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80

抑制剂 & 化合物

20

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
TP2036L	DPDPE TFA (88373-73-3 free base) DPDPE TFA	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	DPDPE TFA 是选择性 δ-阿片受体激动剂肽，在体内具有镇痛作用。
T6277	Doramapimod BIRB 796,达马莫德,度马莫德	Raf; p38 MAPK; Autophagy	Autophagy; MAPK
	Doramapimod (BIRB 796) 是一种具有口服活性的p38 MAPK 抑制剂，Kd 值为0.1nM。它也抑制B-Raf 和 Abl，IC50分别为 83 nM 和 14.6 μM。
T22314	Doripenem	Antibacterial; Antibiotic	Microbiology/Virology
	Doripenem 是对革兰氏阳性菌、阴性菌和厌氧菌有效的β-内酰胺广谱抗生素。
T26760	Bedoradrine sulfate KUR1246,MN 221 sulfate,KUR1246 sulfate,MN221 sulfate,KUR 1246 sulfate,MN-221 sulfate,KUR 1246,KUR-1246 sulfate,MN-221,MN 221,MN221,KUR-1246	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Bedoradrine sulfate（MN-221 sulfate）是一种超选择性β2激动剂，可用于治疗哮喘加重和慢性阻塞性肺病。
T72166	Xanthine oxidoreductase-IN-5	Xanthine Oxidase	Metabolism
	Xanthine oxidoreductase-IN-5 是一种具有口服活性的黄氨酸氧化还原酶 (XOR) 抑制剂（IC50 ： 55 nM）。Xanthine oxidoreductase-IN-5 可用于急性高尿酸血症的研究。
T38193L	β-Endorphin (1-27) (human) acetate β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	β-Endorphin (1-27) (human) acetate 存在于大脑垂体和下丘脑中，具有镇痛活性。 β-Endorphin (1-27) (human) acetate 是一种阿片受体激动剂，对 μ-阿片受体和 δ-阿片受体具有较好的亲和力。
T21511L	alpha-Endorphin acetate α-内啡肽,alpha-Endorphin acetate (59004-96-5 Free base)	Others	Others
	alpha-Endorphin acetate 是具有特征生物活性的原阿片黑皮质素家族的相关肽，从单个人类垂体中纯化至同质。
T1037	Doripenem monohydrate 多尼培南(一水合物),S 4661 monohydrate,Doripenem Hydrate,S-4661	Antibacterial; Antibiotic	Microbiology/Virology
	Doripenem monohydrate (S 4661 monohydrate) 是广谱β-内酰胺抗生素，它对革兰氏阳性，阴性和厌氧菌有抗菌作用。
T15756	Lidorestat IDD-676	Reductase	Endocrinology/Hormones; Metabolism
	Lidorestat (IDD-676) 是一种醛糖还原酶抑制剂(IC50: 5 nM)，具有有效性，选择性和口服活性。Lidorestat 改善神经传导，减少白内障的形成。Lidorestat 可用于治疗慢性糖尿病并发症。
T70047	Bedoradrine Bedoradrine free base	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Bedoradrine free base 是一种新型高选择性 β2-肾上腺素受体激动剂，可用于治疗哮喘和慢性阻塞性肺疾病。
T62839	Dalzanemdor SAGE-718	NMDAR; iGluR	Membrane transporter/Ion channel; Neuroscience
	Dalzanemdor (SAGE-718) 是 NMDA 受体阳性变构调节剂，可用于研究亨廷顿舞蹈病、阿尔茨海默病和认知功能障碍。
T30098	Aplindore Fumarate Aplindore,DAB-452 Fumarate,DAB-452	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Aplindore Fumarate （DAB-452）是一种小分子多巴胺 D2 受体部分激动剂，Aplindore Fumarate 对多巴胺D2 和D3 受体表现出高亲和力，对多巴胺D4、5-羟色胺（5-HT2）和α1-肾上腺素受体表现出低亲和力。Aplindore Fumarate 可用于研究帕金森和精神分裂症。
TP1508L	N-Acetyl-α-Endorphin acetate(88264-63-5 free base)	Others	Others
	N-Acetyl-α-Endorphin acetate(88264-63-5 free base) 是 N 末端乙酰化的 α-Endorphin。 α-内啡肽是一种内源性 opioid 肽。
TP2322L	beta-Neoendorphin acetate(77739-21-0 free base)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	beta-Neoendorphin acetate(77739-21-0 free base) 是 κ-opioid 受体的激动剂
T5500	DORA-22	OX Receptor	GPCR/G Protein; Neuroscience
	DORA-22 是一种双食欲素受体拮抗剂，可改善轻度压力引起的失眠，对记忆的影响很小。
T67888L	Samidorphan HCl Samidorphan HCl（852626-89-2 free base）	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Samidorphan HCl 是一种具有口服活性和高效性的 opioid 系统调节剂，可与 μ‐opioid、 κ‐opioid 和 δ‐opioid 受体结合。Samidorphan HCl 是一种新型 μ‐opioid 受体拮抗剂，是 k-opioid 受体和 δ‐opioid 受体的部分激动剂。Samidorphan HCl 可用于预防和治疗精神分裂。
T1977	Dorsomorphin Compound C,BML-275	AMPK; Autophagy; TGF-beta/Smad	Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Stem Cells
	Dorsomorphin (BML-275) 是一种 AMPK 抑制剂 (Ki=109 nM)，具有选择性和 ATP 竞争性。Dorsomorphin 可以抑制 BMP I 型受体 ALK2、ALK3 和 ALK6。Dorsomorphin 可诱导自噬，具有抗肿瘤活性。
T15159	Dorzagliatin HMS5552	Glucokinase	Metabolism
	Dorzagliatin (HMS5552) 是双重作用的葡萄糖激酶 (glucokinase;GK) 激活剂，可改善 2 型糖尿病的血糖控制，提高胰腺 β 细胞功能。
T2134	Dorzolamide hydrochloride MK507 hydrochloride,L671152 hydrochloride,MK-507 (L-671152) HCl,盐酸多佐胺,Dorzolamide HCl	Carbonic Anhydrase	Metabolism
