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59

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T8239 Cromoglicic acid

Others Others
Cromoglicic acid 可防止肥大细胞释放炎性化学物质,例如组胺。
T0211 Azelastine

Azelastina,Astelin,Azelastinum,氮卓斯汀

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine (Azelastinum) 是一种选择性组胺 1 拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T21404 Fluticasone furoate

Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate

Glucocorticoid Receptor Endocrinology/Hormones
Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇,衍生自氟替卡松,Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。
T3979 Emedastine

LY188695,依美斯汀,Emadine

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Emedastine (LY188695) 是一种可口服的,选择性和高亲和力的组胺 H1受体拮抗剂,Ki 值为 1.3 nM。它是苯并咪唑衍生物,可用于过敏性鼻炎、过敏性皮肤疾病和过敏性结膜炎的研究。
T0118 Mizolastine

SL 850324,咪唑司汀,咪唑斯汀

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mizolastine (SL 850324) 是组胺 H1 受体拮抗剂,IC50为 47 nM。它用于治疗过敏反应,如花粉热和荨麻疹等。
T6242 Rupatadine Fumarate

富马酸卢帕他定,Rinialer,Rupafin,Alergoliber

PAFR; Autophagy; Histamine Receptor Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Rupatadine Fumarate (Rinialer) 是一种可口服的长效PAF/H1受体的双抑制剂,Ki 值分别为 0.55 μM 和 0.1 μM。它可研究过敏性鼻炎和荨麻疹。
T3185 R112

(E)-Elafibranor

Syk Angiogenesis; Tyrosine Kinase/Adaptors
R112 ((E)-Elafibranor) 是ATP 竞争性的 Syk 激酶抑制剂,它能够抑制Syk 激酶活性,Ki=6 nM,IC50=226 nM。
T1030 Triprolidine hydrochloride monohydrate

盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Triprolidine hydrochloride monohydrate 是一种组胺 H1 拮抗剂,用于过敏性鼻炎、哮喘。
T0059 Diphenylpyraline hydrochloride

盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂,抑制多巴胺的吸收。它是可口服的抗组胺试剂,具有抗胆碱和抗过敏作用,可用于缓解过敏性疾病,如鼻炎、花粉热和瘙痒性皮肤疾病等。
T0211L Azelastine hydrochloride

Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine hydrochloride (Astelin) 是一种选择性组胺 1拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T1269 Tripelennamine hydrochloride

Pyribenzamine hydrochloride,去敏灵,Tripelennamine HCl,Pyribenzamine HCl,盐酸曲吡那敏

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) 是一种组胺 H1 拮抗剂,具有低镇静作用,但经常刺激胃肠道。
T3520 Setipiprant

KYTH-105,塞替匹仑,ACT-129968

GPR; Prostaglandin Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation
Setipiprant (ACT-129968) 是一种口服的选择性 CRTH2 拮抗剂,IC50为6.0 nM。
T2335 Ebastine

Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ebastine (Kestine) 是一种可口服的组胺 H1 受体拮抗剂,用于过敏性鼻炎的症状和慢性特发性荨麻疹的研究。
T0188 Fluticasone (propionate)

丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate

Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Microbiology/Virology
Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,亲和力KD 为 0.5 nM。具有抗病毒活性。
T0205 Brompheniramine maleate

Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Brompheniramine maleate (Dimotane) 是一种可口服的丙胺类抗组胺剂,具有抗胆碱能和抗抑郁作用,可用于过敏性鼻炎和缓解疼痛的研究。它是一种选择性组胺 H1 受体拮抗剂,Kd 为 6.06 nM。
T0089 Cetirizine dihydrochloride

盐酸西替利嗪,P071,UCB P071,Cetirizine DiHCl

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Cetirizine dihydrochloride (UCB P071) 是羟嗪的羧化代谢物,是特异性口服有效的 H1 受体长效拮抗剂。它标记抗过敏特性,抑制过敏反应期间嗜酸性粒细胞趋化,可有效治疗过敏性鼻炎、确诊荨麻疹和花粉诱发的哮喘。
T21472 Dimethindene maleate

