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76

抑制剂 & 化合物

14

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Cat. No. Product Name Target Signaling Pathways
T23438 TC LPA5 4

LPA Receptor GPCR/G Protein
TC LPA5 4是LPA5受体的拮抗剂。
T15785 LPA1 receptor antagonist 1

LPA1 R antagonist 1

LPA Receptor GPCR/G Protein
LPA1 receptor antagonist 1(LPA1 R antagonist 1) 是一种具有选择性和高效性的溶血磷脂酸 (LPA1) 受体拮抗剂( IC50 : 25 nM),可用于研究特发性肺纤维化。
T83879 1-Arachidoyl Lysophosphatidic Acid sodium

1-Arachidoyl LPA,LPA(20:0),1-Eicosanoyl-Lysophosphatidic Acid

1-花生四烯酰基溶血磷脂酸(1-arachidoyl LPA)是溶血磷脂酸受体1(LPA1)的激动剂,并且是一种含有花生四烯酸的甘油磷脂,花生四烯酸位于sn-1位置。它能在主要表达LPA1而非LPA2-LPA6的人类肺成纤维细胞中诱导钙离子动员(EC50 = 3.6 µM)。在无细胞试验中,1-Arachidoyl LPA(2.5 µM)还能结合到过氧化物酶体增殖物激活受体γ(PPARγ)的配体结合域。人类尿液中也发现了该化合物。
T77789 Oleoyl-L-alpha-lysophosphatidic acid sodium salt

LPA sodium salt

Oleoyl-L-alpha-lysophosphatidic acid sodium salt为必需的细胞膜生物合成代谢物,可通过与G蛋白偶联受体(GPCR)(即LPA受体)相互作用来介导信号传导,是LPA1和LPA2受体的内源性激动剂。
T31101 CRT0273750

CRT 0273750,CRT-0273750

PDE Metabolism
CRT0273750 是一种 ATX 抑制剂的先导化合物,可调节血浆中 LPA 水平,用于 ATX/LPA 依赖性癌症模型。
T36907 1-Oleoyl Lysophosphatidic Acid

Oleoyl-sn-3-Glycerophosphate,1-Oleoyl LPA,1-Oleoyl Lysophosphatidic Acid

1-Oleoyl lysophosphatidic acid is a species of lysophosphatidic acid (LPA) containing oleic acid at the sn-1 position. Phosphatidic acid is produced either directly through the action of phospholipase D (PLD) or through a two step process involving liberation of diacylglycerol (DAG) by phospholipase C (PLC) followed by phosphorylation of DAG by diglycerol kinase.[1] Hydrolysis of the fatty acid at the sn-2 position by phospholipase A2 (PLA2) yields bioactive LPA. LPA binds to one of five differe...
T22834 H2L 5765834

LPA Receptor; LPL Receptor GPCR/G Protein
H2L 5765834 是溶血磷脂酸受体 LPA1、LPA3和 LPA5拮抗剂,IC50值分别为 94、752 和 463 nM。
T11533 Z-HA155

CS-963

PDE Metabolism
Z-HA155 (CS-963) 是一种高效的 ATX 选择性抑制剂,其 IC50=5.7 nM。
T21654 1-Oleoyl lysophosphatidic acid sodium

1-Oleoyl lysophosphatidic acid sodium salt

LPA Receptor GPCR/G Protein
1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt 是 LPA1 和 LPA2 的内源性激动剂,可通过诱导 DNA 合成促进有丝分裂,参与正常和病理性情绪反应,如焦虑和抑郁。
T83772 1-Linoleoyl Lysophosphatidic Acid sodium

1-Linoleoyl-2-hydroxy-sn-glycero-3-PA,LPA(18:2),PA(18:2(9Z,12Z)/0:0),1-Octadecadienoyl-2-hydroxy-sn-glycero-3-phosphate,18:2 Lyso PA,1-Octadecadienoyl-2-hydroxy-sn-glycero-3-PA,PA(18:2/0:0),1-Linoleoyl-2-hydroxy-sn-glycero-3-phosphate,1-Linoleoyl LPA

