首页 工具
登录
购物车

搜索结果

Search Results for " app "

97

抑制剂 & 化合物

27

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T30103 APP-CHMINACA

PX-3,PX3

APP-CHMINACA is a synthetic cannabinoid (CB) featuring a 1-(cyclohexylmethyl)-1H-indazole-3-carboxamide (CHMINACA) base. It displays a 10-fold greater affinity for the central CB1 receptor than that of JWH 018.
T21890 JLK6

Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
JLK-6 是一种γ分泌酶抑制剂,选择性作用于 HEK293细胞的淀粉样β前体蛋白(APP)的γ-分泌酶裂解 APP,抑制 Aβ的生成,但对不 Notch 受体的裂解无影响。
T9713 δ-secretase inhibitor 11

Beta Amyloid; Caspase Apoptosis; Neuroscience; Proteases/Proteasome
δ-secretase inhibitor 11是一种分泌酶抑制剂,可用作 阿尔茨海默病(AD) 治疗转化开发的先导化合物。
TP1798 Pep-1 (uncapped)

Pep-1 uncapped

Others Others
Pep-1 (uncapped) 是一种能够透过细胞的多肽。
T38570 DMAPP triammonium

Dimethylallyl diphosphate triammonium,Dimethylallyl Pyrophosphate triammonium salt

Others Others
DMAPP triammonium (Dimethylallyl diphosphate triammonium) 是一种异戊二烯类化合物的前提物质之一,参与甲羟戊酸 (MVA) 途径,可用于研究与代谢相关的疾病。
T78337 Mouse IgG2a kappa, Isotype Control

Mouse IgG2a kappa, Isotype Control 是鼠源IIgG2a kappa 抗体的同型抗体。
T126471 3'-Deoxy-4-O-methylepisappanol

3'-Deoxy-4-O-methylepisappanol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126471。
T78612 APPA

Apoptosis Apoptosis
APPA为一种醛糖还原酶抑制剂,能够抑制大鼠多元醇途径,有效预防细胞凋亡及链脲佐菌素引发的糖尿病症状,显示出对糖尿病肾病(DN)研究的应用潜力。
T75859 FTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS

FTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS 是Exendin-4多肽衍生物。
TP1519 Amylin (IAPP), feline

Amylin (IAPP), feline is the peptide subunit of amyloid found in pancreatic islets of type 2 diabetic patients and in insulinomas.
T78244 Human IgG4 kappa, Isotype Control

HumanIgG4kappa Isotype Control为人源化单克隆抗体,用作human IgG4κ抗体的同型对照。
T81756 Mouse IgG3 kappa, Isotype Control

MouseIgG3kappa, Isotype Control为鼠源单克隆抗体,充当mouse IgG3κ抗体的同型对照。
T82161 Human IgG1 (D265A) kappa, Isotype Control

HumanIgG1(D265A) kappa, Isotype Control是一种人鼠嵌合型抗体,用作HumanIgG1(D265A)κ抗体的同型对照。
T126481 Sappanone B

Sappanone B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126481。
T126391 Sappanol

Sappanol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126391。
T81758 Mouse IgG2b kappa, Isotype Control

MouseIgG2bkappa Isotype Control是mouse IgG2bκ抗体的同型对照,属于鼠源单克隆抗体。
T78341 Human IgG1 (F405L) kappa, Isotype Control

HumanIgG1(F405L) kappa, Isotype Control为人-鼠嵌合型单克隆抗体,作为HumanIgG1(F405L)κ抗体的同型对照使用。
T78340 Human IgG1 (N297A) kappa, Isotype Control

HumanIgG1(N297A) kappa, Isotype Control为具有人-鼠嵌合结构的抗体,作为HumanIgG1(N297A)κ 抗体的同型对照物。
T81757 Mouse IgG2c kappa, Isotype Control

MouseIgG2ckappa, Isotype Control为mouse IgG2cκ同型对照的鼠源单克隆抗体。
T81317 Rabbit IgG1 kappa, Isotype Control

RabbitIgG1kappa, Isotype Control为兔源IgG1κ同型对照单克隆抗体,用于科研中作为Rabbit IgG1κ抗体的实验对照。
T66146 (SP-4-4)-2-[2-(Amino-KappaN)ethyl]phenyl-KappaC]chloro[dicyclohexyl[2',4',6'-tris(1-methylethyl)[1,1'-biphenyl]-2-yl]phosphine]-Palladium