	Dorzolamide hydrochloride (MK507 hydrochloride) 是一种碳酸酐酶carbonic anhydrase II 抑制剂，能够抑制红细胞CA-II(IC50:0.18 nM) 和CA-I(IC50:600 nM) 。
T69146	Suksdorfin	PPAR	DNA Damage/DNA Repair; Metabolism
	Suksdorfin 具有降血糖作用，可促进脂肪细胞分化并增强脂联素的产生，可激活过氧化物酶体增殖物激活受体 γ （PPARγ），可促进脂肪细胞对胰岛素依赖性葡萄糖的摄取，可用于肥胖相关研究。
T72165	Xanthine oxidoreductase-IN-3	Xanthine Oxidase	Metabolism
	Xanthine oxidoreductase-IN-3 是一种具有口服活性的黄氨酸氧化还原酶 (XOR) 抑制剂（IC50 ： 26.3 nM）。Xanthine oxidoreductase-IN-3 可用急性高尿酸血症的研究。
T5015	Gonadorelin Acetate (33515-09-2 free base) 醋酸戈那瑞林,Luteinizing Hormone Releasing Hormone (LH-RH),Luteinizing Hormone Releasing Hormone (LH-RH), human,Gonadorelin Acetate	Reductase	Endocrinology/Hormones; Metabolism
	Gonadorelin Acetate (33515-09-2 free base) (Luteinizing Hormone Releasing Hormone (LH-RH)) 是下丘脑神经肽，在控制生殖功能中起关键作用。
T3632	Doravirine 多拉维林,多拉韦林,MK-1439	HIV Protease; Reverse Transcriptase	Microbiology/Virology; Proteases/Proteasome
	Doravirine (MK-1439) 是一种高度特异性的HIV-1非核苷逆转录酶抑制剂，对野生型以及K103N 和Y181C 逆转录酶突变体的IC50值分别为 4.5 nM，5.5 nM 和 6.1 nM。
T7830	Windorphen	Wnt/beta-catenin	Cytoskeletal Signaling; Stem Cells
	Windorphen 是一种 Wnt 抑制剂，可选择性地消除 Wnt 信号传导。
T72078	Xanthine oxidoreductase-IN-4	Xanthine Oxidase	Metabolism
	Xanthine oxidoreductase-IN-4 是一种具有有口服活性黄嘌呤氧化还原酶 (XOR) 抑制剂，对 XOR 具有抑制作用，IC50 值为 29.3 nM。Xanthine oxidoreductase-IN-4 可用于研究高尿酸血症。
T67782	Daridorexant hydrochloride Nemorexant hydrochloride,Quviviq	OX Receptor	GPCR/G Protein; Neuroscience
	Daridorexant hydrochloride (Nemorexant hydrochloride) 是一种新型的双Orexin 受体拮抗剂。Daridorexant hydrochloride 可用于失眠研究。
T6146	Dorsomorphin dihydrochloride BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride	AMPK; Autophagy; TGF-beta/Smad	Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Stem Cells
	Dorsomorphin dihydrochloride (BML-275 2HCl) 是一种选择性和 ATP 竞争性的AMPK 抑制剂，Ki 为 109 nM。它诱导自噬，通过靶向抑制 I 型受体ALK2，ALK3和ALK6来抑制 BMP 途径。
T70072	Aplindore
	Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.
T29818	Aladorian sodium
	Aladorian sodium is used for Treatment of Cardiovascular Diseases.
T14153	Aladorian ARM036	Others	Others
	Aladorian (ARM036) is a benzothiazepine derivative and it has anti-arrhythmia effect. Aladorian is used for the research of heart failure and catecholaminergic polymorphic ventricular tachycardia[1][2].
T80515	β-Endorphin (1-27) (human)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	β-Endorphin (1-27) (human) 是一种 opioid 拮抗剂，与 μ-、δ- 及 κ-阿片受体结合，其 Kis 分别为 5.31、6.17 及 39.82 nM。该化合物还能够抑制由 β-Endorphin 及 etorphine 引起的痛觉消失。
T35460	β-Endorphin (rat)
	β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities. It is produced via piomelanocortin cleavage in the pituitary gland, hypothalamus, and in lymphocytes, then migrates to its sites of action which include plasma, gut, skin, placenta, cerebrospinal fluid, and cardiac tissues. β-EP induces concentration-dependent decreases in electrically stimulated contraction of the mouse vas deferens that can be reversed by the μ-opioid antagonist CTP and δ-opioid antagon...
T25034	Alcindoromycin
	Alcindoromycin 是从bohemic acid complex 中分离得到，具有抗肿瘤活性。
T11656	Indoramin D5 Indoramine D5,Wy-21901 D5	CDK	Cell Cycle/Checkpoint
	Indoramin D5 is a piperidine antiadrenergic agent. Indoramin D5 is deuterium labeled Indoramin.
T32584	Lathodoratin
	Lathodoratin is a bioactive chemical.
T61165	Indoramin
	Indoramin, an orally active antihypertensive agent, exhibits selectivity for the α 1A -adrenoceptor [1].
T82072	Indoramin hydrochloride Indoramine hydrochloride,Wy 21901 hydrochloride
	Indoramin (hydrochloride) is a novel antihypertensive agent that exhibits selectivity for the α1A-adrenergic receptor.
T124290	Doronenine
	Doronenine 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T124290。
T125713	Dorrigocin B

