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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T19609 HP-β-CD

羟丙基-β-环糊精,羟丙基-BETA-环糊精,Hydroxypropyl-β-cyclodextrin,Hydroxypropyl betadex

Others Others
HP-β-CD (HP-β-CD) 是一种药物递送载体,可提高稳定性和利用度。
T19967 Fendosal

芬度柳,HP 129,P 71-0129,P71-0129,P-71-0129,HP129,HP-129

Immunology/Inflammation related Immunology/Inflammation
Fendosal (HP-129) 是一种非甾体抗炎药。在预防性和治疗性辅助诱导的慢性炎症多关节炎模型中,它的活性是阿司匹林的 6.9 至 9.5 倍。
T25507 HP 228

HP-228,Ac-Nle-gln-his-D-phe-arg-D-trp-gly-NH2,HP228

HP 228 is a heptapeptide by inhibits the induction of nitric oxide synthase.
T26778 Besipirdine

HP 749 free base,P-867493,P867493,HP 749,HP749,P 867493

Sodium Channel; Adrenergic Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Besipirdine (HP 749 free base)是一种非受体依赖性拟胆碱化合物,具有α-肾上腺素能活性和心血管活性。Besipirdine 抑制电压依赖性钠钾通道,抑制生物胺的摄取。Besipirdine 可减少大鼠的时间表诱导的烦渴,增强中枢神经系统中的胆碱能和肾上腺素能神经传递。
T1539 Iloperidone

伊潘立酮,HP 873

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Iloperidone (HP 873) 是一种D2/5-HT2受体拮抗剂,是非典型抗精神病药,可治疗精神分裂症。
T21556 Hydroxytacrine maleate

Velnacrine maleate,HP 029 maleate

AChE Neuroscience
Hydroxytacrine maleate (Velnacrine maleate) 是一种胆碱酯酶(cholinesterase) 抑制剂,可增强啮齿动物的记忆力,可用于研究阿尔茨海默型老年性痴呆(SDAT)。
T19333 Gadoteridol

ProHance,SQ-32692,钆特醇,Gd-HP-DO3A

Others Others
Gadoteridol (Gd-HP-DO3A) 是含钆基的 MRI 造影剂,可用于中枢神经系统成像。
T26778L Besipirdine hydrochloride

HP 749 hydrochloride,Besipirdine hydrochloride(119257-34-0 Free base)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Besipirdine hydrochloride 是一种非受体依赖性拟胆碱化合物,具有α-肾上腺素能活性和心血管活性。Besipirdine hydrochloride 抑制电压依赖性钠钾通道,抑制生物胺的摄取。Besipirdine hydrochloride 可减少大鼠的时间表诱导的烦渴,增强中枢神经系统中的胆碱能和肾上腺素能神经传递。
T32125 Hyperphyllin

HP

Hyperphyllin specifically mimics the branch defects of AMP1, including plastid reduction and expansion and proliferation of the branch meristem.
T30590 Brocrinat

HP 522

Brocrinat (HP 522) is an active diuretic with at least one site of action in the medulla oblongata branch of the Henle loop.
T28160 Nerispirdine HCl

HP-184,HP 184,Nerispirdine hydrochloride,HP184

Nerispirdine is a acetylcholine release enhancer, sodium channel blocker and K(V) 2.1 channel blocker. Nerispirdine inhibits voltage-dependent Na(+) channel currents recorded from human SH-SY5Y cells with an IC(50) of 11.9 micromol/L when measured from a
TP1939L1 RVD-Hpα acetate(1193362-76-3 free base)

Cannabinoid Receptor GPCR/G Protein
RVD-Hpα acetate(1193362-76-3 free base) 是人血加压素的 N 末端延伸形式,可作为选择性 CB1 受体激动剂。增加体外表达 CB1 受体的细胞中的细胞内 Ca2+ 水平。也是高亲和力 CB2 正变构调节剂 (Ki = 50 nM)。
T27563 Hydroxypropyl-beta-cyclodextrin

