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73

抑制剂 & 化合物

25

天然产物

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Cat. No. Product Name Target Signaling Pathways
T12854 SBI-797812

NAMPT Metabolism
SBI-797812 是在结构上类似于活性位点定向的 NAMPT 抑制剂的化合物,能够阻断这些抑制剂与 NAMPT 的结合。 它将 NAMPT 反应平衡转向 NMN 形成,提高 NAMPT 对 ATP 的亲和力,稳定 His247 处的磷酸化 NAMPT,增加焦磷酸盐副产物的消耗,并通过 NAD+钝化反馈抑制。
TP1253 Argireline

六胜肽,Acetyl hexapeptide-3,阿基瑞林

Others Others
Argireline (Acetyl hexapeptide-3) 是可渗透皮肤的、无毒的抗皱肽。它对神经肌肉接头处依赖 Ca2+的神经递质释放具有显著的抑制作用。它具有抗皱和抗衰老的活性。
T2004 Ciproxifan maleate

FUB 359 maleate,FUB 359

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ciproxifan maleate (FUB 359) 是一种选择性的,可口服和竞争性的组胺H3受体拮抗剂,IC50值为 9.2 nM。它对其他受体亚型的表观亲和力低,可用于研究衰老性疾病和阿尔兹海默症。
T7823 IDRA-21

7-氯-3-甲基-3,4-二氢-2H-1,2,4-苯并噻二嗪 1,1-二氧化物

GluR Neuroscience
IDRA-21 是一种阳性 AMPA 受体调节剂。
T6164 Ciproxifan

FUB-359,环丙基[4-[3-(1H-咪唑-4-基)丙氧基]苯基]甲酮马来酸盐

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ciproxifan (FUB-359) 是一种高效且特异性的组胺 H3 受体拮抗剂,IC50值为 9.2 nM,可用于研究衰老性疾病和阿尔兹海默症。
T9036 N-Isopropyl-N-Phenyl-1,4-Phenylenediamin

Others Others
N-Isopropyl-N-Phenyl-1,4-Phenylenediamin 是橡胶防老剂
T60503 MFI8

Mitochondrial Metabolism Metabolism
MFI8 是一种调控线粒体裂变的化合物,可用于研究衰老。
T1993 J-147

J147

Epigenetic Reader Domain; Dopamine Receptor; Monoamine Oxidase Chromatin/Epigenetic; GPCR/G Protein; Neuroscience
J-147 是一种高效的、具有口服活性的、可透过血脑屏障神经保护剂,可增强认知能力。它抑制单胺氧化酶 B 和多巴胺转运体,EC50分别为 1.88 μM 和 0.649 μM。它有研究阿尔茨海默氏症的潜力。
TP2491 Palmitoyl Dipeptide-5 Acetate

Palmitoyl Dipeptide-5 Acetate(794590-34-4 Free base)

Others Others
Palmitoyl Dipeptide-5 Acetate 是一种多肽,是一种化妆品原料,可改善皮肤质量,防止皮肤衰老。
T23286 S 24795

Catestatin acetate(142211-96-9 free base),LNAChR

AChR Neuroscience
S 24795 (Catestatin acetate(142211-96-9 free base)) 是一种 α7 nAChR 部分激动剂。 S 24795 改善了老年小鼠的记忆功能,可用于与衰老相关的记忆障碍的研究。
T23667 AGN-201904

AGN201904,AGN 201904

ATPase Membrane transporter/Ion channel
AGN-201904 是质子泵抑制剂,是一种奥美拉唑前药,可延缓衰老,可用于预防和治疗消化性溃疡。
TP1291 Epithalon TFA (307297-39-8 free base)

Epithalon TFA

Others Others
Epithalon TFA (307297-39-8 free base) (Epithalon TFA) 是一种抗衰老剂和端粒酶激活剂。
TP2489 Tetrapeptide-21 Acetate

Tetrapeptide-21 Acetate(960608-17-7 Free base)

Others Others
Tetrapeptide-21 Acetate 是一种新型生物活性纯四肽,具有基于皮肤自身结构的抗衰老特性,可用于护肤配方。
TP2373L Biotinoyl tripeptide-1 Acetate

Biotinoyl tripeptide-1 Acetate(299157-54-3 Free base)

