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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T79125 Protein kinase inhibitor 5

Trk receptor Tyrosine Kinase/Adaptors
Protein kinase inhibitor 5 作为一种有效的TRK-A抑制剂,其IC50值达到1.8 nM,且能抑制细胞活力。
T9034 MK2-IN-3

MK2 Inhibitor III

MAPK MAPK
MK2-IN-3 (MK2 Inhibitor III) 是选择性的 MAPKAP-K2 (MK-2)抑制剂(IC50:8.5 nM),能够抑制 U937 细胞及体内 TNFα 的生成。
T5508 PF-AKT400

(S)-N-[[3-氨基-1-(5-乙基-7H-吡咯并[2,3-D]嘧啶-4-基)吡咯烷-3-基]甲基]-2,4-二氟苯甲酰胺,AKT protein kinase inhibitor

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
PF-AKT400 (AKT protein kinase inhibitor) 是 ATP 竞争性的、选择性的 Akt 抑制剂,对 PKBα(IC50=0.5 nM) 的选择性比 PKA(IC50=450 nM) 高 900 倍。
T79126 Protein kinase inhibitor 5 sulfate hydrate

Trk receptor Tyrosine Kinase/Adaptors
Protein kinase inhibitor 5 sulfate hydrate 作为TRK-A抑制剂,具有高效性,其IC50值仅为1.8 nM,能有效抑制细胞活力。
T60109 Protein kinase inhibitor H-7

5-(2-methylpiperazine-1-sulfonyl)isoquinoline,蛋白激酶抑制剂H-7,1-(5-Isoquinolinylsulfonyl)-2-methylpiperazine

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Protein kinase inhibitor H-7 (5-(2-methylpiperazine-1-sulfonyl)isoquinoline) 是有效的蛋白激酶 C (PKC) 和环核苷酸依赖性蛋白激酶抑制剂,抑制 PKC 的 Ki 值为 6 μM。
T7196 HG-10-102-01

[4-[[5-氯-4-(甲基氨基)-2-嘧啶基]氨基]-3-甲氧基苯基]-4-吗啉基甲酮

LRRK2 Autophagy
HG-10-102-01 是富含亮氨酸重复激酶 2 和突变型G2019S 抑制剂,IC50分别为20.3 nM 和3.2 nM。
T4489 AKT-IN-1

AZD26,AZD-26,6-[4-(1-氨基环丁基)苯基]-5-苯基-3-吡啶甲酰胺,AZD 26

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
AKT-IN-1 (AZD-26) 是一种变构的 AKT 抑制剂,其 IC50=1.042 μM。
T8656 CAY10404

3-(4-METHYLSULPHONYLPHENYL)-4-PHENYL-5-T

Apoptosis; Akt; COX Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Neuroscience; PI3K/Akt/mTOR signaling
CAY10404 (3-(4-METHYLSULPHONYLPHENYL)-4-PHENYL-5-T) 是一种有效且高度选择性的 COX-2 和 COX-1 抑制剂。 它还是 PKB/Akt 和 MAPK 信号通路的有效抑制剂,可诱导 NSC-LC 细胞凋亡,具有镇痛、抗炎和抗癌活性。
T4185 lavendustin C

HDBA,NSC 666251,N-(2,5-二羟基苄基)-5-氨基水杨酸

CaMK; EGFR; Tyrosinase; Src Angiogenesis; JAK/STAT signaling; Neuroscience; Proteases/Proteasome; Tyrosine Kinase/Adaptors
lavendustin C (NSC 666251) 是 Ca2+钙调蛋白依赖性激酶 II 抑制剂,IC50为 0.2 µM。它抑制 EGFR 相关酪氨酸激酶和 pp60c-src(+)激酶,IC50分别为 0.012 和 0.5 µM。
T2287 PIK-75 hydrochloride

PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75

Apoptosis; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK-75 hydrochloride (PIK-75 HCl) 是一种可逆的 DNA-PK 和 p110α-选择性抑制剂,抑制 DNA-PK,p110α和 p110γ,可诱导凋亡。
T6747 8-Bromo-cAMP sodium salt

8-Br-Camp sodium salt,8-溴腺苷-3',5'-环单磷酸钠,8-Bromo-cAMP(sodium salt),8-Bromo-cAMP

PKA Tyrosine Kinase/Adaptors
8-Bromo-cAMP sodium salt (8-Br-Camp sodium salt) 是一种环 AMP 依赖性蛋白激酶 (PKA) 激活剂,是一种环 AMP 类似物。
T62684 Lartesertib

