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99

抑制剂 & 化合物

55

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8507 MAC-545496

Antibacterial Microbiology/Virology
MAC-545496 是一种抗毒剂,可逆转耐甲氧西林的菌株中的 β-内酰胺耐药性。它是糖肽抗性相关蛋白 R 的纳摩尔抑制剂,对全长 GraR 蛋白具有很强的结合亲和力。
T11933 MAC13772

Others Others
MAC13772 是一种 BioA 酶的有效抑制剂,IC50 为 250 nM,从而抑制生物素的生物合成。 MAC13772 具有抗菌活性。
T27971 MAC-0547630

MAC 0547630

MAC-0547630 potent and selective inhibitor of UppS.
T15947 MAC13243 HCl

Antibacterial Microbiology/Virology
MAC13243 HCl 是一种将脂蛋白从内膜运输到外膜的周质伴侣LolA的抑制剂,是一种具有特异性的抗菌剂,对革兰氏阴性菌抑制作用显著。
T71895 MAC-5576

MAC-5576 a SARS-CoV-2 Protease inhibitor (IC50 = 81 nM).
T18230 MAC glucuronide linker-1

Others Others
MAC glucuronide linker-1 is a nonclaevable ADC linker for antibody-drug-conjugations (ADCs).
T18721 MAC-VC-PABC-ST7612AA1

Others Others
MAC-VC-PABC-ST7612AA1 is a part of antibody drug conjugates (ADCs) charged with HDAC inhibitor by a linker, shows antitumor activity[1].
T18231 MAC glucuronide linker-2

Others Others
MAC glucuronide linker-2 is an ADC linker employed in the synthesis of ADCs, offering cleavability [1].
T27972 MAC173979

MAC-173979,MAC 173979

MAC173979 inhibits E. coli de novo PABA biosynthesis and growth.
T18538 MAC glucuronide phenol-linked SN-38

Others Others
MAC glucuronide phenol-linked SN-38, a pH-sensitive lactone and DNA topoisomerase I inhibitor drug linker, exhibits cytotoxicity in L540cy and Ramos cells, with IC50 values of 113 ng/mL and 67 ng/mL, respectively[1].
T18722 MAC glucuronide α-hydroxy lactone-linked SN-38

Others Others
MAC glucuronide α-hydroxy lactone-linked SN-38 (Topoisomerase I inhibitor) is a stabilized lactone MAC glucuronide α-hydroxy lactone-linked SN-38 drug linker. MAC glucuronide α-hydroxy lactone-linked SN-38 is cytotoxic across L540cy cells and Ramos cells
T9915 Eculizumab

Complement System Immunology/Inflammation
Eculizumab 是针对补体 C5 的长效人源化单克隆抗体。它对 C5 裂解为 C5a 和 C5b 具有抑制作用,并抑制了末端补体系统的部署,其中包括膜攻击复合物的形成。它可用于溶血的研究。
T3638 Leukadherin-1

Integrin; Complement System Cytoskeletal Signaling; Immunology/Inflammation
Leukadherin-1 是 CD11b/CD18 的变构激活剂,可增加 CD11b/CD18 依赖性细胞对纤维蛋白原的粘附,减少白细胞运动和跨内皮迁移,具有抗炎作用。
T69305 Milataxel

Milataxel is an orally bioavailable taxane with potential antineoplastic activity. Upon oral administration, milataxel and its major active metabolite M-10 bind to and stabilize tubulin, resulting in the inhibition of microtubule depolymerization and cell division, cell cycle arrest in the G2/M phase, and the inhibition of tumor cell proliferation. Unlike other taxane compounds, milataxel appears to be a poor substrate for the multidrug resistance (MDR) membrane-associated P-glycoprotein (P-gp) ...
T69812 AFN941

AFN941 is a staurosporine analog, acting as a Jak3-specific inhibitor.
T9889 M4 mAChR agonist-1 

4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-

AChR Neuroscience
M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) 是一种有效的 M4 mAChR 激动剂(EC50 >10 μM)。
T21294 Polmacoxib

CG-100649,帕马考昔,CG100649,CG 100649

COX; Carbonic Anhydrase Immunology/Inflammation; Metabolism; Neuroscience
Polmacoxib (CG 100649) 是一流的 NSAID 候选药物,是碳酸酐酶 (CA) 和 COX-2 的双重抑制剂。它在小鼠模型中抑制大肠腺瘤和肿瘤生长。
T2561 Macitentan

