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50

抑制剂 & 化合物

11

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Cat. No. Product Name Target Signaling Pathways
T60006 Aromatase inhibitor 23

Others Others
Aromatase inhibitor 23 是一种针对 RAD51 重组酶家族中蛋白质-蛋白质相互作用的抑制剂。
T60022 Aromatase-IN-2

Others Others
Aromatase-IN-2 具有抗炎、抗肿瘤和平喘作用。
T61444 Nonsteroidal aromatase inhibitor 1

Nonsteroidal aromatase inhibitor 1 (Compound 13h) effectively inhibits the enzyme CYP19A1 with an IC50 value of 0.09 nM. Due to its potent inhibitory activity, Nonsteroidal aromatase inhibitor 1 holds promise for research in the field of breast cancer [1].
T7197 Fadrozole

Aromatase Endocrinology/Hormones
Fadrozole 是一种有效的、非甾体类的、选择性的芳香化酶抑制剂(IC50:6.4 nM)。
T61463 Monoamine oxidase/Aromatase-IN-1

Monoamine oxidase/Aromatase-IN-1 (compound 2q) is a potent dual inhibitor of monoamine oxidase (MAO) and aromatase, with IC50 values of 39 nM and 31 nM for MAO-B and aromatase, respectively. It holds significant potential for research in neurological disorders and breast cancer [1].
T11991 Mefentrifluconazole

P450; Antifungal Metabolism; Microbiology/Virology
Mefentrifluconazole 是一种有效的、选择性的和具有口服活性的真菌 CYP51 (Kd= 0.5 nM) 抑制剂,但对人芳香酶的抑制活性较低,IC50值为0.92 μM。它是一种新型唑类衍生物,用作农用广谱抗真菌剂。
T0393 Anastrozole

阿那曲唑,ZD1033

Aromatase Endocrinology/Hormones
Anastrozole (ZD1033) 是芳香酶的选择性抑制剂,能够抑制胎盘芳香化酶(IC50:15 nM)。
T7556 Fadrozole hydrochloride

CGS 16949A,盐酸法倔唑

Aromatase Endocrinology/Hormones
Fadrozole hydrochloride (CGS 16949A) 是一种选择性的、有效,和非甾体类的芳香化酶抑制剂(IC50:6.4 nM)。
T1103 Aminoglutethimide

DL-Aminoglutethimide,氨鲁米特,BA-16038,NSC-330915

Aromatase Endocrinology/Hormones
Aminoglutethimide (BA-16038) 是一种芳香酶抑制剂,IC50=10 μM,用于治疗晚期 BREAST Y。
T20625 Prochloraz

咪鲜胺,Sporgon,Prelude

Estrogen Receptor/ERR; AhR; Androgen Receptor; Antifungal Endocrinology/Hormones; Immunology/Inflammation; Metabolism; Microbiology/Virology
Prochloraz (Prelude) 是咪唑类抗真菌剂。Prochloraz 抑制羊毛甾醇的细胞色素 P450 依赖性 14α-脱甲基作用,由此抑制麦角固醇的生物合成,从而导致真菌细胞膜破裂和细胞死亡。它也是雌激素受体和 雄激素受体的拮抗剂,IC50分别为25 μM 和4 μM, 并激活芳烃受体,EC50为1μM。
T1587 Exemestane

EXE,依西美坦,FCE 24304,PNU155971

Aromatase Endocrinology/Hormones
Exemestane (EXE) 是一种选择性的、具有口服活性的、不可逆的甾体芳香酶抑制剂,能够作用于人胎盘芳香酶 (IC50:30 nM) 和大鼠卵巢芳香酶 (IC50:40 nM),可用于研究激素依赖性乳腺癌。
T4281 Endoxifen

