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47

抑制剂 & 化合物

19

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T67884	β-catenin modulator IIa-661	Wnt/beta-catenin	Cytoskeletal Signaling; Stem Cells
	β-catenin modulator IIa-661是 Wnt 途径小分子抑制剂，具有抗肿瘤活性。
T13303	Virginiamycin M1 Pristinamycin IIA,Ostreogrycin A	Antibacterial	Microbiology/Virology
	Virginiamycin M1 (Pristinamycin IIA)是一种大环内酯肽类抗生素，是链菌素a 类抗生素的成员。
T126245	1,2-Didehydrotanshinone IIA
	1,2-Didehydrotanshinone IIA 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T126245。
T123833	3alpha-Hydroxytanshinone IIA
	3alpha-Hydroxytanshinone IIA 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T123833。
T123849	Momordin IIa
	Momordin IIa 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T123849。
T81115	sPLA2-IIA Inhibitor
	sPLA2-IIA Inhibitor 是 FLSYK 的环状五肽类似物，具有环2-Nal-Leu-Ser-2-Nal-Arg (c2) 结构，能够特异性结合 hGIIA（人类 IIA 磷脂酶 A2），有效抑制其酯键水解活性。该化合物作为酯酶超家族的一员，主要作用于甘油磷脂 sn-2 位置的酯键，从而阻断游离脂肪酸和花生四烯酸等物质的释放。
T2044	Varespladib LY315920,伐瑞拉地,伐瑞拉迪	Phospholipase	Metabolism
	Varespladib (LY315920) 是选择性group IIA, secretory phospholipase A2(sPLA2)抑制剂，其IC50=9 nM。它对大鼠，兔，豚鼠和人等各种物种血清的sPLA2活性具有明显的抑制作用，IC50分别为 8.1 nM，5.0 nM，3.2 nM 和 6.2 nM。
T82361	FXIIa-IN-1
	XIIa-IN-1-IN-3（Compound 22）作为一种Factor XIIa抑制剂，其Kiapp值为97.8 nM。该化合物主要应用于血栓形成的研究。
T80230	μ-Conotoxin Sx IIIA	Sodium Channel	Membrane transporter/Ion channel
	μ-Conotoxin Sx IIIA是具有生物活性的肽类分子，作为(NaV1.4 通道阻断器)。
T82360	FXIIa-IN-2
	XIIa-IN-1-IN-2（Compound 21）为一种高效的Factor XIIa抑制剂，具有Kiapp为62.2 nM。该化合物适用于血栓形成的研究领域。
T80159	µ-Conotoxin KIIIA	Sodium Channel	Membrane transporter/Ion channel
	μ-Conotoxin KIIIA，一种具有镇痛功能的μ-芋螺毒素，源自Conus kinoshitai。该化合物通过阻断哺乳动物神经元的电压门控钠通道(VGSC) (Nav1.2)，可应用于疼痛研究领域。
T80459	ω-Conotoxin CnVIIA	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	ω-Conotoxin CnVIIA为含27个氨基酸的神经肽类毒素，具有N型钙电流阻滞活性。
T80163	μ-Conotoxin PIIIA	Sodium Channel	Membrane transporter/Ion channel
	μ-Conotoxin PIIIA为钠通道(NaV 1.4)专一性阻断剂，源自紫芋芋螺(Conus purpurascens)。
T80488	µ-Conotoxin SIIIA	Sodium Channel	Membrane transporter/Ion channel
	μ-Conotoxin SIIIA为TTX抗性sodium channel拮抗剂，属于毒性肽类，源自Conus snails毒液。该化合物主要应用于神经系统疾病，尤指神经性疼痛的研究。
T80493	µ-Conotoxin BuIIIA	Sodium Channel	Membrane transporter/Ion channel
	μ-Conotoxin BuIIIA是从Cone snails毒液中提取的一种毒性肽类VGSC阻滞剂，常用于神经系统疾病的研究。
T126467	Atractysucrose IIIa
	Atractysucrose IIIa 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T126467，CAS号为 1053636-75-1。
T3983	TMP195 TFMO 2,TMP 195	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	TMP195 (TFMO 2) 是一种选择性 IIa 类组蛋白脱乙酰酶 (HDAC) 抑制剂。对 HDAC4、HDAC5、HDAC7，HDAC9的 Ki 值分别为59、60、26，5 nM。