Others Others
Biotinoyl tripeptide-1 Acetate 可通过促进头皮微循环产生毛囊,减少毛囊萎缩和衰老。
T77613 SNX7

WAY-323879

CDK Cell Cycle/Checkpoint
SNX7 (WAY-323879) 是细胞周期蛋白依赖性激酶抑制剂 (CDKI) 途径的抑制剂。 SNX7 可用作研究衰老过程和与 CDKI 相关的其他疾病的工具。
T8532 IM156

OXPHOS Apoptosis
IM156 (HL156A; HL271 acetate) 是衍生自二甲双胍的化合物,是一种强效的,具有口服活性的AMPK 激活剂。IM156 在动物模型中可缓解与年龄相关的认知下降。IM156 是一种有效的氧化磷酸化 (OXPHOS) 抑制剂,可用于实体肿瘤的研究。
T23046 N-tert-butyl-α-Phenylnitrone

(Z)-N-benzylidene-2-Methylpropan-2-aMine oxide,N-叔丁基-α-苯基硝酮

ROS; COX Immunology/Inflammation; Neuroscience
N-tert-butyl-α-Phenylnitrone ((Z)-N-benzylidene-2-Methylpropan-2-aMine oxide) 是基于硝酮的自由基清除剂,可形成一氧化氮自旋加合物。它可以穿透血脑屏障,抑制 COX2的催化活性,有 ROS 清除、抗炎、神经保护、抗衰老和抗糖尿病的作用。
T26684 Auten-99 HBr

Auten-99,Auten-99 hydrochloride. Auten-99 HBr,Auten99,Auten 99

Phosphatase Metabolism
Auten-99 HBr (Auten-99) 是新型肌管蛋白磷酸酶 Jumpy( MTMR14) 的抑制剂,可通过血脑屏障,具有强大的神经保护作用。
T77577 SLU-PP-332

Estrogen/progestogen Receptor Endocrinology/Hormones
SLU-PP-332 是一种泛雌激素受体相关受体 (ERR) 激动剂,其对 ERRα, ERRβ 以及 ERRγ 具有很高的亲和力,EC50 值分别为 98、230 以及 430 nM。SLUPP-332 可增强骨骼肌细胞系的线粒体功能和细胞呼吸,增加 IIa 型氧化骨骼肌纤维并增强了运动耐力。SLU-PP-332 具有研究代谢性疾病以及肌肉功能改善的潜力,可能用于改善代谢紊乱和衰老。
T24094 Glycerophosphoinositol lysine

Distinctive gpi lysine,Gpi lysine

Glycerophosphoinositol lysine has an anti-dandruff, anti-inflammatory, anti-aging activity. It significantly suppresses UVB - induced PGE secretion in NHEK keratinocytes.
T11570 HL271

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
HL271, a derivative of metformin, is a potent AMPK activator that increases AMPK phosphorylation. HL271 attenuates aging-associated cognitive impairment.
TP2373 Biotinoyl tripeptide-1

Biotin GHK,BiotinGHK,Biotin-GHK

Biotinoyl tripeptide-1 can produce hair follicles by promoting scalp micro-circulation and reduce follicle atrophy and aging.
T80948 Trifluoroacetyl tripeptide-2

Trifluoroacetyl tripeptide-2,一种生物活性肽,具抗衰老(anti-aging)功能,被报道为化妆品配料。
T83199 Acetyl hexapeptide-37

Acetyl hexapeptide-37是一种生物活性肽,具抗衰老(anti-aging)功能,常作为化妆品成分使用。
T81612 Oligopeptide-68

Oligopeptide-68,生物活性肽,具备抗衰老(anti-aging)特性,报道常用作化妆品成分。
T83190 Acetyltetrapeptide 11

Acetyltetrapeptide-11,生物活性肽,具抗衰老(anti-aging)功效,报道用于化妆品成分。
T81566 Palmitoyl hexapeptide-12

Palmitoyl hexapeptide-12,一种生物活性肽,具抗衰老(anti-aging)功能,常作为化妆品原料。
T81562 Palmitoyl tripeptide-5

Palmitoyl tripeptide-5,一种生物活性肽,具备抗衰老(anti-aging)效果,常用作化妆品成分。
T83203 Acetyl dipeptide-1 cetyl ester