(E/Z)-N-desmethyl-4-hydroxy Tamoxifen,N-去甲基-4-羟基-,(E/Z)-Endoxifen

Estrogen Receptor/ERR; Aromatase; Estrogen/progestogen Receptor; Parasite; Drug Metabolite Endocrinology/Hormones; Metabolism; Microbiology/Virology
Endoxifen ((E/Z)-Endoxifen) 是 Tamoxifen 的关键活性代谢物,能抑制芳香酶的活性,与雌激素受体有较高的亲和力和特异性。它有潜力研究乳腺癌。
T71708 Minamestane

Aromatase Endocrinology/Hormones
Minamestane 是一种新型不可逆芳香化酶抑制剂。Minamestane 引起人胎盘芳香化酶的时间依赖性抑制,半衰期为4分钟,K 为59nM。Minamestane 具有抗肿瘤活性。
T27320 Finrozole

MPV 2213ad,MPV-2213ad,MPV 2213,MPV-2213,MPV2213ad

Aromatase Endocrinology/Hormones
Finrozole (MPV 2213ad) 是一种新型选择性芳香化酶抑制剂,对于乳房发育是部分可逆的。
T23549 YM 511

P450; Aromatase Endocrinology/Hormones; Metabolism
YM 511 是一种高度特异性的非甾体芳香酶 (aromatase) 抑制剂。YM 511 竞争性抑制大鼠卵巢和人胎盘微粒体中的芳香酶活性 (IC50 分别为 0.4 和 0.12 nM)。YM 511 轻微抑制其他类固醇激素的产生。YM 511 具有用于抑制雌激素依赖性作用研究,不会影响其他类固醇激素的血清水平的潜力。
T2280 Endoxifen (Z-isomer)

Z-因多昔芬,Endoxifen Z-isomer,4-[(1E)-1-{4-[2-(甲基氨基)乙氧基]苯基}-2-苯基-1-丁烯-1-基]苯酚

Estrogen Receptor/ERR; EGFR; Potassium Channel; Estrogen/progestogen Receptor; HER Angiogenesis; Endocrinology/Hormones; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
Endoxifen Z-isomer (EDX)是 Tamoxifen 重要的代谢产物,在表达 ERα的乳腺癌细胞中发挥抗雌激素作用。它以浓度依赖的方式抑制 hERG, IC50值为1.6μM。
T72310 Antibacterial agent 132

Antifungal Microbiology/Virology
Antibacterial agent 132 对 C. parapsilosis (ATCC 22019) 和 C. krusei (ATCC 6258) 实验中显示出抗菌作用,MIC90 值分别为 <0.06 μg/mL 和 62.50 μg/mL。Antibacterial agent 132 对芳香化酶 (aromatase enzyme)具有抑制作用,IC50 为 0.047μM。
T27918 LY 43578

LY-43578,LY43578

P450; Aromatase Endocrinology/Hormones; Metabolism
LY 43578 是一种具有口服活性的芳香酶 (aromatase) 抑制剂。LY 43578 对大鼠肝微粒体 P-450依赖的 p-nitroanisole 的 O -去甲基化和 ethylmorphine 的 N -去甲基化有抑制作用,IC50 分别为 0.3 和 5 μΜ。LY 43578 可用于研究神经系统疾病和心血管疾病。
T26322 Vorozole

R83839,R 83839,R-83839,(+)-Vorozole,R83842

P450; Aromatase Endocrinology/Hormones; Metabolism
Vorozole (R83842) 是一种具有口服活性、有效性和选择性的非甾体芳香酶抑制剂。Vorozole 在体内表现出抗肿瘤活性,可用于研究乳腺癌。
T26322L (-)-Vorozole

(-)-Vorozole(Isomer-129731-10-8)

P450; Aromatase Endocrinology/Hormones; Metabolism
(-)-Vorozole 是一种具有口服活性的非甾体芳香酶抑制剂,具有有效性和选择性。(-)-Vorozole在体内实验中表现出抗肿瘤活性。(-)-Vorozole 可用于研究乳腺癌。
T6827L Endoxifen hydrochloride