1-Linoleoyl LPA(1-亚油酰LPA)是LPA2受体的激动剂,属于一种含有亚油酸的甘油磷脂,在sn-1位置含亚油酸。它是小鼠和人体血浆中最丰富的LPA。1-Linoleoyl LPA在表达LPA2受体的Sf9细胞中选择性地增加细胞内钙水平(EC50约为10 nM),相较于表达LPA1和LPA3受体的Sf9细胞(EC50分别约为200和80 nM)。携带NCTC克隆2472肿瘤的小鼠中,1-linoleoyl LPA的血清水平增加。与患有初发进行性多发性硬化症的患者相比,复发缓解型多发性硬化症患者的血浆1-Linoleoyl LPA水平降低,且与神经功能缺损严重程度负相关。
T15786 LPA2 antagonist 1

Hydroxylase Metabolism
LPA2 antagonist 1 is an LPA2 antagonist (IC50: 17 nM).
T11875 LPA2 antagonist 2

LPA Receptor GPCR/G Protein
LPA2 antagonist 2 is >480-fold more selective than LPA3 (IC50 of 13.85 μM).LPA2 antagonist 2 is a selective LPA2 antagonist with an IC50 of 28.3 nM and a Ki of 21.1 nM.
T63231 LPA5 antagonist 1

LPA5 antagonist 1 是选择性的、强效的 lysophosphatidic acid receptor 5(LPA5) 拮抗剂,IC50 值为32 nM。LPA5 antagonist 1 具有高脑渗透性和抗痛活性,能够用于研究炎症性和神经性疼痛。
T63172 LPA5 antagonist 2

LPA5 antagonist 2 (compound 65) 是一种高水溶性的 LPA5 拮抗剂,可明显减轻痛觉。LPA5 antagonist 2 能够用于研究炎症性和神经性疼痛。
T1606 Fasudil

HA-1077,AT877,法舒地尔

ROCK; Serine/threonin kinase; Calcium Channel; PKA; PKC; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
Fasudil (HA-1077) 是一种非特异性 RhoA/ROCK 抑制剂,也是 Ca2+通道拮抗剂和血管扩张剂。它对蛋白激酶有抑制作用,ROCK1 的 Ki 值为 0.33 μM,ROCK2 和 PKA、PKC、PKG 的 IC50值分别 0.158 μM 和 4.58 μM、12.30 μM、1.650 μM。
T3060 Fasudil hydrochloride

Fasudil (HA-1077) HCl,盐酸法舒地尔,HA-1077,Fasudil HCl,HA-1077 hydrochloride,AT-877

ROCK; Serine/threonin kinase; Calcium Channel; HIV Protease; PKA; PKC; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
Fasudil hydrochloride (HA-1077) 是一种非特异性RhoA/ROCK 抑制剂,也抑制蛋白激酶,对 ROCK1、PKA、PKC 和 MLCK 的 Ki 值分别为 0.33 μM、1.0 μM、9.3 μM 和 55 μM。
TP2056L Acetyl-Calpastatin (184-210)(human) acetate

Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )

Cysteine Protease Proteases/Proteasome
Acetyl-Calpastatin (184-210)(human) acetate 是一种有效,选择性和可逆的钙蛋白酶 (calpain) 抑制剂,对 μ-钙蛋白酶和组织蛋白酶 L 的 Ki 值分别为 0.2 nM 和 6 μM。
T4628 Seladelpar

MBX 8025

PPAR DNA Damage/DNA Repair; Metabolism
Seladelpar (MBX 8025) 是一种有效的,具有口服活性的, 特异性PPAR-δ激动剂,EC50为 2 nM。
T5670 Isobutylparaben

Others; Antibacterial Microbiology/Virology; Others
Isobutylparaben 是组成型雄烷受体激活剂,是一种广谱抗菌剂,用于个人护理产品和化妆品中。
T39516 Bocidelpar

PPAR DNA Damage/DNA Repair; Metabolism
Bocidelpar 是一种有效的过氧化物酶体增殖物激活受体 delta 调节剂,可改善杜兴肌营养不良肌肉细胞中的线粒体生物合成和功能。
T12527L Mavodelpar free acid hydrochloride