T24013	DORA 42 DORA42,DORA-42
	DORA 42 is a dual antagonist of the orexin receptor OX1R and OX2R.
T82532	Dorlimomab aritox 4197X-RA,MDX-RA (ricin A chain) immunotoxin
	Dorlimomab aritox（4197X-RA; MDX-RA (ricin A chain) immunotoxin）是一种偶联了蓖麻毒素Ricinus communis ricin A的小鼠源单克隆抗体。
T35733	Doramectin aglycone
	Doramectin aglycone is an acid degradation product of doramectin , a disaccharide-containing anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in nematodes, and its acid-catalyzed hydrolysis product doramectin monosaccharide . Doramectin undergoes one round of acid-catalyzed hydrolysis to form doramectin monosaccharide which is then hydrolyzed again to remove the remaining saccharide unit and form doramectin aglycone.
T126476	Moellendorffilin
	Moellendorffilin 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T126476。
T68929	Lidorestat monohydrate
	Lidorestat monohydrate is an aldose reductase inhibitor potentially for the treatment of diabetic neuropathy and diabetic complications.
T22515	5'-Iodoresiniferatoxin	Others	Others
	TRPV1 (VR1) receptor antagonist
T22527	6'-Iodoresiniferatoxin	Others	Others
	TRPV1 (VR1) vanilloid receptor partial agonist
T32175	Iodorivanol
	Iodorivanol is a cytotoxic agent.
T76913	Avdoralimab
	Avdoralimab (IPH 5401)，一种全人IgGκ单克隆抗体，针对补体C5a受体1 (C5aR1)，阻碍其与C5a结合。该药物适用于研究补体驱动的炎症性疾病及实体瘤。
T75592	Odonthobuthus Doriae Venom
	Odonthobuthus Doriae Venom，一种从Odonthobuthus Doriae获得的蝎子毒液，通过调节离子通道产生神经毒性。
TP1391	β-Endorphin, equine (TFA)
	β-Endorphin, equine (TFA) is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors.

