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119

抑制剂 & 化合物

5

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Cat. No. Product Name Target Signaling Pathways
T37078 VEGFR-2-IN-6

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-6(WO 02/059110)是一种 VEGFR2 的强效抑制剂,这是一种在血管生成调控中起关键作用的受体[1]。
T10123 VEGFR-2-IN-9

KDR-in-4

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-9 (KDR-in-4) 是一种高效的 KDR/VEGFR2 抑制剂(IC50:7 nM),可用于研究乳腺癌。
T9979 VEGFR-2-IN-29

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-29是一种 VEGFR2抑制剂。
T2056 VEGFR-2-IN-5

2, 4-Pyrimidinediamine with linker,UNC0064-12,2,4-Pyrimidinediamine with linker

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-5 (UNC0064-12) 是 VEGFR2 抑制剂。
T40581 TIE-2/VEGFR-2 kinase-IN-2

TIE-2/VEGFR-2 kinase-IN-2 is a powerful inhibitor of both VEGFR2 and Tie-2 kinases, displaying noteworthy pIC 50 values of 8.61 and 8.56, respectively. This compound acts as an anti-angiogenic agent, making it highly relevant for cancer research.
T79860 TIE-2/VEGFR-2 kinase-IN-5

VEGFR; Tie-2 Angiogenesis; Tyrosine Kinase/Adaptors
TIE-2/VEGFR-2 kinase-IN-5 是一种高效的 TIE-2VEGFR-2 酪氨酸激酶受体抑制剂,具有的抗血管生成活性,常用于血管生成相关的生物医学研究领域。
T8817 TIE-2/VEGFR-2 kinase-IN-1

TIE-2/VEGFR-2 kinase-IN-1 用于合成TIE-2或者VEGFR-2抑制剂,可用于研究不适当的血管生成的相关疾病。
TP1474 LXW7

Integrin Cytoskeletal Signaling
LXW7 是一种整合素αvβ3抑制剂,是含 Arg-Gly-Asp (RGD) 的环状肽,对αvβ3整联蛋白具有很高的结合亲和力,IC50为 0.68 μM。它可增强 VEGFR-2 磷酸化和 ERK1/2 活化,具有抗炎活性。
T9724 VEGFR2-IN-2

Others Others
VEGFR2-IN-2 具有抗炎和镇痛活性。
T22432 SU5208

3-[(Thien-2-yl)methylene]-2-indolinone

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
SU5208 (3-[(Thien-2-yl)methylene]-2-indolinone) 对血管内皮生长因子受体2具有抑制作用。
T22349 JNJ-38158471

CS-2660

VEGFR; c-RET; c-Kit Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
JNJ-38158471 (CS-2660) 是一种耐受性好的,有口服活性的、高效的、选择性的 VEGFR-2抑制剂 (IC50:40 nM),还能抑制 Ret (IC50:180 nM) 和 Kit (IC50:500 nM)。
T22431 SU5204

3-[(2-Ethoxyphenyl)methylidene]-1H-indol-2-one

EGFR; VEGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
SU5204 (3-[(2-Ethoxyphenyl)methylidene]-1H-indol-2-one) 是酪氨酸激酶抑制剂,是 SU5025 的类似物,对 FLK-1 (VEGFR-2) 和 HER2 的IC50分别为 4 和 51.5 μM。
T5349 SCR-1481B1

麦他替尼胺丁三醇,c-Met inhibitor 2

VEGFR; c-Met/HGFR Angiogenesis; Tyrosine Kinase/Adaptors
SCR-1481B1 (c-Met inhibitor 2) 能够作用于依赖 Met 激活的癌症,对 VEGFR 具有抑制作用。
T13238 Tyrphostin AG1433

SU1433,AG1433

VEGFR; PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
Tyrphostin AG1433 (AG1433) 是选择性的PDGFRβ和VEGFR-2 (Flk-1/KDR)抑制剂,IC50分别为 5.0 μM 和 9.3 μM。Tyrphostin AG1433有防止血管形成的活性。
T6137 KRN-633

KRN633,N-[2-氯-4-[(6,7-二甲氧基-4-喹唑啉基)氧基]苯基]-N'-丙基脲

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
KRN-633 是一种 VEGFR 抑制剂,能够一种 VEGFR1 (IC50:170 nM)、VEGFR2 (IC50:160 nM)、VEGFR3 (IC50:125 nM)。
T61229 VEGFR-2/DHFR-IN-2

