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96

抑制剂 & 化合物

25

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Cat. No. Product Name Target Signaling Pathways
T23965 DAT 582

DAT582,DAT-582

DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent
T70527 DAT-230

DAT-230 is a promising microtubule inhibitor that has great potential for the treatment of fibrosarcoma in vitro and in vivo. DAT-230 exhibited potent anti-proliferative activity against various cancer cells. DAT-230 -treatment in HT-1080 cells resulted in microtubule de-polymerization and G2/M phase arrest preceding apoptosis. Phosphor-cdc2 (thr14/tyr15) reduction, cyclin B1 accumulation and aberrant spindles denoted the cyclin B1-cdc2 complex active and M phase arrest in HT-1080 cells treated ...
T25290 DAT1

DAT-1,DAT 1

DAT1 is an antimitotic and antiangiogenic that acts by binding to the colchicine binding site of tubulin.
T0322 Fipexide

Dopamine Receptor; AChR GPCR/G Protein; Neuroscience
Fipexide 是对氯苯乙酸衍生物,是哌嗪化学类的精神活性药物,作为促智药物,有用于老年痴呆的研究潜力。它可降低了纹状体腺苷酸环化酶的活性,通过多巴胺能神经传递对认知表现出积极的作用。
T6414 Bisacodyl

比沙可啶,Fenilaxan,Dulcolax,Brocalax

Others Others
Bisacodyl (Fenilaxan) 是刺激性缓泻剂,可直接作用于结肠以产生排便。它能够直接激活结肠巨噬细胞来增加 PGE2的分泌。PGE2充当旁分泌因子并减少结肠中 AQP3 的表达,抑制水从腔向血管一侧的转移,进而产生通便作用。
T22714 Decynium 22

Others Others
Decynium 22 是有机阳离子转运蛋白和单胺转运蛋白的抑制剂,具有抗抑郁作用。
T70525 ARC39

ARC39 is acid sphingomyelinase inhibitor (IC50 =20 nM).
T1871 GBR 12935 dihydrochloride

GBR12935,GBR-12935,GBR 12935

Dopamine Receptor GPCR/G Protein; Neuroscience
GBR 12935 dihydrochloride (GBR 12935) 是一种多巴胺再吸收抑制剂。
T1993 J-147

J147

Epigenetic Reader Domain; Dopamine Receptor; Monoamine Oxidase Chromatin/Epigenetic; GPCR/G Protein; Neuroscience
J-147 是一种高效的、具有口服活性的、可透过血脑屏障神经保护剂,可增强认知能力。它抑制单胺氧化酶 B 和多巴胺转运体,EC50分别为 1.88 μM 和 0.649 μM。它有研究阿尔茨海默氏症的潜力。
T11087 DOV-216,303 Free Base

DOV-216303

Dopamine Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
DOV-216,303 Free Base (DOV-216303) 是血清素、去甲肾上腺素和多巴胺再摄取的抑制剂,IC50 为 14、20 和 78 nM。 DOV-216,303 Free Base 具有抗抑郁作用。
T39429 AHN 1-055 hydrochloride

3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) 与多巴胺转运蛋白具有高亲和力,是多巴胺摄取抑制剂,IC50为 71 nM。
T10758L Centanafadine hydrochloride

EB-1020 hydrochloride

Dopamine Receptor; Serotonin Transporter; Adrenergic Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Centanafadine hydrochloride (EB-1020 hydrochloride) 是一种去甲肾上腺素(NE)/多巴胺(DA)转运的双抑制剂,还能抑制5-羟色胺(serotonin)转运体。它对人 NE,DA 和5-羟色胺转运体的 IC50值分别为6 nM,38 nM 和 83 nM。
T3526 Dasotraline hydrochloride