化合物

DPDPE TFA (88373-73-3 free base)

Cat.No: TP2036L

Synonym: DPDPE TFA

Target: Opioid Receptor

Cat.No: T6277

Synonym: BIRB 796,达马莫德,度马莫德

Target: Raf, p38 MAPK, Autophagy

Cat.No: T22314

Target: Antibacterial, Antibiotic

Bedoradrine sulfate

Cat.No: T26760

Synonym: KUR1246,MN 221 sulfate,KUR1246 sulfate,MN221 sulfate,KUR 1246 sulfate,MN-221 sulfate,KUR 1246,KUR-1246 sulfate,MN-221,MN 221,MN221,KUR-1246

Target: Adrenergic Receptor

Xanthine oxidoreductase-IN-5

Cat.No: T72166

Target: Xanthine Oxidase

β-Endorphin (1-27) (human) acetate

Cat.No: T38193L

Synonym: β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)

Target: Opioid Receptor

alpha-Endorphin acetate

Cat.No: T21511L

Synonym: α-内啡肽,alpha-Endorphin acetate (59004-96-5 Free base)

Target: Others

Doripenem monohydrate

Cat.No: T1037

Synonym: 多尼培南(一水合物),S 4661 monohydrate,Doripenem Hydrate,S-4661

Target: Antibacterial, Antibiotic

Cat.No: T15756

Synonym: IDD-676

Target: Reductase

Cat.No: T70047

Synonym: Bedoradrine free base

Target: Adrenergic Receptor

Cat.No: T62839

Synonym: SAGE-718

Target: NMDAR, iGluR

Aplindore Fumarate

Cat.No: T30098

Synonym: Aplindore,DAB-452 Fumarate,DAB-452

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

N-Acetyl-α-Endorphin acetate(88264-63-5 free base)

Cat.No: TP1508L

Target: Others

beta-Neoendorphin acetate(77739-21-0 free base)

Cat.No: TP2322L

Target: Opioid Receptor

Cat.No: T5500

Target: OX Receptor

Samidorphan HCl

Cat.No: T67888L

Synonym: Samidorphan HCl（852626-89-2 free base）

Target: Opioid Receptor

Cat.No: T1977

Synonym: Compound C,BML-275

Target: AMPK, Autophagy, TGF-beta/Smad

Cat.No: T15159

Synonym: HMS5552

Target: Glucokinase

Dorzolamide hydrochloride

Cat.No: T2134

Synonym: MK507 hydrochloride,L671152 hydrochloride,MK-507 (L-671152) HCl,盐酸多佐胺,Dorzolamide HCl

Target: Carbonic Anhydrase

Cat.No: T69146

Target: PPAR

Xanthine oxidoreductase-IN-3

Cat.No: T72165

Target: Xanthine Oxidase

Gonadorelin Acetate (33515-09-2 free base)

