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329

抑制剂 & 化合物

119

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Cat. No. Product Name Target Signaling Pathways
T22269 Benzyldodecyldimethylammonium Chloride Dihydrate

Antibacterial Microbiology/Virology
Benzyldodecyldimethylammonium chloride dihydrate 可以用作杀虫试剂,可以靶向耐药性细菌,如耐甲氧西林金黄色葡萄球菌、耐多药铜绿假单胞菌等,且具有浓度依赖性。
T36683 Vedaprofen

Quadrisol,PM 150,维达洛芬,CERM 10202

COX; Antibacterial; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Vedaprofen (PM 150) 抑制 COX-1 并通过抗炎活性减少前列腺素 H2 的合成。 Vedaprofen 是一种大肠杆菌滑动钳抑制剂,IC50 为 222 μM,Ki 为 131 μM。
T14864 Caracemide

NSC-253272,卡醋胺

Others; DNA/RNA Synthesis; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Caracemide (NSC-253272) 抑制大肠杆菌的核糖核苷酸还原酶。 Caracemide 可用于抗癌研究。
T9508 MONOCAPRYLIN

Sefsol 318,Glyceryl monocaprylate,辛酸甘油酯

Antibacterial Microbiology/Virology
Monocaprylin (Sefsol 318) 是一种辛酸甘油单辛酸酯,有出色的抗菌活性,可抑制多种食源性致病和腐败微生物,有用于替代食品防腐剂的研究潜力。
T19794 Temafloxacin

替马沙星,Omniflox

Antibiotic Microbiology/Virology
Temafloxacin (Omniflox) 是一种喹诺酮类广谱抗菌剂,对革兰氏阳性菌、革兰氏阴性菌和厌氧菌均有效。
T33828 O-Succinylhomoserine

O-琥珀酰-L-高丝氨酸,O-Succinyl-L-homoserine

Others Others
O-Succinylhomoserine (O-Succinyl-L-homoserine) 是大肠杆菌合成胱硫醚的中间体。
T82462 Enterotoxin STp (E. coli)

Enterotoxin STp (E. coli), 热稳定肠毒素,适用于疫苗研究领域。
T1389 Dyclonine hydrochloride

盐酸达克罗宁,Dyclocaine hydrochloride,Dyclonine HCl

Sodium Channel; Antibacterial; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Dyclonine hydrochloride (Dyclonine HCl) 是润喉片的有效成分,具有显著的杀菌和杀真菌作用。
T0909L Nalidixic acid sodium salt

萘啶酮酸,萘啶酮酸钠,Baktogram,Sodium nalidixate

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Nalidixic acid sodium salt (Baktogram) 是一种喹诺酮类抗生素,对革兰氏阳性和革兰氏阴性细菌均有效。它在较低浓度下有抑菌作用,在较高浓度下有杀菌作用。它抑制 DNA 促旋酶和拓扑异构酶IV 的亚基,并可逆地阻止易感细菌中的 DNA 复制。
T1224 Cefuroxime sodium

Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin

Antibacterial; Antibiotic Microbiology/Virology
Cefuroxime sodium (Cefuroxime sodium salt) 是一种具有口服活性的头孢菌素抗生素,增加了对 β-内酰胺酶的稳定性。
T0788L Spectinomycin dihydrochloride pentahydrate

盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride pentahydrate (Spectogard) 是一种广谱氨基环糊精抗生素,可以抑制多种革兰氏阳性和革兰氏阴性生物的生长。
T6179 Moxalactam sodium salt

Latamoxef sodium,6059 S,拉氧头孢钠,Moxalactam Disodium,LY-127935,Antibiotic 6059S,Shiomarin,FestamoxinLy

Antibacterial; Antibiotic Microbiology/Virology
Moxalactam sodium salt (LY-127935) 是一种抗生素, 对大肠杆菌和绿脓杆菌有作用。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。
T39912 5'-O-(4,4'-Dimethoxytrityl)-2'-deoxyuridine

5'-O-DMT-dU,保护-2'-脱氧尿苷

Others Others
5'-O-(4,4'-Dimethoxytrityl)-2'-deoxyuridine (5'-O-DMT-dU) 是大肠杆菌 dUTP 核苷酸水解酶的竞争性抑制剂,Ki 高于 1000 μM。它通过合成核苷亚磷酰胺嵌段用于机器辅助的 DNA 合成。
T22220 Methyl picolinate

2-吡啶甲酸甲酯,Methyl pyridine-2-carboxylate,2-Pyridinecarboxylic acid methyl ester,2-Carbomethoxypyridine

Others Others
Methyl picolinate (Methyl picolinate) 用作医药中间体。
T12092 Monacolin J

Antibiotic MB 530A,Lovastatin diol lactone,辛伐他汀内酯二醇

HMG-CoA Reductase; Autophagy Autophagy; Metabolism
Monacolin J (Antibiotic MB 530A) 是一种胆固醇生物合成抑制剂,抑制 HMG-CoA 还原酶的活性。
T64334 Glycolithocholic acid, sodium salt