SEP-225289 hydrochloride,达索曲林盐酸盐

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Dasotraline hydrochloride (SEP-225289 hydrochloride) 是具有阻断多巴胺 (IC50=4 nM),去甲肾上腺素 (IC50=6 nM) 和三羟色胺转运蛋白 (IC50=11 nM)的三重再摄取抑制剂。
T7745 Diclofensine hydrochloride

4-(3,4-二氯苯)-7-甲氧基-2-甲基-1,2,3,4-四氢异喹啉盐酸盐,Ro 8-4650 hydrochloride

Others; Dopamine Receptor GPCR/G Protein; Neuroscience; Others
Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。
T2092 Amitifadine hydrochloride

DOV-21947 hydrochloride,EB-1010 hydrochloride

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Amitifadine hydrochloride (EB-1010 hydrochloride) 是一种 5-羟色胺-去甲肾上腺素-多巴胺的再摄取抑制剂(SNDRI),其在 HEK 293 细胞中测得的 IC50值分别为 12, 23, 96 nM。
T69807 EGFR-IN-451

EGFR-IN-451 is an EGFR inhibitor, attenuating Ang II-induced Kidney Fibrosis.
T7153 Vanoxerine dihydrochloride

GBR-12909 dihydrochloride,伐诺司林二盐酸盐,I893 dihydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) 是一种竞争性的、有效的、选择性的多巴胺再摄取抑制剂,能够与多巴胺转运体 (DAT) 上的靶点结合。
T0991 Desipramine hydrochloride

NSC-114901,Desmethylimipramine,盐酸去甲咪嗪,JB-8181,EX-4355,Norimipramine,G-35020

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor GPCR/G Protein; Neuroscience
Desipramine hydrochloride (Norimipramine) 是一种二苯并氮杂类衍生物三环类抗抑郁药,可作为选择性去甲肾上腺素再摄取抑制剂。 它还显示出较弱的 5-羟色胺再摄取抑制、α1 阻断、抗组胺和抗胆碱能作用。
T7341 Diclofensine

Ro 8-4650,(+/-)-双氮奋兴

Dopamine Receptor; Monoamine Transporter GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Diclofensine (Ro 8-4650) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。
T29534 ABT-925 fumarate dihydrate

ABT 925,LU201640,ABT925,ABT-925,BSF201640,DAT201

ABT-925 is a selective dopamine D3 receptor (DRD3) antagonist with an in vitro affinity approximately 100 times higher for dopamine D3 receptors than for D2 receptors.
T1970 Gedatolisib

PF-05212384,PKI-587

PI3K; mTOR PI3K/Akt/mTOR signaling
Gedatolisib (PF-05212384) 是一种高效的双重 PI3Kα (IC50:0.4 nM),PI3Kγ (IC50:5.4 nM) 和 mTOR (IC50:1.6 nM)抑制剂。它在 mTOR 复合物mTORC1和mTORC2中同样有效。
T7747 Datelliptium chloride hydrochloride

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Datelliptium chloride hydrochloride 是一种衍生自玫瑰树碱的 DNA 嵌入剂,具有抗肿瘤活性。
T23631 Adatanserin

WY-50324,WY 50324,WAY SEB 324,WY50324

5-HT Receptor GPCR/G Protein; Neuroscience
Adatanserin (WY 50324) 是一种混合型 5-HT1A 受体部分激动剂,也是一种 5-HT2A 和 5-HT2C 受体拮抗剂,具有潜在的神经保护活性,可用于研究焦虑和抑郁症。
T39630 Zandatrigine

NBI-921352,XEN901

Sodium Channel Membrane transporter/Ion channel
Zandatrigine (NBI-921352) 是钠通道蛋白 8 型亚基 α 的阻断剂,可用于癫痫治疗的神经系统病理学研究。
T13110 Tedatioxetine hydrobromide

Lu AA 24530 hydrobromide

Dopamine Receptor; 5-HT Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) 是一种血清素-去甲肾上腺素-多巴胺再摄取抑制剂 ,也是 5-HT2A、5-HT2C、5-HT3 和 α1A-肾上腺素能受体的拮抗剂,可用于治疗抑郁症和焦虑症。
T19668 Tiomolibdate diammonium