VEGFR-2/DHFR-IN-2 (compound 5b) is a dual inhibitor targeting VEGFR-2 and DHFR, with respective IC50 values of 0.623 μM and 9.085 μM. It demonstrates potent cytotoxicity against C26, HepG2, and MCF7 cancer cell lines, with IC50 values ranging from 3.59 μM to 8.38 μM. VEGFR-2/DHFR-IN-2 holds promise for cancer research [1].
T72608 VEGFR-2/BRAF-IN-2

VEGFR-2/BRAF-IN-2 是一种 VEGFR-2和 BRAF 双重抑制剂,对 VEGFR-2、BRAFV600E、BRAFWT 的 IC50分别为 0.111、0.089 和 0.071 µM。VEGFR-2/BRAF-IN-2 诱导细胞凋亡,在 G1 期阻滞细胞周期。
T74518 PROTAC VEGFR-2 degrader-2

PROTACVEGFR-2降解剂-2(PROTAC-4),作为一种PROTACVEGFR-2降解剂,在VEGFR-2上的抑制作用微乎其微(IC50> 1 μM),但对EA.hy926细胞表现出抗增殖能力(IC50为133.248 μM)。
T7493 AG-13958

AG-013958,N-[2-氟-5-[[3-[(1E)-2-(2-吡啶基)乙烯基]-1H-吲唑-6-基]氨基]苯基]-1,3-二甲基-1H-吡唑-5-甲酰胺

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
AG-13958 (AG-013958) 是 VEGFR 酪氨酸激酶抑制剂,可用于年龄相关性黄斑变性 (AMD) 的脉络膜新生血管形成的研究。
T0263 Chloropyramine hydrochloride

Nilfan,盐酸氯吡胺,Alergosan,Halopyramine hydrochloride

FAK; VEGFR; Histamine Receptor Angiogenesis; Cytoskeletal Signaling; GPCR/G Protein; Immunology/Inflammation; Neuroscience; Tyrosine Kinase/Adaptors
Chloropyramine hydrochloride (Alergosan) 是一种组胺受体 H1 拮抗剂,可抑制VEGFR-3和FAK 的生化功能。
T72607 VEGFR-2/BRAF-IN-1

VEGFR-2/BRAF-IN-1 是一种 VEGFR-2和 BRAF 双重抑制剂,对 VEGFR-2、BRAFV600E 和BRAFWT 的IC50分别为 0.049、0.063 和 0.005 µM。VEGFR-2/BRAF-IN-1 诱导细胞凋亡,在 G1/S 期阻滞细胞周期。
T61489 VEGFR-2/DHFR-IN-1

VEGFR-2/DHFR-IN-1 (compound 8b) 是 VEGFR-2和DHFR 的抑制剂,其IC50值分别为 0.384 和 7.881 μM。VEGFR-2/DHFR-IN-1 对大肠埃希菌,粪链球菌,肠沙门氏菌,金黄色酿脓葡萄球菌,MSSA 和MRSA 显示了良好的抗菌活性,MIC 值分别为 16,16,16,8 和 16 μg/mL。VEGFR-2/DHFR-IN-1 对 C26,HepG2 和 CF7 癌细胞系具有良好的细胞毒性,IC50值为 2.97-7.12 μM。VEGFR-2/DHFR-IN-1 可用于癌症的研究。
T74517 PROTAC VEGFR-2 degrader-1

PROTACVEGFR-2 degrader-1(PROTAC-1),一种 PROTACVEGFR-2降解剂,对 VEGFR-2 的抑制作用很小(IC50> 1 μM),对 EA.hy926 细胞的抗增殖活性也很低(IC50> 100μM)。
T12574 PTC299

Emvododstat,(4-chlorophenyl) (1S)-6-chloro-1-(4-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxylate

VEGFR; Dehydrogenase Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors
PTC299 ((4-chlorophenyl) (1S)-6-chloro-1-(4-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxylate) 是一种口服活性的 VEGFA mRNA 翻译抑制剂,可选择性地抑制转录后水平的 VEGF 蛋白合成。它还是二氢乳酸脱氢酶 (DHODH) 的有效抑制剂,可研究血液系统恶性肿瘤。
T61631 VEGFR-2-IN-23