Mavodelpar free acid hydrochloride(942594-93-6 Free base),Pparδ agonist HCl,HPP593 free acid HCl,REN001 free acid HCl

PPAR DNA Damage/DNA Repair; Metabolism
Mavodelpar free acid hydrochloride (Pparδ agonist HCl) 是一种有效的 PPARδ激动剂。
T5686 Isopropylparaben

Others Others
Isopropylparaben 是一种防腐剂和防腐杀虫剂。
T4165 Delpazolid

LCB01-0371

Antibacterial; Antibiotic Microbiology/Virology
Delpazolid (LCB01-0371) 是一种恶唑烷酮类新型抗生素,能抑制MSSA 和MRSA 的生长,对它们的MIC90值都为 2 μg/mL。
T3334 Velpatasvir

GS-5816,维帕他韦

HCV Protease; SARS-CoV Microbiology/Virology; Proteases/Proteasome
Velpatasvir (GS-5816) 是一种的 HCV NS5A 抑制剂。它也是 SARS-CoV 3CLpro 的抑制剂,IC50为 2.16 μM。
T25076 Amelparib

JPI289,JPI-289,JPI 289

Amelparib (JPI-289) is an inhibitor of the poly-ADP-ribose polymerase.
T126544 3-O-Acetylpadmatin

3-O-Acetylpadmatin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126544,CAS号为 100595-93-5。
T80531 Ac-AAVALLPAVLLALLAP-DEVD-CHO

DEVD-CHO-CPP 32

Caspase Apoptosis; Proteases/Proteasome
DEVD-CHO-CPP 32(Ac-AAVALLPAVLLALLAP-DEVD-CHO)是一种高效且可逆的caspase-3抑制剂。
T75794 Acetyl-Calpastatin(184-210)(human) TFA

Acetyl-Calpastatin(184-210)(human) TFA 是一种有效,选择性和可逆的钙蛋白酶 (calpain) 抑制剂,对 μ-钙蛋白酶和组织蛋白酶 L 的Ki 值分别为 0.2 nM 和 6 μM。
TP2380 Elpamotide

Elpamotide is a vaccine consisting of a VEGFR2-169 peptide.
TP2056 Acetyl-Calpastatin(184-210)(human)

Acetyl-Calpastatin (184-210) (human)

Selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 μM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.
T80537 Ac-AAVALLPAVLLALLAP-LEHD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-LEHD-CHO 是半胱天冬酶4、5和9的抑制剂,能够对Neocarzinostatin处理的MCF-7细胞展现保护效果。
T21949 Calpain Inhibitor XII

(Rac)-Calpain Inhibitor XII是一种可逆的,选择性抑制钙蛋白酶I(calpain I; μ-calpain)的化合物,具有19 nM的Ki值。其对钙蛋白酶II(calpain II; m-calpain; Ki=120 nM)和组织蛋白酶B(cathepsin B; Ki=750 nM)显示出较低的抑制亲和力。(Rac)-Calpain Inhibitor XII用于研究钙蛋白酶在多种生理过程中的角色,如嗜中性粒细胞趋化性、神经元信号传导和心脏对损伤的响应。
T38931 Calpain Inhibitor-1

Calpain Inhibitor-1 (compound 36) is a highly potent and selective inhibitor of Calpain 1 (Cal1), which is a cysteine protease. It exhibits an IC50 value of 100 nM and a Ki value of 2.89 μM.
T26182 Seladelpar lysine

MBX-8025 lysine dihydrate,MBX-8025 Lysine,MBX 8025 Lysine MBX8025 Lysine

Seladelpar lysine, a selective PPAR-δ agonist, is used for the therapy of Homozygous Familial Hypercholesterolemia (HoFH).
T71638 Isomolpan hydrochloride

Isomolpan hydrochloride is a dopamine receptor D2 agonist.
T12876 Seladelpar sodium salt