HP-beta-CyD,VTS-270,HP-beta-CD,Hydroxypropyl-beta-cyclodextri,THPB,HPbCD

Hydroxypropyl-beta-cyclodextrin, also known as Hydroxypropyl-beta-cyclodextrin; THPB; HP-beta-CD; HPbCD; HP-beta-CyD; VTS-270; HPbetaCD; HPbetaCyD, is a drug candidate potentially for the treatment of Niemann-Pick type C diseases. In April 2009, hydroxypr
T34223 Quilostigmine

HP 290,NXX 066,NXX-066

Quilostigmine is a cholinergic.
T32018 Guanoxyfen sulfate

CI-515,C.I. 515,HP 1598,CN-34,799-5A,CI 515

Guanoxyfen sulfate is a bio-active chemical.
T34031 Phosphazide

AZT-5'-Phosphonate,AZT-5'-H2PO3,Nicavir,AZT-HP

Phosphazide is a zidovudine prodrug.
T27635 Isoxepac

伊索克酸,Olopatadine USP Related Compound C

Others Others
Isoxepac (Olopatadine USP Related Compound C) 是非甾体抗炎剂,显示出抗炎、镇痛和解热活性,已在多种动物模型中进行了相关研究。
TP2340 Hemoregulatory peptide 5b

hp 5B,Pglu-glu-asp-cys-lys-OH,Peedck,Glp-glu-asp-cys-lys-OH,SP1 Pentapeptide

Hemoregulatory peptide 5b is a synthetic analog of granulocyte chalone which initially identified in extracts of rodent bone marrow and human leukocytes. Monomer inhibits both formations of GM-CFC colonies and cytotoxic drug-induced recruitment of murine
T75936 RVD-Hpα TFA

RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selectiveCB1receptoragonist. RVD-Hpα TFA increases intracellular Ca2+levels in cells expressingCB1receptors in vitro. RVD-Hpα TFA also high affinityCB2positive allosteric modulator (Ki=50 nM).
T61329 HP1142

HP1142 is a highly effective and specific inhibitor targeting the FLT3 receptor tyrosine kinase, with a particular affinity for its mutant variant FLT3/ITD. It exhibits a benzoimidazole scaffold-based structure, making it a promising compound for investigating and studying the FLT3/ITD mutation in the context of leukemia research [1].
T78073 HP210

Glucocorticoid Receptor Endocrinology/Hormones
HP210是一种选择性糖皮质激素受体调节剂(SGRM),可以抑制IL-1β和IL-6的mRNA表达,有望用于研究炎症相关疾病。
T83865 HP661

HP661是一种针对线粒体复合物I(也称为NADH脱氢酶)的抑制剂,对复合物I具有选择性,以1 µM的浓度抑制其77.6%,而对复合物III抑制率为28.1%,对复合物II和IV则无抑制作用。HP661特异性降低具有高水平氧化磷酸化作用的人类肺癌细胞H460、NCI H441及对trametinib耐药的A549细胞的生存能力(IC50分别为10.6、29.7和15.1 nM),相较于氧化磷酸化水平低的NCI H358人类肺癌细胞(IC50 >10,000 nM)以及非癌性人类胰腺正常上皮细胞(HPNE)和MRC-5人类胎肺成纤维细胞(两者的IC50均>10,000 nM)。当以每天两次,每次30 mg/kg的剂量给药时,HP661在H460小鼠异种移植模型中减少肿瘤体积,并对trametinib引导的肿瘤生长减少产生加成效应。
T64182 HP590

HP590 是一种新型的、强效的、口服具有活力的 STAT3 抑制剂 (STAT3 荧光素酶活性:IC50=27.8 nM; ATP 抑制:IC50=24.7 nM)。HP590 具有抗胃癌细胞增殖的作用,能够诱导细胞凋亡。
T61758 HP1328

HP1328 is a highly effective inhibitor of FLT3 receptor tyrosine kinase with a specific focus on FLT3/ITD mutation. It belongs to the benzoimidazole scaffold-based compound family. Significantly reducing the leukemia burden, HP1328 effectively extends the survival of mice afflicted with FLT3/ITD leukemia [1].
T62253 S-HP210