T14947	CHDI-390576	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	CHDI-390576 is a CNS penetrant class IIa HDAC inhibitor (IC50s: 54 nM, 60 nM, 31 nM, 50 nM for class IIa HDAC4, HDAC5, HDAC7, HDAC9). It shows >500-fold selectivity over class I HDACs (1, 2, 3) and ~150-fold selectivity over HDAC8 and the class IIb HDAC6 isoform.
T1857	TMP269	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	TMP269 是一种有效的特异性 IIa 类 HDAC 抑制剂，分别抑制 HDAC 4/HDAC 5/HDAC 7/HDAC 9，IC50值分别为 157 nM，97 nM，43 nM 和 23 nM。
T77577	SLU-PP-332	Estrogen/progestogen Receptor	Endocrinology/Hormones
	SLU-PP-332 是一种泛雌激素受体相关受体 (ERR) 激动剂，其对 ERRα, ERRβ 以及 ERRγ 具有很高的亲和力，EC50 值分别为 98、230 以及 430 nM。SLUPP-332 可增强骨骼肌细胞系的线粒体功能和细胞呼吸，增加 IIa 型氧化骨骼肌纤维并增强了运动耐力。SLU-PP-332 具有研究代谢性疾病以及肌肉功能改善的潜力，可能用于改善代谢紊乱和衰老。
T22323	Enoxaparin sodium	Thrombin	Proteases/Proteasome
	Enoxaparin sodium 是一种低分子量肝素 (LMWH)，已获得美国 FDA 批准，可用于医疗管理的 ST 段心肌梗死 (STEMI) 或 STEMI 及随后的经皮冠状动脉介入治疗 (PCI) 患者。它与抗凝血酶结合并增强其作用，并抑制凝血因子 XIa、IXa、Xa 和 IIa（凝血酶），从而防止血栓形成。
T6531	Heparin sodium salt 肝素钠,Sodium heparinate,Heparin sodium	Factor Xa; Thrombin; Autophagy	Autophagy; Metabolism; Proteases/Proteasome
	Heparin sodium salt (Sodium heparinate) 是一种抗凝剂，可与抗凝血酶 III 可逆地结合，使凝血酶因子 IIa 和 Xa 的失活速度加快，显着抑制外泌体-细胞相互作用。
T30831	Cgp 43182 Cgp-43182,Cgp43182
	CGP 43182 is an effective inhibitor of group IIA secretory phospholipase A2 (Group IIA sPLA2) activity in vitro, which can be used to prevent the synergistic effect of pro-inflammatory genes stimulated by cytokines mediated by NFkappaB.
T27731	sPLA2 inhibitor 1 KH-064,KH 064,KH064,5-BPP acid
	KH064 is a sPLA2-IIA inhibitor of oral activity.
T79100	β-Catenin modulator-1
	β-Cateninmodulator-1（IIa-650）是一种癌症研究中使用的β-Catenin调节剂。
T12990	sPLA2-X Inhibitor 31	Others	Others
	sPLA2-X Inhibitor 31 is a selective inhibitor of secreted phospholipase A2 type X (sPLA2-X) (IC50s of 26 nM, 310 nM, and 2230 nM for sPLA2-X, sPLA2-IIa, and sPLA2-V, respectively).
T78709	NT160	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	NT160，一种IIa类HDAC高效抑制剂，IC50为0.046 μM，适用于中枢神经系统疾病研究。
T32011	GSK945237 GSK-945237,GSK 945237
	GSK945237 is an effective bacterial type IIA topoisomerase inhibitor with good efficacy against both Gram-positive and Gram-negative, and shows good PK and in vivo efficacy characteristics.
T79104	β-Catenin modulator-5
	β-Cateninmodulator-5 (compound IIa-84) 为一种融合恶唑与噻唑结构的化合物，兼具高效与选择性的β-Catenin调控活性。
T71459	PD 163449
	PD 163449 is a bioactive molecule of 4-pyridone group that inhibits bacterial type IIA topoisomerase (DNA gyrase and topoisomerase IV).
T83946	CHDI 00484077
	CHDI 00484077是一种强效且选择性的IIa类组蛋白去乙酰化酶(HDAC)抑制剂，其体内IC50值为10-30 nM，而在HEK293和Jurkat细胞中的IC50值分别为0.01 nM和0.04 nM。在细胞中对IIa类HDACs具有150倍的选择性，优于I/IIb类HDACs。具有口服生物可用性和中枢神经系统(CNS)穿透能力。