Ammonium molybdenum sulfide,Ammonium tetrathiomolybdate,NSC 286644,ATTM,四硫钼酸铵,Coprexa

Others Others
Tiomolibdate diammonium (NSC-286644) 是超氧化物歧化酶 1 (SOD1) 的抑制剂,具有抗血管生成和抗肿瘤活性。 Tiomolibdate diammonium 抑制铜酶的活性,包括 SOD1 和 COX。
T5159 Olodaterol hydrochloride

BI-1744 HCl,盐酸奥达特罗,BI 1744 hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Olodaterol hydrochloride (BI-1744 HCl) 是一种长效的、选择性 β2-adrenoceptor(β2-AR) 激动剂 (EC50=0.1 nM;pKi= 9.14 for human β2-adrenoceptor),可用于慢性阻塞性肺疾病 (COPD) 和肺纤维化的研究。
T23445 Anxiolytic/nonsedative agent-1

TCS 1205

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Anxiolytic/nonsedative agent-1 (TCS 1205) 是一种有效的选择性 GABAA 激动剂。Anxiolytic/nonsedative agent-1 对牛脑膜中的 BzR 显示出明显的亲和力,对 α1β2γ2、α2β2γ2、α5β3γ2 的 Kis 分别为 14、121、239 nM。Anxiolytic/nonsedative agent-1 在体外表现出 α2 选择性功效,在体内表现出抗焦虑选择性作用。
T2189 Sodium orthovanadate

Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate

ATPase; Phosphatase Membrane transporter/Ion channel; Metabolism
Sodium orthovanadate 是一种蛋白酪氨酸磷酸酶,碱性磷酸酶和一些ATP 酶的抑制剂,有可能充当磷酸盐类似物。它具有胰岛素样作用、对心室肌的正性肌力作用和其他代谢作用。
T34795 Tedatioxetine

Lu AA-24530,Lu AA24530,Lu AA 24530

Tetaxetine( LU AA24530) has been reported as a triple reuptake inhibitor (5-HT > NE > DA) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist.Meanwhile, it is an antidepressant agent.
T15378L Gemcitabine elaidate hydrochloride

CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride

Others Others
Gemcitabine elaidate (CP-4126) hydrochloride 是 Gemcitabine 的亲脂性前药。Gemcitabine elaidate hydrochloride 通过酯酶转化为 Gemcitabine 以被磷酸化。Gemcitabine elaidate hydrochloride 可以口服给药,具有抗肿瘤活性。
T74398 DATPT

Reactive Oxygen Species; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
DATPT 是一种小分子 12WLVSKF17 肽模拟分子。DATPT 抑制 SNX9-p47phox 相互作用,抑制活性氧和炎性细胞因子的产生。DATPT 具有抗炎和抗菌活性,通过减少 ATP 的产生发挥作用。DATPT 是治疗脓毒症的潜在化合物。
T29645 Adatanserin hydrochloride

WY50324 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Adatanserin hydrochloride (WY50324 hydrochloride) 是一种新型 5-HT(1A)/5-HT(2) 受体配体,具有潜在的神经保护作用,抑制内源性氨基酸缺血性外排,可用于研究抑郁症和焦虑症。
T9901A-007 Datopotamab

Others Others
Datopotamab (CDP7657) 是一种靶向 TROP2 的抗体,是 Datopotamab deruxtecan 的裸抗,可用于合成抗体活性分子偶联物( Datopotamab deruxtecan)。
T22867 Indatraline hydrochloride

Others Others
Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)
T38630 Ludaterone

Ludaterone is an antiandrogen agent, with potent antiandrogenic activity.
T70323 Diethanolamine Fusidate