VEGFR-2-IN-23 (compound 11b) is a highly potent and selective inhibitor of VEGFR-2, with an impressive IC 50 value of 0.34 nM. This compound exhibits notable antitumor activity, capable of inducing apoptosis and cell cycle arrest specifically at the G1 phase [1].
T4315 Ki20227

N-[4-[(6,7-二甲氧基-4-喹啉基)氧基]-2-甲氧基苯基]-N'-[1-(2-噻唑基)乙基]脲

c-Fms; VEGFR; CSF-1R; PDGFR; c-Kit Angiogenesis; Tyrosine Kinase/Adaptors
Ki20227 是一种高效的、口服具有活性的、选择性的CSF1R(c-Fms 酪氨酸激酶)抑制剂,对 CSF1R,VEGFR2,c-Kit 和PDGFRβ的IC50分别为 2 nM,12 nM,451 nM 和 217 nM。它可以阻止破骨细胞分化和溶骨性破坏。
T79859 TIE-2/VEGFR-2 kinase-IN-4

TIE-2/VEGFR-2 kinase-IN-4,一种苯并咪唑衍生物,作为有效的TIE-2VEGFR-2酪氨酸激酶受体抑制剂,其IC50值分别为5.2 nM和5.1 nM,适用于血管生成相关研究。
T79858 TIE-2/VEGFR-2 kinase-IN-3

TIE-2/VEGFR-2 kinase-IN-3,为苯并咪唑衍生物,具备高效的抑制作用于TIE-2VEGFR-2受体酪氨酸激酶,其IC50值分别达到6.9 nM和3.5 nM。本化合物主要用于血管生成相关研究。
T80874 VEGFR-2/c-Met-IN-1

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2/c-Met-IN-1为VEGFR-2及c-Met的双重抑制剂,IC50值为138 nM和74 nM,显示出抗肿瘤活性。
T63804 VEGFR-2-IN-28

VEGFR-2-IN-28 是 VEGFR-2 的有效抑制剂 (IC50: 0.83 μM)。VEGFR-2-IN-28 能够诱导细胞凋亡 (apoptosis),表现出抗肿瘤效果。
T64060 VEGFR-2-IN-21

VEGFR-2-IN-21 是 VEGFR-2 的有效抑制剂 (IC50: 0.10 μM),表现出抗癌作用。
T62796 VEGFR-2-IN-13

VEGFR-2-IN-13 (Compound 19a) 是一种有效的 VEGFR-2 抑制剂 (IC50: 3.4 nM)。VEGFR-2-IN-13 能够将 HepG2 的细胞周期停滞在 G2/M 期,诱导细胞凋亡 (apoptosis)。
T62439 VEGFR-2-IN-14

VEGFR-2-IN-14 (Compound 5) 是一种 VEGFR-2 的有效抑制剂。VEGFR-2-IN-14 对 HepG2 细胞在 Pre-G1 期的生长具有抑制作用,并能够诱导细胞凋亡 (apoptosis)。
T63900 VEGFR-2-IN-11

VEGFR-2-IN-11 是 VEGFR-2 的有效抑制剂 (IC50: 60.27 nM),其IC50值为 60.27 nM,能够诱导细胞凋亡 (apoptosis),具有抗癌活性。
T79494 VEGFR-2-IN-31

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-31(compound 3i)是一款针对VEGFR-2的高效抑制剂(IC50=8.93 nM),具有抗前列腺癌的活性。该化合物能够导致细胞周期在S期停滞,并诱导细胞发生凋亡(apoptosis)。
T80872 VEGFR-2-IN-37

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-37(化合物12)是一种VEGFR-2抑制剂,其在200 μM浓度下的抑制率为56.9%。该化合物也是潜在的HUVEC增殖抑制剂。
T79587 hCA/VEGFR-2-IN-2

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
hCA/VEGFR-2-IN-2 (compound 8g) 是一种具有吲哚酮基苯磺酰胺结构的化合物,目标是癌症相关的hCA IX/XII 及VEGFR-2 的双重抑制剂。该化合物对VEGFR-2 表现出强效的抑制作用(IC50=204 nM),且对hCAs有高亲和力,Ki 值分别为 hCA IX 3.6 nM、hCA II 16.1 nM、hCA XII 16.7 nM 以及hCA I 75.3 nM。hCA/VEGFR-2-IN-2 还展现出针对过表达VEGFR-2 的乳腺癌细胞的抗增殖活性。
T62901 VEGFR-2-IN-27