T80024	Cationic Bovine Serum Albumin cBSA, chemically modified cationic bovine serum albumin
	Cationic Bovine Serum Albumin（带正电荷的牛血清白蛋白）是由583个氨基酸组成的蛋白质，具有三个同源的全α结构域。该蛋白质与Tanshinone IIA联用，在缺血性脑卒中中展现出显著的神经保护作用。
T79103	β-Catenin modulator-4
	β-Cateninmodulator-4 (compound IIa-92) 为恶唑与噻唑类化合物，兼具高效性与选择性，作为β-Catenin调节剂。
T79102	β-Catenin modulator-3
	β-Cateninmodulator-3 (compound IIa-112) 是一种结合了恶唑和噻唑结构的高效选择性β-Catenin调节剂。
T39173	Varespladib sodium LY315920 sodium,伐瑞拉迪钠；伐瑞拉地钠
	Varespladib sodium (LY315920 sodium) is a highly potent and selective inhibitor of group IIA secretory phospholipase A2 (sPLA2), with an IC50 of 9 nM. It demonstrates significant inhibitory activity against sPLA2 in serum samples from multiple species, including rat, rabbit, guinea pig, and human, with IC50 values of 8.1 nM, 5.0 nM, 3.2 nM, and 6.2 nM, respectively.
T79101	β-Catenin modulator-2
	β-Cateninmodulator-2 (compound IIa-130) 是一种融合了恶唑和噻唑结构的化合物，具有高效的β-Catenin选择性调控作用。
T39310	Sofigatran 索非加群,MCC-977
	Sofigatran (MCC-977) is an orally active inhibitor of factor IIa, also known as thrombin, and functions as an anticoagulant. It is primarily utilized in cardiovascular disease research.
T37785	1-Palmitoyl-2-linoleoyl PE
	Phosphatidylethanolamines are important components of cell membranes and biochemical pathways of fatty acid synthesis. 1-Palmitoyl-2-linoleoyl PE (PLPE) is one of the many phosphatidylethanolamines that may be present in cellular membranes. It has been used in studies involving the biosynthesis of anandamide via the phospholipase A2 (PLA2) and lysoPLD pathways. PLPE can also be used as a specific substrate to assess the activity of sPLA2-IIA in the presence of other phospholipids.
TQ0319	Ripasudil K-115,瑞舒地尔盐酸二水合物,Ripasudil hydrochloride dihydrate	ROCK	Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
	Ripasudil (Ripasudil hydrochloride dihydrate) 是一种 ROCK 特异性抑制剂，能够抑制 ROCK1和 ROCK2的活性，IC50值分别为 51 和 19 nM。
T83947	HDAC4 CHDI Degrader 11
	HDAC4 CHDI Degrader 11是一种高效且选择性的HDAC4降解剂（PROTAC），其在Jurkat E6-1细胞和Jurkat细胞中的DC50值分别为4 nM和6 nM。该化合物由类IIa HDAC抑制剂三氟甲基噁二唑通过连接体与Von Hippel-Lindau (VHL) 蛋白的配体连接而成。在亨廷顿病小鼠细胞模型中，HDAC4 CHDI Degrader 11能强效地降解HDAC4（DC50= 1nM）。在神经母细胞瘤细胞系中，可与P-糖蛋白抑制剂Elacridar联用以实现更有效的降解。
T14144	AGN-195183	Others	Others
	AGN 195183 is a potent and selective agonist of RARα(Kd=3 nM) with improved binding selectivity relative to AGN 193836; no activity on RARβ/γ. IC50 value: 3 nM (Kd); 200 nM (EC80, RAR Trans.) Target: RARα agonist Compound 4(AGN-195183) inhibited the growt
T37331	Pyrrophenone