马西替坦,ACT-064992

Apoptosis; Endothelin Receptor Apoptosis; GPCR/G Protein
Macitentan (ACT-064992) 是一种内皮素受体拮抗剂,用于治疗肺动脉高压。
T2381 Abemaciclib

CDK4/6 dual inhibitor,LY2835219

CDK Cell Cycle/Checkpoint
Abemaciclib (LY2835219) 是一种 CDK4/6 的双重抑制剂 (IC50=2/10 nM),具有选择性和特异性。Abemaciclib 具有抗肿瘤活性,被用于治疗晚期或转移性乳腺癌。
T10738 Abemaciclib metabolite M20

CDK4/6-IN-4,LSN3106726

CDK Cell Cycle/Checkpoint
Abemaciclib metabolite M20 (CDK4/6-IN-4) 是 Abemaciclib 的活性代谢物。 Abemaciclib metabolite M20 是一种特异性 CDK4/6 抑制剂,可用于癌症治疗的相关研究。
T24214 Phenamacril

JS39919,苯那普利,JS399 19

Myosin; Antifungal Cytoskeletal Signaling; Microbiology/Virology
Phenamacril (JS39919) 是一种氰基丙烯酸酯类杀菌剂,对镰刀菌,特别是禾谷镰刀菌有很强的抑制作用。它是一种特异性镰刀菌肌球蛋白 I 抑制剂。
T76776 Emactuzumab

RO 5509554,RG 7155

c-Fms; TAM Receptor Tyrosine Kinase/Adaptors
Emactuzumab(RG 7155) 是一种针对集落刺激因子-1 受体的单克隆抗体,靶向肿瘤相关巨噬细胞 (TAM)。Emactuzumab 具有抗肿瘤活性,可抑制集落刺激因子 1 受体 (CSF1R) 的激活。Emactuzumab 对 CSF-1R 具有高亲和力,Ki 值为 0.2 nM。Emactuzumab 可阻断 CSF-1R 二聚化,可用于研究如弥漫型腱鞘巨细胞瘤(dt-GCT)类的癌症。
T8827 EMAC10101d

Carbonic Anhydrase Metabolism
EMAC10101d 是 hCA II 选择性抑制剂(Ki:8.1 nM)。
T11938L Macropa-NH2

Others Others
Macropa-NH2 是 macropa 双功能类似物,是一种常与抗体偶联的载体分子,常作为螯合剂使用,参与癌症研究。
T3111 Abemaciclib methanesulfonate

abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate)

CDK Cell Cycle/Checkpoint
Abemaciclib methanesulfonate (LY2835219) 是一种选择性的CDK4/6抑制剂,能够抑制 CDK4/CDK6 的活性,IC50分别为 2 nM 和 10 nM。
T77099 Nimacimab

JNJ 2463,RYI-018

Others Others
Nimacimab是一种重组人源化单克隆抗体可改善糖尿病和非酒精性脂肪性肝炎。
T5655 mAChR-IN-1 hydrochloride

AChR Neuroscience
mAChR-IN-1 hydrochloride 是一种毒蕈碱胆碱能受体抑制剂,IC50值为17nM。
T3510 Olumacostat Glasaretil

Acetyl-CoA Carboxylase Metabolism
Olumacostat glasaretil 是乙酰辅酶A 羧化酶的有效抑制剂。
T2595 Lumacaftor

鲁玛卡托,VX-809,VRT 826809

CFTR; Autophagy Autophagy; Membrane transporter/Ion channel
Lumacaftor (VRT 826809) 是一种 CFTR 调节剂,可纠正 CFTR 蛋白的折叠和运输。它增强了 FRT 细胞中 F508del-CFTR 蛋白的成熟,EC50为100 nM。
T3583 Macozinone

PBTZ169

Antibacterial; DprE1 Microbiology/Virology; Others
Macozinone (PBTZ169) 是具有杀菌作用的苯并噻嗪酮,也有抗结核作用。它也是一种 DprE1有效抑制剂,可通过与活性位点 Cys387 残基形成共价键来抑制必需的黄素蛋白 DprE1。
T10220 Abemaciclib metabolite M2

Abemaciclib Metabolites M2

CDK Cell Cycle/Checkpoint
Abemaciclib Metabolites M2 is a metabolite of abemaciclib, acts as a potent CDK4 and CDK6 inhibitor (IC50s: 1-3 nM) with anti-cancer activity.
T0867 Bufexamac

