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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T8708 Paroxetine

Serotonin Transporter Neuroscience
Paroxetine 是选择性血清素再摄取抑制剂,是苯基哌啶的衍生物。 它对于甲肾上腺素摄取抑制功能较弱,但比该位点其他SSRIs 更有效。
T12232 Nitroxazepine

CIBA 2330Go

Serotonin Transporter Neuroscience
Nitroxazepine (CIBA 2330Go) 是三环抗抑郁化合物,是一种 5-羟色胺去甲肾上腺素再摄取抑制剂,可用于抗抑郁的研究。
T7061 Duloxetine

Serotonin Transporter Neuroscience
Duloxetine 是一种 5 羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂,Ki=4.6 nM,可作用于广泛性焦虑症的研究。
T0450 Fluoxetine

氟西汀,LY-110140

5-HT Receptor; Serotonin Transporter; MRP; Autophagy Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Fluoxetine (LY-110140) 是一种高度特异性的血清素摄取抑制剂,是选择性 5-羟色胺 (5-HT) 再吸收抑制剂。Fluoxetine 具有抗抑郁活性。
T22714 Decynium 22

Others Others
Decynium 22 是有机阳离子转运蛋白和单胺转运蛋白的抑制剂,具有抗抑郁作用。
T1189 Milnacipran hydrochloride

盐酸米那普仑,Milnacipran HCl,Savella,Dalcipran

Serotonin Transporter; Norepinephrine Neuroscience
Milnacipran hydrochloride (Savella) 是一种5-羟色胺-去甲肾上腺素重吸收抑制剂(SNRI),可用于纤维肌痛的研究。
T2594 Dextromilnacipran

Levomilnacipran,左旋米那普仑

Serotonin Transporter; Norepinephrine Neuroscience
Dextromilnacipran (Levomilnacipran) 是米那普仑的对映体,是一种选择性 5- 羟色胺和去甲肾上腺素(5-HT/NE)再摄取抑制剂,也是一种人类 α 肾上腺素能受体拮抗剂,IC50=3.4 μM。
T22453 Venlafaxine

Wy 45030,文拉法辛

Serotonin Transporter Neuroscience
Venlafaxine (Wy 45030) 是一种口服有效的 5-羟色胺 (5-HT)/去甲肾上腺素 (NE) 重摄取的双重抑制剂,具有抗抑郁活性。
T11087 DOV-216,303 Free Base

DOV-216303

Dopamine Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
DOV-216,303 Free Base (DOV-216303) 是血清素、去甲肾上腺素和多巴胺再摄取的抑制剂,IC50 为 14、20 和 78 nM。 DOV-216,303 Free Base 具有抗抑郁作用。
T7940 Milnacipran ((1S-cis) hydrochloride)

左旋米那普林,Levomilnacipran Hydrochloride

Serotonin Transporter Neuroscience
Milnacipran (1S-cis) hydrochloride (Levomilnacipran Hydrochloride) 是 5-羟色胺去甲肾上腺素再摄取抑制剂,用于研究纤维肌痛。
T0482 Sertraline hydrochloride

Sertraline HCl,CP-51974-1 HCl,盐酸舍曲林

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Sertraline hydrochloride (Sertraline HCl) 是选择性 5- 羟色胺再吸收抑制剂类的抗抑郁剂,可用于多种疾病的研究,如重度抑郁症和强迫症。
T10758L Centanafadine hydrochloride

EB-1020 hydrochloride

Dopamine Receptor; Serotonin Transporter; Adrenergic Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Centanafadine hydrochloride (EB-1020 hydrochloride) 是一种去甲肾上腺素(NE)/多巴胺(DA)转运的双抑制剂,还能抑制5-羟色胺(serotonin)转运体。它对人 NE,DA 和5-羟色胺转运体的 IC50值分别为6 nM,38 nM 和 83 nM。
T3526 Dasotraline hydrochloride