马来酸二甲茚定,UNII-6LL60J9E0O,SU 6518,SU-6518

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Dimethindene maleate (SU 6518) 是一种组胺 H1 拮抗剂,可用于治疗过敏反应、瘙痒和鼻炎的研究。
T6660 SB-705498

TRP/TRPV Channel Membrane transporter/Ion channel
SB705498 是一种口服有效的 TRPV1选择性拮抗剂,pIC50值为 7.1。
T1553 Chlorpheniramine maleate

马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Chlorpheniramine maleate (NCI-C55265) 是一种组胺 H1 拮抗剂,IC50为12 nM,用于过敏反应、花粉热、鼻炎、荨麻疹和哮喘。
T1531 Mometasone furoate

糠酸莫美他松,糠酸莫米松,Sch32088

Glucocorticoid Receptor Endocrinology/Hormones
Mometasone furoate (Sch32088) 是糖皮质激素受体激动剂,具有抗炎和抗过敏作用。它是皮质固醇类试剂,动物模型中,可局部应用于气道炎症、慢性皮肤湿疹、哮喘。
T2396 Ramatroban

BAY u3405,雷马曲班

GPR; Prostaglandin Receptor; PPAR DNA Damage/DNA Repair; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism
Ramatroban (BAY u3405) 是一种血栓素 A(2) (TxA(2)) 拮抗剂,IC50为 14 nM。它还通过抑制PGD2结合从而拮抗CRTH2,IC50为113 nM。它用于治疗过敏性鼻炎,可用于治疗哮喘的研究。
T22354 Levocetirizine Dihydrochloride

Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydrochloride is the R-enantiomer of Cetirizine, which gives it a higher affinity for the H1-receptor than the S-enantiomer. Due to this enhanced affinity, Levocetirizine Dihydrochloride is effective in treating allergic rhinitis and chronic idiopathic urticaria.
T1097 Loratadine

氯雷他定,SCH 29851,Loratidine

Influenza Virus; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Loratadine (SCH 29851) 是一种组胺 H1受体反向激动剂,IC50>32 μM。它抑制炎症介质的免疫释放,具有抗登革热病毒的活性。
T61213 PF-03654764

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
PF-03654764 是一种具有口服活性、高效性和选择性的组胺 H3 受体拮抗剂,对人 H3 和大鼠 H3 具有抑制作用, Ki 值分别为 1.2 nM 和 7.9 nM。PF-03654764 常与 Fexofenadine 一起联合用药来治疗过敏性鼻炎。
T77601 (2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid

GPR Endocrinology/Hormones; GPCR/G Protein
(2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid是一种前列腺素类 CRTH2拮抗剂,其IC50< 10 μM,可用于研究鼻炎、慢性阻塞性肺疾病、类风湿性关节炎、湿疹和结膜炎。
T77426 Pascolizumab

SB-240683

IL Receptor Immunology/Inflammation
Pascolizumab (SB-240683) 是一种人源化抗 IL-4 单克隆抗体。Pascolizumab 具有哮喘作用,可用于研究过敏性鼻炎。
T1470 Fexofenadine hydrochloride

Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,盐酸非索非那定,Telfast,Fexofenadine HCl,Allegra,MDL 16455A

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) 是一种抗组胺药,用于治疗过敏性鼻炎、血管性水肿和慢性荨麻疹。
T0098 Ipratropium bromide monohydrate

Ipratropium bromide hydrate,溴化异丙托品单水合物

AChR Neuroscience
Ipratropium bromide monohydrate (Ipratropium bromide hydrate) 是一种毒蕈碱拮抗剂,结构上与阿托品相关,但它通常被认为对吸入使用更安全、更有效。它用于各种支气管疾病、鼻炎和抗心律失常。
T2270 Trans-Tranilast

Tranilast trans-,反式-曲尼司特,反-曲尼司特

RAAS Endocrinology/Hormones
Trans-Tranilast 是抗过敏剂,可用于过敏性鼻炎、支气管哮喘和特应性皮炎的研究。
T1278 Astemizole