S-HP210 是一种选择性的、有效的糖皮质激素受体 (GR) 调节剂,能够抑制 NF-κB 转录 (IC50: 1.92 μM)。S-HP210 对于 LPS 诱导的多种促炎基因(如 IL-1β、IL-6 和 COX-2)的转录具有抑制作用。S-HP210 在有效剂量下对小鼠成纤维细胞 3T3 没有毒性。
T62252 R-HP210

R-HP210 能够抑制 LPS 诱导的多种促炎基因(IL-1β、IL-6 和 COX-2)的转录。R-HP210 对 NF-κB 介导的栓系反式抑制功能的 IC50 值为 3.80 μM。R-HP210 不诱导糖皮质激素 (GCs) 的反式激活功能。
T71279 BPR1K653

BPR1K653 is a potent Aurora kinase inhibitor with potential anticancder activity. BPR1K653 specifically inhibited the activity of Aurora-A and Aurora-B kinase at low nano-molar concentrations in vitro. BPR1K653 was potent in targeting a variety of cancer cell lines regardless of the tissue origin, p53 status, or expression of MDR1. At the cellular level, BPR1K653 induced endo-replication and subsequent apoptosis in both MDR1-negative and MDR1-positive cancer cells. Importantly, it showed potent ...
T22021 ACHP

IKK-2 Inhibitor VIII

IκB/IKK NF-κB
ACHP(IKK-2 Inhibitor VIII) 是一种新型具有选择性和高效性的 IKK 抑制剂,对IKK-α和IKK-β 具有抑制作用。ACHP 具有抗 HIV-1 活性,通过抑制 NF-κB 激活来抑制 HIV-1 长末端重复序列 (LTR) 驱动的基因表达,抑制 TNF-α 诱导的 NF-κB (p65)募集到 HIV-1 LTR。
T17909 (S,R,S)-AHPC-PEG3-N3

VHL Ligand-Linker Conjugates 8,VH032-PEG3-N3,E3 ligase Ligand-Linker Conjugates 12

Others; E3 Ligase Ligand-Linker Conjugate; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-PEG3-N3 (VHL Ligand-Linker Conjugates 8) 包含基于 (S,R,S)-AHPC 的 VHL 配体和 3 个单元 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物。
T17924 (S,R,S)-AHPC-PEG2-NH2 hydrochloride

VH032-PEG2-NH2 hydrochloride,VHL Ligand-Linker Conjugates 3 hydrochloride,E3 ligase Ligand-Linker Conjugates 6

Others; E3 Ligase Ligand-Linker Conjugate Others; PROTAC
(S,R,S)-AHPC-PEG2-NH2 hydrochloride (E3 ligase Ligand-Linker Conjugates 6) 包含基于 (S,R,S)-AHPC 的 VHL 配体和 2 个单元 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物,可用于 PROTAC 的合成分子。
T10809L CHPG hydrochloride

CHPG hydrochloride(170846-74-9 Free base)

ERK; NF-κB; GluR MAPK; Neuroscience; NF-κB
CHPG hydrochloride 是 mGluR5 的选择性激动剂。
T28410 PHPS1

PHPS-1,PHPS 1

Phosphatase Metabolism
PHPS1 是 Shp2的选择性抑制剂,对 Shp2,Shp2-R362K,Shp1,PTP1B 和 PTP1B-Q 的 Ki 分别为 0.73,5.8,10.7,5.8 和 0.47 μM。
T18675 (S,R,S)-AHPC-PEG2-NH2 dihydrochloride

VH032 amide-PEG2-amine,VH032-PEG2-NH2 dihydrochloride,(S,R,S)-AHPC-PEG2-NH2二盐酸盐,VH032-linker 12

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-PEG2-NH2 dihydrochloride (VH032-linker 12) 包含基于 (S,R,S)-AHPC 的 VHL 配体和 2 个单元 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物,可用于 PROTAC 分子的合成。
T1804 HPGDS inhibitor 1