(SP-4-4)-2-[2-(Amino-KappaN)ethyl]phenyl-KappaC]chloro[dicyclohexyl[2',4',6'-tris(1-methylethyl)[1,1'-biphenyl]-2-yl]phosphine]-Palladium 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66146,CAS号为 1028206-56-5。
T28818 SMAPP1

SMAPP1 is an activator of protein phosphatase 1 (PP1). SMAPP1 induces PP1 activity in vitro and activates latent HIV-1 provirus in cultured and primary T cells.
T82160 Human IgG1 (D270N) kappa, Isotype Control

HumanIgG1(D270N) kappa, Isotype Control为人-鼠嵌合型抗体, 作为HumanIgG1(D270N)κ 抗体的同型对照品。
T82158 Human IgG1 (S239D/I332E) kappa, Isotype Control

HumanIgG1(S239D/I332E) kappa, Isotype Control为一种人源-鼠源嵌合型单克隆抗体,作为HumanIgG1(S239D/I332E)κ抗体之同型对照物。
T82156 Human IgG3 kappa, Isotype Control

HumanIgG3kappa, Isotype Control为人-鼠嵌合型抗体,作为human IgG3κ抗体同型对照使用。
T78242 Human IgG1 kappa, Isotype Control

HumanIgG1kappa, Isotype Control为人源化单克隆抗体,作为human IgG1κ抗体的同型对照物。
T22856 IgG light chain variable region [Homo sapiens]/IgM/kappa antibody [Mus musculus]

Others Others
IgG has four forms, provides the majority of antibody-based immunity against invading pathogens. The only antibody capable of crossing the placenta to give passive immunity to the fetus. Eliminates pathogens in the early stages of B cell-mediated (humoral
T2806L Lappaconitine HCl

Lappaconitine hydrochloride

Lappaconitine HCl is a centrally acting non-opioid analgesic and class-I antiarrhythmic. It acts by binding to the site-2 receptor and irreversibly blocking hH1 sodium channels.
T36760 KQMEEEAVRLFIEWLKNGGPSSGAPPPS

KQMEEEAVRLFIEWLKNGGPSSGAPPPS is a Exendin-4 peptide derivative. Exendin-4 is a pure GLP-1 receptor agonist. Exendin-4 peptide derivatives are structurally derived from Exendin-4 and may relates to dual GLP-1/glucagon receptor agonists. Their medical use, for example in the treatment of disorders of the metabolic syndrome, including diabetes and obesity, as well as for reduction of excess food intake. These dual GLP-1/glucagon receptor agonists show reduced activity on the GIP receptor to reduce ...
T76028 Amylin (IAPP), feline TFA

Amylin (IAPP), feline TFA,一种来自猫科动物、含37个氨基酸的多肽,为胰岛β细胞的主要分泌物之一。作为调节肽,它能够抑制胰岛素和胰高血糖素的分泌。
T13663 Ds-HAPP

Others Others
Ds-HAPP is an anthrancenyl and dansyl fluorophore ligand.
T78339 Human IgG4 (S228P) kappa, Isotype Control

HumanIgG4(S228P) kappa, Isotype Control为人-鼠嵌合型单克隆抗体,作为humanIgG4(S228P)κ抗体的同型对照使用。
T82159 Human IgG1 (K214R) kappa, Isotype Control

HumanIgG1(K214R) kappa, Isotype Control为HumanIgG1(K214R)κ 抗体的人源化同型对照,属于人-鼠嵌合型抗体。
T78336 Mouse IgG1 kappa, Isotype Control

MouseIgG1kappa Isotype Control 为 mouse IgG1κ 抗体的同型对照鼠源单克隆抗体。
T81760 Mouse IgG1 (D265A) kappa, Isotype Control

MouseIgG1(D265A) kappa, Isotype Control 为鼠源IgG1 κ类同型对照单克隆抗体,适用作为mouse IgG1(D265A)κ抗体的实验对照。
T38039 (E)-C-HDMAPP (ammonium salt)

Synthetic and natural alkyl phosphates, also known as phosphoantigens, stimulate the proliferation of γδ-T lymphocytes. Isopentenyl pyrophosphate, and related derivatives including (E)-hydroxy-dimethyl-allyl pyrophosphate ((E)-HDMAPP), are particularly effective activators of γδ-T cells. (E)-C-HDMAPP is the pyrophosphonate form of (E)-HDMAPP. The pyrophosphonate moiety in (E)-C-HDMAPP is much less susceptible to chemical or enzymatic hydrolysis than its pyrophosphate counterpart. As a result, (E...
T126375 4-O-Methylepisappanol