Calmosensine

Acetyl dipeptide-1 cetyl ester(Calmosensine)为一种具抗衰老(anti-aging)功能的生物活性肽,常作为化妆品成分。
T81978 KLKKTETQ

KLKKTETQ 是一种生物活性肽,具有抗衰老(anti-aging)功效,已报导应用于化妆品成分。
T80944 Tripeptide-10 citrulline

T10-C

Tripeptide-10 citrulline(T10-C),一种生物活性肽,具备抗衰老(anti-aging)功能,广泛应用于化妆品成分。
T80201 Tripeptide-32

Caspase Apoptosis; Proteases/Proteasome
Tripeptide-32,一种生物活性肽,具备抗衰老(anti-aging)功能,已报告作为化妆品成分使用。
T81006 Tetrapeptide-26

Tetrapeptide-26,一种生物活性肽,具抗衰老(anti-aging)功能,常用作化妆品成分。
T81230 SA1-III

KP1

SA1-III(KP1)为具抗衰老(anti-aging)功能的生物活性肽,已报道作为化妆品成分使用。
T83198 Acetyl sh-heptapeptide-1

Acetyl sh-heptapeptide-1,一种多肽,有效对抗面部老化。
T21035 Rufloxacin

MF 934

Rufloxacin is a drug that belongs to the class of fluoroquinolones, which act mainly as specific inhibitors of bacterial Topoisomerase II. These drugs involve in various diseases including cutaneous reactions, aging, etc.
T81518 Pentapeptide-31

Pentapeptide-31,一种生物活性肽,具抗衰老(anti-aging)功能,已报道应用于化妆品成分。
T83194 Acetylarginyltryptophyl diphenylglycine

Acetylarginyltryptophyl diphenylglycine 是抗衰老(anti-aging)生物活性肽,已报道作为化妆品成分使用。
T81568 Palmitoyl dipeptide-5 diaminobutyroyl hydroxythreonine

Palmitoyl dipeptide-7, 一种化妆品成分,以其生物活性肽特性作用于抗衰老。
T82206 Hexapeptide-12

Hexapeptide-12为一生物活性肽,具抗衰老功能,现报道应用于化妆品成分中。
T83202 Acetyl dipeptide-3 aminohexanoate

Acetyl dipeptide-3 aminohexanoate为生物活性肽,具抗衰老(anti-aging)功能,广泛应用于化妆品成分。
T81567 Palmitoyl dipeptide-5 diaminohydroxybutyrate

Palmitoyl dipeptide-5 diaminohydroxybutyrate,一种生物活性肽,具有抗衰老 (anti-aging) 功能,常作为化妆品成分使用。
T80027 Palmitoyl tripeptide-38

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Palmitoyl tripeptide-38是生物活性肽,具有抗老化效果。
TP2354 Tetrapeptide-11

Pro-pro-tyr-leu

Tetrapeptide-11 is the reaction product of Acetic Acid and tetrapeptide-11, containing leucine, proline, and tyrosine residues. It boosts cell growth, Syndecan-1, and Collagen XVII synthesis. Tetrapeptide-11 has a face and body anti-wrinkle and anti-aging
T61684 S 17092

S 17092 (S 17092-1) is a highly effective inhibitor of cerebral prolyl-endopeptidase (PEP), displaying an IC50 value of 1.2 nM. It is utilized in research focused on understanding memory impairment and cognitive disorders associated with cerebral aging [1].
T35892 Q134R

Q134R

Q134R, a neuroprotective hydroxyquinoline derivative that suppresses nuclear factor of activated T cell (NFAT) signaling. Q134R can across blood-brain barrier. Q134R has the potential for Alzheimer’s disease (AD) and aging-related disorders research[1]. Q134R (1-10 μM) suppresses NFAT signaling, without inhibiting calcineurin activity. Q134R partially inhibits NFAT activity in primary rat astrocytes, but does not prevent calcineurin-mediated dephosphorylation of a non-NFAT target, either in vivo...
T81564 Palmitoyl tetrapeptide-10

Palmitoyl tetrapeptide-10,一种生物活性肽,具有抗衰老功能,已报道用于化妆品成分。
T38116 Fmoc-Ala-Glu-Asn-Lys-NH2