Cat.No: T5015

Synonym: 醋酸戈那瑞林,Luteinizing Hormone Releasing Hormone (LH-RH),Luteinizing Hormone Releasing Hormone (LH-RH), human,Gonadorelin Acetate

Target: Reductase

Cat.No: T3632

Synonym: 多拉维林,多拉韦林,MK-1439

Target: HIV Protease, Reverse Transcriptase

Cat.No: T7830

Target: Wnt/beta-catenin

Xanthine oxidoreductase-IN-4

Cat.No: T72078

Target: Xanthine Oxidase

Daridorexant hydrochloride

Cat.No: T67782

Synonym: Nemorexant hydrochloride,Quviviq

Target: OX Receptor

Dorsomorphin dihydrochloride

Cat.No: T6146

Synonym: BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride

Target: AMPK, Autophagy, TGF-beta/Smad

Cat.No: T70072

Aladorian sodium

Cat.No: T29818

Cat.No: T14153

Synonym: ARM036

Target: Others

β-Endorphin (1-27) (human)

Cat.No: T80515

Target: Opioid Receptor

β-Endorphin (rat)

Cat.No: T35460

Cat.No: T25034

Cat.No: T11656

Synonym: Indoramine D5,Wy-21901 D5

Target: CDK

Cat.No: T32584

Cat.No: T61165

Indoramin hydrochloride

Cat.No: T82072

Synonym: Indoramine hydrochloride,Wy 21901 hydrochloride

Cat.No: T124290

Cat.No: T125713

Cat.No: T24013

Synonym: DORA42,DORA-42

Dorlimomab aritox

Cat.No: T82532

Synonym: 4197X-RA,MDX-RA (ricin A chain) immunotoxin

Doramectin aglycone

Cat.No: T35733

Moellendorffilin

Cat.No: T126476

Lidorestat monohydrate

Cat.No: T68929

5'-Iodoresiniferatoxin

Cat.No: T22515

Target: Others

6'-Iodoresiniferatoxin

Cat.No: T22527

Target: Others

Cat.No: T32175

Cat.No: T76913

Odonthobuthus Doriae Venom

Cat.No: T75592

β-Endorphin, equine (TFA)