HPGDS-inhibitor-1

PGE Synthase Immunology/Inflammation
HPGDS inhibitor 1 是口服具有活性的HPGDS 选择性抑制剂,在酶和细胞分析中的IC50值分别为 0.6 nM 和 32 nM,但对 L-PGDS、mPGES、COX-1、COX-2 、5-LOX 无抑制作用。
T8412 (S,R,S)-AHPC

VH032-NH2,MDK7526,VHL ligand 1

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC (VH032-NH2) 是一种 VH032-based VHL ligand,可用于募集 von Hippel-Lindau (VHL)蛋白。它能够利用 linker 与靶蛋白配体连接,得到 PROTAC 分子。
T18640 (S,R,S)-AHPC-C4-NH2 hydrochloride

VH032-C4-NH2 hydrochloride,E3 ligase Ligand-Linker Conjugates 28,VHL Ligand-Linker Conjugates 13

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-C4-NH2 hydrochloride (E3 ligase Ligand-Linker Conjugates 28) 是一种合成的 E3 连接酶配体- linker 偶联物,包含基于 (S,R,S)-AHPC 的 VHL 配体和 linker。
T9777 THP104c

Mitochondrial Metabolism Metabolism
THP104c 是有效的线粒体分裂抑制剂。
T77668 hPL-IN-1

Others Others
hPL-IN-1 是一种有效的可逆胰脂肪酶 (PL) 抑制剂 (IC50=1.86 μM),可用于研究与肥胖相关的疾病。
T17920 (S,R,S)-AHPC-PEG1-N3

VHL Ligand-Linker Conjugates 9,VH032-PEG1-N3,E3 ligase Ligand-Linker Conjugates 3

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-PEG1-N3 (E3 ligase Ligand-Linker Conjugates 3) 是 E3 连接酶配体和linker 连接得到的 偶联物,包含基于 (S,R,S)-AHPC 的 VHL 配体和 1 个单元 PEG linker。
T19955 Biotin-HPDP

Pyridyldisulfide-biotin,Pyridyldithiol-biotin

Others Others
Biotin-HPDP (Pyridyldithiol-biotin) 是一种巯基反应性生物素化试剂。
T17921 (S,R,S)-AHPC-PEG4-N3

VH032-PEG4-N3,VHL Ligand-Linker Conjugates 5,E3 ligase Ligand-Linker Conjugates 4

Others; PROTAC Linker Others; PROTAC
(S,R,S)-AHPC-PEG4-N3 (VHL Ligand-Linker Conjugates 5) is a synthesized conjugate that functions as a ligand-linker in E3 ligase-based systems. It is composed of the (S,R,S)-AHPC VHL ligand and a 4-unit PEG linker, both commonly employed in PROTAC technology.
T18912 ADHP

10-乙酰基-3,7-二羟基吩嗪,10-Acetyl-3,7-dihydroxyphenoxazine

Others Others
ADHP (10-Acetyl-3,7-dihydroxyphenoxazine) 是荧光过氧化物酶底物,其λex=530 nm,λem=590 nm。
T10237 ACHP Hydrochloride

IKK-2 Inhibitor VIII

IκB/IKK NF-κB
ACHP Hydrochloride (IKK-2 Inhibitor VIII) 是选择性的IKK-β抑制剂 (IC50=5.8 nM)。
T2430 HPOB

Apoptosis; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
HPOB 是一种高选择性HDAC6抑制剂,IC50为 56 nM,其选择性是其他 HDAC 的 30 倍以上。它提高 DNA 损伤抗癌药物在转化细胞中的有效性。
T4658 MHP

Methyl caprooyl tyrosinate

S1P Receptor GPCR/G Protein
MHP (Methyl caprooyl tyrosinate) 是一种鞘氨醇激酶 (SPHK1) 激活剂,可显著增加 CAMP mRNA 和蛋白水平,还可增强抗微生物防御能力和先天免疫力。
T2681 hPGDS-IN-1