	The group IVA phospholipase A2 (PLA2), known as calcium-dependent cytosolic PLA2 (cPLA2), selectively releases arachidonic acid (AA) from membrane phospholipids, playing a central role in initiating the synthesis of prostaglandins (PGs) and leukotrienes (LTs). Pyrrophenone inhibits cPLA2α with an IC50 of 4.2 nM in enzyme assays and potently blocks the release of AA and the production of PGE2 and LTC4 in cells (IC50 = 24, 25, and 14 nM, respectively). Its action is reversible and selective, as py...
T36335	(S)-nitro-Blebbistatin
	(S)-nitro-Blebbistatin is a more stable form of (-)-blebbistatin , which is a selective cell-permeable inhibitor of non-muscle myosin II ATPases. (-)-Blebbistatin rapidly and reversibly inhibits Mg-ATPase activity and in vitro motility of non-muscle myosin IIA and IIB for several species (IC50s = 0.5-5 μM), while poorly inhibiting smooth muscle myosin (IC50 = 80 μM). Through these effects, it blocks apoptosis-related bleb formation, directed cell migration, and cytokinesis in vertebrate cells. H...
T35762	MC1742
	MC1742 is an inhibitor of class I histone deacetylases (HDACs; IC50s = 0.1, 0.11, 0.02, and 0.61 μM for HDAC1, -2, -3, and -8, respectively) and class IIb HDACs (IC50s = 7 and 40 nM for HDAC6 and HDAC10, respectively).1 It is selective for class I and class IIb over class IIa HDACs (IC50s = >50 μM for HDAC4, -5, -7, and -9). MC1742 reduces proliferation of HOS, MG-63, RD, A204, SK-ES-1, and A673 sarcoma cancer stem cells (CSCs). It increases levels of acetylated histone H3 and acetylated tubulin...
T36400	para-amino-Blebbistatin
	para-amino-Blebbistatin is a more water-soluble form of (S)-4'-nitro-blebbistatin , which is a more stable and less phototoxic form of (-)-blebbistatin .1,2,3 (-)-Blebbistatin is a selective cell-permeable inhibitor of non-muscle myosin II ATPases that rapidly and reversibly inhibits Mg-ATPase activity and in vitro motility of non-muscle myosin IIA and IIB for several species (IC50s = 0.5-5 μM), while poorly inhibiting smooth muscle myosin (IC50 = 80 μM).2,3,4 Through these effects, it blocks ap...
T36195	CAY10744
	CAY10744 is a topoisomerase II-α poison.1 It inhibits topoisomerase II-α by 78.9% when used at a concentration of 20 μM. CAY10744 is selective for topoisomerase II-α over topoisomerase I providing 100 and 0% inhibition, respectively, at 100 μM. It inhibits proliferation of HCT15 colon, T47D breast, DU145 prostate, and HeLa cervical cancer cells (IC50s = 0.014, 0.00267, 0.072, and 2.46 μM, respectively). CAY10744 induces apoptosis in T47D cells when used at concentrations of 10 and 30 μM. CAY1074...
T7492	Ripasudil free base K-115 (free base)	ROCK; Antibacterial	Cell Cycle/Checkpoint; Cytoskeletal Signaling; Microbiology/Virology; Stem Cells
	Ripasudil free base (K-115 (free base)) 是一种ROCK 特异性抑制剂，能够抑制ROCK1和ROCK2的活性，IC50值分别为 51 和 19 nM。