Others Others
Glycolithocholic acid, sodium salt 是 Glycolithocholic acid 的钠盐。Glycolithocholic acid 是一种甘氨酸结合的次级胆汁酸。Glycolithocholic acid 可用于诊断溃疡性结肠炎 (UC),非酒精性脂肪性肝炎 (NASH0) 和原发性硬化性胆管炎 (PSC)。
T77426 Pascolizumab

SB-240683

IL Receptor Immunology/Inflammation
Pascolizumab (SB-240683) 是一种人源化抗 IL-4 单克隆抗体。Pascolizumab 具有哮喘作用,可用于研究过敏性鼻炎。
TP1856 Colivelin

Beta Amyloid; STAT JAK/STAT signaling; Neuroscience; Stem Cells
Colivelin 是一种神经保护肽和 STAT3 的激活剂,是一种合成的杂合肽,可增强 humanin (HN) 的神经保护作用。它通过激活 STAT3 在体外抑制神经元死亡,具有潜力用于阿尔茨海默病和缺血性脑损伤的相关研究。
T2489 Ricolinostat

ACY-1215,Rocilinostat

Apoptosis; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Ricolinostat (Rocilinostat) 是一种选择性HDAC6抑制剂,IC50为 5 nM。它还抑制HDAC1,HDAC2和HDAC3,IC50分别为 58,48 和 51 nM。
T66390 4-(4-Amino-3-fluorophenoxy)-N-methylpicolinamide

4-(4-Amino-3-fluorophenoxy)-N-methylpicolinamide 是芳香谜,是是抗肿瘤药物瑞非尼的代谢产物。
T4575 Chromium picolinate

DNA; p38 MAPK DNA Damage/DNA Repair; MAPK
Chromium picolinate 具有降低胰岛素抵抗的作用,对 2 型糖尿病具有潜在的研究价值。
T74465 Colibactin

Colibactin 是一种复杂的次级代谢产物,由一些具有遗传毒性的肠道大肠杆菌菌株产生。Colibactin 具有研究结直肠癌的潜力。
T11429 Glycolic acid oxidase inhibitor 1

Others Others
Glycolic acid oxidase inhibitor 1 is a glycolate oxidase inhibitor.
T64672 Colivelin TFA

Colivelin (sequence SALLRSIPAPAGASRLLLLTGEIDLP) is composed of activity-dependent neurotrophic factor (ADNF) C-terminally fused to AGA-(C8R)HNG17, a potent HN derivative. It works as a neuroprotective peptide and activator of STAT3. Colivelin-induced neuroprotection has been confirmed to occur via two neuroprotective pathways: one mediated by Ca2+/calmodulin-dependent protein kinase IV, triggered by ADNF, and one mediated by signal transducer and activator of transcription 3, triggered by HN. Co...
T78551 Glycolithocholic acid 3-sulfate disodium

Glycolithocholate sulfate disodium,SLCG disodium,Sulfolithocholylglycine disodium

Glycolithocholic acid 3-sulfate (disodium) 是抑制HIV-1复制的化合物,同时它也被用于HIV感染和胆囊疾病的研究。
T31858 Foscolic acid

PDLA,Phoscolic acid

Foscolic acid is a bioactive chemical.
T64568 4,6-Dichloro-N-methylpicolinamide

4,6-Dichloro-N-methylpicolinamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64568,CAS号为 1379324-09-0。
T31518 Dipinacoline glutamate

L-Glutamic acid dipinacoline ester,DiPG

Dipinacoline glutamate is a bioactive chemical.
T126341 Sambacolignoside

Sambacolignoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126341,CAS号为 114449-12-6。
T67100 N-Methyl-4-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenoxy)picolinamide

N-Methyl-4-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenoxy)picolinamide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67100。
T64459 4-(4-Formamidophenoxy)-N-methylpicolinamide

4-(4-Formamidophenoxy)-N-methylpicolinamide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64459。
T124339 Caleurticolide 2-methylacrylate

Caleurticolide 2-methylacrylate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124339,CAS号为 71652-12-5。
T61154 Colistin adjuvant-2

Colistin adjuvant-2 is a compound that acts as a potentiation agent for colistin, effectively enhancing its activity against Gram-negative bacteria [1].
T62125 Colistin adjuvant-1

Colistin adjuvant-1 是一种粘菌素佐剂 (colistin adjuvant),对革兰氏阴性细菌具有增强的粘菌素增强活性。Colistin adjuvant-1 对 NF-κB 表现出抑制作用 (IC50: 0.209 μM)。
TP1278 Colivelin TFA (867021-83-8 free base)

Colivelin TFA

Colivelin (TFA) is a hybrid peptide composed of ADNF and AGA-(C8R)HNG17, a potent Humanin (HN) derivative.
T73798 Colistin