Fmoc-Ala-Glu-Asn-Lys-NH2

Fmoc-Ala-Glu-Asn-Lys-NH2 is a peptide inhibitor that selectively targets asparagine endopeptidase (AEP) and inhibits the cleavage of amyloid precursor protein (APP). AEP, a pH-controlled cysteine proteinase, plays a crucial role in the proteolytic processing of APP, and its activity is enhanced during the aging process [1].
T10029 1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine

Endogenous Metabolite Metabolism
1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine 是内源性代谢产物的一种。
T80521 Caveolin-1 (82-101) amide (human, mouse, rat)

Caveolin-1 scaffolding domain peptide

c-Met/HGFR Tyrosine Kinase/Adaptors
Caveolin-1 (82-101) amide (human, mouse, rat) (Caveolin-1 scaffolding domain peptide) 是抑制酪氨酸激酶的肽,可逆转多器官衰老相关的有害变化。

化合物

SBI-797812
Cat.No: T12854
Synonym:
Target: NAMPT
Argireline
Cat.No: TP1253
Synonym: 六胜肽,Acetyl hexapeptide-3,阿基瑞林
Target: Others
Ciproxifan maleate
Cat.No: T2004
Synonym: FUB 359 maleate,FUB 359
Target: Histamine Receptor
IDRA-21
Cat.No: T7823
Synonym: 7-氯-3-甲基-3,4-二氢-2H-1,2,4-苯并噻二嗪 1,1-二氧化物
Target: GluR
Ciproxifan
Cat.No: T6164
Synonym: FUB-359,环丙基[4-[3-(1H-咪唑-4-基)丙氧基]苯基]甲酮马来酸盐
Target: Histamine Receptor
N-Isopropyl-N-Phenyl-1,4-Phenylenediamin
Cat.No: T9036
Synonym:
Target: Others
MFI8
Cat.No: T60503
Synonym:
Target: Mitochondrial Metabolism
J-147
Cat.No: T1993
Synonym: J147
Target: Epigenetic Reader Domain, Dopamine Receptor, Monoamine Oxidase
Palmitoyl Dipeptide-5 Acetate
Cat.No: TP2491
Synonym: Palmitoyl Dipeptide-5 Acetate(794590-34-4 Free base)
Target: Others
S 24795
Cat.No: T23286
Synonym: Catestatin acetate(142211-96-9 free base),LNAChR
Target: AChR
AGN-201904
Cat.No: T23667
Synonym: AGN201904,AGN 201904
Target: ATPase
Epithalon TFA (307297-39-8 free base)
Cat.No: TP1291
Synonym: Epithalon TFA
Target: Others
Tetrapeptide-21 Acetate
Cat.No: TP2489
Synonym: Tetrapeptide-21 Acetate(960608-17-7 Free base)
Target: Others
Biotinoyl tripeptide-1 Acetate
Cat.No: TP2373L
Synonym: Biotinoyl tripeptide-1 Acetate(299157-54-3 Free base)
Target: Others
SNX7
Cat.No: T77613
Synonym: WAY-323879
Target: CDK
IM156
Cat.No: T8532
Synonym:
Target: OXPHOS
N-tert-butyl-α-Phenylnitrone
Cat.No: T23046
Synonym: (Z)-N-benzylidene-2-Methylpropan-2-aMine oxide,N-叔丁基-α-苯基硝酮
Target: ROS, COX
Auten-99 HBr
Cat.No: T26684
Synonym: Auten-99,Auten-99 hydrochloride. Auten-99 HBr,Auten99,Auten 99
Target: Phosphatase
SLU-PP-332
Cat.No: T77577
Synonym:
Target: Estrogen/progestogen Receptor
Glycerophosphoinositol lysine
Cat.No: T24094
Synonym: Distinctive gpi lysine,Gpi lysine
Target:
HL271
Cat.No: T11570
Synonym:
Target: AMPK
Biotinoyl tripeptide-1
Cat.No: TP2373
Synonym: Biotin GHK,BiotinGHK,Biotin-GHK
Target:
Trifluoroacetyl tripeptide-2
Cat.No: T80948
Synonym:
Target:
Acetyl hexapeptide-37
Cat.No: T83199
Synonym:
Target:
Oligopeptide-68
Cat.No: T81612
Synonym:
Target:
Acetyltetrapeptide 11
Cat.No: T83190
Synonym:
Target:
Palmitoyl hexapeptide-12
Cat.No: T81566
Synonym:
Target:
Palmitoyl tripeptide-5
Cat.No: T81562
Synonym:
Target:
Acetyl dipeptide-1 cetyl ester
Cat.No: T83203
Synonym: Calmosensine
Target:
KLKKTETQ
Cat.No: T81978
Synonym:
Target:
Tripeptide-10 citrulline
Cat.No: T80944
Synonym: T10-C
Target:
Tripeptide-32
Cat.No: T80201
Synonym:
Target: Caspase
Tetrapeptide-26
Cat.No: T81006
Synonym:
Target:
SA1-III
Cat.No: T81230
Synonym: KP1
Target:
Acetyl sh-heptapeptide-1
Cat.No: T83198
Synonym:
Target:
Rufloxacin
Cat.No: T21035
Synonym: MF 934
Target:
Pentapeptide-31
Cat.No: T81518
Synonym:
Target:
Acetylarginyltryptophyl diphenylglycine
Cat.No: T83194
Synonym:
Target:
Palmitoyl dipeptide-5 diaminobutyroyl hydroxythreonine
Cat.No: T81568
Synonym:
Target:
Hexapeptide-12
Cat.No: T82206
Synonym:
Target:
Acetyl dipeptide-3 aminohexanoate
Cat.No: T83202
Synonym:
Target:
Palmitoyl dipeptide-5 diaminohydroxybutyrate
Cat.No: T81567
Synonym:
Target:
Palmitoyl tripeptide-38
Cat.No: T80027
Synonym:
Target: Reactive Oxygen Species
Tetrapeptide-11
Cat.No: TP2354
Synonym: Pro-pro-tyr-leu
Target:
S 17092
Cat.No: T61684
Synonym:
Target:
Q134R
Cat.No: T35892
Synonym: Q134R
Target:
Palmitoyl tetrapeptide-10
Cat.No: T81564
Synonym:
Target:
Fmoc-Ala-Glu-Asn-Lys-NH2
Cat.No: T38116
Synonym: Fmoc-Ala-Glu-Asn-Lys-NH2
Target:
1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine
Cat.No: T10029
Synonym:
Target: Endogenous Metabolite
Caveolin-1 (82-101) amide (human, mouse, rat)
Cat.No: T80521
Synonym: Caveolin-1 scaffolding domain peptide
Target: c-Met/HGFR
Cat. No. Product Name Target Signaling Pathways
T3S1265 Liriopesides B