Endoxifen hydrochloride,Tamoxifen的主要活性代谢产物,具备较高的对雌激素受体(estrogen receptor)的亲和力和特异性,并能抑制芳香酶活性。它在乳腺癌研究中表现出潜在应用价值。
T11847L Liarozole

R75251 dihydrochloride,利阿唑

P450; Retinoid Receptor Metabolism
Liarozole (R75251 dihydrochloride) 是一种咪唑衍生物,是一种具有口服活性的维甲酸 (RA) 代谢阻断剂(RAMBA),具有抗肿瘤作用。它能够抑制维甲酸依赖的细胞色素P450(CYP26) 4- 羟基化 (IC50=7 μM),导致组织维甲酸水平增加。
T70558 Org 33201

Org 33201 is a potent aromatase inhibitor.
T27868 LY 113174

LY-113174,LY113174

LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.
T71897 Vatalanib succinate

Vatalanib succinate is a VEGFR, PDGFR-β, c-Kit, c-Fms, and aromatase inhibitor.
T27369 FR 901537

FR901537,FR-901537

FR 901537 is a new aromatase inhibitor with antitumor effects.
T70404 MPV-2213AD

MPV-2213AD is an aromatase inhibitor.
T20683 Letrozole related compound B

Letrozole specified impurity A

Letrozole related compound B is an impurity of aromatase inhibitor.
T71410 Cgs 18320B

Cgs 18320B is a non-steroidal aromatase inhibitor
T7197L Fadrozole HCl hydrate

Fadrozole,CGS-16949A,Fadrozole hydrochloride hemihydrate,CGS16949A,CGS 16949A

Fadrozole is a selective inhibitor of aromatase. It also effective in the treatment of estrogen-dependent diseases including breast cancer.
T27922 LY 56110

LY56110,LY-56110

LY 56110 is a novel nonsteroidal aromatase inhibitor.
T25716 Liarozole fumarate

Liazal,R85246,R-85246,R 85246

Liarozole fumarate is used as a retinoic acid metabolism blocking agent (RAMBA) and an aromatase inhibitor.
T12319 Org30958

Aromatase Endocrinology/Hormones
Org30958 is a potent inhibitor of aromatase in vivo.
T30837 Cgp 47645

Leflutrozole,Cgp-47645,Cgp47645

CGP 47645 (Leflurozole) is an oral active non-steroidal aromatase inhibitor and antitumor agent with anti-tumor and endocrine effects.
T30834 Cgp 45688

Cgp45688,Cgp-45688

CGP 45688 is an oral active non-steroidal aromatase inhibitor with anti-tumor and endocrine effects on rat breast tumors.
T61787 SYN20028567

SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].
T81012 Testololactone

Testololactone,一种芳香酶抑制剂,常用于乳腺癌研究。
T71073 Tan 931

Tan 931 is a nonsteroidal aromatase inhibitor that was first isolated from the culture filtrate of a soil isolate fungus, No. 8974
T6060L Anabasine HCl

BB-NC-0036,CCG-38440,H-8174,AR-1H7273,ZX-BK000320,ST-24041653

Anabasine HCl is used as a clinical biomarker for tobacco smoke exposure and as an insecticide. It is also a depolarizing NMJ blocker, aromatase inhibitor, nAChr antagonist, and teratogen found in species of Nicotiana.
T38424 (R)-Fadrozole

FAD286,(R)-CGS 16949A free base,(R)-Fadrozole

(R)-Fadrozole ((R)-CGS 16949A; FAD286) is a potent nonsteroidal inhibitor. (R)-Fadrozole also inhibits human placental aromatase (pIC 50 = 6.17) and aldosterone biosynthesis. (R)-Fadrozole reverses cardiac fibrosis in spontaneously hypertensive heart failure rats..
T71010 Norendoxifen

Norendoxifen, also known as 4-hydroxy-N, N-didesmethyltamoxifen, is a nonsteroidal aromatase inhibitor of the triphenylethylene group that was never marketed. It is an active metabolite of the selective estrogen receptor modulator tamoxifen.
T80057 Cytochrome P450 reductase