VEGFR-2-IN-27 (compound 7a) 是一种 VEGFR-2 的高效抑制剂 (IC50: 14.8 nM),能够用于抗癌研究。
T63168 VEGFR-2-IN-26

VEGFR-2-IN-26 (compound 5h) 是一种 VEGFR-2 的高效抑制剂 (IC50: 15.5 nM)。VEGFR-2-IN-26 对白血病、中枢神经系统、非小肺、卵巢、肾、前列腺和乳腺癌细胞表现出良好的抗增殖作用。
T61561 VEGFR-2-IN-18

VEGFR-2-IN-18 (Compound 15d) is a high-potency inhibitor of VEGFR-2, with an IC 50 value of 60 nM. This compound effectively initiates cell apoptosis and demonstrates significant antitumor properties [1].
T61137 VEGFR-2-IN-19

VEGFR-2-IN-19 (Compound 15b) is a highly efficacious inhibitor of VEGFR2, a receptor involved in angiogenesis. Its mechanism of action involves the induction of cellular apoptosis and elevation of intracellular reactive oxygen species. Due to these properties, VEGFR-2-IN-19 holds promise as an effective anticancer agent [1].
T62314 VEGFR-2-IN-25

VEGFR-2-IN-25 (compound 5d) 是一种 VEGFR-2 的高效抑制剂 (IC50: 12.1 nM)。VEGFR-2-IN-25 能够用于研究抗癌。
T63002 VEGFR-2-IN-15

VEGFR-2-IN-15 (Compound 14b) 是一种 VEGFR-2 的有效抑制剂。VEGFR-2-IN-15 能够抑制 HepG2 细胞在 Pre-G1 期的生长,诱导细胞凋亡。
T79495 VEGFR-2-IN-32

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-32(Comp 3a)作为一种VEGFR-2的抑制剂,其IC50值为8.93 nM。该化合物对PC-3细胞表现出细胞毒性,IC50为1.22 μM,适用于前列腺癌研究。
T79403 VEGFR-2-IN-36

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-36(compound 15)是一种具有抗癌活性的VEGFR-2抑制剂(IC50:0.067 μM)和凋亡诱导剂。该化合物能够上调BAX水平和下调Bcl-2水平,对MCF-7(IC50=0.42 μM)和HepG2(IC50=0.22 μM)癌细胞展现出明显的毒性效果。
T37079 VEGFR2 Kinase Inhibitor II

Vascular endothelial growth factor receptor 2 (VEGFR2, also known as KDR and FLK1) is a receptor tyrosine kinase that regulates angiogenesis, vascular development, and embryonic hematopoiesis in response to VEGF isoforms A, C, and D. VEGFR2 kinase inhibitor II is a reversible, cell-permeable inhibitor of VEGFR2's kinase activity (IC50 = 70 nM). It less potently inhibits the platelet-derived growth factor receptor β (PDGFRβ; IC50 = 920 nM) and related receptor and non-receptor tyrosine kinases. V...
T63822 VEGFR-2-IN-22

VEGFR-2-IN-22 (Compound 25) 是 VEGFR-2 和 β-tubulin 聚合抑制剂,对 VEGFR-2 的 IC50=19.82 nM。VEGFR-2-IN-22 能够诱导细胞凋亡 (apoptosis)。
T62763 VEGFR-2-IN-12

VEGFR-2-IN-12 (compound 6g) 是一种 2-oxoquinoxalinyl-1,2,4-triazole,是一种 VEGFR-2 的有效抑制剂 (IC50: 0.037 μM)。VEGFR-2-IN-12 能够高度抑制 MCF-7 细胞的生长 (GI50: 1.6 μM)。VEGFR-2-IN-12 具有抗肿瘤作用。
T63722 VEGFR-2-IN-24