山麦冬皂苷B,Nolinospiroside F

Others Others
Liriopesides B (Nolinospiroside F) 是一种甾体皂苷,分离自 Ophiopogon japonicas 中,具有抗氧化和抗衰老活性。
T3416 Aucubin

Aucuboside,桃叶珊瑚苷,Rhinanthin

IL Receptor; NF-κB; Antibacterial Immunology/Inflammation; Microbiology/Virology; NF-κB
Aucubin (Rhinanthin) 是一种可从许多传统的草药中提取的环烯醚萜苷,有许多生物学活性。
TN2019 Orobol

3'-Hydroxygenistein,3’,4’,5,7-tetrahydroxy-isoflavon,3',4',5,7-四羟基异黄酮

BCL; Caspase; PI3K Apoptosis; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) 是酪氨酸特异性蛋白激酶和磷脂酰肌醇转换的抑制剂。Orobol 抑制 PI3K,对 PI3K α/β/γ/K/δ 的 IC50 为 3.46-5.27 μM。 Orobol 具有抗皮肤老化和抗肥胖的作用。
T3768 Epifriedelanol

表木栓醇,Epifriedelinol

Others Others
Epifriedelanol (Epifriedelinol) 是一种分离自 Ulmus davidiana 根皮中的三萜类化合物,具有抗肿瘤作用,可以减缓人原始细胞的衰老。
T3018 Protocatechualdehyde

Protocatechuic aldehyde,3,4-Dihydroxybenzaldehyde,Rancinamycin IV,Catechaldehyde,原儿茶醛