Diethanolamine Fusidate is a bacteriostatic antibiotic with similar activity and better absorption after oral administration (in animals) than the sodium salt of Fusidic Acid. This product inhibits protein synthesis in prokaryotes by inhibiting the ribosome-dependent activity of G factor and translocation of peptidyl-tRNA.
T76875 Zanidatamab

Zanidatamab (ZW25) 是一种针对 2 个不同 HER2表位 (ECD2 和 ECD4) 的人源双特异性单克隆抗体。Zanidatamab 具有抗肿瘤活性。
T77104 Obrindatamab

Obrindatamab 是一种人源化抗 B7-H3/CD3双特异性抗体。Obrindatamab 结合 B7-H3和 CD3,从而介导针对表达 B7-H3的癌细胞的重定向细胞毒性 T 淋巴细胞 (CTL) 活性。Obrindatamab 可用于癌症研究。
T68661 Edatrexate

CGP 30694

Edatrexate (CGP 30694),即 10-乙基-10-去甲氨基蝶呤,是甲氨蝶呤Methotrexate 的类似物,对耐 MTX 肿瘤具有抗肿瘤活性。Edatrexate 是一种抗叶酸抗代谢物,可用于研究非小细胞肺癌,乳腺癌,非霍奇金淋巴瘤和头颈部癌症的研究。
T80434 Heteropodatoxin-2

Potassium Channel Membrane transporter/Ion channel
Heteropodatoxin-2为含30个氨基酸的肽,归属于异足毒素类。它能电压依赖性地阻断非洲爪蟾卵母细胞表达的Kv4.2电流,并在正电位较高时显示出较低的阻断效应。
T14339 Athidathion

GS-13006

Others Others
Thiophos (GS-13006) is an insecticide, which is an organic phosphate ester.
T40670 7-Deaza-7-propargylamino-dATP

7-Deaza-7-propargylamino-dATP is a deoxyadenosine triphosphate (dATP) analog utilized in the field of gene sequencing.
T38532 7-Deaza-7-propargylamino-ddATP

7-Deaza-7-propargylamino-ddATP, an analog of ddATP, serves as a viable option for gene sequencing purposes due to its chemical composition.
T75026 PROTAC TYK2 degradation agent1

PROTACs PROTAC
PROTACTYK2 degradation agent1为亚型选择性TYK2降解剂,表现出杰出的TYK2降解活性,其DC50为14 nM,适用于自身免疫性疾病研究。
T24604 PDAT

Propyl Dimethyl Amino Tryptamine

PDAT is a noncompetitive Indolethylamine N-methyltransferase inhibitor.
T64510 Hexan-3-yl carbonochloridate

Hexan-3-yl carbonochloridate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64510。
T20679 Pyridate

P1 3419,CL-11344,Fenpyrate,Pyron,CL11344,CL 11344

Pyridate is mainly used as a selective post seedling herbicide.
T15378 Gemcitabine elaidate

Gemcitabine 5'-elaidate,反油酸吉西他滨,吉西他滨反油酸酯,Gemcitabine (elaidate),CO-101,CP-4126

Apoptosis; Nucleoside Antimetabolite/Analog; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Gemcitabine elaidate (CP-4126) 是 Gemcitabine 的亲脂性前药。它通过酯酶转化为 Gemcitabine 以被磷酸化。它具有抗肿瘤活性。
T10982 ddATP

2',3'-Dideoxyadenosine 5'-triphosphate

Others Others
ddATP is a dideoxynucleotide, used as a chain extension inhibitor for DNA polymerase, and used for DNA sequencing by the Sanger method.