Cat.No: TP1391

Cat. No.	Product Name	Target	Signaling Pathways
T0969	Doramectin Dectomax,Cyclohexylavermectin B1,多拉菌素	Others; Antibiotic; Parasite	Microbiology/Virology; Others
	Doramectin (Dectomax) 是 Ivermectin 的衍生物。它是一种抗寄生虫抗生素。它具有在 NMRI 小鼠感染模型中抗曼氏链球菌作用。
T81621	Odoratisol B
	Odoratisol B为从Machilus odoratissimaNEES分离获得的天然化合物。
TN4695	Odorine	Others	Others
	Odorine has potent anti-carcinogenic effect by inhibiting both the initiation and promotion stages of two-stage skin carcinogenesis. It was found to inhibit the growth of the vinblastine-resistant KB cells by enhancing the anticancer activity of vinblastine.
TN4285	Isodorsmanin A	Others	Others
	Isodorsmanin A 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN4285，CAS号为 118266-99-2。
T13433	β-Endorphin, human	Others	Others
	β-Endorphin, human, a prominent endogenous peptide, existing in the hypophysis cerebri and hypothalamus,and is an agonist of opioid receptor.
TN3284	8-Hydroxyodoroside A	Others	Others
	An antitumor agent containing at least one compound selected from the group consisting of nerigoside, oleandrigenin, sarmentoside, oleaside A, oleandrin, 8β-hydroxy odoroside A, narciclasine, trans-dihydronarciclasine and bisdeoxynarciclasine is provided, this antitumor agent has an advantage of having an excellent therapeutic effect of tumor and less side effects.
TN4697	Odoroside H	ATPase; Potassium Channel; Sodium Channel	Membrane transporter/Ion channel
	Odoroside H has anticancer activities, the cytotoxic effects are induced by the inhibition of the plasma membrane bound Na(+)/K(+)-ATPase.
TN4694	Odoratone	Others	Others
	Odoratone shows insecticidal activities, it shows mortality on fourth instar larvae of mosquitoes (Anopheles stephensi) with LC(50) values of 154 ppm. Odoratone exhibits strong antifeedant activity against Pieris brassicae.
T76027	β-Endorphin, equine TFA
	β-Endorphin, equine TFA，是具备强效亲和力于μ和δ阿片受体(μ/δ opioid receptors)的内源性阿片类多肽，主要功能包括止痛。
TN2006	Odoriflavene	Others	Others
	Odoriflavene has antioxidant activity, and it also shows inhibition effects on the decrease of glutathione level of rat lens induced by UV irradiation. Odoriflavene shows cytotoxic activity against a SH-SY5Y cell line in vitro.
TN3888	Dorsmanin A	Others	Others
	Dorsmanin A is a natural product from Psoralea corylifolia.
TN5234	Vindorosine	Calcium Channel; Sodium Channel	Membrane transporter/Ion channel; Metabolism
	Vindorosine has blood vessel relaxation effect, possible underlying mechanisms involving the inhibition of Ca(2+) entry via L-type Ca(2+) channels in vascular smooth muscles.
TN3835	Desacetyldoronine	Others	Others
	Desacetyldoronine is a hepatotoxic pyrrolizidine alkaloid.
TN4696	Odorinol	Antifection	Microbiology/Virology
	Odorine and odorinol inhibit both the initiation and promotion stages of two-stage skin carcinogenesis. (+)-Odorinol exhibits strong antiviral activity against Ranikhet disease virus (RVD) in chick embryo.
TN5589	6α-Hydroxynidorellol
	6alpha-Hydroxynidorellol is a natural product from Callicarpa macrophylla.
T75669	Odoroside A
	Odoroside A，一种自夹竹桃叶中提取的有效成分，具抗癌活性。它通过ROS/p53信号通路诱导细胞凋亡及细胞周期阻滞，进而引发肿瘤细胞死亡。
TN6351	Dorsmanin I
	Dorsmanin I 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN6351，CAS号为 329703-46-0。
TN3159	6-Deoxy-9alpha-hydroxycedrodorin	Others	Others
	6-Deoxy-9alpha-hydroxycedrodorin shows potential value in the selection of insect-resistant clones for timber plantations.
TN2005	Odoratisol A	Others	Others
	Odoratisol A is a natural product from Myristica fragrans Houtt.
T83913	Mitraciliatine
	Mitraciliatine是一种在M. speciosa（泰国称为Kratom）中发现的生物碱，是μ-阿片受体（MOR）部分激动剂和κ-阿片受体（KOR）激动剂。该化合物对MOR和KOR具有选择性，与δ-阿片受体（DOR; EC50s分别为228, 218, 和 >1,000 nM，针对小鼠受体在GTPγS结合实验中的表现）。Mitraciliatine（100 nmol/动物，脑室内注射）在小鼠的热水尾部缩回实验中延长了撤回潜伏期，这一效果可以通过敲除MOR而非KOR来逆转。与吗啡不同，Mitraciliatine不会诱发过度活动或呼吸抑制。

天然产物

Cat.No: T0969

Synonym: Dectomax,Cyclohexylavermectin B1,多拉菌素

Target: Others, Antibiotic, Parasite

Cat.No: T81621

Cat.No: TN4695

Target: Others

Cat.No: TN4285

Target: Others

β-Endorphin, human

Cat.No: T13433

Target: Others

8-Hydroxyodoroside A

Cat.No: TN3284

Target: Others

Cat.No: TN4697

Target: ATPase, Potassium Channel, Sodium Channel

Cat.No: TN4694

Target: Others

β-Endorphin, equine TFA

Cat.No: T76027

Cat.No: TN2006

Target: Others

Cat.No: TN3888

Target: Others

Cat.No: TN5234

Target: Calcium Channel, Sodium Channel

Desacetyldoronine

Cat.No: TN3835

Target: Others

Cat.No: TN4696

Target: Antifection

6α-Hydroxynidorellol

Cat.No: TN5589

Cat.No: T75669

Cat.No: TN6351

6-Deoxy-9alpha-hydroxycedrodorin

Cat.No: TN3159

Target: Others

Cat.No: TN2005

Target: Others

Cat.No: T83913

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