4-O-Methylepisappanol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126375。
T125353 Apparicine

Apparicine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125353。
T69053 ANAPP3

ANAPP3 is a P2x-purinoceptor antagonist. It affects contractions in various muscle groups and tissues.
T78243 Human IgG2 kappa, Isotype Control

HumanIgG2kappa, Isotype Control为人源化单克隆抗体,作为human IgG2κ抗体的标准同型对照使用。
T73416 BiCAPPA

BiCAPPA 是一个二价抗朊病毒配体。BiCAPPA 可以减少痒病感染细胞中传染性构象形式的朊病毒蛋白 (PrPSc),EC50值为 0.32 μM。
T75860 GTFTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS

GTFTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS 是 Exendin-4多肽衍生物。
T78338 Rat IgG1 kappa, Isotype Control

RatIgG1kappa(Isotype Control)是Rat IgG1κ抗体同型对照的鼠源性单克隆抗体。
T81759 Mouse IgG1 (N297A) kappa, Isotype Control

MouseIgG1(N297A) kappa,Isotype Control 为特定mouse IgG1(N297A)κ 抗体之同型对照,属鼠源单克隆抗体。
T81755 Mouse lgG2a (D265A) kappa, Isotype Control

Mouse lgG2a (D265A) kappa, Isotype Control 为 mouse lgG2a (D265A) 的鼠源单克隆同型对照抗体。
T22069 D-NMAPPD

D-NMAPPD ((1R,2R)-B13) 是一种酸性神经酰胺酶 (acid ceramidase) 抑制剂。D-NMAPPD 通过增强神经酰胺的内源性产生来调节 NMDA 受体特性。D-NMAPPD 具有肠癌治疗的潜力。
T37056 D-erythro-MAPP

D-erythro-MAPP is a derivative of ceramide and an inhibitor of alkaline ceramidase (Ki = 2-13 μM; IC50 = 1-5 μM). It is selective for alkaline ceramidase over acid ceramidase (IC50 = >500 μM) as well as the serine/threonine protein phosphatase CAPP at concentrations up to 10 μM. D-erythro-MAPP increases intracellular ceramide levels, induces cell cycle arrest at the G0/G1 phase, and inhibits growth of HL-60 promyelocytic leukemia cells in a time- and concentration-dependent manner.
T125730 Glucocapparin

Glucocapparin 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125730。
T7490 ARN2966

Beta Amyloid Neuroscience
ARN2966 是高效的,针对 APP 表达的转录后调节剂,能够抑制 APP 的表达从而使 Aβ的量降低。
T28441 PPI-1019

PPI1019,Apan

Beta Amyloid Neuroscience
PPI-1019 是一种 APP( β -淀粉状蛋白 A4 )抑制剂,可用于治疗神经系统疾病和研究阿尔茨海默病(AD)。