Bufexamic acid,丁苯羟酸

COX; HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Neuroscience
Bufexamac (Bufexamic acid) 是 HDAC6 和 HDAC10 的抑制剂,也是一种COX 抑制剂,用于释放 IFN-α,具有抗炎、镇痛和解热作用。
T22202 iMAC2

iMAC2 是一种有效的MAC 抑制剂,IC50为 28 nM,LD50为15000 nM。iMAC2 显示出抗凋亡作用,并且iMAC2 阻断细胞色素 c 的释放。
T32726 L-FMAC

L FMAC,LFMAC

L-FMAC is a bioactive chemical.
T23725 Amicoumacin A

Amicoumacin A has antibacterial activity. It also strongly suppresses inflammatory and ulcer activity.
T20616 Coumachlor

G-23133,Ratilan,G23133,Tomorin,G 23133

Coumachlor, a first-generation anticoagulant rodenticide, blocks the formation of prothrombin and inhibits blood coagulation causing internal haemorrhage.
T11934 Macitentan-d4

Macitentan D4,ACT-064992 D4

Endothelin Receptor GPCR/G Protein
Macitentan-d4 (ACT-064992 D4) 是一种 Macitentan 氘代物,可被当作非多肽 ETA 和 ETB  (内皮素受体)双拮抗剂。Macitentan-d4 比 Macitentan 毒性更低,半衰期更长,可用于研究由内皮素受体介导介导的疾病。
T16752 Rimacalib

SMP 114

CaMK Neuroscience
Rimacalib is an inhibitor of Ca2+/calmodulin-dependent protein kinase II (IC50s: ~1 μM for CaMKIIα and ~30 μM for CaMKIIγ).
T22960 Macbecin I

Others Others
Hsp90 inhibitor
T71969 Remacemide

Remacemide is a low-affinity NMDA antagonist with sodium channel blocking properties. It has been studied for the treatment of acute ischemic stroke, epilepsy, Huntington's disease, and Parkinson's disease.
T23231 Remacemide hydrochloride

Others Others
NMDA receptor antagonist
T33157 Macrocalin B

Macrocalin B is a diterpenoid against tumor cell proliferation and telomerase activity.
T33961 Phenamacide hydrochloride

Aklonine

Phenamacide hydrochloride is a biochemical.
T70043 Valomaciclovir

Valomaciclovir is a DNA polymerase inhibitor potentially for treatment of acute herpes zoster and EB virus infection.
T73909 Abemaciclib metabolite M18

LSN3106729

Ligands for Target Protein for PROTAC PROTAC
Abemaciclibmetabolite M18 (LSN3106729) 是一种CDK抑制剂,具有抗肿瘤活性。作为Abemaciclib的代谢物,Abemaciclibmetabolite M18 能与CRBN配体结合,用于设计PROTAC CDK4/6降解剂。
TP2283 parathyroid hormone (7-34) [Homo sapiens]/[Macaca fascicularis]

Others Others
parathyroid hormone (7-34) [Homo sapiens] [Macaca fascicularis] is a peptide with the sequence H2N-LMHNLGKHLNSMERVEWLRKKLQDVHNF-OH, MW= 3474.03. Parathyroid hormone (PTH) is secreted by the chief cells of the parathyroid glands as a polypeptide containing
T40765 DMAC-SPDB-sulfo

DMAC-SPDB-sulfo is a cleavable linker vital in ADC synthesis. DMAC-SPDB-sulfo joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T24406 L-FMAC F-18

L-(18F)-FMAC

L-FMAC F-18 has potential diagnostic activity during positron emission tomography (PET) imaging. After phosphorylation by DCK, the 18F moiety can be visualized by PET imaging.
T5476 mAChr-in-1