Laridal,Histaminos,Paralergin,阿司咪唑

Potassium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Astemizole (Laridal) 是一种长效、非镇静抗组胺药,用于治疗季节性过敏性鼻炎、哮喘、过敏性结膜炎和慢性特发性荨麻疹。它是组胺 H1 受体的拮抗剂,IC50值为 4 nM,还阻断 hERG K+通道,IC50值为 0.9 nM,具有抗胆碱能和止痒作用。
T4563 Thonzylamine

neohetramine,松齐拉敏

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Thonzylamine (neohetramine) 是可口服的H1组胺受体拮抗剂,具有抗组胺和抗过敏特性,可用于鼻充血、过敏性结膜炎和其他过敏性疾病的研究。
T2392 Nafamostat mesylate

甲磺酸萘莫司他,FUT-175

Apoptosis; Serine/threonin kinase; SARS-CoV; Serine Protease Apoptosis; Cell Cycle/Checkpoint; Metabolism; Microbiology/Virology; Proteases/Proteasome
Nafamostat mesylate (FUT-175) 是一种广谱丝氨酸蛋白酶抑制剂,血管舒缓素抑制剂,能抑制血液凝固。它通过降低颗粒酶活性和 CTL 细胞溶解抑制T 细胞自身反应活性,可抑制SARS-CoV-2 的激活。它还是潜在的补体抑制剂。
T10437 AZD8848

TLR Immunology/Inflammation
AZD8848 is a selective antedrug agonist of toll-like receptor 7 (TLR7). It is developed for the research of asthma and allergic rhinitis.
T69737 SCH-79687

SCH-79687 is a histamine antagonist selective for the H3 subtype. This H3 antagonist may play a role in allergic rhinitis.
T20630 M 12325

Lasamide,M12325,M-12325

M 12325 is used in the production of furosemide; rhinitis and occupational asthma were observed in workers from a lasamide production line.
T21112 Triprolidine hydrochloride

295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil

Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.
T29951 Ambicromil

Ambicromil is used for allergic rhinitis.
T69025 Ipratropium Free Base

Ipratropium Free Base is a muscarinic antagonist structurally related to ATROPINE but often considered safer and more effective for inhalation use. It is used for various bronchial disorders, in rhinitis, and as an antiarrhythmic.
T37386 Dihydro Montelukast

Dihydro montelukast is a potential impurity found in commercial montelukast preparations. Montelukast (sodium salt) is a potent and selective cysteinyl leukotriene 1 (CysLT1) receptor antagonist. Formulations containing montelukast are used for the treatment of asthma as well as for the symptoms associated with allergic rhinitis.
T27556 HSR-609

HSR609,FY609,FY-609,FY 609

HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.
T0785L Dexchlorpheniramine free base

Polaramine,Dexchlorpheniramine Maleate,Mylaramine

Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.
T27445 GSK-1004723

GSK 1004723

GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.
T73789 5(S)-HETE

5(S)-HETE 是存在于血液中的内源代谢物,可用于研究风湿性关节炎,鼻炎和哮喘。
T21247 Carbinoxamine

Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine

Carbinoxamine, an anticholinergic and antihistamine agent, is used for hay fever, angioedema, vasomotor rhinitis, mild urticaria, dermatographism and allergic conjunctivitis. It is a histamine antagonist, specifically an H1-antagonist.
T16476 PF-03654746

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。
T60514 Triprolidine

Triprolidine 是一种口服活性的组胺H1受体拮抗剂,可用于过敏性鼻炎的研究 。Triprolidine 具有脊髓运动和知觉阻止的作用。
T26770 Bencycloquidium Bromide

BCQB

Bencycloquidium Bromide is a muscarinic M3 antagonist. Bencycloquidium bromide inhibits nasal hypersecretion in a rat model of allergic rhinitis. Bencycloquidium Bromide showed high affinity toward the M(3) receptor in Chinese hamster ovary (CHO) cells (M
T62604 Flunisolide hemihydrate

Flunisolide hemihydrate 是一种皮质类固醇,是一种口服具有活力的糖皮质激素受体 (Glucocorticoid receptor) 激活剂,具有抗炎作用。Flunisolide hemihydrate 能够诱导嗜酸性粒细胞凋亡 (apoptosis),能够用于研究哮喘或鼻炎、炎症。
T62654 Fluocortin butyl ester