Cytochrome P450reductase,一种NADPH-细胞色素还原酶,发挥作用于促进芳香酶构象,以最适合底物结合。
T61919 Anticancer agent 78

Anticancer agent 78 具有抗芳香酶活性(IC50= 0.9 μM)。Anticancer agent 78 是一种有效的抗癌剂,显示细胞毒性。Anticancer agent 78 在乳腺癌中有研究潜力。
T35676 17β-hydroxy Exemestane

17β-hydroxy Exemestane is the primary active metabolite of exemestane . It is formed by metabolism of exemestane by the cytochrome P450 (CYP) isoforms CYP1A and CYP4A11. 17β-hydroxy Exemestane is an aromatase inhibitor (IC50 = 69 nM using human placental microsomes) and an androgen receptor (AR) agonist (IC50 = 39.6 nM) that is selective for AR over estrogen receptor α (ERα; IC50 = 21.2 μM). It stimulates growth of AR- and ERα-positive MCF-7 (EC50 = 2.7 μM) and T47D breast cancer cells (EC50s = ...
T11847 Liarozole dihydrochloride

R75251 dihydrochloride

Others Others
Liarozole dihydrochloride is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase).Liarozole dihydrochloride is an imidazole derivative; it is being investigated as a non-hormonal agent in prostate cancer and in the treatment of various other cancers and skin disorders.
T37560 Nidulin

Nidulin is a depsidone originally isolated from A. nidulans. It is active against the bacteria M. tuberculosis and M. ranoe, as well as the fungi T. tonsurans and M. audouini. It also inhibits the growth of methicillin-resistant S. aureus (MRSA; MIC = 4 μg/ml) and has larvicidal activity toward Artemia (LC50 = 2.8 μg/ml). Nidulin is cytotoxic to MOLT-3 cells (IC50 = 21.2 μM) but not HuCCA-1, HepG2, or A549 cells (IC50s = >112.7 μM). It inhibits aromatase with an IC50 value of 11.2 μM.
T25716L Liarozole HCl

R75251,Liarozole hydrochloride,R 75251,R-75251

Liarozole HCl is a benzimidazole derivative with antineoplastic activity. As a retinoic acid metabolism blocking agent, liarozole inhibits CYP450-dependent all-trans-retinoic acid (ATRA)-4-hydroxylase, leading to an increase in endogenous ATRA production,
T83907 10-Chloroestra-1,4-diene-3,17-dione

10-chloro-1,4-Estradiene

10-Chloroestra-1,4-diene-3,17-dione 是一个对雌性激素受体α (ERα) 具有激动作用的类固醇。它能增加在S. cerevisiae 中报告基因的表达(对人类受体的EC50 = 0.36 nM)。同时,它也是一种芳香化酶抑制剂(IC50 = 2.4 µM)。
T78590 Dibenzylfluorescein

DBF

Dibenzylfluorescein(DBF)是一款荧光探针,作为细胞色素P450(CYP)亚型,包括CYP3A4、CYP2C8、CYP2C9、CYP2C19和CYP19的特异性底物,常在Km值0.87-1.9 µM(Ex=485nm,Em=535nm)范围内应用。该探针主要用于监测药物或疾病导致的CYP催化活性变化。
T71578 Endoxifen mesylate

Endoxifen, also known as N-desmethyl-4-hydroxytamoxifen, is a chemical that is under development for estrogen receptor-positive breast cancer. It is also being evaluated as an antipsychotic for treatment of mania and other psychotic disorders. Endoxifen is a nonsteroidal selective estrogen receptor modulator (SERM) of the triphenylethylene group. It is an active metabolite of tamoxifen and has been found to be effective in patients that have failed previous hormonal therapies (tamoxifen, aromat...