AChR Neuroscience
mAChR-IN-1 是一种毒蕈碱胆碱能受体拮抗剂,IC50为17 nM。
T131600 Maculine

Maculine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131600。

化合物

MAC-545496
Cat.No: T8507
Synonym:
Target: Antibacterial
MAC13772
Cat.No: T11933
Synonym:
Target: Others
MAC-0547630
Cat.No: T27971
Synonym: MAC 0547630
Target:
MAC13243 HCl
Cat.No: T15947
Synonym:
Target: Antibacterial
MAC-5576
Cat.No: T71895
Synonym:
Target:
MAC glucuronide linker-1
Cat.No: T18230
Synonym:
Target: Others
MAC-VC-PABC-ST7612AA1
Cat.No: T18721
Synonym:
Target: Others
MAC glucuronide linker-2
Cat.No: T18231
Synonym:
Target: Others
MAC173979
Cat.No: T27972
Synonym: MAC-173979,MAC 173979
Target:
MAC glucuronide phenol-linked SN-38
Cat.No: T18538
Synonym:
Target: Others
MAC glucuronide α-hydroxy lactone-linked SN-38
Cat.No: T18722
Synonym:
Target: Others
Eculizumab
Cat.No: T9915
Synonym:
Target: Complement System
Leukadherin-1
Cat.No: T3638
Synonym:
Target: Integrin, Complement System
Milataxel
Cat.No: T69305
Synonym:
Target:
AFN941
Cat.No: T69812
Synonym:
Target:
M4 mAChR agonist-1 
Cat.No: T9889
Synonym: 4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-
Target: AChR
Polmacoxib
Cat.No: T21294
Synonym: CG-100649,帕马考昔,CG100649,CG 100649
Target: COX, Carbonic Anhydrase
Macitentan
Cat.No: T2561
Synonym: 马西替坦,ACT-064992
Target: Apoptosis, Endothelin Receptor
Abemaciclib
Cat.No: T2381
Synonym: CDK4/6 dual inhibitor,LY2835219
Target: CDK
Abemaciclib metabolite M20
Cat.No: T10738
Synonym: CDK4/6-IN-4,LSN3106726
Target: CDK
Phenamacril
Cat.No: T24214
Synonym: JS39919,苯那普利,JS399 19
Target: Myosin, Antifungal
Emactuzumab
Cat.No: T76776
Synonym: RO 5509554,RG 7155
Target: c-Fms, TAM Receptor
EMAC10101d
Cat.No: T8827
Synonym:
Target: Carbonic Anhydrase
Macropa-NH2
Cat.No: T11938L
Synonym:
Target: Others
Abemaciclib methanesulfonate
Cat.No: T3111
Synonym: abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate)
Target: CDK
Nimacimab
Cat.No: T77099
Synonym: JNJ 2463,RYI-018
Target: Others
mAChR-IN-1 hydrochloride
Cat.No: T5655
Synonym:
Target: AChR
Olumacostat Glasaretil
Cat.No: T3510
Synonym:
Target: Acetyl-CoA Carboxylase
Lumacaftor
Cat.No: T2595
Synonym: 鲁玛卡托,VX-809,VRT 826809
Target: CFTR, Autophagy
Macozinone
Cat.No: T3583
Synonym: PBTZ169
Target: Antibacterial, DprE1
Abemaciclib metabolite M2
Cat.No: T10220
Synonym: Abemaciclib Metabolites M2
Target: CDK
Bufexamac
Cat.No: T0867
Synonym: Bufexamic acid,丁苯羟酸
Target: COX, HDAC
iMAC2
Cat.No: T22202
Synonym:
Target:
L-FMAC
Cat.No: T32726
Synonym: L FMAC,LFMAC
Target:
Amicoumacin A
Cat.No: T23725
Synonym:
Target:
Coumachlor
Cat.No: T20616
Synonym: G-23133,Ratilan,G23133,Tomorin,G 23133
Target:
Macitentan-d4
Cat.No: T11934
Synonym: Macitentan D4,ACT-064992 D4
Target: Endothelin Receptor
Rimacalib
Cat.No: T16752
Synonym: SMP 114
Target: CaMK
Macbecin I
Cat.No: T22960
Synonym:
Target: Others
Remacemide
Cat.No: T71969
Synonym:
Target:
Remacemide hydrochloride
Cat.No: T23231
Synonym:
Target: Others
Macrocalin B
Cat.No: T33157
Synonym:
Target:
Phenamacide hydrochloride
Cat.No: T33961
Synonym: Aklonine
Target:
Valomaciclovir
Cat.No: T70043
Synonym:
Target:
Abemaciclib metabolite M18
Cat.No: T73909
Synonym: LSN3106729
Target: Ligands for Target Protein for PROTAC
parathyroid hormone (7-34) [Homo sapiens]/[Macaca fascicularis]
Cat.No: TP2283
Synonym:
Target: Others
DMAC-SPDB-sulfo
Cat.No: T40765
Synonym:
Target:
L-FMAC F-18
Cat.No: T24406
Synonym: L-(18F)-FMAC
Target:
mAChr-in-1
Cat.No: T5476
Synonym:
Target: AChR
Maculine
Cat.No: T131600
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1966 N-(3-Methoxybenzyl)Oleamide