RWJ-800025 sodium salt,MBX-8025 sodium salt

Others Others
Seladelpar sodium salt (MBX-8025) 是一种具有口服活性、有效且特异性的PPARδ激动剂,EC50值为 2 nM。它对 PPARδ 的选择性分别是对 PPARα 和 PPARγ 的 750 和 2500 多倍。
T80241 Calpastatin subdomain B

Proteasome Proteases/Proteasome; Ubiquitination
Calpastatin subdomain B为具有生物活性的肽,其作用为抑制钙蛋白酶活性。
T80551 Calpain inhibitor V

Mu-Val-HPh-FMK

Antibiotic Microbiology/Virology
Calpain inhibitor V (Mu-Val-HPh-FMK) 为具抗衣原体活性的细胞渗透性不可逆钙蛋白酶抑制剂。
T63391 Calpain Inhibitor-2

Calpain Inhibitor-2 是具有亲脂性的钙蛋白酶抑制剂,与黑色素瘤细胞系(A-375和B-16F1)和PC-3前列腺癌细胞相比,他们在体外具有中等到良好的抗增殖效果。Calpain Inhibitor-2 中的化合物3,在基质胶细胞侵袭测定中以2μM 浓度能够抑制了80%的DU-145细胞侵袭。
T33793 Olpadronic acid

Me2 APD,Me2-APD,Me2APD

Olpadronic acid is a biochemical.
T75158 Olpasiran

Olpasiran 是一种siRNA,可减少肝脏中脂蛋白 lipoprotein(a) 的合成。
T125997 17-Methylparsonsianidine

17-Methylparsonsianidine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125997。
T77140 Ralpancizumab

Ralpancizumab 是一种 PCSK9选择性抑制剂,在出血性中风中有潜在应用。
T20590 Zilpaterol hydrochloride

Zilpaterol hydrochloride is a agonist of β-adrenergic receptor (AR). It is used to increase the feeding efficiency and the size of cattle.
T72439 Calpain Inhibitor XI

Calpain Inhibitor XI,一种可逆的calpain-1共价抑制剂,适用于神经退行性疾病的研究。
T15336 Fonadelpar

NPS-005,SJP-0035

PPAR DNA Damage/DNA Repair; Metabolism
Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.
T124098 12a-Hydroxydalpanol

12a-Hydroxydalpanol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124098,CAS号为 85042-77-9。
T39577 Fostroxacitabine bralpamide

MIV-818

Fostroxacitabine bralpamide (MIV-818) is an orally active Troxacitabine-based nucleotide prodrug. Fostroxacitabine bralpamide has anticancer effects.
T77157 Dilpacimab

Dilpacimab (ABT165) 是一种有效的双可变结构域免疫球蛋白,靶向 delta 样配体 4 (DLL4) 和VEGF 通路。Dilpacimab 可用于癌症研究。
T73088 Mavodelpar

HPP593,REN001,REN001 ; HPP593

Mavodelpar (REN001) 是一种选择性的 PPARδ激动剂。Mavodelpar 抑制肾小球损伤和肾纤维化。Mavodelpar 可用于原发性线粒体肌病 (PMM) 和长链脂肪酸氧化障碍 (LC-FAOD) 的研究。

