fexofenadine Impurity F

Fexofenadine Impurity F 是 Fexofenadine 的杂质。 Fexofenadine 是一种H1R 拮抗剂,可用于研究季节性过敏性鼻炎和慢性特发性荨麻疹。
T60514 Triprolidine

Triprolidine 是一种口服活性的组胺H1受体拮抗剂,可用于过敏性鼻炎的研究 。Triprolidine 具有脊髓运动和知觉阻止的作用。
T62669 Tripelennamine citrate

Tripelennamine citrate 是一种乙二胺衍生物,是一种有效的组胺 H1 受体拮抗剂。Tripelennamine citrate 能够减少组织胺引起的机体过敏反应。Tripelennamine citrate 能够用于研究鼻炎、结膜炎、过敏性和过敏性反应。
T73129 STAT6-IN-1

STAT6-IN-1(化合物19a)是一种针对STAT6的SH2结构域表现出较高亲和力(IC50=0.028 µM)的STAT6抑制剂。该化合物主要用于研究过敏性肺病、过敏性鼻炎、慢性阻塞性肺病或癌症。
T60392 Tripelennamine

Tripelennamine 是一种乙二胺衍生物,是一种有效的组胺 H1受体拮抗剂,可减轻由组织胺引起的机体过敏反应。Tripelennamine 可用于鼻炎、结膜炎、过敏性和过敏性反应的研究。
T38350 TAS 205

TAS 205 is an inhibitor of hematopoietic prostaglandin D synthase (H-PGDS; IC50= 55.8 nM).1It is selective for H-PGDS over lipocalin-type PGDS (L-PGDS) at 100 μM, as well as over enzyme and receptor panels at 10 μM. TAS 205 inhibits production of prostaglandin D2induced by A23187 in KU812 human and RBL-2H3 rat basophils with IC50values of 78.3 and 181.3 nM, respectively. It inhibits ovalbumin-induced nasal lavage fluid eosinophil infiltration and late-phase nasal obstruction in an ovalbumin-sens...
T69918 Adriforant tartrate hydrate

Adriforant tartrate hydrate, also known as ZPL-3893787 tartrate hydrate, PF-3893787 tartrate hydrate and ZPL-389 tartrate hydrate, is a novel histamine H4 receptor antagonist. Adriforant tartrate hydrate shows an excellent in vitro profile that warrants their further investigation in relevant models of human disease. Histamine H4 receptor (H4R) has become a promising target for immuno-inflammatory diseases, such as allergic rhinitis, asthma or dermal allergies.
T60843 Brompheniramine

Brompheniramine ((±)-Brompheniramine) 是具有口服活性的烷基胺类抗组胺药。Brompheniramine 是组胺 H1 受体的选择性拮抗剂 (Kd = 6.06 nM)。Brompheniramine 可用于过敏性鼻炎,它具有抗胆碱能、抗抑郁和麻醉作用。Brompheniramine 可阻断钙离子通道、钠离子通道和 hERG 通道,IC50分别为 16.12 μM, 21.26 μM 和 0.90 μM。
T74583 Desmethylazelastine

Desmethylazelastine是Azelastine经由细胞色素P450酶系统的氧化代谢形成的主要活性代谢物,具有97%的蛋白结合率和54小时的消除半衰期。Azelastine作为一种口服活性的组胺H1受体拮抗剂,特点是选择性高和亲和力强。它主要用于治疗过敏性鼻炎、哮喘、糖尿病高脂血症以及用于SARS-CoV-2的研究。