N-Benzyloleamide,MAC 18:1

Antioxidant oxidation-reduction
N-(3-Methoxybenzyl)Oleamide (MAC 18:1) 是一种从 Lepidium meyenii 中分离出来的玛瑙酰胺,对运动引起的疲劳具有药理作用,可能与调节能量代谢和改善抗氧化状态有关。
T20578 Maclurin

Fustic extract,Morintannic acid,NSC 83240

Free radical scavengers; Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Maclurin (NSC-83240) 是桑枝的酚类成分,具有抗转移作用。 Maclurin 可有效防止 OH 诱导的 DNA 和 MSCs 损伤,可用于预防多种疾病或 MSCs 移植的研究。
T3866 Macelignan

安五脂素,Anwuligan,(+)-Anwulignan

Others; COX Immunology/Inflammation; Neuroscience; Others
Macelignan (Anwuligan) 是一种从肉豆蔻中分离得到的木脂素,具有抗炎、抗癌、抗糖尿病和神经保护活性。
T2945 Germacrone

P450; Antiviral; Influenza Virus Immunology/Inflammation; Metabolism; Microbiology/Virology
Germacrone 提取自姜黄,具有抗炎、抗雄激素和抗病毒活性。 它还通过促进细胞凋亡来抑制胶质瘤细胞的增殖。
T5787 Macranthoside B

金银花,灰毡毛忍冬次皂苷乙

Antibacterial Microbiology/Virology
Macranthoside B 是一种从金银花中分离出来的天然产物,具有抗菌活性。
TN1831 Macranthoside A

Kalopanaxsaponin H

Antioxidant oxidation-reduction
Macranthoside A (Kalopanaxsaponin H) 是一种从地黄中提取的三萜糖苷,属于环烯醚萜类化合。Macranthoside A 具有抗炎、抗氧化、抗菌和神经保护活性,抑制促炎细胞因子的产生和抑制炎症信号通路的激活,有助于中和有害的自由基,保护细胞免受氧化损伤,可以促进神经元的存活和生长,并防止氧化应激或神经毒性化合物引起的神经元细胞死亡,具有治疗神经退行性疾病、心血管疾病和肝损伤的潜力。
T3367 Macranthoidin B

灰毡毛忍冬皂苷乙,金银花,Macranthoiside I

Others Others
Macranthoidin B (Macranthoiside I) 是一种活性天然皂苷。
TN1159 (1(10)E,2R*,4R*)-2-Methoxy-8,12-epoxygermacra-1(10),7,11-trien-6-one

[(1(10)E,2R,4R)]-2-Methoxy-8,12-epoxygemacra-1(10),7,11-trien-6-one

Others Others
(1(10)E,2R*,4R*)-2-Methoxy-8,12-epoxygermacra-1(10),7,11-trien-6-one ([(1(10)E,2R,4R)]-2-Methoxy-8,12-epoxygemacra-1(10),7,11-trien-6-one) 是一种来自姜黄的倍半萜。
T19412 Macrozamin

甲基氧化偶氮甲醇樱草糖苷,大泽明素

Others Others
Macrozamin 是苏铁的一种主要成分,表现出致癌,致畸,诱变和神经毒性作用。
T3858 macranthoidin A

灰毡毛忍冬皂苷甲,金银花

Others Others
Macranthoidin A 是一种具有口服活性的、提取于金银花中的皂苷。它对四氯化碳,对乙酰氨基酚和镉所致的肝损伤具有保护作用,对耳巴豆油的溶胀具有明显的抑制作用。
T81890 Macedonoside A

Macedonoside A是从鳞片甘草的匍匐茎中分离出来的皂苷。
T81887 Macrostemonoside I

Macrostemonoside I,一种从Allium macrostemon分离得到的呋甾烷醇皂苷。
TN4478 Macrocarpal H

Antifection Microbiology/Virology
Macrocarpal H has anti-glucosyltransferase, and anti-bacterial activities.
TN6086 Machigline

Machigline 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6086,CAS号为 87264-30-0。
TN5912 Macluraxanthone