化合物

DAT 582
Cat.No: T23965
Synonym: DAT582,DAT-582
Target:
DAT-230
Cat.No: T70527
Synonym:
Target:
DAT1
Cat.No: T25290
Synonym: DAT-1,DAT 1
Target:
Fipexide
Cat.No: T0322
Synonym:
Target: Dopamine Receptor, AChR
Bisacodyl
Cat.No: T6414
Synonym: 比沙可啶,Fenilaxan,Dulcolax,Brocalax
Target: Others
Decynium 22
Cat.No: T22714
Synonym:
Target: Others
ARC39
Cat.No: T70525
Synonym:
Target:
GBR 12935 dihydrochloride
Cat.No: T1871
Synonym: GBR12935,GBR-12935,GBR 12935
Target: Dopamine Receptor
J-147
Cat.No: T1993
Synonym: J147
Target: Epigenetic Reader Domain, Dopamine Receptor, Monoamine Oxidase
DOV-216,303 Free Base
Cat.No: T11087
Synonym: DOV-216303
Target: Dopamine Receptor, Serotonin Transporter, Norepinephrine
AHN 1-055 hydrochloride
Cat.No: T39429
Synonym: 3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride
Target: Dopamine Receptor
Centanafadine hydrochloride
Cat.No: T10758L
Synonym: EB-1020 hydrochloride
Target: Dopamine Receptor, Serotonin Transporter, Adrenergic Receptor, Norepinephrine
Dasotraline hydrochloride
Cat.No: T3526
Synonym: SEP-225289 hydrochloride,达索曲林盐酸盐
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine
Diclofensine hydrochloride
Cat.No: T7745
Synonym: 4-(3,4-二氯苯)-7-甲氧基-2-甲基-1,2,3,4-四氢异喹啉盐酸盐,Ro 8-4650 hydrochloride
Target: Others, Dopamine Receptor
Amitifadine hydrochloride
Cat.No: T2092
Synonym: DOV-21947 hydrochloride,EB-1010 hydrochloride
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine
EGFR-IN-451
Cat.No: T69807
Synonym:
Target:
Vanoxerine dihydrochloride
Cat.No: T7153
Synonym: GBR-12909 dihydrochloride,伐诺司林二盐酸盐,I893 dihydrochloride
Target: Dopamine Receptor
Desipramine hydrochloride
Cat.No: T0991
Synonym: NSC-114901,Desmethylimipramine,盐酸去甲咪嗪,JB-8181,EX-4355,Norimipramine,G-35020
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor
Diclofensine
Cat.No: T7341
Synonym: Ro 8-4650,(+/-)-双氮奋兴
Target: Dopamine Receptor, Monoamine Transporter
ABT-925 fumarate dihydrate
Cat.No: T29534
Synonym: ABT 925,LU201640,ABT925,ABT-925,BSF201640,DAT201
Target:
Gedatolisib
Cat.No: T1970
Synonym: PF-05212384,PKI-587
Target: PI3K, mTOR
Datelliptium chloride hydrochloride
Cat.No: T7747
Synonym:
Target: DNA/RNA Synthesis
Adatanserin
Cat.No: T23631
Synonym: WY-50324,WY 50324,WAY SEB 324,WY50324
Target: 5-HT Receptor
Zandatrigine
Cat.No: T39630
Synonym: NBI-921352,XEN901
Target: Sodium Channel
Tedatioxetine hydrobromide
Cat.No: T13110
Synonym: Lu AA 24530 hydrobromide
Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine
Tiomolibdate diammonium
Cat.No: T19668
Synonym: Ammonium molybdenum sulfide,Ammonium tetrathiomolybdate,NSC 286644,ATTM,四硫钼酸铵,Coprexa
Target: Others
Olodaterol hydrochloride
Cat.No: T5159
Synonym: BI-1744 HCl,盐酸奥达特罗,BI 1744 hydrochloride
Target: Adrenergic Receptor
Anxiolytic/nonsedative agent-1
Cat.No: T23445
Synonym: TCS 1205
Target: GABA Receptor
Sodium orthovanadate
Cat.No: T2189
Synonym: Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate
Target: ATPase, Phosphatase
Tedatioxetine
Cat.No: T34795
Synonym: Lu AA-24530,Lu AA24530,Lu AA 24530
Target:
Gemcitabine elaidate hydrochloride
Cat.No: T15378L
Synonym: CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride
Target: Others
DATPT
Cat.No: T74398
Synonym:
Target: Reactive Oxygen Species, Antibacterial
Adatanserin hydrochloride
Cat.No: T29645
Synonym: WY50324 hydrochloride
Target: 5-HT Receptor
Datopotamab
Cat.No: T9901A-007
Synonym:
Target: Others
Indatraline hydrochloride
Cat.No: T22867
Synonym:
Target: Others
Ludaterone
Cat.No: T38630
Synonym:
Target:
Diethanolamine Fusidate
Cat.No: T70323
Synonym:
Target:
Zanidatamab
Cat.No: T76875
Synonym:
Target:
Obrindatamab
Cat.No: T77104
Synonym:
Target:
Edatrexate
Cat.No: T68661
Synonym: CGP 30694
Target:
Heteropodatoxin-2
Cat.No: T80434
Synonym:
Target: Potassium Channel
Athidathion
Cat.No: T14339
Synonym: GS-13006
Target: Others
7-Deaza-7-propargylamino-dATP
Cat.No: T40670
Synonym:
Target:
7-Deaza-7-propargylamino-ddATP
Cat.No: T38532
Synonym:
Target:
PROTAC TYK2 degradation agent1
Cat.No: T75026
Synonym:
Target: PROTACs
PDAT
Cat.No: T24604
Synonym: Propyl Dimethyl Amino Tryptamine
Target:
Hexan-3-yl carbonochloridate
Cat.No: T64510
Synonym:
Target:
Pyridate
Cat.No: T20679
Synonym: P1 3419,CL-11344,Fenpyrate,Pyron,CL11344,CL 11344
Target:
Gemcitabine elaidate
Cat.No: T15378
Synonym: Gemcitabine 5'-elaidate,反油酸吉西他滨,吉西他滨反油酸酯,Gemcitabine (elaidate),CO-101,CP-4126
Target: Apoptosis, Nucleoside Antimetabolite/Analog, Autophagy
ddATP
Cat.No: T10982
Synonym: 2',3'-Dideoxyadenosine 5'-triphosphate
Target: Others
Cat. No. Product Name Target Signaling Pathways
T5165 10-Deacetyltaxol