化合物

β-catenin modulator IIa-661

Cat.No: T67884

Target: Wnt/beta-catenin

Virginiamycin M1

Cat.No: T13303

Synonym: Pristinamycin IIA,Ostreogrycin A

Target: Antibacterial

1,2-Didehydrotanshinone IIA

Cat.No: T126245

3alpha-Hydroxytanshinone IIA

Cat.No: T123833

Cat.No: T123849

sPLA2-IIA Inhibitor

Cat.No: T81115

Cat.No: T2044

Synonym: LY315920,伐瑞拉地,伐瑞拉迪

Target: Phospholipase

Cat.No: T82361

μ-Conotoxin Sx IIIA

Cat.No: T80230

Target: Sodium Channel

Cat.No: T82360

µ-Conotoxin KIIIA

Cat.No: T80159

Target: Sodium Channel

ω-Conotoxin CnVIIA

Cat.No: T80459

Target: Calcium Channel

μ-Conotoxin PIIIA

Cat.No: T80163

Target: Sodium Channel

µ-Conotoxin SIIIA

Cat.No: T80488

Target: Sodium Channel

µ-Conotoxin BuIIIA

Cat.No: T80493

Target: Sodium Channel

Atractysucrose IIIa

Cat.No: T126467

Cat.No: T3983

Synonym: TFMO 2,TMP 195

Target: HDAC

Cat.No: T14947

Target: HDAC

Cat.No: T1857

Target: HDAC

Cat.No: T77577

Target: Estrogen/progestogen Receptor

Enoxaparin sodium

Cat.No: T22323

Target: Thrombin

Heparin sodium salt

Cat.No: T6531

Synonym: 肝素钠,Sodium heparinate,Heparin sodium

Target: Factor Xa, Thrombin, Autophagy

Cat.No: T30831

Synonym: Cgp-43182,Cgp43182

sPLA2 inhibitor 1

Cat.No: T27731

Synonym: KH-064,KH 064,KH064,5-BPP acid

β-Catenin modulator-1

Cat.No: T79100

sPLA2-X Inhibitor 31

Cat.No: T12990

Target: Others

Cat.No: T78709

Target: HDAC

Cat.No: T32011

Synonym: GSK-945237,GSK 945237

β-Catenin modulator-5

Cat.No: T79104

Cat.No: T71459

Cat.No: T83946

Cationic Bovine Serum Albumin

Cat.No: T80024

Synonym: cBSA, chemically modified cationic bovine serum albumin

β-Catenin modulator-4

Cat.No: T79103

β-Catenin modulator-3

Cat.No: T79102

Varespladib sodium

Cat.No: T39173

Synonym: LY315920 sodium,伐瑞拉迪钠；伐瑞拉地钠

β-Catenin modulator-2

Cat.No: T79101

Cat.No: T39310

Synonym: 索非加群,MCC-977

1-Palmitoyl-2-linoleoyl PE

Cat.No: T37785

Cat.No: TQ0319

Synonym: K-115,瑞舒地尔盐酸二水合物,Ripasudil hydrochloride dihydrate

Target: ROCK

HDAC4 CHDI Degrader 11

Cat.No: T83947

Cat.No: T14144

Target: Others

Cat.No: T37331

(S)-nitro-Blebbistatin

Cat.No: T36335

Cat.No: T35762

para-amino-Blebbistatin

Cat.No: T36400

Cat.No: T36195

Ripasudil free base

Cat.No: T7492

Synonym: K-115 (free base)