化合物

Aromatase inhibitor 23
Cat.No: T60006
Synonym:
Target: Others
Aromatase-IN-2
Cat.No: T60022
Synonym:
Target: Others
Nonsteroidal aromatase inhibitor 1
Cat.No: T61444
Synonym:
Target:
Fadrozole
Cat.No: T7197
Synonym:
Target: Aromatase
Monoamine oxidase/Aromatase-IN-1
Cat.No: T61463
Synonym:
Target:
Mefentrifluconazole
Cat.No: T11991
Synonym:
Target: P450, Antifungal
Anastrozole
Cat.No: T0393
Synonym: 阿那曲唑,ZD1033
Target: Aromatase
Fadrozole hydrochloride
Cat.No: T7556
Synonym: CGS 16949A,盐酸法倔唑
Target: Aromatase
Aminoglutethimide
Cat.No: T1103
Synonym: DL-Aminoglutethimide,氨鲁米特,BA-16038,NSC-330915
Target: Aromatase
Prochloraz
Cat.No: T20625
Synonym: 咪鲜胺,Sporgon,Prelude
Target: Estrogen Receptor/ERR, AhR, Androgen Receptor, Antifungal
Exemestane
Cat.No: T1587
Synonym: EXE,依西美坦,FCE 24304,PNU155971
Target: Aromatase
Endoxifen
Cat.No: T4281
Synonym: (E/Z)-N-desmethyl-4-hydroxy Tamoxifen,N-去甲基-4-羟基-,(E/Z)-Endoxifen
Target: Estrogen Receptor/ERR, Aromatase, Estrogen/progestogen Receptor, Parasite, Drug Metabolite
Minamestane
Cat.No: T71708
Synonym:
Target: Aromatase
Finrozole
Cat.No: T27320
Synonym: MPV 2213ad,MPV-2213ad,MPV 2213,MPV-2213,MPV2213ad
Target: Aromatase
YM 511
Cat.No: T23549
Synonym:
Target: P450, Aromatase
Endoxifen (Z-isomer)
Cat.No: T2280
Synonym: Z-因多昔芬,Endoxifen Z-isomer,4-[(1E)-1-{4-[2-(甲基氨基)乙氧基]苯基}-2-苯基-1-丁烯-1-基]苯酚
Target: Estrogen Receptor/ERR, EGFR, Potassium Channel, Estrogen/progestogen Receptor, HER
Antibacterial agent 132
Cat.No: T72310
Synonym:
Target: Antifungal
LY 43578
Cat.No: T27918
Synonym: LY-43578,LY43578
Target: P450, Aromatase
Vorozole
Cat.No: T26322
Synonym: R83839,R 83839,R-83839,(+)-Vorozole,R83842
Target: P450, Aromatase
(-)-Vorozole
Cat.No: T26322L
Synonym: (-)-Vorozole(Isomer-129731-10-8)
Target: P450, Aromatase
Endoxifen hydrochloride
Cat.No: T6827L
Synonym:
Target:
Liarozole
Cat.No: T11847L
Synonym: R75251 dihydrochloride,利阿唑
Target: P450, Retinoid Receptor
Org 33201
Cat.No: T70558
Synonym:
Target:
LY 113174
Cat.No: T27868
Synonym: LY-113174,LY113174
Target:
Vatalanib succinate
Cat.No: T71897
Synonym:
Target:
FR 901537
Cat.No: T27369
Synonym: FR901537,FR-901537
Target:
MPV-2213AD
Cat.No: T70404
Synonym:
Target:
Letrozole related compound B
Cat.No: T20683
Synonym: Letrozole specified impurity A
Target:
Cgs 18320B
Cat.No: T71410
Synonym:
Target:
Fadrozole HCl hydrate
Cat.No: T7197L
Synonym: Fadrozole,CGS-16949A,Fadrozole hydrochloride hemihydrate,CGS16949A,CGS 16949A
Target:
LY 56110
Cat.No: T27922
Synonym: LY56110,LY-56110
Target:
Liarozole fumarate
Cat.No: T25716
Synonym: Liazal,R85246,R-85246,R 85246
Target:
Org30958
Cat.No: T12319
Synonym:
Target: Aromatase
Cgp 47645
Cat.No: T30837
Synonym: Leflutrozole,Cgp-47645,Cgp47645
Target:
Cgp 45688
Cat.No: T30834
Synonym: Cgp45688,Cgp-45688
Target:
SYN20028567
Cat.No: T61787
Synonym:
Target:
Testololactone
Cat.No: T81012
Synonym:
Target:
Tan 931
Cat.No: T71073
Synonym:
Target:
Anabasine HCl
Cat.No: T6060L
Synonym: BB-NC-0036,CCG-38440,H-8174,AR-1H7273,ZX-BK000320,ST-24041653
Target:
(R)-Fadrozole
Cat.No: T38424
Synonym: FAD286,(R)-CGS 16949A free base,(R)-Fadrozole
Target:
Norendoxifen
Cat.No: T71010
Synonym:
Target:
Cytochrome P450 reductase
Cat.No: T80057
Synonym:
Target:
Anticancer agent 78
Cat.No: T61919
Synonym:
Target:
17β-hydroxy Exemestane
Cat.No: T35676
Synonym:
Target:
Liarozole dihydrochloride
Cat.No: T11847
Synonym: R75251 dihydrochloride
Target: Others
Nidulin
Cat.No: T37560
Synonym:
Target:
Liarozole HCl
Cat.No: T25716L
Synonym: R75251,Liarozole hydrochloride,R 75251,R-75251
Target:
10-Chloroestra-1,4-diene-3,17-dione
Cat.No: T83907
Synonym: 10-chloro-1,4-Estradiene
Target:
Dibenzylfluorescein
Cat.No: T78590
Synonym: DBF
Target:
Endoxifen mesylate
Cat.No: T71578
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T7999 7-Hydroxyflavanone