ATM Inhibitor-5,M4076

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Lartesertib (ATM Inhibitor-5) 是一种丝氨酸/苏氨酸蛋白激酶 ATM 的抑制剂,具有潜在的抗癌活性,可用于研究肺癌。
T10727 Cdc7-IN-5

CDK Cell Cycle/Checkpoint
Cdc7-IN-5 是一种有效的 Cdc7 激酶抑制剂。Cdc7 是一种丝氨酸苏氨酸蛋白激酶酶,在细胞周期中对 DNA 复制的启动至关重要。
T77570 AP-C2

PKA Tyrosine Kinase/Adaptors
AP-C2 是一种有效的小分子鸟苷 3',5'-环单磷酸 (cGMP) 依赖性蛋白激酶 II (cGKII) 抑制剂,对 cGKII 的 pIC50 为 5.2。
T6250 H-89 dihydrochloride

Protein kinase inhibitor H-89 dihydrochloride,H 89 2HCl,5-Isoquinolinesulfonamide

PKA; S6 Kinase; Autophagy Autophagy; MAPK; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
H-89 dihydrochloride (5-Isoquinolinesulfonamide) 是一种选择性 cAMP 依赖性蛋白激酶A(PKA) 抑制剂,IC50值为 48 nM。也可轻微抑制 PKG、PKC 和酪蛋白激酶活性。
T9609 GRK5-IN-2

GRK GPCR/G Protein
GRK5-IN-2 是基于吡啶的双环化合物,抑制 G 蛋白偶联受体激酶 5 。它调节胰岛素的表达和/或释放,在代谢疾病中有研究价值。
TP1897L1 JIP-1 (153-163) acetate(438567-88-5 free base)

JNK MAPK
JIP-1 (153-163) acetate(438567-88-5 free base) 是c-Jun N-末端激酶 (JNK) 的肽抑制剂,基于 JNK-interacting protein-1 (JIP-1) 的残基 153-163。以微摩尔范围内的亲和力与 JNK 结合,并抑制 p38 和 ERK。
T72322 R 59-022 hydrochloride

DKGI-I hydrochloride,Diacylglycerol kinase inhibitor I hydrochloride,DKGI-I hydrochloride ; Diacylglycerol kinase inhibitor I hydrochloride

5-HT Receptor; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; GPCR/G Protein; Neuroscience
R 59-022 hydrochloride (DKGI-I hydrochloride) 是一种 5-HT Receptor 拮抗剂,可激活蛋白激酶 C (PKC)。R 59-022 hydrochloride 是一种 DGK 抑制剂 (IC50:2.8 µM),可抑制 OAG 磷酸化为 OAPA。R 59-022 增强血小板中凝血酶诱导的甘油二酯的产生,并抑制嗜中性粒细胞中磷脂酸的产生。
T27416 GLPG0259

GLPG-0259,GLPG 0259

GLPG-0259 is an inhibitor of mitogen-activated protein kinase-activated protein kinase 5 (MAPKAPK5).
T71274 GLPG0259 A

GLPG0259 A is a small-molecule inhibitor of mitogen-activated protein kinase-activated protein kinase 5 (MAPKAPK5), a kinase enzyme that plays a role in important inflammatory pathways.
T75739 PKI(5-24) TFA

PKI(5-24) TFA 是一种强效、竞争性、合成的PKA(cAMP 依赖性蛋白激酶) 抑制剂,Ki 为 2.3 nM。PKI(5-24) TFA 对应于天然存在的热稳定蛋白激酶抑制剂中的 5-24 残基。
T16709 R 59-022

Diacylglycerol kinase inhibitor I,DKGI-I

Others Others
R 59-022 is a 5-HTR antagonist and activates protein kinase C (PKC). R 59-022 is a diacylglycerol kinase inhibitor (IC50=2.8 μM). R 59-022 potentiates thrombin-induced diacylglycerol production in platelets and inhibits phosphatidic acid production in neu
T82258 GRL018-21

GRL018-21为一种高效、高选择性G蛋白偶联受体激酶5 (GRK5) 抑制剂,其IC50值仅为10 nM。
T36019 PKA Inhibitor (5-24) (trifluoroacetate salt)

PKI PKA Inhibitor (5-24) is a synthetic peptide inhibitor of PKA (cAMP-dependent protein kinase) (Ki= 2.3 nM) derived from the active site of the skeletal muscle inhibitor protein.1It mimics the protein substrate by binding to the catalytic site through the arginine-cluster basic subsite.1The prominent enzyme-substrate interaction site occurs where PKA catalytic subunit residues Tyr235and Phe239form a sandwich-like structure with residue Phe10of PKI (5-24).2
T40395 ζ-Stat trisodium