3-Hydroxyblancoxanthone

Antioxidant; TNF Apoptosis; oxidation-reduction
Macluraxanthone (3-Hydroxyblancoxanthone) 具有许多生物活性,包括抗胆碱酯酶、抗氧化、抗癌、抗疟疾、抗炎和免疫调节作用。Macluraxanthone 通过增加表达CD86的巨噬细胞的百分比,同时减少其CD14、CD11b 和CD80的表达,来促进M1类促炎症巨噬细胞的极化。Macluraxanthone 在促炎症刺激物脂多糖的存在下明显减少了TNF-α和IL-10细胞因子的产生。
TN2997 4(15),5,10(14)-Germacratrien-1-ol

Others Others
4(15),5,10(14)-Germacratrien-1-ol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2997,CAS号为 81968-62-9。
T81889 Machilin A

Machilin A,作为一种木酚素类化合物,能从润楠树皮的甲醇提取物中分离提取。该化合物能有效抑制B-16小鼠黑色素瘤细胞的黑色素生物合成,其半抑制浓度(IC50)为39.9 μM。
TN4474 Macrocarpal B

c-Met/HGFR Tyrosine Kinase/Adaptors
The intestinal absorption of M-A, Macrocarpal B, and Cy-C was passive diffusion as the dominating process and Cy-C was partly ATP-dependent.
TN5390 Macarangioside D

Macarangioside D 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5390,CAS号为 819870-23-0。
TN6917 Macrostemonoside J

Macrostemonoside J is a natural product.
TN2608 13-Acetoxy-3beta-hydroxygermacra-1(10)E,4E,7(11)-trien-12,6alpha-olide

Others Others
13-Acetoxy-3beta-hydroxygermacra-1(10)E,4E,7(11)-trien-12,6alpha-olide is a natural product from Artemisia myriantha.
T33158 Macrocalyxin C

Macrocalyxin C is extracted from the stems and leaves of Isodon albopilosus.
TN4130 Germacrone 4,5-epoxide

gp120/CD4; IL Receptor; P450 Immunology/Inflammation; Metabolism
(4S,5S)-(+)-Germacrone-4,5-epoxide inhibits certain subtypes of cytochrome P450 (CYP).
TN4484 Macrophylline

Others Others
Macrophylline A shows weak inhibitory action on KCl-induced contraction.
TN2476 1,10:4,5-Diepoxy-7(11)-germacren-8-one

Others Others
1,10:4,5-Diepoxy-7(11)-germacren-8-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2476,CAS号为 32179-18-3。
T79977 Maceneolignan A

Maceneolignan A,一种可从肉豆蔻(肉豆蔻科)假种皮分离的天然产品,有能力抑制RBL-2H3细胞内β-己糖胺酶释放,其IC50值为48.4 μM。同样,Maceneolignan A对抗原激活的RBL-2H3细胞中TNF-α释放的抑制作用,其IC50为63.7 μM。
TN4483 Macrocarpal N

Others Others
Macrocarpal N是一种天然产物,属于桃金娘科桉属,其产品编号为 TN4483,CAS号为 221899-21-4。Macrocarpal N可用作对照参考。
TN6050 Macusine B

Macusine B is a dual inhibitor, has almost equal inhibitory activity on both acetylcholinesterase (AChE) and butyrylcholinesterase (BChE).
TN6565 Maculosidin

Maculosidine affect the PS I electron acceptors on leaf discs, it can inhibit ATP synthesis, basal, phosphorylating and uncoupled electron transport acting as Hill reaction inhibitors on spinach chloroplasts.
TN6000 Macedonic acid

Macedonic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6000,CAS号为 39022-00-9。
TN4473 Macrocarpal A

Antifection Microbiology/Virology
Macrocarpal A is the key component that stimulates the synthesis of ceramide in the stratum corneum. Macrocarpal A has cytotoxic, and antibacterial activities.
TN4475 Macrocarpal C

ROS; Antifection Immunology/Inflammation; Microbiology/Virology
Macrocarpal C, isolated from the fresh leaves of Eucalyptus globulus Labill. (Lan An) and identified as its major antifungal component by bioassay-guided purification, the antifungal action of macrocarpal C was associated with increases of membrane permea
T75499 Maceneolignan H

Maceneolignan H (Compound 8)是一种新的木脂素化合物,从肉豆蔻假种皮中分离而来。它表现为选择性CCR3拮抗剂(EC50=1.4 μM),具有研究过敏性疾病潜力。
TN4477 Macrocarpal E