Anti-infection Microbiology/Virology
7-Hydroxyflavanone 对肺炎链球菌临床分离株显示出抗菌活性。
T1590 Letrozole

CGS 20267,来曲唑

Aromatase; Autophagy Autophagy; Endocrinology/Hormones
Letrozole (CGS 20267) 是一种可口服的,选择性可逆的非甾体类芳香化酶抑制剂,IC50值为 11.5 nM。它选择性抑制雌激素的生物合成,可研究乳腺癌。
T6917 Oleuropein

洋橄榄苦甙,橄榄苦苷

Apoptosis; Aromatase; ROS; PPAR Apoptosis; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Oleuropein 在橄榄叶和油中发现的天然产物,通过 p53 依赖性途径以及 Bax 和 Bcl2基因的调控来诱导乳腺癌细胞凋亡,还抑制芳香化酶。它可通过直接抑制 PPARγ转录活性来发挥抗氧化,抗炎和抗动脉粥样硬化作用。
T2O2744 alpha-Naphthoflavone

苯并黄素;α-萘黄酮;7,8-苯并黄酮,7,8-benzoflavone,α-萘黄酮

Aromatase Endocrinology/Hormones
alpha-Naphthoflavone (7,8-benzoflavone) 是合成的黄酮类化合物,是一种竞争性芳香酶抑制剂,其IC50=0.5 μM,Ki=0.2 μM。
TN3987 Eriodictyol chalcone

Anti-infection; Aromatase Endocrinology/Hormones; Microbiology/Virology
Eriodictyol chalcone 具有抗芳香化酶和抗 17β-HSD 的活性。它对恶性疟原虫的生长具有抗疟原虫作用。
T0530 Flavanone

2-Phenyl-4-chromanone,4-Flavanone,2,3-Dihydroflavone,黄烷酮,2-Phenylchroman-4-one

Others; Aromatase Endocrinology/Hormones; Others
Flavanone (2-Phenylchroman-4-one) 是天然的黄酮类化合物,对人类雌激素合成酶芳香化酶具有抑制作用。
T3390 Obacunone