VEGFR-2-IN-24 是 VEGFR-2 的有效抑制剂 (IC50: 0.22 μM),能够用于研究肿瘤。
T62071 VEGFR-2-IN-16

VEGFR-2-IN-16 (Compound 15b) 是一种 VEGFR-2 的有效抑制剂 (IC50: 86.36 nM),表现出抗肿瘤效果。

化合物

VEGFR-2-IN-6
Cat.No: T37078
Synonym:
Target: VEGFR
VEGFR-2-IN-9
Cat.No: T10123
Synonym: KDR-in-4
Target: VEGFR
VEGFR-2-IN-29
Cat.No: T9979
Synonym:
Target: VEGFR
VEGFR-2-IN-5
Cat.No: T2056
Synonym: 2, 4-Pyrimidinediamine with linker,UNC0064-12,2,4-Pyrimidinediamine with linker
Target: VEGFR
TIE-2/VEGFR-2 kinase-IN-2
Cat.No: T40581
Synonym:
Target:
TIE-2/VEGFR-2 kinase-IN-5
Cat.No: T79860
Synonym:
Target: VEGFR, Tie-2
TIE-2/VEGFR-2 kinase-IN-1
Cat.No: T8817
Synonym:
Target:
LXW7
Cat.No: TP1474
Synonym:
Target: Integrin
VEGFR2-IN-2
Cat.No: T9724
Synonym:
Target: Others
SU5208
Cat.No: T22432
Synonym: 3-[(Thien-2-yl)methylene]-2-indolinone
Target: VEGFR
JNJ-38158471
Cat.No: T22349
Synonym: CS-2660
Target: VEGFR, c-RET, c-Kit
SU5204
Cat.No: T22431
Synonym: 3-[(2-Ethoxyphenyl)methylidene]-1H-indol-2-one
Target: EGFR, VEGFR, HER
SCR-1481B1
Cat.No: T5349
Synonym: 麦他替尼胺丁三醇,c-Met inhibitor 2
Target: VEGFR, c-Met/HGFR
Tyrphostin AG1433
Cat.No: T13238
Synonym: SU1433,AG1433
Target: VEGFR, PDGFR
KRN-633
Cat.No: T6137
Synonym: KRN633,N-[2-氯-4-[(6,7-二甲氧基-4-喹唑啉基)氧基]苯基]-N'-丙基脲
Target: VEGFR
VEGFR-2/DHFR-IN-2
Cat.No: T61229
Synonym:
Target:
VEGFR-2/BRAF-IN-2
Cat.No: T72608
Synonym:
Target:
PROTAC VEGFR-2 degrader-2
Cat.No: T74518
Synonym:
Target:
AG-13958
Cat.No: T7493
Synonym: AG-013958,N-[2-氟-5-[[3-[(1E)-2-(2-吡啶基)乙烯基]-1H-吲唑-6-基]氨基]苯基]-1,3-二甲基-1H-吡唑-5-甲酰胺
Target: VEGFR
Chloropyramine hydrochloride
Cat.No: T0263
Synonym: Nilfan,盐酸氯吡胺,Alergosan,Halopyramine hydrochloride
Target: FAK, VEGFR, Histamine Receptor
VEGFR-2/BRAF-IN-1
Cat.No: T72607
Synonym:
Target:
VEGFR-2/DHFR-IN-1
Cat.No: T61489
Synonym:
Target:
PROTAC VEGFR-2 degrader-1
Cat.No: T74517
Synonym:
Target:
PTC299
Cat.No: T12574
Synonym: Emvododstat,(4-chlorophenyl) (1S)-6-chloro-1-(4-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carboxylate
Target: VEGFR, Dehydrogenase
VEGFR-2-IN-23
Cat.No: T61631
Synonym:
Target:
Ki20227
Cat.No: T4315
Synonym: N-[4-[(6,7-二甲氧基-4-喹啉基)氧基]-2-甲氧基苯基]-N'-[1-(2-噻唑基)乙基]脲
Target: c-Fms, VEGFR, CSF-1R, PDGFR, c-Kit
TIE-2/VEGFR-2 kinase-IN-4
Cat.No: T79859
Synonym:
Target:
TIE-2/VEGFR-2 kinase-IN-3
Cat.No: T79858
Synonym:
Target:
VEGFR-2/c-Met-IN-1
Cat.No: T80874
Synonym:
Target: VEGFR
VEGFR-2-IN-28
Cat.No: T63804
Synonym:
Target:
VEGFR-2-IN-21
Cat.No: T64060
Synonym:
Target:
VEGFR-2-IN-13
Cat.No: T62796
Synonym:
Target:
VEGFR-2-IN-14
Cat.No: T62439
Synonym:
Target:
VEGFR-2-IN-11
Cat.No: T63900
Synonym:
Target:
VEGFR-2-IN-31
Cat.No: T79494
Synonym:
Target: VEGFR
VEGFR-2-IN-37
Cat.No: T80872
Synonym:
Target: VEGFR
hCA/VEGFR-2-IN-2
Cat.No: T79587
Synonym:
Target: VEGFR
VEGFR-2-IN-27
Cat.No: T62901
Synonym:
Target:
VEGFR-2-IN-26
Cat.No: T63168
Synonym:
Target:
VEGFR-2-IN-18
Cat.No: T61561
Synonym:
Target:
VEGFR-2-IN-19
Cat.No: T61137
Synonym:
Target:
VEGFR-2-IN-25
Cat.No: T62314
Synonym:
Target:
VEGFR-2-IN-15
Cat.No: T63002
Synonym:
Target:
VEGFR-2-IN-32
Cat.No: T79495
Synonym:
Target: VEGFR
VEGFR-2-IN-36
Cat.No: T79403
Synonym:
Target: VEGFR
VEGFR2 Kinase Inhibitor II
Cat.No: T37079
Synonym:
Target:
VEGFR-2-IN-22
Cat.No: T63822
Synonym:
Target:
VEGFR-2-IN-12
Cat.No: T62763
Synonym:
Target:
VEGFR-2-IN-24
Cat.No: T63722
Synonym:
Target:
VEGFR-2-IN-16
Cat.No: T62071
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8213 Isolinderalactone