Antibacterial Microbiology/Virology
Macrocarpal E 是一种来自蓝桉的间苯三酚二醛二萜衍生物,具有抗菌活性。
T11392 Germacrene D

Antibacterial Microbiology/Virology
Germacrene D has antibacterial and antifungal activities and can be used as an adjuvant agent in the application of aminoglycosides and azoles. Germacrene D is isolated from Bursera species.
TN6974 (-)-Isobicyclogermacrenal

(-)-Isobicyclogermacrenal is a natural product.
TN4482 Macrocarpal L

Others Others
Macrocarpal L 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4482,CAS号为 327601-97-8。
TN6491 1,2-Epoxy-10(14)-furanogermacren-6-one

1,2-Epoxy-10(14)-furanogermacren-6-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6491,CAS号为 383368-24-9。
T82362 Furanogermacra-1(10)Z,4Z-dien-6-one

Furanogermacra-1(10)Z,4Z-dien-6-one为呋喃倍半萜类化合物,源自Commiphora myrrha。
TN6558 Macrophylloside D

Macrophylloside D 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6558,CAS号为 179457-69-3。
TN1214 2-Methoxy-5-acetoxy-fruranogermacr-1(10)-en-6-one

2-Methoxy-5-acetoxy-furanogermacr-1(10)-en-6-one

Others Others
2-Methoxy-5-acetoxy-furanogermacr-1(10)-en-6-one is a natural product
TN5363 Macrocarpal O

Macrocarpal O is a natural product from Eucalyptus globulus.
T81896 Lysimachigenoside C

Lysimachigenoside C为从Lysimachia foenum-graecum Hance 中分离的三萜皂苷。
T37552 (+)-Macrosphelide A

(+)-Macrosphelide A is a fungal metabolite originally isolated from Microsphaeropsis. It inhibits adhesion of HL-60 human leukemia cells to human umbilical vein endothelial cells (HUVECs) in a concentration-dependent manner. It also inhibits the growth of SKOV3 ovarian cancer cells in a concentration-dependent manner. (+)-Macrosphelide A inhibits the growth of Gram-positive bacteria, including B. subtilis, M. luteus, B. thuringiensis, and S. aureus (MICs = 143, 143, 57, and 57 μg/ml, respectivel...
T21032 Germacrene D

1(10),4(14),5-Germacratriene

Germacrene D, a natural essential oil, has antioxidant activity and cytotoxicity on tumor cells.
TN4479 Macrocarpal I

Antifection Microbiology/Virology
Macrocarpal I has anti-glucosyltransferase, and anti-bacterial activities.
TN4481 Macrocarpal K

Others Others
Macrocarpal K 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4481,CAS号为 218290-59-6。
T4479 Isomaculosidine

Others Others
Isomaculosidine can significantly inhibit nitric oxide (NO) production in lipopolysaccharide (LPS)-stimulated BV2 cells.
T82335 Ganodermacetal

Ganodermacetal是从G. amboinense中分离的高度氧化羊毛甾烷三萜类化合物,对丰年虾幼虫表现出显著毒性。
TN6492 (1E)-3-methoxy-8,12-epoxygermacra-1,7,10,11-tetraen-6-one

(1E)-3-methoxy-8,12-epoxygermacra-1,7,10,11-tetraen-6-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6492,CAS号为 1393342-06-7。
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天然产物