PGE Synthase Immunology/Inflammation
hPGDS-IN-1是 hPGDS 抑制剂,使用荧光偏振检测或通过 EIA 法测得的 IC50值为12 nM。
T38948 MS-PEG4-THP

PROTAC Linker PROTAC
MS-PEG4-THP 是PEG 类PROTAC linker,可用于合成 PROTAC 分子。
T40028 (S,R,S)-AHPC

Ligand for E3 Ligase PROTAC
(S,R,S)-AHPC 是一种 VHL 配体,用于募集 VHL 蛋白。
T13671 (S,R,S)-AHPC-Me hydrochloride

VHL ligand 2 hydrochloride,E3 ligase Ligand 1

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-Me hydrochloride (VHL ligand 2 hydrochloride) is a chemical compound utilized in the synthesis of ARV-771, an exceptionally potent BET protein degrader. This compound selectively degrades BET protein in cells resistant to castration, exhibiting a remarkable DC50 <1 nM. Recognized as VHL ligand 2 hydrochloride, (S,R,S)-AHPC-Me hydrochloride serves as the VHL ligand derived from (S,R,S)-AHPC for the recruitment of von Hippel-Lindau (VHL) protein.
T6967 RHPS4

RHPS 4 methosulfate,NSC714187

Apoptosis; Telomerase Apoptosis; DNA Damage/DNA Repair
RHPS4 (RHPS 4 methosulfate) 是 DNA 损伤诱导剂,是一种有效的亚微摩尔端粒酶抑制剂,IC50为0.33 μM。