Fluocortin butyl ester 是一种发达的皮质类固醇化合物,局部使用时无法检测到全身性的皮质类固醇活性。Fluocortin butyl ester 似乎是一种有效的、耐受性良好的局部类固醇,能够用于常年性鼻炎的研究。
T74646 PM-81I

PM-81I为一种高效STAT6抑制剂(针对SH2结构域),可显著减少STAT6的磷酸化水平。适用于研究过敏性肺病、过敏性鼻炎、慢性阻塞性肺病或癌症。

化合物

Cromoglicic acid
Cat.No: T8239
Synonym:
Target: Others
Azelastine
Cat.No: T0211
Synonym: Azelastina,Astelin,Azelastinum,氮卓斯汀
Target: SARS-CoV, Histamine Receptor
Fluticasone furoate
Cat.No: T21404
Synonym: Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate
Target: Glucocorticoid Receptor
Emedastine
Cat.No: T3979
Synonym: LY188695,依美斯汀,Emadine
Target: Histamine Receptor
Mizolastine
Cat.No: T0118
Synonym: SL 850324,咪唑司汀,咪唑斯汀
Target: Histamine Receptor
Rupatadine Fumarate
Cat.No: T6242
Synonym: 富马酸卢帕他定,Rinialer,Rupafin,Alergoliber
Target: PAFR, Autophagy, Histamine Receptor
R112
Cat.No: T3185
Synonym: (E)-Elafibranor
Target: Syk
Triprolidine hydrochloride monohydrate
Cat.No: T1030
Synonym: 盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride
Target: Histamine Receptor
Diphenylpyraline hydrochloride
Cat.No: T0059
Synonym: 盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride
Target: Histamine Receptor
Azelastine hydrochloride
Cat.No: T0211L
Synonym: Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin
Target: SARS-CoV, Histamine Receptor
Tripelennamine hydrochloride
Cat.No: T1269
Synonym: Pyribenzamine hydrochloride,去敏灵,Tripelennamine HCl,Pyribenzamine HCl,盐酸曲吡那敏
Target: Histamine Receptor
Setipiprant
Cat.No: T3520
Synonym: KYTH-105,塞替匹仑,ACT-129968
Target: GPR, Prostaglandin Receptor
Ebastine
Cat.No: T2335
Synonym: Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305
Target: Histamine Receptor
Fluticasone (propionate)
Cat.No: T0188
Synonym: 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate
Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite
Brompheniramine maleate
Cat.No: T0205
Synonym: Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane
Target: 5-HT Receptor, Histamine Receptor
Cetirizine dihydrochloride
Cat.No: T0089
Synonym: 盐酸西替利嗪,P071,UCB P071,Cetirizine DiHCl
Target: Histamine Receptor
Dimethindene maleate
Cat.No: T21472
Synonym: 马来酸二甲茚定,UNII-6LL60J9E0O,SU 6518,SU-6518
Target: Histamine Receptor
SB-705498
Cat.No: T6660
Synonym:
Target: TRP/TRPV Channel
Chlorpheniramine maleate
Cat.No: T1553
Synonym: 马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate
Target: Histamine Receptor
Mometasone furoate
Cat.No: T1531
Synonym: 糠酸莫美他松,糠酸莫米松,Sch32088
Target: Glucocorticoid Receptor
Ramatroban
Cat.No: T2396
Synonym: BAY u3405,雷马曲班
Target: GPR, Prostaglandin Receptor, PPAR
Levocetirizine Dihydrochloride
Cat.No: T22354
Synonym: Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride
Target: Histamine Receptor
Loratadine
Cat.No: T1097
Synonym: 氯雷他定,SCH 29851,Loratidine
Target: Influenza Virus, Histamine Receptor
PF-03654764
Cat.No: T61213
Synonym:
Target: Histamine Receptor
(2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid
Cat.No: T77601
Synonym:
Target: GPR
Pascolizumab
Cat.No: T77426
Synonym: SB-240683
Target: IL Receptor
Fexofenadine hydrochloride
Cat.No: T1470
Synonym: Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,盐酸非索非那定,Telfast,Fexofenadine HCl,Allegra,MDL 16455A
Target: Histamine Receptor
Ipratropium bromide monohydrate
Cat.No: T0098
Synonym: Ipratropium bromide hydrate,溴化异丙托品单水合物
Target: AChR
Trans-Tranilast
Cat.No: T2270
Synonym: Tranilast trans-,反式-曲尼司特,反-曲尼司特
Target: RAAS
Astemizole
Cat.No: T1278
Synonym: Laridal,Histaminos,Paralergin,阿司咪唑
Target: Potassium Channel, Histamine Receptor
Thonzylamine
Cat.No: T4563
Synonym: neohetramine,松齐拉敏
Target: Histamine Receptor
Nafamostat mesylate
Cat.No: T2392
Synonym: 甲磺酸萘莫司他,FUT-175
Target: Apoptosis, Serine/threonin kinase, SARS-CoV, Serine Protease
AZD8848
Cat.No: T10437
Synonym:
Target: TLR
SCH-79687
Cat.No: T69737
Synonym:
Target:
M 12325
Cat.No: T20630
Synonym: Lasamide,M12325,M-12325
Target:
Triprolidine hydrochloride
Cat.No: T21112
Synonym: 295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil
Target:
Ambicromil
Cat.No: T29951
Synonym:
Target:
Ipratropium Free Base
Cat.No: T69025
Synonym:
Target:
Dihydro Montelukast
Cat.No: T37386
Synonym:
Target:
HSR-609
Cat.No: T27556
Synonym: HSR609,FY609,FY-609,FY 609
Target:
Dexchlorpheniramine free base
Cat.No: T0785L
Synonym: Polaramine,Dexchlorpheniramine Maleate,Mylaramine
Target:
GSK-1004723
Cat.No: T27445
Synonym: GSK 1004723
Target:
5(S)-HETE
Cat.No: T73789
Synonym:
Target:
Carbinoxamine
Cat.No: T21247
Synonym: Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine
Target:
PF-03654746
Cat.No: T16476
Synonym:
Target: Histamine Receptor
Triprolidine
Cat.No: T60514
Synonym:
Target:
Bencycloquidium Bromide
Cat.No: T26770
Synonym: BCQB
Target:
Flunisolide hemihydrate
Cat.No: T62604
Synonym:
Target:
Fluocortin butyl ester
Cat.No: T62654
Synonym:
Target:
PM-81I
Cat.No: T74646
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S0878 Prunetin