10-DAT,10-Desacetyl Paclitaxel,去乙酰紫衫醇,Deacetyltaxol,10-去乙酰紫杉醇,10-deacetyl-paclitaxel,Deacetyl Paclitaxel

Others; Microtubule Associated Cytoskeletal Signaling; Others
10-Deacetyltaxol (10-DAT) 是从红豆杉中分离得到的一种紫杉醇衍生物,对人脑胶质细胞瘤和神经母细胞瘤细胞具有细胞毒性。它能促进微管蛋白的聚合,在体外抑制由钙离子诱导的微管解聚。
TN6552 5,7-Dimethoxyluteolin

Dopamine Receptor GPCR/G Protein; Neuroscience
5,7-Dimethoxyluteolin 是 5,7-二甲基木犀草素的一种衍生物,可以活化多巴胺转运蛋白,EC50为 3.417 μM。
T3273 Bifendate

联苯双酯,Bifendatatum

HBV; Reverse Transcriptase Microbiology/Virology
Bifendate (Bifendatatum) 是 Schisandrin C 的合成中间体,在慢性 B 型肝炎的研究中具有抗HBV 功效,用于治疗病毒性肝炎和药物性肝损伤引起的转氨酶升高。
TN3831 (-)-Denudatin B

Denudatin B

ATPase; Potassium Channel; Calcium Channel; PAFR GPCR/G Protein; Membrane transporter/Ion channel; Metabolism
(-)-Denudatin B (Denudatin B) 源自 Magnolia fargesii。 (-)-Denudatin B 通过抑制胶原蛋白和凝血酶诱导的磷酸肌醇分解,在高浓度下具有非特异性抗血小板作用。
T2736 Sodium Demethylcantharidate