化合物

APP-CHMINACA
Cat.No: T30103
Synonym: PX-3,PX3
Target:
JLK6
Cat.No: T21890
Synonym:
Target: Gamma-secretase
δ-secretase inhibitor 11
Cat.No: T9713
Synonym:
Target: Beta Amyloid, Caspase
Pep-1 (uncapped)
Cat.No: TP1798
Synonym: Pep-1 uncapped
Target: Others
DMAPP triammonium
Cat.No: T38570
Synonym: Dimethylallyl diphosphate triammonium,Dimethylallyl Pyrophosphate triammonium salt
Target: Others
Mouse IgG2a kappa, Isotype Control
Cat.No: T78337
Synonym:
Target:
3'-Deoxy-4-O-methylepisappanol
Cat.No: T126471
Synonym:
Target:
APPA
Cat.No: T78612
Synonym:
Target: Apoptosis
FTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS
Cat.No: T75859
Synonym:
Target:
Amylin (IAPP), feline
Cat.No: TP1519
Synonym:
Target:
Human IgG4 kappa, Isotype Control
Cat.No: T78244
Synonym:
Target:
Mouse IgG3 kappa, Isotype Control
Cat.No: T81756
Synonym:
Target:
Human IgG1 (D265A) kappa, Isotype Control
Cat.No: T82161
Synonym:
Target:
Sappanone B
Cat.No: T126481
Synonym:
Target:
Sappanol
Cat.No: T126391
Synonym:
Target:
Mouse IgG2b kappa, Isotype Control
Cat.No: T81758
Synonym:
Target:
Human IgG1 (F405L) kappa, Isotype Control
Cat.No: T78341
Synonym:
Target:
Human IgG1 (N297A) kappa, Isotype Control
Cat.No: T78340
Synonym:
Target:
Mouse IgG2c kappa, Isotype Control
Cat.No: T81757
Synonym:
Target:
Rabbit IgG1 kappa, Isotype Control
Cat.No: T81317
Synonym:
Target:
(SP-4-4)-2-[2-(Amino-KappaN)ethyl]phenyl-KappaC]chloro[dicyclohexyl[2',4',6'-tris(1-methylethyl)[1,1'-biphenyl]-2-yl]phosphine]-Palladium
Cat.No: T66146
Synonym:
Target:
SMAPP1
Cat.No: T28818
Synonym:
Target:
Human IgG1 (D270N) kappa, Isotype Control
Cat.No: T82160
Synonym:
Target:
Human IgG1 (S239D/I332E) kappa, Isotype Control
Cat.No: T82158
Synonym:
Target:
Human IgG3 kappa, Isotype Control
Cat.No: T82156
Synonym:
Target:
Human IgG1 kappa, Isotype Control
Cat.No: T78242
Synonym:
Target:
IgG light chain variable region [Homo sapiens]/IgM/kappa antibody [Mus musculus]
Cat.No: T22856
Synonym:
Target: Others
Lappaconitine HCl
Cat.No: T2806L
Synonym: Lappaconitine hydrochloride
Target:
KQMEEEAVRLFIEWLKNGGPSSGAPPPS
Cat.No: T36760
Synonym:
Target:
Amylin (IAPP), feline TFA
Cat.No: T76028
Synonym:
Target:
Ds-HAPP
Cat.No: T13663
Synonym:
Target: Others
Human IgG4 (S228P) kappa, Isotype Control
Cat.No: T78339
Synonym:
Target:
Human IgG1 (K214R) kappa, Isotype Control
Cat.No: T82159
Synonym:
Target:
Mouse IgG1 kappa, Isotype Control
Cat.No: T78336
Synonym:
Target:
Mouse IgG1 (D265A) kappa, Isotype Control
Cat.No: T81760
Synonym:
Target:
(E)-C-HDMAPP (ammonium salt)
Cat.No: T38039
Synonym:
Target:
4-O-Methylepisappanol
Cat.No: T126375
Synonym:
Target:
Apparicine
Cat.No: T125353
Synonym:
Target:
ANAPP3
Cat.No: T69053
Synonym:
Target:
Human IgG2 kappa, Isotype Control
Cat.No: T78243
Synonym:
Target:
BiCAPPA
Cat.No: T73416
Synonym:
Target:
GTFTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS
Cat.No: T75860
Synonym:
Target:
Rat IgG1 kappa, Isotype Control
Cat.No: T78338
Synonym:
Target:
Mouse IgG1 (N297A) kappa, Isotype Control
Cat.No: T81759
Synonym:
Target:
Mouse lgG2a (D265A) kappa, Isotype Control
Cat.No: T81755
Synonym:
Target:
D-NMAPPD
Cat.No: T22069
Synonym:
Target:
D-erythro-MAPP
Cat.No: T37056
Synonym:
Target:
Glucocapparin
Cat.No: T125730
Synonym:
Target:
ARN2966
Cat.No: T7490
Synonym:
Target: Beta Amyloid
PPI-1019
Cat.No: T28441
Synonym: PPI1019,Apan
Target: Beta Amyloid
Cat. No. Product Name Target Signaling Pathways
T13589 Caesappanin C

Others Others
Caesappanin C 是一种联苯二聚体,提取自印度尼西亚 Caesalpinia sappan L. 的心材中,具有刺激骨形成和再生的潜力。它在体外显示出对原代成骨细胞的强增殖刺激活性。
T32570 Lappaconine

20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol,O(sup 1)-Methyllappaconidine

Others Others
Lappaconine (20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol) 衍生自去甲二萜生物碱。
TJS1779 Protosappanin A

原苏木素A,PTA

NADPH-oxidase; IL Receptor; IκB/IKK; TNF; NF-κB; TLR; ROS; COX; HIV Protease; JAK; NO Synthase; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome; Stem Cells
Protosappanin A (PTA) 是从苏木中分离得到的免疫抑制成分和主要联苯化合物,通过下调 JAK2和 STAT3的磷酸化,抑制 JAK2/STAT3依赖的炎症通路。
T2806 Lappaconitine