化合物

Cromoglicic acid
Cat.No: T8239
Synonym:
Target: Others
Azelastine
Cat.No: T0211
Synonym: Azelastina,Astelin,Azelastinum,氮卓斯汀
Target: SARS-CoV, Histamine Receptor
Emedastine
Cat.No: T3979
Synonym: LY188695,依美斯汀,Emadine
Target: Histamine Receptor
Mizolastine
Cat.No: T0118
Synonym: SL 850324,咪唑司汀,咪唑斯汀
Target: Histamine Receptor
Fluticasone furoate
Cat.No: T21404
Synonym: Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate
Target: Glucocorticoid Receptor
Rupatadine Fumarate
Cat.No: T6242
Synonym: 富马酸卢帕他定,Rinialer,Rupafin,Alergoliber
Target: PAFR, Autophagy, Histamine Receptor
Diphenylpyraline hydrochloride
Cat.No: T0059
Synonym: 盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride
Target: Histamine Receptor
R112
Cat.No: T3185
Synonym: (E)-Elafibranor
Target: Syk
Azelastine hydrochloride
Cat.No: T0211L
Synonym: Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin
Target: SARS-CoV, Histamine Receptor
Triprolidine hydrochloride monohydrate
Cat.No: T1030
Synonym: 盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride
Target: Histamine Receptor
Tripelennamine hydrochloride
Cat.No: T1269
Synonym: Pyribenzamine hydrochloride,去敏灵,Tripelennamine HCl,Pyribenzamine HCl,盐酸曲吡那敏
Target: Histamine Receptor
Ebastine
Cat.No: T2335
Synonym: Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305
Target: Histamine Receptor
Brompheniramine maleate
Cat.No: T0205
Synonym: Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane
Target: 5-HT Receptor, Histamine Receptor
Fluticasone (propionate)
Cat.No: T0188
Synonym: 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate
Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite
Cetirizine dihydrochloride
Cat.No: T0089
Synonym: 盐酸西替利嗪,P071,UCB P071,Cetirizine DiHCl
Target: Histamine Receptor
Chlorpheniramine maleate
Cat.No: T1553
Synonym: 马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate
Target: Histamine Receptor
SB-705498
Cat.No: T6660
Synonym:
Target: TRP/TRPV Channel
Mometasone furoate
Cat.No: T1531
Synonym: 糠酸莫美他松,糠酸莫米松,Sch32088
Target: Glucocorticoid Receptor
Astemizole
Cat.No: T1278
Synonym: Laridal,Histaminos,Paralergin,阿司咪唑
Target: Potassium Channel, Histamine Receptor
Trans-Tranilast
Cat.No: T2270
Synonym: Tranilast trans-,反式-曲尼司特,反-曲尼司特
Target: RAAS
Pascolizumab
Cat.No: T77426
Synonym: SB-240683
Target: IL Receptor
Fexofenadine hydrochloride
Cat.No: T1470
Synonym: Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,盐酸非索非那定,Telfast,Fexofenadine HCl,Allegra,MDL 16455A
Target: Histamine Receptor
PF-03654764
Cat.No: T61213
Synonym:
Target: Histamine Receptor
Ramatroban
Cat.No: T2396
Synonym: BAY u3405,雷马曲班
Target: GPR, Prostaglandin Receptor, PPAR
Levocetirizine Dihydrochloride
Cat.No: T22354
Synonym: Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride
Target: Histamine Receptor
Loratadine
Cat.No: T1097
Synonym: 氯雷他定,SCH 29851,Loratidine
Target: Influenza Virus, Histamine Receptor
Nafamostat mesylate
Cat.No: T2392
Synonym: 甲磺酸萘莫司他,FUT-175
Target: Apoptosis, Serine/threonin kinase, SARS-CoV, Serine Protease
Thonzylamine
Cat.No: T4563
Synonym: neohetramine,松齐拉敏
Target: Histamine Receptor
Triprolidine hydrochloride
Cat.No: T21112
Synonym: 295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil
Target:
AZD8848
Cat.No: T10437
Synonym:
Target: TLR
SCH-79687
Cat.No: T69737
Synonym:
Target:
Ambicromil
Cat.No: T29951
Synonym:
Target:
Dexchlorpheniramine free base
Cat.No: T0785L
Synonym: Polaramine,Dexchlorpheniramine Maleate,Mylaramine
Target:
HSR-609
Cat.No: T27556
Synonym: HSR609,FY609,FY-609,FY 609
Target:
Dihydro Montelukast
Cat.No: T37386
Synonym:
Target:
GSK-1004723
Cat.No: T27445
Synonym: GSK 1004723
Target:
PM-81I
Cat.No: T74646
Synonym:
Target:
Carbinoxamine
Cat.No: T21247
Synonym: Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine
Target:
Adriforant
Cat.No: T68280
Synonym:
Target:
Bencycloquidium Bromide
Cat.No: T26770
Synonym: BCQB
Target:
PF-03654746
Cat.No: T16476
Synonym:
Target: Histamine Receptor
Fexofenadine Impurity F
Cat.No: T73972
Synonym:
Target:
Triprolidine
Cat.No: T60514
Synonym:
Target:
Tripelennamine citrate
Cat.No: T62669
Synonym:
Target:
STAT6-IN-1
Cat.No: T73129
Synonym:
Target:
Tripelennamine
Cat.No: T60392
Synonym:
Target:
TAS 205
Cat.No: T38350
Synonym:
Target:
Adriforant tartrate hydrate
Cat.No: T69918
Synonym:
Target:
Brompheniramine
Cat.No: T60843
Synonym:
Target:
Desmethylazelastine
Cat.No: T74583
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S0878 Prunetin

樱黄素,Prunusetin

ERK; Dehydrogenase; NF-κB MAPK; Metabolism; NF-κB
Prunetin (Prunusetin) 是一种O-甲基化异黄酮,具有抗炎的作用。它是人醛脱氢酶的有效抑制剂。
T4038 Ectoine

THP(B),L-Ectoine,四氢甲基嘧啶羧酸

Others; Antibacterial Microbiology/Virology; Others
Ectoine (L-Ectoine) 是生活在极其恶劣环境中的细菌所产生的氨基酸衍生物,是一种天然的细胞保护剂。它具有良好的安全性,可研究过敏性鼻炎。它用作渗透调节相容性溶质,可增加皮肤表面的水合作用并稳定脂质层,常用于皮肤护理。

天然产物

Prunetin
Cat.No: T4S0878
Synonym: 樱黄素,Prunusetin
Target: ERK, Dehydrogenase, NF-κB
Ectoine
Cat.No: T4038
Synonym: THP(B),L-Ectoine,四氢甲基嘧啶羧酸
Target: Others, Antibacterial
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