N-(3-Methoxybenzyl)Oleamide
Cat.No: TN1966
Synonym: N-Benzyloleamide,MAC 18:1
Target: Antioxidant
Maclurin
Cat.No: T20578
Synonym: Fustic extract,Morintannic acid,NSC 83240
Target: Free radical scavengers, Reactive Oxygen Species
Macelignan
Cat.No: T3866
Synonym: 安五脂素,Anwuligan,(+)-Anwulignan
Target: Others, COX
Germacrone
Cat.No: T2945
Synonym:
Target: P450, Antiviral, Influenza Virus
Macranthoside B
Cat.No: T5787
Synonym: 金银花,灰毡毛忍冬次皂苷乙
Target: Antibacterial
Macranthoside A
Cat.No: TN1831
Synonym: Kalopanaxsaponin H
Target: Antioxidant
Macranthoidin B
Cat.No: T3367
Synonym: 灰毡毛忍冬皂苷乙,金银花,Macranthoiside I
Target: Others
(1(10)E,2R*,4R*)-2-Methoxy-8,12-epoxygermacra-1(10),7,11-trien-6-one
Cat.No: TN1159
Synonym: [(1(10)E,2R,4R)]-2-Methoxy-8,12-epoxygemacra-1(10),7,11-trien-6-one
Target: Others
Macrozamin
Cat.No: T19412
Synonym: 甲基氧化偶氮甲醇樱草糖苷,大泽明素
Target: Others
macranthoidin A
Cat.No: T3858
Synonym: 灰毡毛忍冬皂苷甲,金银花
Target: Others
Macedonoside A
Cat.No: T81890
Synonym:
Target:
Macrostemonoside I
Cat.No: T81887
Synonym:
Target:
Macrocarpal H
Cat.No: TN4478
Synonym:
Target: Antifection
Machigline
Cat.No: TN6086
Synonym:
Target:
Macluraxanthone
Cat.No: TN5912
Synonym: 3-Hydroxyblancoxanthone
Target: Antioxidant, TNF
4(15),5,10(14)-Germacratrien-1-ol
Cat.No: TN2997
Synonym:
Target: Others
Machilin A
Cat.No: T81889
Synonym:
Target:
Macrocarpal B
Cat.No: TN4474
Synonym:
Target: c-Met/HGFR
Macarangioside D
Cat.No: TN5390
Synonym:
Target:
Macrostemonoside J
Cat.No: TN6917
Synonym:
Target:
13-Acetoxy-3beta-hydroxygermacra-1(10)E,4E,7(11)-trien-12,6alpha-olide
Cat.No: TN2608
Synonym:
Target: Others
Macrocalyxin C
Cat.No: T33158
Synonym:
Target:
Germacrone 4,5-epoxide
Cat.No: TN4130
Synonym:
Target: gp120/CD4, IL Receptor, P450
Macrophylline
Cat.No: TN4484
Synonym:
Target: Others
1,10:4,5-Diepoxy-7(11)-germacren-8-one
Cat.No: TN2476
Synonym:
Target: Others
Maceneolignan A
Cat.No: T79977
Synonym:
Target:
Macrocarpal N
Cat.No: TN4483
Synonym:
Target: Others
Macusine B
Cat.No: TN6050
Synonym:
Target:
Maculosidin
Cat.No: TN6565
Synonym:
Target:
Macedonic acid
Cat.No: TN6000
Synonym:
Target:
Macrocarpal A
Cat.No: TN4473
Synonym:
Target: Antifection
Macrocarpal C
Cat.No: TN4475
Synonym:
Target: ROS, Antifection
Maceneolignan H
Cat.No: T75499
Synonym:
Target:
Macrocarpal E
Cat.No: TN4477
Synonym:
Target: Antibacterial
Germacrene D
Cat.No: T11392
Synonym:
Target: Antibacterial
(-)-Isobicyclogermacrenal
Cat.No: TN6974
Synonym:
Target:
Macrocarpal L
Cat.No: TN4482
Synonym:
Target: Others
1,2-Epoxy-10(14)-furanogermacren-6-one
Cat.No: TN6491
Synonym:
Target:
Furanogermacra-1(10)Z,4Z-dien-6-one
Cat.No: T82362
Synonym:
Target:
Macrophylloside D
Cat.No: TN6558
Synonym:
Target:
2-Methoxy-5-acetoxy-fruranogermacr-1(10)-en-6-one
Cat.No: TN1214
Synonym: 2-Methoxy-5-acetoxy-furanogermacr-1(10)-en-6-one
Target: Others
Macrocarpal O
Cat.No: TN5363
Synonym:
Target:
Lysimachigenoside C
Cat.No: T81896
Synonym:
Target:
(+)-Macrosphelide A
Cat.No: T37552
Synonym:
Target:
Germacrene D
Cat.No: T21032
Synonym: 1(10),4(14),5-Germacratriene
Target:
Macrocarpal I
Cat.No: TN4479
Synonym:
Target: Antifection
Macrocarpal K
Cat.No: TN4481
Synonym:
Target: Others
Isomaculosidine
Cat.No: T4479
Synonym:
Target: Others
Ganodermacetal
Cat.No: T82335
Synonym:
Target:
(1E)-3-methoxy-8,12-epoxygermacra-1,7,10,11-tetraen-6-one
Cat.No: TN6492
Synonym:
Target:
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