化合物

HP-β-CD
Cat.No: T19609
Synonym: 羟丙基-β-环糊精,羟丙基-BETA-环糊精,Hydroxypropyl-β-cyclodextrin,Hydroxypropyl betadex
Target: Others
Fendosal
Cat.No: T19967
Synonym: 芬度柳,HP 129,P 71-0129,P71-0129,P-71-0129,HP129,HP-129
Target: Immunology/Inflammation related
HP 228
Cat.No: T25507
Synonym: HP-228,Ac-Nle-gln-his-D-phe-arg-D-trp-gly-NH2,HP228
Target:
Besipirdine
Cat.No: T26778
Synonym: HP 749 free base,P-867493,P867493,HP 749,HP749,P 867493
Target: Sodium Channel, Adrenergic Receptor
Iloperidone
Cat.No: T1539
Synonym: 伊潘立酮,HP 873
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Hydroxytacrine maleate
Cat.No: T21556
Synonym: Velnacrine maleate,HP 029 maleate
Target: AChE
Gadoteridol
Cat.No: T19333
Synonym: ProHance,SQ-32692,钆特醇,Gd-HP-DO3A
Target: Others
Besipirdine hydrochloride
Cat.No: T26778L
Synonym: HP 749 hydrochloride,Besipirdine hydrochloride(119257-34-0 Free base)
Target: Adrenergic Receptor
Hyperphyllin
Cat.No: T32125
Synonym: HP
Target:
Brocrinat
Cat.No: T30590
Synonym: HP 522
Target:
Nerispirdine HCl
Cat.No: T28160
Synonym: HP-184,HP 184,Nerispirdine hydrochloride,HP184
Target:
RVD-Hpα acetate(1193362-76-3 free base)
Cat.No: TP1939L1
Synonym:
Target: Cannabinoid Receptor
Hydroxypropyl-beta-cyclodextrin
Cat.No: T27563
Synonym: HP-beta-CyD,VTS-270,HP-beta-CD,Hydroxypropyl-beta-cyclodextri,THPB,HPbCD
Target:
Quilostigmine
Cat.No: T34223
Synonym: HP 290,NXX 066,NXX-066
Target:
Guanoxyfen sulfate
Cat.No: T32018
Synonym: CI-515,C.I. 515,HP 1598,CN-34,799-5A,CI 515
Target:
Phosphazide
Cat.No: T34031
Synonym: AZT-5'-Phosphonate,AZT-5'-H2PO3,Nicavir,AZT-HP
Target:
Isoxepac
Cat.No: T27635
Synonym: 伊索克酸,Olopatadine USP Related Compound C
Target: Others
Hemoregulatory peptide 5b
Cat.No: TP2340
Synonym: hp 5B,Pglu-glu-asp-cys-lys-OH,Peedck,Glp-glu-asp-cys-lys-OH,SP1 Pentapeptide
Target:
RVD-Hpα TFA
Cat.No: T75936
Synonym:
Target:
HP1142
Cat.No: T61329
Synonym:
Target:
HP210
Cat.No: T78073
Synonym:
Target: Glucocorticoid Receptor
HP661
Cat.No: T83865
Synonym:
Target:
HP590
Cat.No: T64182
Synonym:
Target:
HP1328
Cat.No: T61758
Synonym:
Target:
S-HP210
Cat.No: T62253
Synonym:
Target:
R-HP210
Cat.No: T62252
Synonym:
Target:
BPR1K653
Cat.No: T71279
Synonym:
Target:
ACHP
Cat.No: T22021
Synonym: IKK-2 Inhibitor VIII
Target: IκB/IKK
(S,R,S)-AHPC-PEG3-N3
Cat.No: T17909
Synonym: VHL Ligand-Linker Conjugates 8,VH032-PEG3-N3,E3 ligase Ligand-Linker Conjugates 12
Target: Others, E3 Ligase Ligand-Linker Conjugate, Ligand for E3 Ligase
(S,R,S)-AHPC-PEG2-NH2 hydrochloride
Cat.No: T17924
Synonym: VH032-PEG2-NH2 hydrochloride,VHL Ligand-Linker Conjugates 3 hydrochloride,E3 ligase Ligand-Linker Conjugates 6
Target: Others, E3 Ligase Ligand-Linker Conjugate
CHPG hydrochloride
Cat.No: T10809L
Synonym: CHPG hydrochloride(170846-74-9 Free base)
Target: ERK, NF-κB, GluR
PHPS1
Cat.No: T28410
Synonym: PHPS-1,PHPS 1
Target: Phosphatase
(S,R,S)-AHPC-PEG2-NH2 dihydrochloride
Cat.No: T18675
Synonym: VH032 amide-PEG2-amine,VH032-PEG2-NH2 dihydrochloride,(S,R,S)-AHPC-PEG2-NH2二盐酸盐,VH032-linker 12
Target: Others, Ligand for E3 Ligase
HPGDS inhibitor 1
Cat.No: T1804
Synonym: HPGDS-inhibitor-1
Target: PGE Synthase
(S,R,S)-AHPC
Cat.No: T8412
Synonym: VH032-NH2,MDK7526,VHL ligand 1
Target: Others, Ligand for E3 Ligase
(S,R,S)-AHPC-C4-NH2 hydrochloride
Cat.No: T18640
Synonym: VH032-C4-NH2 hydrochloride,E3 ligase Ligand-Linker Conjugates 28,VHL Ligand-Linker Conjugates 13
Target: Others, Ligand for E3 Ligase
THP104c
Cat.No: T9777
Synonym:
Target: Mitochondrial Metabolism
hPL-IN-1
Cat.No: T77668
Synonym:
Target: Others
(S,R,S)-AHPC-PEG1-N3
Cat.No: T17920
Synonym: VHL Ligand-Linker Conjugates 9,VH032-PEG1-N3,E3 ligase Ligand-Linker Conjugates 3
Target: Others, Ligand for E3 Ligase
Biotin-HPDP
Cat.No: T19955
Synonym: Pyridyldisulfide-biotin,Pyridyldithiol-biotin
Target: Others
(S,R,S)-AHPC-PEG4-N3
Cat.No: T17921
Synonym: VH032-PEG4-N3,VHL Ligand-Linker Conjugates 5,E3 ligase Ligand-Linker Conjugates 4
Target: Others, PROTAC Linker
ADHP
Cat.No: T18912
Synonym: 10-乙酰基-3,7-二羟基吩嗪,10-Acetyl-3,7-dihydroxyphenoxazine
Target: Others
ACHP Hydrochloride
Cat.No: T10237
Synonym: IKK-2 Inhibitor VIII
Target: IκB/IKK
HPOB
Cat.No: T2430
Synonym:
Target: Apoptosis, HDAC
MHP
Cat.No: T4658
Synonym: Methyl caprooyl tyrosinate
Target: S1P Receptor
hPGDS-IN-1
Cat.No: T2681
Synonym:
Target: PGE Synthase
MS-PEG4-THP
Cat.No: T38948
Synonym:
Target: PROTAC Linker
(S,R,S)-AHPC
Cat.No: T40028
Synonym:
Target: Ligand for E3 Ligase
(S,R,S)-AHPC-Me hydrochloride
Cat.No: T13671
Synonym: VHL ligand 2 hydrochloride,E3 ligase Ligand 1
Target: Others, Ligand for E3 Ligase
RHPS4
Cat.No: T6967
Synonym: RHPS 4 methosulfate,NSC714187
Target: Apoptosis, Telomerase
Cat. No. Product Name Target Signaling Pathways
T4797 DEHP