Reactive Oxygen Species; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Protocatechualdehyde (3,4-Dihydroxybenzaldehyde), a natural polyphenol compound derived from radix Salviae Miltiorrhizae roots, exhibits diverse biological activities and finds extensive medicinal applications as an antioxidant, anti-aging, antibacterial, and anti-inflammatory agent.
T22218 2'-Deoxyguanosine

Deoxyguanosine,Guanine deoxyriboside

Endogenous Metabolite Metabolism
2'-Deoxyguanosine (Guanine deoxyriboside) 是一种嘌呤核苷,可被2'-dG-II家族的成员识别。2'-Deoxyguanosine 与衰老、突变和致癌有关,可被分子氧氧化。
T2813 Madecassoside

Asiaticoside A,羟基积雪草苷

Apoptosis; Antioxidant; Endogenous Metabolite Apoptosis; Metabolism; oxidation-reduction
Madecassoside (Asiaticoside A) 是从崩大碗中分离出来的一种五环三萜,有抗炎症,抗氧化和抗衰老的作用。
TN1296 5-Feruloylquinic acid

5-O-Feruloylquinic acid,5-FQA,5-O-阿魏酰奎尼酸

Tyrosinase; Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome
5-Feruloylquinic acid (5-FQA) 表现出抗氧化作用和酪氨酸酶抑制作用。
T4732 L-Carnosine

Karnozin,L-肌肽,beta-Alanyl-L-histidine

Antioxidant; Endogenous Metabolite Metabolism; oxidation-reduction
L-Carnosine (Karnozin) 是 由beta-丙氨酸和组氨酸组成的二肽,具有抑制衰老的作用。
TMS0418 Dihydroergotoxine mesylate

甲磺酸二氢麦角碱,Ergoloid mesylates,甲磺酸双氢麦角毒碱

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Dihydroergotoxine mesylate (Ergoloid mesylates) 是系列生物碱盐混合物,对GABAA 受体高结合活性。它主要用于改善与衰老相关的精神退化的症状和身体症状。
TJO2691 (-)-Fucose

L-岩藻糖,Madecassic acid,L-(-)-Fucose,L-Galactomethylose,Brahmic acid,6-Desoxygalactose

Endogenous Metabolite; Parasite Metabolism; Microbiology/Virology
(-)-Fucose (6-Desoxygalactose) 是己糖中的一种,有抗感染、抗癌、增强免疫力、皮肤保湿和延缓皮肤衰老作用。
T2S0842 Scutellarin methyl ester

Scutellarin methylester,野黄芩苷甲酯

Others Others
Scutellarin methyl ester (3-Oxotirucallenoic Acid) 是一种灯盏花素的成分, 其中灯盏花素是灯盏花中几种黄酮类化合物的粗提物。
T3812 (20R)-Ginsenoside Rg3

人参皂甙 RG3,(20R)-人参皂苷Rg3,20(R)-Ginsenoside Rg3,(20R)Ginsenoside Rg3,20(R)-Propanaxadiol

Others Others
(20R)-Ginsenoside Rg3 (20(R)-Propanaxadiol) 是一种人参根中的化合物,具有抑制血管内皮细胞增生(IC50= 10 nM)和抗肿瘤作用。
T3911 Pulchinenoside A

白头翁皂苷A,Anemoside A3

Others Others
Pulchinenoside A (Anemoside A3) 是一种天然的白头翁皂苷 A,也是 NMDA 受体的非竞争性的调节器,能够提高成年老鼠的海马体突触可塑性和醋精成年老鼠的空间记忆。
TMS2182 trans-Zeatinriboside

Ribosylzeatin,Zeatin Riboside,Trans-Zeatin Riboside,玉米素核苷

Others Others
trans-Zeatinriboside (Ribosylzeatin) 是一种细胞分裂素前体,是木质素导管中主要的长距离信号形式,能够调节叶片大小和分生组织活性相关形状。
T0591 D-Galactose

D-(+)-Galactose,alpha-D-半乳糖,D-半乳糖,D-Galactopyranose,Alpha-D-galactose

Endogenous Metabolite Metabolism
D-Galactose (Alpha-D-galactose) 是一种天然的己糖,是葡萄糖的C-4差向异构体。
TN1088 3,​5,​6,​7,​8,​3',​4'-​Heptemthoxyflavone