樱黄素,Prunusetin

ERK; Dehydrogenase; NF-κB MAPK; Metabolism; NF-κB
Prunetin (Prunusetin) 是一种O-甲基化异黄酮,具有抗炎的作用。它是人醛脱氢酶的有效抑制剂。
T0861 Tylosin tartrate

酒石酸泰洛星,酒石酸泰乐菌素

Antibacterial; Antibiotic Microbiology/Virology
Tylosin tartrate 是一种大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高效的抗菌活性。它作为饲料添加剂可促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
T1003 Tylosin

Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine

Antibacterial; Antibiotic Microbiology/Virology
Tylosin (Tylosine) 是一种兽医用大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高抗菌活性。它是饲料添加剂用于促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
T4038 Ectoine

THP(B),L-Ectoine,四氢甲基嘧啶羧酸

Others; Antibacterial Microbiology/Virology; Others
Ectoine (L-Ectoine) 是生活在极其恶劣环境中的细菌所产生的氨基酸衍生物,是一种天然的细胞保护剂。它具有良好的安全性,可研究过敏性鼻炎。它用作渗透调节相容性溶质,可增加皮肤表面的水合作用并稳定脂质层,常用于皮肤护理。

天然产物

Prunetin
Cat.No: T4S0878
Synonym: 樱黄素,Prunusetin
Target: ERK, Dehydrogenase, NF-κB
Tylosin tartrate
Cat.No: T0861
Synonym: 酒石酸泰洛星,酒石酸泰乐菌素
Target: Antibacterial, Antibiotic
Tylosin
Cat.No: T1003
Synonym: Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine
Target: Antibacterial, Antibiotic
Ectoine
Cat.No: T4038
Synonym: THP(B),L-Ectoine,四氢甲基嘧啶羧酸
Target: Others, Antibacterial
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