高乌甲素,(+)-Lappaconitine

P2X Receptor; Sodium Channel Membrane transporter/Ion channel; Neuroscience
Lappaconitine ((+)-Lappaconitine) 是从高乌头中分离得到的一种天然产物,可用于缓解疼痛的研究。
TMA1570 Sappanone A

NF-κB; Nrf2 Immunology/Inflammation; NF-κB
Sappanone A 是一种高异黄烷酮,通过调节 Nrf2 和 NF-κB 表现出抗炎作用。Sappanone A 可以减轻卵清蛋白引起的哮喘中的过敏性气道炎症。
T6S1780 Protosappanin B

原苏木素B,Q-100961,FT-0689654

Apoptosis Apoptosis
Protosappanin B (Q-100961) 是从苏木中提取的一种多酚类天然产物,具有抗肿瘤作用。它通过激活 MDM2 依赖性泛素化过程诱导 p53 蛋白降解。它显著提高细胞活力,抑制细胞凋亡并上调生长相关蛋白 43 的表达。
T6560 Lappaconitine hydrobromide

氢溴酸高乌甲素,Lappaconite HBr,Allapinine

Others Others
Lappaconitine hydrobromide (Allapinine) 是天然生物碱类化合物,具有抗心律失常作用。
T82338 Ganoapplanoid F

Ganoapplanoid F,一种三萜类化合物,源自Ganoderma applanatum,具有抑制脂肪细胞脂质积累的功能,适用于肥胖研究领域。
TN4410 Lappaol C

P-gp; JNK MAPK; Membrane transporter/Ion channel; Neuroscience
Lappaol C has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. Lappaol C also has potential chemosensitizing activity, it may be candidates for developing novel adjuvant an
TN6463 Lappaol B

Lappaol B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6463,CAS号为 62359-60-8。
TN1245 3-Deoxysappanchalcone

Others; Akt; mTOR Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling
3-Deoxysappanchalcone is an effective HO-1 inducer at the translational level.
TN3063 4-O-Methylsappanol

Antifection Microbiology/Virology
4-O-Methylsappanol shows activity against this fungus against Beauveria bassiana.
TN2923 3'-Deoxy-4-O-methylsappanol

Tyrosinase Proteases/Proteasome
3'-Deoxy-4-O-methylsappanol shows moderate cytotoxicities against cultured human melanoma HMV-II cells with the IC50 value of 872.0 uM ± 2.4.
TN6461 Isolappaol A

Isolappaol A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6461,CAS号为 131400-96-9。
T40454 DMAPP

Dimethylallyl diphosphate

DMAPP, also known as Dimethylallyl pyrophosphate, is an isoprenoid precursor found in all life forms. It serves as an isomer of isopentenyl pyrophosphate (IPP).
TMA2576 Episappanol

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Episappanol has anti-inflammatory activity , it can significantly inhibit the secretion of the pro-inflammatory cytokines interleukin (IL-6) and tumor necrosis factor-alpha (TNF-α).
TN2180 Sappanchalcone

苏木查耳酮

IL Receptor; BCL; TNF Apoptosis; Immunology/Inflammation
Sappanchalcone shows xanthine oxidase inhibitory activity, is a xanthine oxidase inhibitor.
TN5673 10-O-Methylprotosappanin B

10-O-Methylprotosappanin B是一种天然产物,属于豆科云实属,其产品编号为 TN5673,CAS号为 111830-77-4。10-O-Methylprotosappanin B可用作对照参考。
TN1246 3-Deoxysappanone B

Others Others
3-Deoxysappanone B has vasorelaxation effects, it can mediate endothelium- independent vasodilator action in rat thoracic aortic rings.
TN5670 Protosappanin A dimethyl acetal

Protosappanin A dimethyl acetal shows significant xanthine oxidase inhibitory activity in a concentration-dependent manner.
TN1072 Lappaol A

P-gp; JNK MAPK; Membrane transporter/Ion channel; Neuroscience
Lappaol A has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. Lappaol A also has potential chemosensitizing activity, it may be candidates for developing novel adjuvant an
TN6462 Isolappaol C

Isolappaol C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6462,CAS号为 929905-15-7。
TN4411 Lappaol F

CDK; P-gp; JNK Cell Cycle/Checkpoint; MAPK; Membrane transporter/Ion channel; Neuroscience
1. Lappaol F has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. <br/> 2. Lappaol F has potential chemosensitizing activity, it may be candidates for developing novel adju
T14305 Apicidin