Sodium norcantharidin,去甲斑蝥酸钠

Others; Endogenous Metabolite Metabolism; Others
Sodium Demethylcantharidate (Sodium norcantharidin) 是内源性代谢产物的一种。
T5735 Methyl deacetylasperulosidate

Deacetyl asperulosidic acid methyl ester,6α-Hydroxygeniposide,去乙酰车叶草苷酸甲酯

Others Others
Methyl deacetylasperulosidate (6α-Hydroxygeniposide) 是环烯醚萜类化合物,能够降低正常小鼠的血糖水平,对小鼠具有通便作用。
T3150 Caudatin

告达亭苷元,告达庭

Apoptosis; Others Apoptosis; Others
Caudatin 是白首乌中的一种甾体类天然产物,具有抗肿瘤和抗血管生成作用。它是一种 C-21 甾体糖苷,可使细胞周期停滞,诱导细胞凋亡。
T2938 (E/Z)-Polydatin

云杉新甙,(E/Z)-虎杖苷,Polydatin,(E/Z)-Piceid

Phospholipase Metabolism
(E/Z)-Polydatin (Polydatin) 是从虎杖的根和根茎中分离得到的一种单晶化合物。它具有抗血小板聚集、心脏保护作用、抗低密度脂蛋白 (LDL) 氧化作用、抗炎和免疫调节功能。
T7958 Methyl arachidate

花生酸甲酯,Methyl Icosanoate

Others; Aminopeptidase Metabolism; Others
Methyl arachidate (Methyl Icosanoate) 是一种天然化合物,具有白三烯 A4 水解酶 (LTA4H) 抑制活性。
T3427 Polydatin

Piceid,虎杖苷,Polydotin Peceid

Apoptosis; Mitophagy; NF-κB; Autophagy Apoptosis; Autophagy; NF-κB
Polydatin (Piceid) 是从传统中药虎杖根中提取的一种天然产物,在多个实验模型中具有抗炎作用。它可抑制 G6PD,并诱导氧化和内质网应激。
TN3774 Daturametelin I

Others Others
Daturametelin I 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3774,CAS号为 904667-65-8。
T38415 Adenosine 5′-monophosphoramidate sodium

Adenosine 5′-monophosphoramidate sodium is a derivative of adenosine used as an intermediate for nucleotide synthesis. It significantly influences the accumulation of cyclic AMP.
T75637 Demethylcantharidate disodium

Demethylcantharidate disodium 是一种内源性代谢产物,能通过诱导内质网应激来促进肝癌细胞的凋亡,并且对多种类型的癌症展现出良好的抗癌活性。
TN3775 Daturataturin A aglycone

Others Others
Daturataturin A aglycone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3775,CAS号为 904665-71-0。
TN3772 Datiscin

Others Others
Datiscin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3772,CAS号为 16310-92-2。
TN7002 Methyl linolelaidate

Methyl linolelaidate is a natural product.
T3S0626 Denudatine

光翠雀碱;裸翠雀亭,光翠雀碱

Others Others
Denudatine 是分离自乌头属和翠雀属植物中,能够影响心室纤维的动作电位,并抑制乌头碱的致心律失常作用。
TN6570 Daturaolone

Daturaolone has potency in reducing the harmful effects or in maintaining the normal hepatic physiological mechanisms in both acute and chronic hepato-toxic induced liver damage in rats. Daturaolone also possesses in vivo anti-inflammatory and antinocicep
TN3773 Daturabietatriene

Others Others
Daturabietatriene is a natural product from Pinus yunnanensis.
TN3776 Daturataturin A

Others Others
Daturataturin A是一种天然产物,属于茄科曼陀罗属,其产品编号为 TN3776,CAS号为 133360-51-7。Daturataturin A可用作对照参考。
TN5218 Valerosidate

Others Others
Valerosidate is a natural product from Valeriana jatamansi.
TN6027 Pedatisectine F