Colistin (Polymyxin E) 是一种具有口服活性的多肽类抗生素。它对包括多重耐药铜绿假单胞菌、鲍曼不动杆菌和肺炎克雷伯菌在内的多种革兰氏阴性杆菌表现出良好的抑制作用。此外,Colistin 与肾毒性相关,常用于研究革兰氏阴性菌感染。
T65881 Methyl 4-chloropicolinate

Methyl 4-chloropicolinate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65881,CAS号为 24484-93-3。
T125288 Ilicicolin B

Ilicicolin B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125288,CAS号为 22581-07-3。
T126034 4,15-Isoatriplicolide methylacrylate

4,15-Isoatriplicolide methylacrylate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126034。
T67664 4-Chloro-N,N-dimethylpicolinamide

4-Chloro-N,N-dimethylpicolinamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67664,CAS号为 114780-06-2。
T64454 4-Bromo-N-methylpicolinamide

4-Bromo-N-methylpicolinamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64454,CAS号为 1209459-88-0。
T67103 2-Bromo-N-(4-bromo-2-picolinoylphenyl)acetamide

2-Bromo-N-(4-bromo-2-picolinoylphenyl)acetamide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67103。
T25269 Colistin A

Polymixin E1,Polymyxin E1,Colistin IV

Colistin A is an antibiotic generated by certain strains of the bacteria Paenibacillus polymyxa. Colistin is a mixture of the cyclic polypeptides colistin A and B and belongs to the class of polypeptide antibiotics known as polymyxins. Colistin is effecti
T20580 Picolinamidoxime

RA7,RA-7,RA 7,Picolinamide oxime

Picolinamidoxime is a biochemical substance.
T124005 Gingerglycolipid B

Gingerglycolipid B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124005,CAS号为 88168-90-5。
T125289 Ilicicolin A

Ilicicolin A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125289,CAS号为 22581-06-2。
T66513 4-Chloro-N-methylpicolinamide

4-Chloro-N-methylpicolinamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66513,CAS号为 220000-87-3。
T81723 N-(2-Hydroxyphenyl)picolinamide

N-(2-Hydroxyphenyl)picolinamide是一种用于生化反应研究的活性分子。
T31962 Glycolic acid, (5-nitrofurfurylidene)hydrazide

Glycolic acid, (5-nitrofurfurylidene)hydrazide is a bioactive chemical.