SEP-225289 hydrochloride,达索曲林盐酸盐

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Dasotraline hydrochloride (SEP-225289 hydrochloride) 是具有阻断多巴胺 (IC50=4 nM),去甲肾上腺素 (IC50=6 nM) 和三羟色胺转运蛋白 (IC50=11 nM)的三重再摄取抑制剂。
T1279 Vilazodone

维拉佐酮,SB659746A,EMD 68843

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Vilazodone (SB659746A) 是一种可口服的选择性 5 -羟色胺再摄取抑制剂 (SSRI) 和部分5-HT1A 受体激动剂。它有抗抑郁作用,可用于抑郁症和情绪性疾病的研究。
T0450L Fluoxetine hydrochloride

Fluoxetine HCl,盐酸氟西汀,LY-110140,Lilly110140

5-HT Receptor; Serotonin Transporter; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Fluoxetine hydrochloride (Lilly110140) 是一种高度特异性血清素摄取抑制剂。它被用作抗抑郁药,并且通常比传统的抗抑郁药具有更可接受的副作用特征。
T2395 Vortioxetine

沃替西汀,Lu AA 21004

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Vortioxetine (Lu AA 21004) 是5-HT1A、5-HT1B、5-HT3A、5-HT7受体和 5-羟色胺转运体抑制剂,Ki 值分别为 15、33、3.7、19 和 1.6 nM。它作为抗抑郁药,用于治疗重度抑郁症。
T7941 Imipramine hydrochloride

盐酸丙咪嗪,Imipramine (hydrochloride),Tofranil,G 22355,Imipramine HCl,Melipramine

Serotonin Transporter Neuroscience
Imipramine hydrochloride (Imipramine HCl) 可抑制血清素转运蛋白,IC50=32 nM。它可阻止胰酶的易位,阻碍 MV 和外泌体的分泌。
T0472 Venlafaxine hydrochloride

Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Venlafaxine hydrochloride (Wy 45030 hydrochloride) 是一种口服有效的 5-羟色胺 (5-HT)/去甲肾上腺素 (NE) 重摄取的双重抑制剂,具有抗抑郁活性。
T6232 Vilazodone Hydrochloride

盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl

Others; 5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience; Others
Vilazodone Hydrochloride (EMD 68843) 是 5-HT1A 受体和特异性 5-羟色胺再摄取抑制剂(SSRI) 的部分激动剂,用于治疗重度抑郁症。
T1077 Fluvoxamine maleate

氟伏沙明马来酸盐,马来酸氟伏沙明,MK-264,DU-23000 (maleate)

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Fluvoxamine maleate (DU-23000 (maleate)) 是一种5-羟色胺再吸收抑制剂,有抗抑郁作用。
T6493 Escitalopram Oxalate

草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate

Others; 5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience; Others
Escitalopram Oxalate ((S)-(+)Citalopram oxalate) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。
T2092 Amitifadine hydrochloride

DOV-21947 hydrochloride,EB-1010 hydrochloride

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Amitifadine hydrochloride (EB-1010 hydrochloride) 是一种 5-羟色胺-去甲肾上腺素-多巴胺的再摄取抑制剂(SNDRI),其在 HEK 293 细胞中测得的 IC50值分别为 12, 23, 96 nM。
T0255 Clomipramine hydrochloride

Clomipramine HCl,Anafranil,盐酸氯米帕明

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine; GST GPCR/G Protein; Neuroscience; oxidation-reduction
Clomipramine hydrochloride (Anafranil) 是一种5-羟色胺转运体(Ki:0.14 nM)、去甲肾上腺素转运体(Ki:54 nM)和多巴胺转运体(Ki:3 nM)阻断剂。
T21013 Clomipramine

Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明

5-HT Receptor GPCR/G Protein; Neuroscience
Clomipramine (Clomicalm) 是一种三环类抗抑郁药,能够有效阻断 5-HT 再摄取 (IC50:1.5 nM) ,可用于研究强迫症 (OCD) 及抑郁症。
T1636 Paroxetine hydrochloride