Apoptosis; Aromatase; p38 MAPK Apoptosis; Endocrinology/Hormones; MAPK
Obacunone 是从沼泽白葡萄柚种子中分离得到的,通过诱导凋亡发挥抗癌作用。它在雄激素依赖性人前列腺 Y 细胞中具有细胞毒性。它对鼠伤寒沙门氏菌具有抗毒作用,可作为开发鼠伤寒沙门氏菌抗毒策略的先导化合物。
T3899 Calceolarioside B

Desrhamnosyl isoacteoside,木通苯乙醇苷 B,Nuomioside A,木通苯乙醇苷B

Aromatase Endocrinology/Hormones
Calceolarioside B (Desrhamnosyl isoacteoside) 是一种分离自Stauntonia hexaphylla 叶片中的天然产物。它抑制 DPPH 自由基清除活性(IC50:94.60 μM)。它显著抑制大鼠晶状体醛糖还原酶(RLAR)活性(C50:23.99 μM。
TN1674 Garcinone D

伽升沃 D

Reactive Oxygen Species; Nrf2; STAT Immunology/Inflammation; JAK/STAT signaling; Metabolism; NF-κB; Stem Cells
Garcinone D 是来自山竹的一种呫吨酮,可促进 C17.2 神经干细胞的增殖。它以浓度和时间依赖的方式增加磷酸化信号转导和转录激活因子 3 (p-STAT3)、Cyclin D1 和核因子红细胞 2 相关因子 (Nrf2)、以及血红素加氧酶-1 (HO-1) 的蛋白质水平。
TN4605 Myriceric acid B

HIV Protease Microbiology/Virology; Proteases/Proteasome
Myriceric acid B is a potent HIV-1 entry inhibitor targeting gp41 and can serve as a lead compound for developing novel anti-HIV-1 drug. Myriceric acid B scavenges DPPH free radicals with IC50 value of 21.8 uM, it inhibits aromatase activity with IC50 val
TN4307 Isolimonexic acid

BCL; Caspase; COX; p53 Apoptosis; Immunology/Inflammation; Neuroscience; Proteases/Proteasome
Isolimonexic acid exhibits cytotoxicity on MCF-7 cell lines, it also inhibits Panc-28 cancer cell growth.

天然产物

7-Hydroxyflavanone
Cat.No: T7999
Synonym:
Target: Anti-infection
Letrozole
Cat.No: T1590
Synonym: CGS 20267,来曲唑
Target: Aromatase, Autophagy
Oleuropein
Cat.No: T6917
Synonym: 洋橄榄苦甙,橄榄苦苷
Target: Apoptosis, Aromatase, ROS, PPAR
alpha-Naphthoflavone
Cat.No: T2O2744
Synonym: 苯并黄素;α-萘黄酮;7,8-苯并黄酮,7,8-benzoflavone,α-萘黄酮
Target: Aromatase
Eriodictyol chalcone
Cat.No: TN3987
Synonym:
Target: Anti-infection, Aromatase
Flavanone
Cat.No: T0530
Synonym: 2-Phenyl-4-chromanone,4-Flavanone,2,3-Dihydroflavone,黄烷酮,2-Phenylchroman-4-one
Target: Others, Aromatase
Obacunone
Cat.No: T3390
Synonym:
Target: Apoptosis, Aromatase, p38 MAPK
Calceolarioside B
Cat.No: T3899
Synonym: Desrhamnosyl isoacteoside,木通苯乙醇苷 B,Nuomioside A,木通苯乙醇苷B
Target: Aromatase
Garcinone D
Cat.No: TN1674
Synonym: 伽升沃 D
Target: Reactive Oxygen Species, Nrf2, STAT
Myriceric acid B
Cat.No: TN4605
Synonym:
Target: HIV Protease
Isolimonexic acid
Cat.No: TN4307
Synonym:
Target: BCL, Caspase, COX, p53
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