化合物

Benzyldodecyldimethylammonium Chloride Dihydrate
Cat.No: T22269
Synonym:
Target: Antibacterial
Vedaprofen
Cat.No: T36683
Synonym: Quadrisol,PM 150,维达洛芬,CERM 10202
Target: COX, Antibacterial, Prostaglandin Receptor
Caracemide
Cat.No: T14864
Synonym: NSC-253272,卡醋胺
Target: Others, DNA/RNA Synthesis, Antibacterial
MONOCAPRYLIN
Cat.No: T9508
Synonym: Sefsol 318,Glyceryl monocaprylate,辛酸甘油酯
Target: Antibacterial
Temafloxacin
Cat.No: T19794
Synonym: 替马沙星,Omniflox
Target: Antibiotic
O-Succinylhomoserine
Cat.No: T33828
Synonym: O-琥珀酰-L-高丝氨酸,O-Succinyl-L-homoserine
Target: Others
Enterotoxin STp (E. coli)
Cat.No: T82462
Synonym:
Target:
Dyclonine hydrochloride
Cat.No: T1389
Synonym: 盐酸达克罗宁,Dyclocaine hydrochloride,Dyclonine HCl
Target: Sodium Channel, Antibacterial, Antifungal
Nalidixic acid sodium salt
Cat.No: T0909L
Synonym: 萘啶酮酸,萘啶酮酸钠,Baktogram,Sodium nalidixate
Target: Topoisomerase, Antibacterial, Antibiotic
Cefuroxime sodium
Cat.No: T1224
Synonym: Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin
Target: Antibacterial, Antibiotic
Spectinomycin dihydrochloride pentahydrate
Cat.No: T0788L
Synonym: 盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
Moxalactam sodium salt
Cat.No: T6179
Synonym: Latamoxef sodium,6059 S,拉氧头孢钠,Moxalactam Disodium,LY-127935,Antibiotic 6059S,Shiomarin,FestamoxinLy
Target: Antibacterial, Antibiotic
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
5'-O-(4,4'-Dimethoxytrityl)-2'-deoxyuridine
Cat.No: T39912
Synonym: 5'-O-DMT-dU,保护-2'-脱氧尿苷
Target: Others
Methyl picolinate
Cat.No: T22220
Synonym: 2-吡啶甲酸甲酯,Methyl pyridine-2-carboxylate,2-Pyridinecarboxylic acid methyl ester,2-Carbomethoxypyridine
Target: Others
Monacolin J
Cat.No: T12092
Synonym: Antibiotic MB 530A,Lovastatin diol lactone,辛伐他汀内酯二醇
Target: HMG-CoA Reductase, Autophagy
Glycolithocholic acid, sodium salt
Cat.No: T64334
Synonym:
Target: Others
Pascolizumab
Cat.No: T77426
Synonym: SB-240683
Target: IL Receptor
Colivelin
Cat.No: TP1856
Synonym:
Target: Beta Amyloid, STAT
Ricolinostat
Cat.No: T2489
Synonym: ACY-1215,Rocilinostat
Target: Apoptosis, HDAC
4-(4-Amino-3-fluorophenoxy)-N-methylpicolinamide
Cat.No: T66390
Synonym:
Target:
Chromium picolinate
Cat.No: T4575
Synonym:
Target: DNA, p38 MAPK
Colibactin
Cat.No: T74465
Synonym:
Target:
Glycolic acid oxidase inhibitor 1
Cat.No: T11429
Synonym:
Target: Others
Colivelin TFA
Cat.No: T64672
Synonym:
Target:
Glycolithocholic acid 3-sulfate disodium
Cat.No: T78551
Synonym: Glycolithocholate sulfate disodium,SLCG disodium,Sulfolithocholylglycine disodium
Target:
Foscolic acid
Cat.No: T31858
Synonym: PDLA,Phoscolic acid
Target:
4,6-Dichloro-N-methylpicolinamide
Cat.No: T64568
Synonym:
Target:
Dipinacoline glutamate
Cat.No: T31518
Synonym: L-Glutamic acid dipinacoline ester,DiPG
Target:
Sambacolignoside
Cat.No: T126341
Synonym:
Target:
N-Methyl-4-(4-(3-(3-(trifluoromethyl)phenyl)ureido)phenoxy)picolinamide
Cat.No: T67100
Synonym:
Target:
4-(4-Formamidophenoxy)-N-methylpicolinamide
Cat.No: T64459
Synonym:
Target:
Caleurticolide 2-methylacrylate
Cat.No: T124339
Synonym:
Target:
Colistin adjuvant-2
Cat.No: T61154
Synonym:
Target:
Colistin adjuvant-1
Cat.No: T62125
Synonym:
Target:
Colivelin TFA (867021-83-8 free base)
Cat.No: TP1278
Synonym: Colivelin TFA
Target:
Colistin
Cat.No: T73798
Synonym:
Target:
Methyl 4-chloropicolinate
Cat.No: T65881
Synonym:
Target:
Ilicicolin B
Cat.No: T125288
Synonym:
Target:
4,15-Isoatriplicolide methylacrylate
Cat.No: T126034
Synonym:
Target:
4-Chloro-N,N-dimethylpicolinamide
Cat.No: T67664
Synonym:
Target:
4-Bromo-N-methylpicolinamide
Cat.No: T64454
Synonym:
Target:
2-Bromo-N-(4-bromo-2-picolinoylphenyl)acetamide
Cat.No: T67103
Synonym:
Target:
Colistin A
Cat.No: T25269
Synonym: Polymixin E1,Polymyxin E1,Colistin IV
Target:
Picolinamidoxime
Cat.No: T20580
Synonym: RA7,RA-7,RA 7,Picolinamide oxime
Target:
Gingerglycolipid B
Cat.No: T124005
Synonym:
Target:
Ilicicolin A
Cat.No: T125289
Synonym:
Target:
4-Chloro-N-methylpicolinamide
Cat.No: T66513
Synonym:
Target:
N-(2-Hydroxyphenyl)picolinamide
Cat.No: T81723
Synonym:
Target:
Glycolic acid, (5-nitrofurfurylidene)hydrazide
Cat.No: T31962
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T41078 Lipopolysaccharides, Escherichiacoli

Lipopolysaccharide, E. coli O111:B4

Others Others
Lipopolysaccharides, Escherichiacoli (E. coli O111:B4)是革兰阴性菌外膜的大分子成分,由脂质a、寡糖核心和o -特异性多糖(O-antigen) 3个区域组成。
T2904 Sclareolide

香紫苏内酯,Norambreinolide

Others; Antibacterial Microbiology/Virology; Others
Sclareolide (Norambreinolide) 是一种从Salvia sclarea 的花中分离得到的天然产物,具有抗菌和细胞毒性作用。
T1313 Nitrofurantoin

Furadantine,呋喃妥因,Macrodantin,Furadonine

Antibacterial; Antibiotic Microbiology/Virology
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。
T0909 Nalidixic acid

萘啶酸,NSC-82174

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Nalidixic acid (NSC-82174) 是一种喹诺酮类抗生素,对革兰氏阳性和革兰氏阴性细菌有效。它在较低浓度下有抑菌作用,而在较高浓度下有杀菌作用。它抑制 DNA 促旋酶和拓扑异构酶 IV 的亚基,并可逆地阻止易感细菌中的 DNA 复制。
T1079 Metronidazole

Flagyl,Metronidazol,甲硝唑,Anagiardil

Apoptosis; NADPH; Hydrogenase; Antibacterial; Antibiotic; Parasite; Antifection Apoptosis; Metabolism; Microbiology/Virology
Metronidazole (Metronidazol) 是一种合成的硝基咪唑衍生物,具有抗原生动物和抗菌活性。
T0788 Spectinomycin dihydrochloride

淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride (Actinospectacin) 是一种能与细菌核糖体的30S 亚基结合,干扰蛋白质合成的抗生素。
T1100 Polymyxin B Sulfate

Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX

Antibacterial; Antibiotic Microbiology/Virology
Polymyxin B Sulfate (Poly-RX) 是一个阳离子型表面活性剂抗生素剂,能够提高细胞膜的渗透性。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
T3501 Colistimethate Sodium

Colistin-1,3,5,9-tetramethanesulfonic A acid,多粘菌素E甲磺酸钠

Others Others
Colistin-1,3,5,9-tetramethanesulfonic A acid 用于治疗选择有限的患者因选定的需氧革兰氏阴性病原体引起的严重感染。
T19458 N-Hydroxypipecolic acid

1-Hydroxy-2-piperidinecarboxylic acid,NHP

Others Others
N-Hydroxypipecolic acid (NHP) 是植物代谢产物和系统性获得性抗性调节剂,可与免疫信号水杨酸协调建立系统性获得性抗性,诱导系统获得性耐药对细菌和卵菌感染。它在植物叶片中系统地积累,以应对病原菌的侵袭。
T68953 Arecoline

Reactive Oxygen Species; AChR Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Arecoline 是一种来自棕榈科植物槟榔的天然生物碱,是有效的烟碱和毒蕈碱乙酰胆碱受体的部分激动剂。Arecoline 具有抗焦虑和抗寄生虫活性,可诱导氧化应激,可用于研究阿尔茨海默病和老年性痴呆。
T1245 Colistin sulfate

Colistin sulfate (1066-17-7 free base),Polymixin E Sulfate,Polymyxin E Sulfate,硫酸粘杆菌素

Cell wall; Antibacterial; Antibiotic; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology
Colistin sulfate (Colistin sulfate (1066-17-7 free base)) 是抑制革兰氏阴性细菌的一种多肽抗生素,与革兰氏阴性细菌的外细胞膜中的脂多糖和磷脂结合起作用。
T0136 Citicoline

CDP-Choline,Citicholine,尼古林,cytidine 5'-diphosphocholine,cytidine diphosphate-choline

Apoptosis; Dopamine Receptor; Endogenous Metabolite Apoptosis; GPCR/G Protein; Metabolism; Neuroscience
Citicoline (CDP-Choline) 是一种合成细胞膜组分磷脂酰胆碱的中间体,有神经保护作用。
TN1833 Karacoline

NF-κB NF-κB
Karacoline 是发现于植物Aconitum kusnezoffii 中的一种二萜生物碱,通过 NF-κB 信号通路,抑制椎间盘退变中细胞外基质的降解。
TN1405 Arnicolide D

山金车内酯 D,山金车内酯D

Akt; Caspase; PI3K; STAT; mTOR Apoptosis; Cytoskeletal Signaling; JAK/STAT signaling; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Arnicolide D 是从石胡荽中分离出的一种倍半萜内酯,以浓度和时间依赖性方式抑制鼻咽癌细胞活力。它调节细胞周期,激活 caspase 信号通路并抑制 PI3K/AKT/mTOR 和 STAT3 信号通路。
T4819 Pipecolic acid

DL-哌啶甲酸,(±)-Piperidine-2-carboxylic acid,呢可酸,2-Piperidinecarboxylic acid,Pipecolinic acid,Homoproline

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
Pipecolic acid (2-Piperidinecarboxylic acid) 是一种赖氨酸代谢物,是许多微生物次级代谢物的重要前体,可用作吡哆醇依赖性癫痫的诊断标记。
T5986 3-Hydroxypicolinic acid

3-羟基-2-吡啶甲酸,Picolinic acid, 3-hydroxy- (6CI,7CI,8CI),2-Carboxy-3-hydroxypyridine

Endogenous Metabolite Metabolism
3-Hydroxypicolinic acid (Picolinic acid, 3-hydroxy- (6CI,7CI,8CI)) 是一种内源性代谢物,属于吡啶甲酸的衍生物。
T13634 D-Pipecolinic acid

(R)-Piperidine-2-carboxylic acid

Endogenous Metabolite Metabolism
D-Pipecolinic acid ((R)-Piperidine-2-carboxylic acid) 是一种存在于人体生物液体中的正常人体代谢物。
T31964 Glycolithocholic acid

Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine

Others Others
Glycolithocholic acid (Lithocholic acid glycine conjugate) 属于内源性代谢产物,是甘氨酸结合的次级胆汁酸。它可用于诊断非酒精性脂肪性肝炎,溃疡性结肠炎和原发性硬化性胆管炎。
T5985 Glycolic acid

Tyrosinase; Endogenous Metabolite Metabolism; Proteases/Proteasome
Glycolic acid 是一种酪氨酸酶抑制剂,可以抑制黑色素的形成,从而减淡皮肤的颜色。
T21518 Colistin methanesulfonate sodium salt

粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)

Cell wall; Antibacterial Immunology/Inflammation; Microbiology/Virology
Colistin methanesulfonate sodium salt (Colistimethate Sodium) 是一种来自 Bacillus colistinus 的环状多肽抗生素,由多粘菌素 E1 和 E2 组成。
T4762 L-Pipecolic acid

L-哌啶酸,L-Homoproline,H-HoPro-OH

Endogenous Metabolite Metabolism
L-Pipecolic acid (L-Homoproline) 是赖氨酸的分解产物,它能在患有常染色体遗传性疾病的婴儿体液中积累,比如新生儿肾上腺机能障碍, Zellweger 综合征等。
T14304 Aphidicolin

Others Others
Aphidicolin is a potent inhibitor of cellular deoxyribonucleic acid synthesis and inhibits the growth of herpes simplex virus[2]. Aphidicolin is an inhibitor of DNA polymerase α and δ, prevents mitotic cell division by interfering with the activity of DNA
T5805 Guvacoline hydrochloride

1,2,5,6-四氢吡啶-3-甲酸甲酯盐酸盐,Norarecoline hydrochloride,去甲槟榔碱

AChR Neuroscience
Guvacoline hydrochloride (Norarecoline hydrochloride) 是从三药槟榔中发现的一种吡啶生物碱,可作为心房和回肠的毒蕈碱激动剂。
T6942 Picolinamide

2-Pyridinecarboxamide,2-Carbamoylpyridine,2-吡啶甲酰胺,2-Picolinamide,Picolinoylamide

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Picolinamide (Picolinoylamide) 被发现是大鼠胰岛细胞核聚 (ADP-核糖) 合成酶的强抑制剂。
T2198 Arecoline hydrobromide

Arecoline HBr,氢溴酸槟榔碱,Arecoline bromide

AChR Neuroscience
Arecoline hydrobromide (Arecoline HBr) 是从槟榔中得到的一种生物碱,具有刺激、警觉、抗焦虑和抗寄生虫作用。它是烟碱和毒蕈碱乙酰胆碱受体的部分激动剂,可诱导氧化应激。
TN4145 Glucoliquiritin

Others Others
Glucoliquiritin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4145,CAS号为 93446-18-5。
T19457 N-Hydroxypipecolic acid potassium

NHP potassium,1-Hydroxy-2-piperidinecarboxylic acid potassium

Others Others
N-Hydroxypipecolic acid potassium is a metabolite of plant and a systemic acquired resistance (SAR) regulator.
TN5322 Minisecolide C

Minisecolide C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5322,CAS号为 1967030-77-8。
TN4144 Glucolimnanthin

Others Others
Glucolimnanthin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4144,CAS号为 111810-95-8。
TMA2544 Angelicolide

Others Others
Angelicolide是一种天然产物,属于伞形科当归属,其产品编号为 TMA2544,CAS号为 90826-58-7。Angelicolide可用作对照参考。
TN5323 Minisecolide D

Minisecolide D 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5323,CAS号为 1967030-78-9。
TN1404 ArnicolideC

山金车内酯C,山金车内酯 C,Arnicolide C

Others Others
Arnicolide C exhibits significant antiallergy activity.
TN2163 Rubioncolin C

NF-κB NF-κB
Rubioncolin C shows good cytotoxicity with IC50 value of 1.53 μM and NF-κB inhibitory activity with IC50 value of 2.97 μM.
T38837 Microcolin B

Microcolin B, an acylpeptide immunosuppressant, is a highly potent and biologically unique compound containing proline. It is derived from the blue-green alga Lyngbya majuscule.
T38949 Gingerglycolipid A

Gingerglycolipid A is a monoacyldigalactosyl glycerol.
T1208 Citicoline sodium

Citicoline sodium salt,CDP-choline,胞磷胆碱钠

Apoptosis; Others; Endogenous Metabolite Apoptosis; Metabolism; Others
Citicoline sodium (CDP-choline) 是一种合成细胞膜组分磷脂酰胆碱的中间体,有神经保护作用。
T73758 Glycolithocholic acid 3-sulfate

Glycolithocholic acid 3-sulfate (SLCG) 为一种胆汁酸衍生物及甘胆酸的代谢产物,具有抑制HIV-1复制的作用。该化合物在HIV感染和胆囊疾病的研究中有潜在应用价值。
T72965 Inuviscolide

Inuviscolide,一种诱导细胞凋亡(apoptosis)的化合物,能够引起人黑素瘤细胞系在G2/M期的停滞,并展现出抗肿瘤和抗炎活性。
TN3026 4-Epi-isoinuviscolide

Others Others
4-Epi-isoinuviscolide是一种天然产物,属于菊科旋覆花属,其产品编号为 TN3026,CAS号为 68832-39-3。4-Epi-isoinuviscolide可用作对照参考。
T13708 Glycol chitosan