Paroxetine HCl,BRL29060 hydrochloride,FG-7051,BRL29060A,盐酸帕罗西汀

5-HT Receptor; Serotonin Transporter; GRK; AChR; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Paroxetine hydrochloride (Paroxetine HCl) 是一种血清素摄取抑制剂,能抑制 GRK2 活性,IC50值为 14 μM。它可研究抑郁症。
T6188 Desvenlafaxine succinate hydrate

O-Desmethylvenlafaxine succinate hydrate,WY 45233 Succinate,琥珀酸去甲文拉法辛,Desvenlafaxine Succinate

5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Desvenlafaxine succinate hydrate (WY 45233 Succinate) 是 Venlafaxine 主要代谢物的丁二酸盐形式,在人多巴胺转运体上显示弱的结合亲和力。它是具有口服活性的、能透过血脑屏障的5-HT 和 去甲肾上腺素再摄取的抑制剂,对 hSERT 和 hNET 的IC50值分别为47.3 nM 和531.3 nM。
T6461 Dapoxetine hydrochloride

LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Dapoxetine hydrochloride (LY-210448 hydrochloride) 是一种具有口服活性的、选择性的血清素再摄取 (serotonin reuptake) 抑制剂 (SSRI),可用于研究早泄 (PE) 。
T0991 Desipramine hydrochloride

NSC-114901,Desmethylimipramine,盐酸去甲咪嗪,JB-8181,EX-4355,Norimipramine,G-35020

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor GPCR/G Protein; Neuroscience
Desipramine hydrochloride (Norimipramine) 是一种二苯并氮杂类衍生物三环类抗抑郁药,可作为选择性去甲肾上腺素再摄取抑制剂。 它还显示出较弱的 5-羟色胺再摄取抑制、α1 阻断、抗组胺和抗胆碱能作用。
T1471 Duloxetine hydrochloride

Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Duloxetine hydrochloride ((S)-Duloxetine hydrochloride) 是一种 5-羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂 (SNRI),Ki=4.6 nM,可用于广泛性焦虑症的研究。
T2395L Vortioxetine hydrobromide

氢溴酸沃替西汀,Vortioxetine (Lu AA21004) HBr,Vortioxetine HBr,盐酸沃替西汀,Lu AA21004 hydrobromide

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Vortioxetine hydrobromide (Lu AA21004 hydrobromide) 是5-HT1A、5-HT1B、5-HT3A、5-HT7受体和5-羟色胺转运体(SERT)的抑制剂,Ki 值分别为 15、33、3.7、19 和 1.6 nM。
T0678 Amitriptyline hydrochloride

Amitriptyline HCl,Tryptizol,盐酸阿米替林,Domical,Annoyltin

Trk receptor; Sigma receptor; 5-HT Receptor; Serotonin Transporter; Sodium Channel; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; Tyrosine Kinase/Adaptors
Amitriptyline hydrochloride (Annoyltin) 是血清素再摄取转运体和去甲肾上腺素再摄取转运体抑制剂,还与多巴胺再摄取转运体结合,其Ki 为 2.58 μM。它也抑制肾上腺素能受体、毒蕈碱受体、组胺受体、5-羟色胺受体。它是TrkA 和TrkA 受体的激动剂,具有强神经营养活性和有抗抑郁作用。
T1483 Citalopram hydrobromide

Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,氢溴酸西酞普兰,Citalopram HBr

5-HT Receptor; Serotonin Transporter; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Citalopram hydrobromide (XU-62-320) 是一种选择性 5-羟色胺再摄取抑制剂,可选择性地抑制 CNS 神经元对 5-羟色胺的再摄取,从而增强中枢神经系统中的 5-羟色胺能活性,也具有抗抑郁活性。它抑制兔血小板中 5-HT 的摄取,IC50为 14 nM。
T0039 Dapoxetine