Target: ROCK, Antibacterial

Cat. No.	Product Name	Target	Signaling Pathways
T3S1471	Cucurbitacin IIA 葫芦素Iia,Dihydrocucurbitacin Q1,Hemslecin A,Curcurbitacin IIA	Apoptosis; Survivin	Apoptosis
	Cucurbitacin IIA (Dihydrocucurbitacin Q1) 是从园果雪胆中分离得到的一种三萜烯，可诱导细胞凋亡和增强自噬，有助于葫芦素IIA 对炎症相关疾病的抗炎活性。它可降低癌细胞中生存素的表达，降低磷酸化组蛋白 H3 的水平，增加裂解的 PARP 的水平。
T2946	Tanshinone IIA sulfonate sodium 丹参酮IIA磺酸盐,丹参酮IIA-磺酸钠,Tanshinone IIA sulfonate,Sodium Tanshinone IIA sulfonate,Tanshinone IIA sodium sulfonate,sodium	CaMK; P450; Calcium Channel	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Tanshinone IIA sulfonate sodium (Tanshinone IIA sodium sulfonate) 是从丹参中提取的丹参酮IIA 的水溶性衍生物，是SOCE 抑制剂，用于心血管疾病的研究。
T2906	Tanshinone IIA 丹参酮IIA,Tanshinone B,Dan Shen ketone	VEGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	Tanshinone IIA (Tanshinone B) 是红根丹参根系中的一种主要组合物。它能够利用靶向 VEGF/VEGFR2的蛋白激酶结构域，抑制血管生成。
TN1358	Escin IIa 七叶皂苷C,Aescin IIA	Others	Others
	Aescin IIA is a natural product
TN3657	Cinchonain IIa	Others	Others
	Cinchonain IIa has antioxidant activity, it shows high radical scavenging activity and reducing power.
TN4239	Hydroxytanshinone IIA	Others	Others
	Hydroxytanshinone ⅡA has good antiproliferative effect on SGC-7901,HeLa, and HepG 2 cell, the values of IC50 are 4.18, 6.08 and10.20 uM, respectively; it has tumor cell proliferation inhibition significantly stronger than the tanshinoneⅡA.
T10042	11-Oxomogroside IIa	Others	Others
	11-Oxomogroside IIa is a cucurbitane glycoside extracted from the fruits of Siraitia grosVenorii. It has inhibitory effects against the EBV-EA activation induced by TPA, shows weak inhibitory effects on activation of NOR 1, a nitric oxide (NO) donor.
T13740	Isotanshinone IIA	Others	Others
	Isotanshinone IIA, could non-competitively inhibit Protein Tyrosine Phosphatase 1B (PTP1B) activity with an IC50 0f 11.4 μM. is an abietane-type diterpene metabolite.
TN5995	Cucurbitacin IIa 2-O-glucoside Hemslecin A 2-O-glucoside,雪胆甲素苷
	Cucurbitacin IIa 2-O-glucoside 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5995，CAS号为 77704-34-8。
T83424	1-Oxotanshinone IIA
	1-Oxotanshinone IIA（Compound 6），一种从Perovskia artemisioides中提取的化合物，显示出显著的抗炎活性。
T75541	Tanshinone IIA anhydride
	Tanshinone IIA anhydride 是一种有效且不可逆的人羧酸酯酶 (CE) 抑制剂，对人 CE1 和人肠道 CE (hiCE) 的Ki 值分别为 1.9 nM 和 1.4 nM。
TN1934	Mogroside IIA1 Mogroside II-A1,罗汉果苷II A1	Others; NO Synthase	Immunology/Inflammation; Others
	Mogroside IIA1 (Mogroside II-A1) 是从罗汉果的果实中分离得到的。Mogroside IIA1 是一种无糖甜味剂，比蔗糖更甜。 Mogroside IIA1 具有抗氧化、抗糖尿病和抗癌活性。
TN5989	Hemslecin D 雪胆甲素-16-乙酸酯,Cucurbitacin IIa 16-acetate,23,24-Dihydrocucurbitacin F 16,25-diacetate
	Hemslecin D 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5989，CAS号为 586960-44-3。
TN6624	11-Oxomogroside IIA2
	11-Oxomogroside IIA2 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN6624，CAS号为 2170761-37-0。
TN3486	Bakkenolide IIIa	ERK; BCL; IκB/IKK; NF-κB; Akt	Apoptosis; Cytoskeletal Signaling; MAPK; NF-κB; PI3K/Akt/mTOR signaling
	Bakkenolide IIIa has antioxidant, and neuroprotective effects, it protects against cerebral damage by inhibiting AKT and ERK1/2 activation and inactivated NF-ÎºB signaling.
TN6118	Aristolactam IIIa N-β-glucoside
	Aristolactam IIIa N-β-glucoside 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN6118，CAS号为 80311-26-8。
TL0017	Aristolactam AIIIa	MAPK; CDK	Cell Cycle/Checkpoint; MAPK
	Aristolactam AIIIa is a new type of Plk1 inhibitors, targeting the Polo Box domain (PBD), it has anti-tumor activity. Aristolactam IIIa shows inhibition of platelet aggregation induced by collagen or arachidonic acid.
T75619	Aristololactam IIIa
	Aristololactam IIIa 对超氧阴离子生成和弹性蛋白酶的释放有显著抑制作用，其 IC50值分别为 0.12 和 0.20 μg/mL。
T2907	Tanshinone I 丹参酮I,Tanshinone A	Phospholipase	Metabolism
	Tanshinone I (Tanshinone A) 是IIA 型人重组sPLA2(IC50=11 μM)和兔重组cPLA2(IC50=82 μM)抑制剂。