羟乙基脱乙酰壳多糖,乙二醇壳聚糖

Antibacterial Microbiology/Virology
Glycol chitosan 是具有亲水性乙二醇支链的壳聚糖衍生物。它抑制大肠杆菌,金黄色葡萄球菌和肠炎链球菌的生长,MIC 值分别为 4 μg/mL,32 μg/m L 和 <0.5 μg/mL。它可增强 Glycine max Harosoy 63W 细胞的膜通透性和渗漏。
T19146 5,6-Dihydrouridine

Endogenous Metabolite Metabolism
5,6-Dihydrouridine 是一种修饰碱基,存在于真核生物、细菌和某些古细菌tRNA D 环的保守位置。
T4913 Maleic acid

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
Maleic Acid 是大肠杆菌和单核细胞增生李斯特菌的谷氨酸脱羧酶抑制剂。
T7565 3-Hydroxycapric acid

Endogenous Metabolite Metabolism
3-Hydroxycapric acid 是有丝分裂抑制剂。
T10941 D-Ribonolactone

D-(+)-核糖酸-1,4-内酯,D-核糖内酯

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
D-Ribonolactone 是一种大肠杆菌 β-半乳糖苷酶的抑制剂,Ki 为 26 mM。它也一种糖内酯。
T13750 L-Fucitol

L-岩藻糖醇,1-Deoxy-D-galactitol

Others Others
L-Fucitol (1-Deoxy-D-galactitol) 是一种糖醇,从肉豆蔻 (Nutmeg) 中分离得到。
TF0083 POPE

POPE 是从大肠杆菌中发现的化合物,是细胞膜的一部分,可用来研究改变细胞膜通透性。
T6S2116 Ginkgolic acid C17:1

银杏酸 C17:1,银杏酸C17:1

Phosphatase; PTEN Metabolism; PI3K/Akt/mTOR signaling
Ginkgolic acid C17:1 是分离自银杏叶中,通过诱导PTEN 和SHP-1酪氨酸磷酸酶抑制组成型和诱导型 STAT3 活化。它具有抗癌活性。
TN2281 Sinapaldehyde

trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde,TRANS-3,5-二甲氧基-4-羟基肉桂醛,芥子醛

Antibacterial Microbiology/Virology
Sinapaldehyde (trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde) 对耐甲氧西林的金黄色葡萄球菌和大肠杆菌有抗菌作用,MIC 值都为 128 μg/mL。
TN2898 Kaempferol-7,4'-dimethyl ether

3,5-Dihydroxy-4',7-dimethoxyflavone

Antioxidant; Antifection Microbiology/Virology; oxidation-reduction
Kaempferol-7,4'-dimethyl ether 是从 Zingiber phillipseae 的根茎中分离得到的,对金黄色葡萄球菌和大肠杆菌具有抗氧化活性,MIC 分别为 200 和 225 μg/ml。
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天然产物