化合物

TC LPA5 4
Cat.No: T23438
Synonym:
Target: LPA Receptor
LPA1 receptor antagonist 1
Cat.No: T15785
Synonym: LPA1 R antagonist 1
Target: LPA Receptor
1-Arachidoyl Lysophosphatidic Acid sodium
Cat.No: T83879
Synonym: 1-Arachidoyl LPA,LPA(20:0),1-Eicosanoyl-Lysophosphatidic Acid
Target:
Oleoyl-L-alpha-lysophosphatidic acid sodium salt
Cat.No: T77789
Synonym: LPA sodium salt
Target:
CRT0273750
Cat.No: T31101
Synonym: CRT 0273750,CRT-0273750
Target: PDE
1-Oleoyl Lysophosphatidic Acid
Cat.No: T36907
Synonym: Oleoyl-sn-3-Glycerophosphate,1-Oleoyl LPA,1-Oleoyl Lysophosphatidic Acid
Target:
H2L 5765834
Cat.No: T22834
Synonym:
Target: LPA Receptor, LPL Receptor
Z-HA155
Cat.No: T11533
Synonym: CS-963
Target: PDE
1-Oleoyl lysophosphatidic acid sodium
Cat.No: T21654
Synonym: 1-Oleoyl lysophosphatidic acid sodium salt
Target: LPA Receptor
1-Linoleoyl Lysophosphatidic Acid sodium
Cat.No: T83772
Synonym: 1-Linoleoyl-2-hydroxy-sn-glycero-3-PA,LPA(18:2),PA(18:2(9Z,12Z)/0:0),1-Octadecadienoyl-2-hydroxy-sn-glycero-3-phosphate,18:2 Lyso PA,1-Octadecadienoyl-2-hydroxy-sn-glycero-3-PA,PA(18:2/0:0),1-Linoleoyl-2-hydroxy-sn-glycero-3-phosphate,1-Linoleoyl LPA
Target:
LPA2 antagonist 1
Cat.No: T15786
Synonym:
Target: Hydroxylase
LPA2 antagonist 2
Cat.No: T11875
Synonym:
Target: LPA Receptor
LPA5 antagonist 1
Cat.No: T63231
Synonym:
Target:
LPA5 antagonist 2
Cat.No: T63172
Synonym:
Target:
Fasudil
Cat.No: T1606
Synonym: HA-1077,AT877,法舒地尔
Target: ROCK, Serine/threonin kinase, Calcium Channel, PKA, PKC, Autophagy
Fasudil hydrochloride
Cat.No: T3060
Synonym: Fasudil (HA-1077) HCl,盐酸法舒地尔,HA-1077,Fasudil HCl,HA-1077 hydrochloride,AT-877
Target: ROCK, Serine/threonin kinase, Calcium Channel, HIV Protease, PKA, PKC, Autophagy
Acetyl-Calpastatin (184-210)(human) acetate
Cat.No: TP2056L
Synonym: Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )
Target: Cysteine Protease
Seladelpar
Cat.No: T4628
Synonym: MBX 8025
Target: PPAR
Isobutylparaben
Cat.No: T5670
Synonym:
Target: Others, Antibacterial
Bocidelpar
Cat.No: T39516
Synonym:
Target: PPAR
Mavodelpar free acid hydrochloride
Cat.No: T12527L
Synonym: Mavodelpar free acid hydrochloride(942594-93-6 Free base),Pparδ agonist HCl,HPP593 free acid HCl,REN001 free acid HCl
Target: PPAR
Isopropylparaben
Cat.No: T5686
Synonym:
Target: Others
Delpazolid
Cat.No: T4165
Synonym: LCB01-0371
Target: Antibacterial, Antibiotic
Velpatasvir
Cat.No: T3334
Synonym: GS-5816,维帕他韦
Target: HCV Protease, SARS-CoV
Amelparib
Cat.No: T25076
Synonym: JPI289,JPI-289,JPI 289
Target:
3-O-Acetylpadmatin
Cat.No: T126544
Synonym:
Target:
Ac-AAVALLPAVLLALLAP-DEVD-CHO
Cat.No: T80531
Synonym: DEVD-CHO-CPP 32
Target: Caspase
Acetyl-Calpastatin(184-210)(human) TFA
Cat.No: T75794
Synonym:
Target:
Elpamotide
Cat.No: TP2380
Synonym:
Target:
Acetyl-Calpastatin(184-210)(human)
Cat.No: TP2056
Synonym: Acetyl-Calpastatin (184-210) (human)
Target:
Ac-AAVALLPAVLLALLAP-LEHD-CHO
Cat.No: T80537
Synonym:
Target: Caspase
Calpain Inhibitor XII
Cat.No: T21949
Synonym:
Target:
Calpain Inhibitor-1
Cat.No: T38931
Synonym:
Target:
Seladelpar lysine
Cat.No: T26182
Synonym: MBX-8025 lysine dihydrate,MBX-8025 Lysine,MBX 8025 Lysine MBX8025 Lysine
Target:
Isomolpan hydrochloride
Cat.No: T71638
Synonym:
Target:
Seladelpar sodium salt
Cat.No: T12876
Synonym: RWJ-800025 sodium salt,MBX-8025 sodium salt
Target: Others
Calpastatin subdomain B
Cat.No: T80241
Synonym:
Target: Proteasome
Calpain inhibitor V
Cat.No: T80551
Synonym: Mu-Val-HPh-FMK
Target: Antibiotic
Calpain Inhibitor-2
Cat.No: T63391
Synonym:
Target:
Olpadronic acid
Cat.No: T33793
Synonym: Me2 APD,Me2-APD,Me2APD
Target:
Olpasiran
Cat.No: T75158
Synonym:
Target:
17-Methylparsonsianidine
Cat.No: T125997
Synonym:
Target:
Ralpancizumab
Cat.No: T77140
Synonym:
Target:
Zilpaterol hydrochloride
Cat.No: T20590
Synonym:
Target:
Calpain Inhibitor XI
Cat.No: T72439
Synonym:
Target:
Fonadelpar
Cat.No: T15336
Synonym: NPS-005,SJP-0035
Target: PPAR
12a-Hydroxydalpanol
Cat.No: T124098
Synonym:
Target:
Fostroxacitabine bralpamide
Cat.No: T39577
Synonym: MIV-818
Target:
Dilpacimab
Cat.No: T77157
Synonym:
Target:
Mavodelpar
Cat.No: T73088
Synonym: HPP593,REN001,REN001 ; HPP593
Target:
Cat. No. Product Name Target Signaling Pathways
T0834 Ethylparaben