Bis(2-ethylhexyl) phthalate,邻苯二甲酸二(2-乙基己)酯

Others; Endogenous Metabolite Metabolism; Others
DEHP (Bis(2-ethylhexyl) phthalate) 是内源性代谢产物的一种。
TN6684 Cyclo(Tyr-Hpro)

Cyclo(Tyr-Hpro) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6684,CAS号为 813461-21-1。
T36560 (±)9-HpODE

(±)9-HpODE is a racemic mixture of the fatty acid hydroperoxide product (9(S)-HpODE) formed from lipoxygenase action on linoleic acid. It shows antimicrobial activity against various fungal and bacterial pathogens and thus may play a role in plant defense. In mammalian species, monocyte-induced oxidization of LDL generates significant amounts of esterified 9-HpODE, which is rapidly reduced to 9-HODE.
TN3118 5-Hydroxy-7-(4'-hydroxy-3'-methoxyphenyl)-1-phenyl-3-heptanone (DHPA)

Others Others
5-Hydroxy-7-(4'-hydroxy-3'-methoxyphenyl)-1-phenyl-3-heptanone (DHPA) is a pancreatic lipase inhibitor, it shows antihyperlipidemic activity.
TN7019 DNHP

DNHP is a natural product.
TN6429 Cyclo(Phe-Hpro)

Cyclo(Phe-Hpro) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6429,CAS号为 1016899-94-7。
TN6680 Cyclo(Hpro-Leu)

Cyclo(Hpro-Leu) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6680,CAS号为 1016899-93-6。
T74193 (R)-IDHP

(R)-IDHP为IDHP异构体,属于丹参代谢物。该化合物能通过抑制血管平滑肌细胞电压依赖性钙通道与受体操作钙通道的Ca2+释放和Ca2+内流,发挥血管松弛作用,适用于心脑血管疾病研究。

天然产物

DEHP
Cat.No: T4797
Synonym: Bis(2-ethylhexyl) phthalate,邻苯二甲酸二(2-乙基己)酯
Target: Others, Endogenous Metabolite
Cyclo(Tyr-Hpro)
Cat.No: TN6684
Synonym:
Target:
(±)9-HpODE
Cat.No: T36560
Synonym:
Target:
5-Hydroxy-7-(4'-hydroxy-3'-methoxyphenyl)-1-phenyl-3-heptanone (DHPA)
Cat.No: TN3118
Synonym:
Target: Others
DNHP
Cat.No: TN7019
Synonym:
Target:
Cyclo(Phe-Hpro)
Cat.No: TN6429
Synonym:
Target:
Cyclo(Hpro-Leu)
Cat.No: TN6680
Synonym:
Target:
(R)-IDHP
Cat.No: T74193
Synonym:
Target:
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