Lipopolysaccharides, Escherichiacoli
Cat.No: T41078
Synonym: Lipopolysaccharide, E. coli O111:B4
Target: Others
Sclareolide
Cat.No: T2904
Synonym: 香紫苏内酯,Norambreinolide
Target: Others, Antibacterial
Nitrofurantoin
Cat.No: T1313
Synonym: Furadantine,呋喃妥因,Macrodantin,Furadonine
Target: Antibacterial, Antibiotic
Nalidixic acid
Cat.No: T0909
Synonym: 萘啶酸,NSC-82174
Target: Topoisomerase, Antibacterial, Antibiotic
Metronidazole
Cat.No: T1079
Synonym: Flagyl,Metronidazol,甲硝唑,Anagiardil
Target: Apoptosis, NADPH, Hydrogenase, Antibacterial, Antibiotic, Parasite, Antifection
Spectinomycin dihydrochloride
Cat.No: T0788
Synonym: 淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin
Target: ribosome, Antibacterial, Antibiotic
Polymyxin B Sulfate
Cat.No: T1100
Synonym: Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX
Target: Antibacterial, Antibiotic
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
Colistimethate Sodium
Cat.No: T3501
Synonym: Colistin-1,3,5,9-tetramethanesulfonic A acid,多粘菌素E甲磺酸钠
Target: Others
N-Hydroxypipecolic acid
Cat.No: T19458
Synonym: 1-Hydroxy-2-piperidinecarboxylic acid,NHP
Target: Others
Arecoline
Cat.No: T68953
Synonym:
Target: Reactive Oxygen Species, AChR
Colistin sulfate
Cat.No: T1245
Synonym: Colistin sulfate (1066-17-7 free base),Polymixin E Sulfate,Polymyxin E Sulfate,硫酸粘杆菌素
Target: Cell wall, Antibacterial, Antibiotic, Autophagy
Citicoline
Cat.No: T0136
Synonym: CDP-Choline,Citicholine,尼古林,cytidine 5'-diphosphocholine,cytidine diphosphate-choline
Target: Apoptosis, Dopamine Receptor, Endogenous Metabolite
Karacoline
Cat.No: TN1833
Synonym:
Target: NF-κB
Arnicolide D
Cat.No: TN1405
Synonym: 山金车内酯 D,山金车内酯D
Target: Akt, Caspase, PI3K, STAT, mTOR
Pipecolic acid
Cat.No: T4819
Synonym: DL-哌啶甲酸,(±)-Piperidine-2-carboxylic acid,呢可酸,2-Piperidinecarboxylic acid,Pipecolinic acid,Homoproline
Target: Others, Endogenous Metabolite, Antibacterial
3-Hydroxypicolinic acid
Cat.No: T5986
Synonym: 3-羟基-2-吡啶甲酸,Picolinic acid, 3-hydroxy- (6CI,7CI,8CI),2-Carboxy-3-hydroxypyridine
Target: Endogenous Metabolite
D-Pipecolinic acid
Cat.No: T13634
Synonym: (R)-Piperidine-2-carboxylic acid
Target: Endogenous Metabolite
Glycolithocholic acid
Cat.No: T31964
Synonym: Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine
Target: Others
Glycolic acid
Cat.No: T5985
Synonym:
Target: Tyrosinase, Endogenous Metabolite
Colistin methanesulfonate sodium salt
Cat.No: T21518
Synonym: 粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)
Target: Cell wall, Antibacterial
L-Pipecolic acid
Cat.No: T4762
Synonym: L-哌啶酸,L-Homoproline,H-HoPro-OH
Target: Endogenous Metabolite
Aphidicolin
Cat.No: T14304
Synonym:
Target: Others
Guvacoline hydrochloride
Cat.No: T5805
Synonym: 1,2,5,6-四氢吡啶-3-甲酸甲酯盐酸盐,Norarecoline hydrochloride,去甲槟榔碱
Target: AChR
Picolinamide
Cat.No: T6942
Synonym: 2-Pyridinecarboxamide,2-Carbamoylpyridine,2-吡啶甲酰胺,2-Picolinamide,Picolinoylamide
Target: PARP
Arecoline hydrobromide
Cat.No: T2198
Synonym: Arecoline HBr,氢溴酸槟榔碱,Arecoline bromide
Target: AChR
Glucoliquiritin
Cat.No: TN4145
Synonym:
Target: Others
N-Hydroxypipecolic acid potassium
Cat.No: T19457
Synonym: NHP potassium,1-Hydroxy-2-piperidinecarboxylic acid potassium
Target: Others
Minisecolide C
Cat.No: TN5322
Synonym:
Target:
Glucolimnanthin
Cat.No: TN4144
Synonym:
Target: Others
Angelicolide
Cat.No: TMA2544
Synonym:
Target: Others
Minisecolide D
Cat.No: TN5323
Synonym:
Target:
ArnicolideC
Cat.No: TN1404
Synonym: 山金车内酯C,山金车内酯 C,Arnicolide C
Target: Others
Rubioncolin C
Cat.No: TN2163
Synonym:
Target: NF-κB
Microcolin B
Cat.No: T38837
Synonym:
Target:
Gingerglycolipid A
Cat.No: T38949
Synonym:
Target:
Citicoline sodium
Cat.No: T1208
Synonym: Citicoline sodium salt,CDP-choline,胞磷胆碱钠
Target: Apoptosis, Others, Endogenous Metabolite
Glycolithocholic acid 3-sulfate
Cat.No: T73758
Synonym:
Target:
Inuviscolide
Cat.No: T72965
Synonym:
Target:
4-Epi-isoinuviscolide
Cat.No: TN3026
Synonym:
Target: Others
Glycol chitosan
Cat.No: T13708
Synonym: 羟乙基脱乙酰壳多糖,乙二醇壳聚糖
Target: Antibacterial
5,6-Dihydrouridine
Cat.No: T19146
Synonym:
Target: Endogenous Metabolite
Maleic acid
Cat.No: T4913
Synonym:
Target: Endogenous Metabolite, Antibacterial
3-Hydroxycapric acid
Cat.No: T7565
Synonym:
Target: Endogenous Metabolite
D-Ribonolactone
Cat.No: T10941
Synonym: D-(+)-核糖酸-1,4-内酯,D-核糖内酯
Target: Endogenous Metabolite, Antibacterial
L-Fucitol
Cat.No: T13750
Synonym: L-岩藻糖醇,1-Deoxy-D-galactitol
Target: Others
POPE
Cat.No: TF0083
Synonym:
Target:
Ginkgolic acid C17:1
Cat.No: T6S2116
Synonym: 银杏酸 C17:1,银杏酸C17:1
Target: Phosphatase, PTEN
Sinapaldehyde
Cat.No: TN2281
Synonym: trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde,TRANS-3,5-二甲氧基-4-羟基肉桂醛,芥子醛
Target: Antibacterial
Kaempferol-7,4'-dimethyl ether
Cat.No: TN2898
Synonym: 3,5-Dihydroxy-4',7-dimethoxyflavone
Target: Antioxidant, Antifection
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