达波西汀,Dapoxetina,Dapoxetinum

Others; 5-HT Receptor GPCR/G Protein; Neuroscience; Others
Dapoxetine (Dapoxetina) 是一种选择性5-羟色胺再摄取抑制剂,用于治疗早泄。
T1580 Desvenlafaxine

去甲文拉法辛,WY 45233 Succinate,O-Desmethylvenlafaxine

5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Desvenlafaxine (O-Desmethylvenlafaxine) 是 Venlafaxine 主要代谢物的丁二酸盐形式,在人多巴胺转运体上显示弱的结合亲和力。它是一种具有口服活性的、能透过血脑屏障的5-HT 和去甲肾上腺素再摄取的抑制剂,对 hSERT 和 hNET 的IC50值分别为 47.3 nM 和 531.3 nM。

化合物

Paroxetine
Cat.No: T8708
Synonym:
Target: Serotonin Transporter
Nitroxazepine
Cat.No: T12232
Synonym: CIBA 2330Go
Target: Serotonin Transporter
Duloxetine
Cat.No: T7061
Synonym:
Target: Serotonin Transporter
Fluoxetine
Cat.No: T0450
Synonym: 氟西汀,LY-110140
Target: 5-HT Receptor, Serotonin Transporter, MRP, Autophagy
Decynium 22
Cat.No: T22714
Synonym:
Target: Others
Milnacipran hydrochloride
Cat.No: T1189
Synonym: 盐酸米那普仑,Milnacipran HCl,Savella,Dalcipran
Target: Serotonin Transporter, Norepinephrine
Dextromilnacipran
Cat.No: T2594
Synonym: Levomilnacipran,左旋米那普仑
Target: Serotonin Transporter, Norepinephrine
Venlafaxine
Cat.No: T22453
Synonym: Wy 45030,文拉法辛
Target: Serotonin Transporter
DOV-216,303 Free Base
Cat.No: T11087
Synonym: DOV-216303
Target: Dopamine Receptor, Serotonin Transporter, Norepinephrine
Milnacipran ((1S-cis) hydrochloride)
Cat.No: T7940
Synonym: 左旋米那普林,Levomilnacipran Hydrochloride
Target: Serotonin Transporter
Sertraline hydrochloride
Cat.No: T0482
Synonym: Sertraline HCl,CP-51974-1 HCl,盐酸舍曲林
Target: 5-HT Receptor, Serotonin Transporter
Centanafadine hydrochloride
Cat.No: T10758L
Synonym: EB-1020 hydrochloride
Target: Dopamine Receptor, Serotonin Transporter, Adrenergic Receptor, Norepinephrine
Dasotraline hydrochloride
Cat.No: T3526
Synonym: SEP-225289 hydrochloride,达索曲林盐酸盐
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine
Vilazodone
Cat.No: T1279
Synonym: 维拉佐酮,SB659746A,EMD 68843
Target: 5-HT Receptor, Serotonin Transporter
Fluoxetine hydrochloride
Cat.No: T0450L
Synonym: Fluoxetine HCl,盐酸氟西汀,LY-110140,Lilly110140
Target: 5-HT Receptor, Serotonin Transporter, Autophagy
Vortioxetine
Cat.No: T2395
Synonym: 沃替西汀,Lu AA 21004
Target: 5-HT Receptor, Serotonin Transporter
Imipramine hydrochloride
Cat.No: T7941
Synonym: 盐酸丙咪嗪,Imipramine (hydrochloride),Tofranil,G 22355,Imipramine HCl,Melipramine
Target: Serotonin Transporter
Venlafaxine hydrochloride
Cat.No: T0472
Synonym: Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride
Target: 5-HT Receptor, Serotonin Transporter
Vilazodone Hydrochloride
Cat.No: T6232
Synonym: 盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl
Target: Others, 5-HT Receptor, Serotonin Transporter
Fluvoxamine maleate
Cat.No: T1077
Synonym: 氟伏沙明马来酸盐,马来酸氟伏沙明,MK-264,DU-23000 (maleate)
Target: 5-HT Receptor, Serotonin Transporter
Escitalopram Oxalate
Cat.No: T6493
Synonym: 草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate
Target: Others, 5-HT Receptor, Serotonin Transporter
Amitifadine hydrochloride
Cat.No: T2092
Synonym: DOV-21947 hydrochloride,EB-1010 hydrochloride