3,3',4',5,6,7,8-heptamethoxyflavone,3,5,6,7,8,3',4'-七甲氧基黄酮

Others Others
3,5,6,7,8,3',4'-Heptemthoxyflavone 是来自蜜柑皮中的黄酮,具有抗肿瘤起始活性和抗神经炎症作用。它能通过 cAMP/ERK/CREB 信号诱导脑源性神经营养因子表达,降低 C6 细胞磷酸二酯酶活性。它能抑制胶原酶的活性,增加人真皮成纤维细胞新生细胞中 I 型前胶原含量。
TMS1461 Qingyangshengenin B

青阳参甙元B,青阳参苷元B,Otophylloside B

Beta Amyloid Neuroscience
Qingyangshengenin B (Otophylloside B) 是一种分离自 Qingyangshen 的 C-21 甾体苷。它能够在 mRNA 水平上抑制 Aβ 的表达来减少 Aβ 的沉积,对 Aβ 的毒性有保护作用。它具有抗癫痫作用。
T4971 5'-DEOXYADENOSINE

5′-dAdo,5-脱氧腺嘌呤核苷

Endogenous Metabolite Metabolism
5'-Deoxyadenosine (5′-dAdo) 是正常受试者尿液中发现的氧化核苷,氧化核苷代表了用于确定遗传物质损伤程度的生物标志物。
T2O2733 L-Cystine

Cystine Acid,cystine,胱氨酸,L-胱氨酸

Antioxidant; Ferroptosis; Endogenous Metabolite Apoptosis; Metabolism; oxidation-reduction
L-Cystine (Cystine Acid) 是一种从半胱氨酸氨基酸硫醇侧链氧化获得的含硫衍生物。它起到抗氧化剂的作用,保护组织免受辐射和污染,减缓衰老过程。它还有助于蛋白质合成。
TN1594 DL-Syringaresinol

(±)-Syringaresinol

Antioxidant; Antifungal Microbiology/Virology; oxidation-reduction
DL-Syringaresinol ( (±)-Syringaresinol) 是一种来自与人参浆果的木质素,具有抗炎、抗氧化、镇痛活性和较弱的抗分枝杆菌活性。DL-Syringaresinol 可通过自噬延缓氧化应激诱导的皮肤老化,通过抑制炎症反应来缓解奥沙利铂诱导的神经性疼痛和脓毒症引起的心功能障碍。
T2864 Lycopene

番茄红素,ψ,ψ-Carotene

Reactive Oxygen Species; ROS Immunology/Inflammation; Metabolism; NF-κB
Lycopene (ψ,ψ-Carotene) 是一种番茄及其产品和其他红色水果和蔬菜中天然存在的类胡萝卜素,具有抗氧化活性。
TN3968 Epifriedelanol acetate

Others Others
Epifriedelanol exhibits antibacterial activities. It also can reduce cellular senescence in human primary cells and may be used to develop dietary supplements or cosmetics that modulate tissue aging or aging-associated diseases. Epifriedelanol and friedel
T78539 (+)-Coclaurine hydrochloride

d-Coclaurine hydrochloride,(R)-Coclaurine hydrochloride,(+)-(R)-Coclaurine hydrochloride

Others Others
(+)-Coclaurine ((+)-(R)-Coclaurine) hydrochloride 是从多种植物中分离得到的四氢异喹啉类生物碱,具有抗衰老活性。
TN1543 Cynaropicrin

IL Receptor; Others; TNF Apoptosis; Immunology/Inflammation; Others
Cynaropicrin is a potent activator of the AhR-Nrf2-Nqo1 pathway, and could therefore be applied to prevention of UVB-induced photo aging; it may be a potential anticancer agent against some leukocyte cancer cells such as lymphoma or leukemia, through pro-