Ethyl 4-hydroxybenzoate,Ethyl parahydroxybenzoate,羟苯乙酯,尼泊金乙酯

Antibacterial; Antifungal Microbiology/Virology
Ethylparaben (Ethyl parahydroxybenzoate) 是一种标准化的化学过敏原。 对羟基苯甲酸乙酯的生理作用是通过增加组胺释放和细胞介导免疫来实现的。
T3S2105 N-Benzylpalmitamide

Macamide 1,玛卡酰胺 B,N-苄基十六烷酰胺,N-Benzylhexadecanamide

Others; FAAH; Autophagy Autophagy; Metabolism; Neuroscience; Others
N-Benzylpalmitamide (Macamide 1) 是从玛卡中得到的一种生物碱,可以时间依赖性方式抑制脂肪酸酰胺水解酶,有治疗疼痛、炎症和中枢神经系统退行性疾病的研究潜力。
T5557 Propylparaben

羟苯丙酯,Propyl 4-hydroxybenzoate,尼泊金丙酯,Propyl parahydroxybenzoate

Apoptosis; Endogenous Metabolite; Antibacterial Apoptosis; Metabolism; Microbiology/Virology
Propylparaben (Propyl parahydroxybenzoate) 是一种由植物和细菌产生的抗菌防腐剂。它普遍用于化妆品,药品和食品中。它通过改变细胞周期,细胞凋亡和类固醇生成途径来破坏卵泡的生长和类固醇生成功能。它还可降低大鼠的精子数量和活动能力。
T6S1652 Benzoylpaeoniflorin

COX Immunology/Inflammation; Neuroscience
Benzoylpaeoniflorin 是一种从白芍中提取的天然化合物,可以降低细胞凋亡,对冠心病具有潜在的研究价值。
TN1067 Galloylpaeoniflorin

6'-O-Galloyl paeoniflorin,没食子酰芍药苷

NF-κB; Androgen Receptor; ROS Endocrinology/Hormones; Immunology/Inflammation; NF-κB
Galloylpaeoniflorin (6'-O-Galloyl paeoniflorin) 是 NF-κB 抑制剂,同时也是 DNA 裂解抑制剂。
T0927 Butylparaben

Butyl 4-hydroxybenzoate,Butyl parahydroxybenzoate,尼泊金丁酯,对羟基苯甲酸丁酯

Endogenous Metabolite; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
Butylparaben (Butyl 4-hydroxybenzoate) 是一种标准化的化学过敏原,可增加组胺释放和细胞介导的免疫。
TN4688 O-Methylpallidine