NOS; STAT Immunology/Inflammation; JAK/STAT signaling; Stem Cells
Isolinderalactone 具有抗炎和抗癌能力,具有中等的 iNOS 抑制活性,IC50 值为 0.30 uM。
T13108 Pamufetinib

H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115

VEGFR; c-Met/HGFR Angiogenesis; Tyrosine Kinase/Adaptors
Pamufetinib (TAS-115) 是VEGFR 和c-Met/HGFR 抑制剂,能够抑制 rVEGFR2 (IC50:30 nM)和 rMET (IC50:32 nM)的活性。
T14055 5Z-7-Oxozeaenol

FR148083,L783279,LL-Z 1640-2

VEGFR; FLT; MEK; MAPK; PDGFR; Antibiotic; Src Angiogenesis; MAPK; Microbiology/Virology; Tyrosine Kinase/Adaptors
5Z-7-Oxozeaenol (FR148083) 是一种天然抗原生动物抑制剂,不可逆的选择性抑制 TAK1和 VEGF-R2,IC50值分别为 8 nM 和 52 nM。
TN1557 Decursinol angelate

ERK; VEGFR; PKC; JNK Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Tyrosine Kinase/Adaptors
Decursinol angelate 是从朝鲜当归根部分离得到的一种天然产物,是 PKC 激酶的激活剂,有细胞毒性,抗肿瘤和抗炎活性。
T38250 L-Sepiapterin

L-Sepiapterin, also known as Sepiapterin, is a precursor compound crucial for the production of tetrahydrobiopterin (BH4), which serves as a coenzyme for endothelial nitric oxide synthase (eNOS). This compound demonstrates its efficacy by improving endothelial dysfunction in small mesenteric arteries from db/db mice and promoting angiogenesis. Moreover, L-Sepiapterin exerts inhibitory effects on cellular proliferation and migration in ovarian cancer cells through the down-regulation of p70S6K-de...

天然产物

Isolinderalactone
Cat.No: T8213
Synonym:
Target: NOS, STAT
Pamufetinib
Cat.No: T13108
Synonym: H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115
Target: VEGFR, c-Met/HGFR
5Z-7-Oxozeaenol
Cat.No: T14055
Synonym: FR148083,L783279,LL-Z 1640-2
Target: VEGFR, FLT, MEK, MAPK, PDGFR, Antibiotic, Src
Decursinol angelate
Cat.No: TN1557
Synonym:
Target: ERK, VEGFR, PKC, JNK
L-Sepiapterin
Cat.No: T38250
Synonym:
Target:
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