OSI 2040

Apoptosis; HDAC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair
Apicidin (OSI 2040) 是组蛋白去乙酰化酶(HDAC)抑制剂,具有抗寄生虫活性和抗增殖活性。Apicidin 通过减少 APP/PS1 小鼠中的 Abeta 负荷来减轻记忆缺陷,抑制细胞生长增殖,诱导细胞凋亡和自噬,可用于研究白血病。
TN1420 Bacopaside I

Others Others
Bacopaside I 是一种皂苷,分离自 Bacopa monniera 中,具有抗氧化活性和清除自由基的功能,有抗抑郁作用。
T79994 7-Deoxy-trans-dihydronarciclasine

7-Deoxy-trans-dihydronarciclasine 作为生物碱,担任烟草花叶病毒(TMV)抑制剂(IC50: 1.80 μM),亦具有抗神经炎症作用,能够降低Tg2576小鼠大脑皮质中Aβ与APP水平。
TN4399 Kushenol C

SGLT; NF-κB; ROS; BACE; Antifection GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience; NF-κB
Kushenol C is a good 1,1-diphenyl-2-picrylhydrazyl (DPPH) scavenger, and it exhibits inhibitory activity against Sodium-dependent glucose cotransporter 2(SGLT2). Kushenol C shows antimicrobial activity against Staphylococcus aureus and Streptococcus mutan

天然产物

Caesappanin C
Cat.No: T13589
Synonym:
Target: Others
Lappaconine
Cat.No: T32570
Synonym: 20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol,O(sup 1)-Methyllappaconidine
Target: Others
Protosappanin A
Cat.No: TJS1779
Synonym: 原苏木素A,PTA
Target: NADPH-oxidase, IL Receptor, IκB/IKK, TNF, NF-κB, TLR, ROS, COX, HIV Protease, JAK, NO Synthase, STAT
Lappaconitine
Cat.No: T2806
Synonym: 高乌甲素,(+)-Lappaconitine
Target: P2X Receptor, Sodium Channel
Sappanone A
Cat.No: TMA1570
Synonym:
Target: NF-κB, Nrf2
Protosappanin B
Cat.No: T6S1780
Synonym: 原苏木素B,Q-100961,FT-0689654
Target: Apoptosis
Lappaconitine hydrobromide
Cat.No: T6560
Synonym: 氢溴酸高乌甲素,Lappaconite HBr,Allapinine
Target: Others
Ganoapplanoid F
Cat.No: T82338
Synonym:
Target:
Lappaol C
Cat.No: TN4410
Synonym:
Target: P-gp, JNK
Lappaol B
Cat.No: TN6463
Synonym:
Target:
3-Deoxysappanchalcone
Cat.No: TN1245
Synonym:
Target: Others, Akt, mTOR
4-O-Methylsappanol
Cat.No: TN3063
Synonym:
Target: Antifection
3'-Deoxy-4-O-methylsappanol
Cat.No: TN2923
Synonym:
Target: Tyrosinase
Isolappaol A
Cat.No: TN6461
Synonym:
Target:
DMAPP
Cat.No: T40454
Synonym: Dimethylallyl diphosphate
Target:
Episappanol
Cat.No: TMA2576
Synonym:
Target: IL Receptor, TNF
Sappanchalcone
Cat.No: TN2180
Synonym: 苏木查耳酮
Target: IL Receptor, BCL, TNF
10-O-Methylprotosappanin B
Cat.No: TN5673
Synonym:
Target:
3-Deoxysappanone B
Cat.No: TN1246
Synonym:
Target: Others
Protosappanin A dimethyl acetal
Cat.No: TN5670
Synonym:
Target:
Lappaol A
Cat.No: TN1072
Synonym:
Target: P-gp, JNK
Isolappaol C
Cat.No: TN6462
Synonym:
Target:
Lappaol F
Cat.No: TN4411
Synonym:
Target: CDK, P-gp, JNK
Apicidin
Cat.No: T14305
Synonym: OSI 2040
Target: Apoptosis, HDAC, Autophagy
Bacopaside I
Cat.No: TN1420
Synonym:
Target: Others
7-Deoxy-trans-dihydronarciclasine
Cat.No: T79994
Synonym:
Target:
Kushenol C
Cat.No: TN4399
Synonym:
Target: SGLT, NF-κB, ROS, BACE, Antifection
共97条,每页50条 1 2
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