天然产物

Cucurbitacin IIA

Cat.No: T3S1471

Synonym: 葫芦素Iia,Dihydrocucurbitacin Q1,Hemslecin A,Curcurbitacin IIA

Target: Apoptosis, Survivin

Tanshinone IIA sulfonate sodium

Cat.No: T2946

Synonym: 丹参酮IIA磺酸盐,丹参酮IIA-磺酸钠,Tanshinone IIA sulfonate,Sodium Tanshinone IIA sulfonate,Tanshinone IIA sodium sulfonate,sodium

Target: CaMK, P450, Calcium Channel

Tanshinone IIA

Cat.No: T2906

Synonym: 丹参酮IIA,Tanshinone B,Dan Shen ketone

Target: VEGFR

Cat.No: TN1358

Synonym: 七叶皂苷C,Aescin IIA

Target: Others

Cinchonain IIa

Cat.No: TN3657

Target: Others

Hydroxytanshinone IIA

Cat.No: TN4239

Target: Others

11-Oxomogroside IIa

Cat.No: T10042

Target: Others

Isotanshinone IIA

Cat.No: T13740

Target: Others

Cucurbitacin IIa 2-O-glucoside

Cat.No: TN5995

Synonym: Hemslecin A 2-O-glucoside,雪胆甲素苷

1-Oxotanshinone IIA

Cat.No: T83424

Tanshinone IIA anhydride

Cat.No: T75541

Mogroside IIA1

Cat.No: TN1934

Synonym: Mogroside II-A1,罗汉果苷II A1

Target: Others, NO Synthase

Cat.No: TN5989

Synonym: 雪胆甲素-16-乙酸酯,Cucurbitacin IIa 16-acetate,23,24-Dihydrocucurbitacin F 16,25-diacetate

11-Oxomogroside IIA2

Cat.No: TN6624

Bakkenolide IIIa

Cat.No: TN3486

Target: ERK, BCL, IκB/IKK, NF-κB, Akt

Aristolactam IIIa N-β-glucoside

Cat.No: TN6118

Aristolactam AIIIa

Cat.No: TL0017

Target: MAPK, CDK

Aristololactam IIIa

Cat.No: T75619

Cat.No: T2907

Synonym: 丹参酮I,Tanshinone A

Target: Phospholipase

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