天然产物

Liriopesides B
Cat.No: T3S1265
Synonym: 山麦冬皂苷B,Nolinospiroside F
Target: Others
Aucubin
Cat.No: T3416
Synonym: Aucuboside,桃叶珊瑚苷,Rhinanthin
Target: IL Receptor, NF-κB, Antibacterial
Orobol
Cat.No: TN2019
Synonym: 3'-Hydroxygenistein,3’,4’,5,7-tetrahydroxy-isoflavon,3',4',5,7-四羟基异黄酮
Target: BCL, Caspase, PI3K
Epifriedelanol
Cat.No: T3768
Synonym: 表木栓醇,Epifriedelinol
Target: Others
Protocatechualdehyde
Cat.No: T3018
Synonym: Protocatechuic aldehyde,3,4-Dihydroxybenzaldehyde,Rancinamycin IV,Catechaldehyde,原儿茶醛
Target: Reactive Oxygen Species, Antibacterial
2'-Deoxyguanosine
Cat.No: T22218
Synonym: Deoxyguanosine,Guanine deoxyriboside
Target: Endogenous Metabolite
Madecassoside
Cat.No: T2813
Synonym: Asiaticoside A,羟基积雪草苷
Target: Apoptosis, Antioxidant, Endogenous Metabolite
5-Feruloylquinic acid
Cat.No: TN1296
Synonym: 5-O-Feruloylquinic acid,5-FQA,5-O-阿魏酰奎尼酸
Target: Tyrosinase, Sirtuin
L-Carnosine
Cat.No: T4732
Synonym: Karnozin,L-肌肽,beta-Alanyl-L-histidine
Target: Antioxidant, Endogenous Metabolite
Dihydroergotoxine mesylate
Cat.No: TMS0418
Synonym: 甲磺酸二氢麦角碱,Ergoloid mesylates,甲磺酸双氢麦角毒碱
Target: GABA Receptor
(-)-Fucose
Cat.No: TJO2691
Synonym: L-岩藻糖,Madecassic acid,L-(-)-Fucose,L-Galactomethylose,Brahmic acid,6-Desoxygalactose
Target: Endogenous Metabolite, Parasite
Scutellarin methyl ester
Cat.No: T2S0842
Synonym: Scutellarin methylester,野黄芩苷甲酯
Target: Others
(20R)-Ginsenoside Rg3
Cat.No: T3812
Synonym: 人参皂甙 RG3,(20R)-人参皂苷Rg3,20(R)-Ginsenoside Rg3,(20R)Ginsenoside Rg3,20(R)-Propanaxadiol
Target: Others
Pulchinenoside A
Cat.No: T3911
Synonym: 白头翁皂苷A,Anemoside A3
Target: Others
trans-Zeatinriboside
Cat.No: TMS2182
Synonym: Ribosylzeatin,Zeatin Riboside,Trans-Zeatin Riboside,玉米素核苷
Target: Others
D-Galactose
Cat.No: T0591
Synonym: D-(+)-Galactose,alpha-D-半乳糖,D-半乳糖,D-Galactopyranose,Alpha-D-galactose
Target: Endogenous Metabolite
3,​5,​6,​7,​8,​3',​4'-​Heptemthoxyflavone
Cat.No: TN1088
Synonym: 3,3',4',5,6,7,8-heptamethoxyflavone,3,5,6,7,8,3',4'-七甲氧基黄酮
Target: Others
Qingyangshengenin B
Cat.No: TMS1461
Synonym: 青阳参甙元B,青阳参苷元B,Otophylloside B
Target: Beta Amyloid
5'-DEOXYADENOSINE
Cat.No: T4971
Synonym: 5′-dAdo,5-脱氧腺嘌呤核苷
Target: Endogenous Metabolite
L-Cystine
Cat.No: T2O2733
Synonym: Cystine Acid,cystine,胱氨酸,L-胱氨酸
Target: Antioxidant, Ferroptosis, Endogenous Metabolite
DL-Syringaresinol
Cat.No: TN1594
Synonym: (±)-Syringaresinol
Target: Antioxidant, Antifungal
Lycopene
Cat.No: T2864
Synonym: 番茄红素,ψ,ψ-Carotene
Target: Reactive Oxygen Species, ROS
Epifriedelanol acetate
Cat.No: TN3968
Synonym:
Target: Others
(+)-Coclaurine hydrochloride
Cat.No: T78539
Synonym: d-Coclaurine hydrochloride,(R)-Coclaurine hydrochloride,(+)-(R)-Coclaurine hydrochloride
Target: Others
Cynaropicrin
Cat.No: TN1543
Synonym:
Target: IL Receptor, Others, TNF
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