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine
Clomipramine hydrochloride
Cat.No: T0255
Synonym: Clomipramine HCl,Anafranil,盐酸氯米帕明
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine, GST
Clomipramine
Cat.No: T21013
Synonym: Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明
Target: 5-HT Receptor
Paroxetine hydrochloride
Cat.No: T1636
Synonym: Paroxetine HCl,BRL29060 hydrochloride,FG-7051,BRL29060A,盐酸帕罗西汀
Target: 5-HT Receptor, Serotonin Transporter, GRK, AChR, Autophagy
Desvenlafaxine succinate hydrate
Cat.No: T6188
Synonym: O-Desmethylvenlafaxine succinate hydrate,WY 45233 Succinate,琥珀酸去甲文拉法辛,Desvenlafaxine Succinate
Target: 5-HT Receptor, Serotonin Transporter, Norepinephrine
Dapoxetine hydrochloride
Cat.No: T6461
Synonym: LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy
Target: 5-HT Receptor, Serotonin Transporter
Desipramine hydrochloride
Cat.No: T0991
Synonym: NSC-114901,Desmethylimipramine,盐酸去甲咪嗪,JB-8181,EX-4355,Norimipramine,G-35020
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor
Duloxetine hydrochloride
Cat.No: T1471
Synonym: Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine
Vortioxetine hydrobromide
Cat.No: T2395L
Synonym: 氢溴酸沃替西汀,Vortioxetine (Lu AA21004) HBr,Vortioxetine HBr,盐酸沃替西汀,Lu AA21004 hydrobromide
Target: 5-HT Receptor, Serotonin Transporter
Amitriptyline hydrochloride
Cat.No: T0678
Synonym: Amitriptyline HCl,Tryptizol,盐酸阿米替林,Domical,Annoyltin
Target: Trk receptor, Sigma receptor, 5-HT Receptor, Serotonin Transporter, Sodium Channel, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
Citalopram hydrobromide
Cat.No: T1483
Synonym: Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,氢溴酸西酞普兰,Citalopram HBr
Target: 5-HT Receptor, Serotonin Transporter, Autophagy
Dapoxetine
Cat.No: T0039
Synonym: 达波西汀,Dapoxetina,Dapoxetinum
Target: Others, 5-HT Receptor
Desvenlafaxine
Cat.No: T1580
Synonym: 去甲文拉法辛,WY 45233 Succinate,O-Desmethylvenlafaxine
Target: 5-HT Receptor, Serotonin Transporter, Norepinephrine
Cat. No. Product Name Target Signaling Pathways
T7521 Azaphen

Pipofezin hydrochloride,阿扎吩,Pipofezine hydrochloride,Azafen

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Azaphen (Pipofezin hydrochloride) 是一种 5-羟色胺重吸收抑制剂。
T1317 Cinchonidine

奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine

5-HT Receptor; Serotonin Transporter; Parasite GPCR/G Protein; Microbiology/Virology; Neuroscience
Cinchonidine (L-Cinchonidine) 是在金鸡纳和角蒿中发现的一种生物碱,有抗疟活性。 它是用于有机化学中不对称合成的砌块,是血清素转运蛋白的弱抑制剂。
T0185 Escitalopram

Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。

天然产物

Azaphen
Cat.No: T7521
Synonym: Pipofezin hydrochloride,阿扎吩,Pipofezine hydrochloride,Azafen
Target: 5-HT Receptor, Serotonin Transporter
Cinchonidine
Cat.No: T1317
Synonym: 奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine
Target: 5-HT Receptor, Serotonin Transporter, Parasite
Escitalopram
Cat.No: T0185
Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
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