2-Methyl-6-(1,2,3,4-tetrahydroxybutyl)pyrazine

Pedatisectine F是一种天然产物,属于天南星科半夏属,其产品编号为 TN6027,CAS号为 206757-32-6。Pedatisectine F可用作对照参考。
TN3262 8(17),12E,14-Labdatrien-20-oic acid

Others Others
8(17),12E,14-Labdatrien-20-oic acid is a natural product from Isodon yuennanensis.
TN3788 Decursidate

Others Others
Decursidate是一种天然产物,属于伞形科前胡属,其产品编号为 TN3788,CAS号为 272122-56-2。Decursidate可用作对照参考。
TN2161 Rotundatin

Others Others
Rotundatin is a natural product from Dendrobium rotundatum.

天然产物

10-Deacetyltaxol
Cat.No: T5165
Synonym: 10-DAT,10-Desacetyl Paclitaxel,去乙酰紫衫醇,Deacetyltaxol,10-去乙酰紫杉醇,10-deacetyl-paclitaxel,Deacetyl Paclitaxel
Target: Others, Microtubule Associated
5,7-Dimethoxyluteolin
Cat.No: TN6552
Synonym:
Target: Dopamine Receptor
Bifendate
Cat.No: T3273
Synonym: 联苯双酯,Bifendatatum
Target: HBV, Reverse Transcriptase
(-)-Denudatin B
Cat.No: TN3831
Synonym: Denudatin B
Target: ATPase, Potassium Channel, Calcium Channel, PAFR
Sodium Demethylcantharidate
Cat.No: T2736
Synonym: Sodium norcantharidin,去甲斑蝥酸钠
Target: Others, Endogenous Metabolite
Methyl deacetylasperulosidate
Cat.No: T5735
Synonym: Deacetyl asperulosidic acid methyl ester,6α-Hydroxygeniposide,去乙酰车叶草苷酸甲酯
Target: Others
Caudatin
Cat.No: T3150
Synonym: 告达亭苷元,告达庭
Target: Apoptosis, Others
(E/Z)-Polydatin
Cat.No: T2938
Synonym: 云杉新甙,(E/Z)-虎杖苷,Polydatin,(E/Z)-Piceid
Target: Phospholipase
Methyl arachidate
Cat.No: T7958
Synonym: 花生酸甲酯,Methyl Icosanoate
Target: Others, Aminopeptidase
Polydatin
Cat.No: T3427
Synonym: Piceid,虎杖苷,Polydotin Peceid
Target: Apoptosis, Mitophagy, NF-κB, Autophagy
Daturametelin I
Cat.No: TN3774
Synonym:
Target: Others
Adenosine 5′-monophosphoramidate sodium
Cat.No: T38415
Synonym:
Target:
Demethylcantharidate disodium
Cat.No: T75637
Synonym:
Target:
Daturataturin A aglycone
Cat.No: TN3775
Synonym:
Target: Others
Datiscin
Cat.No: TN3772
Synonym:
Target: Others
Methyl linolelaidate
Cat.No: TN7002
Synonym:
Target:
Denudatine
Cat.No: T3S0626
Synonym: 光翠雀碱;裸翠雀亭,光翠雀碱
Target: Others
Daturaolone
Cat.No: TN6570
Synonym:
Target:
Daturabietatriene
Cat.No: TN3773
Synonym:
Target: Others
Daturataturin A
Cat.No: TN3776
Synonym:
Target: Others
Valerosidate
Cat.No: TN5218
Synonym:
Target: Others
Pedatisectine F
Cat.No: TN6027
Synonym: 2-Methyl-6-(1,2,3,4-tetrahydroxybutyl)pyrazine
Target:
8(17),12E,14-Labdatrien-20-oic acid
Cat.No: TN3262
Synonym:
Target: Others
Decursidate
Cat.No: TN3788
Synonym:
Target: Others
Rotundatin
Cat.No: TN2161
Synonym:
Target: Others
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