Others Others
O-Methylpallidine是一种天然产物,属于番荔枝科索木属,其产品编号为 TN4688,CAS号为 27510-33-4。O-Methylpallidine可用作对照参考。
T82594 Debenzoylpaeoniflorgenin

Debenzoylpaeoniflorgenin是从Paeonia lactiflora中分离得到的天然化合物,该植物是Guizhitang的一个组成成份。
TN2416 8-Debenzoylpaeoniflorin

Others Others
8-Debenzoylpaeoniflorin is a natural product from plants
T40442 Propylparaben sodium

Propyl4-hydroxybenzoatesodium,羟苯丙酯钠,Propylparahydroxybenzoatesodium

Propylparaben sodium (propyl parahydroxybenzoate) is a naturally occurring antimicrobial preservative found in plants and bacteria. Widely utilized in cosmetics, pharmaceuticals, and foods, this compound impairs antral follicle growth and steroidogenic function by modifying the cell-cycle, apoptosis, and steroidogenesis pathways. Additionally, propylparaben sodium reduces sperm count and motility in rats.
TN5857 Debenzoylgalloylpaeoniflorin

Debenzoylgalloylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5857,CAS号为 262350-51-6。
T83310 4-O-Methyldebenzoylpaeoniflorin

4-O-Methyldebenzoylpaeoniflorin为自Paeonia albiflora提取的自然化合物。
TN3607 Catalpalactone

cAMP GPCR/G Protein
Catalpalactone exhibits high antitermitic, and cytotoxic activities, it exhibits potent inhibitory effects on lipopolysaccharide-induced NO synthesis in RAW 264.7 cells , with IC50 values of 9.80 microM. Catalpalactone can inhibit dopamine biosynthesis by
TN5855 2'-O-Benzoylpaeoniflorin

2'-O-Benzoylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5855,CAS号为 1456598-64-3。

天然产物

Ethylparaben
Cat.No: T0834
Synonym: Ethyl 4-hydroxybenzoate,Ethyl parahydroxybenzoate,羟苯乙酯,尼泊金乙酯
Target: Antibacterial, Antifungal
N-Benzylpalmitamide
Cat.No: T3S2105
Synonym: Macamide 1,玛卡酰胺 B,N-苄基十六烷酰胺,N-Benzylhexadecanamide
Target: Others, FAAH, Autophagy
Propylparaben
Cat.No: T5557
Synonym: 羟苯丙酯,Propyl 4-hydroxybenzoate,尼泊金丙酯,Propyl parahydroxybenzoate
Target: Apoptosis, Endogenous Metabolite, Antibacterial
Benzoylpaeoniflorin
Cat.No: T6S1652
Synonym:
Target: COX
Galloylpaeoniflorin
Cat.No: TN1067
Synonym: 6'-O-Galloyl paeoniflorin,没食子酰芍药苷
Target: NF-κB, Androgen Receptor, ROS
Butylparaben
Cat.No: T0927
Synonym: Butyl 4-hydroxybenzoate,Butyl parahydroxybenzoate,尼泊金丁酯,对羟基苯甲酸丁酯
Target: Endogenous Metabolite, Antibacterial, Antibiotic
O-Methylpallidine
Cat.No: TN4688
Synonym:
Target: Others
Debenzoylpaeoniflorgenin
Cat.No: T82594
Synonym:
Target:
8-Debenzoylpaeoniflorin
Cat.No: TN2416
Synonym:
Target: Others
Propylparaben sodium
Cat.No: T40442
Synonym: Propyl4-hydroxybenzoatesodium,羟苯丙酯钠,Propylparahydroxybenzoatesodium
Target:
Debenzoylgalloylpaeoniflorin
Cat.No: TN5857
Synonym:
Target:
4-O-Methyldebenzoylpaeoniflorin
Cat.No: T83310
Synonym:
Target:
Catalpalactone
Cat.No: TN3607
Synonym:
Target: cAMP
2'-O-Benzoylpaeoniflorin
Cat.No: TN5855
Synonym:
Target:
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