NSC37044 trisodium,ζ-Stat trisodium

ζ-Stat trisodium (NSC37044 trisodium) is a potent and selective inhibitor of protein kinase C-ζ (PKC-ζ), exhibiting an IC50 of 5 μM. It effectively suppresses the proliferation of melanoma cell lines and promotes apoptosis. Moreover, ζ-Stat trisodium demonstrates notable antitumor activity in vitro.
T83640 RIPK2-IN-5

RIP kinase Apoptosis; NF-κB
RIPK2-IN-5 是一种受体相互作用蛋白激酶 2 (RIPK2) 抑制剂,具有潜在的抗炎活性,可用于研究免疫功能异常引起的疾病。
T64116 B-Raf IN 5

B-Raf IN 5 是蛋白激酶 B-Raf 的有效抑制剂 (IC50: 2.0 nM)。B-Raf IN 5 可抵抗快速代谢,切不结合二级靶点 PXR。B-Raf IN 5 对癌症疾病表现出研究潜力。
T76399 PKI(5-22)amide

PKI(5-22)amide 是环 AMP 依赖性蛋白激酶 (PKA) 抑制剂的活性片段。PKI(5-22)amide 抑制PKA 激活,但不能减弱 CRF1 受体的同源脱敏作用。
T62599 GRK5-IN-3

GRK5-IN-3 是一种 G 蛋白偶联受体激酶 5 (GRK5) 的共价抑制剂。GRK5-IN-3 对 GRK5 (IC50: 0.22 μM) 和 GRK6 (IC50: 0.41 μM)有显著的抑制作用。
T63008 PERK-IN-5

PERK-IN-5 是一种高度选择性的、高效的、口服具有活力的蛋白激酶 R 样内质网 (ER) 激酶 (PERK) 抑制剂,能够作用于 PERK (IC50: 2 nM) 与 p-eIF2α (IC50: 9 nM)。在 786-O 肾细胞癌异种移植瘤模型中,PERK-IN-5 可以明显抑制肿瘤生长。
T74374 ERK1/2 inhibitor 4

ERK1/2 inhibitor 5 是一种有效的ERK1/2抑制剂。丝裂原活化蛋白激酶 (MAPK) 在信号转导通路中起着极其重要的作用,而细胞外信号调节激酶 (ERK) 是MAPK 家族的成员。ERK1/2 inhibitor 5 具有研究或预防癌症、炎症或其他增殖性疾病的潜力。
T63340 CCG-273220

CCG-273220 是 G 蛋白偶联受体 (GPCR) 激酶 5 (GRK5) 共价抑制剂 (IC50: 220 nM)。CCG-273220 可以共价结合GRK5亚家族特异性残基 Cys474 ,而对GRK5的选择性比 GRK2 高。
T76482 PKI (5-24),amide

PKI (5-24),amide (IP20-amide)为对应于cAMP依赖性蛋白激酶热稳定抑制蛋白活性部分的20残基肽。该化合物是一种高效的cAMP依赖性蛋白激酶(PKA)抑制剂,具有2.3 nM的Ki值。
T82990 AP-C4

AP-C4是cGMP依赖性蛋白激酶II(cGKII)的抑制剂,具有pIC50值为5.2,但不影响cGKII依赖性阴离子分泌。
T35541 Lipoxygenin

Lipoxygenin is an inhibitor of 5-lipoxygenase (5-LO) with an IC50value of 5 μM for inhibition of 5-LO product synthesis in isolated human granulocytes stimulated with the cation ionophore A23187 .1It inhibits hedgehog-dependent signaling in Shh-LIGHT2 cells and TGF-β-, activin A-, bone morphogenic protein (BMP)-, or Wnt-dependent signaling in HEK293T cells (IC50s = 9.3, 3.2, 8.2, 9.6, and 3.7 μM, respectively, in luciferase reporter assays). Lipoxygenin (5 and 10 μM) increases levels of troponin...
T35827 Epsilon-V1-2

PKCε Inhibitor Peptide,Protein KinaseInhibitor Peptide,ɛV1-2

Protein kinase C (PKC ) is a calcium-independent, phospholipid- and diacylglycerol-dependent serine/threonine kinase involved in diverse signaling pathways, including those involved in neuronal signaling, cytoskeletal function, and inflammation.[1] PKC inhibitor peptide is a synthetic peptide corresponding to an amino acid sequence found in the amino terminal C2 domain of most mammalian forms of PKC .[2] It selectively and reversibly inhibits the translocation of PKC to intracellular membrane...
T63203 GRK5-IN-4

GRK5-IN-4 是选择性的、有效的、共价 GRK5(G 蛋白偶联受体激酶 5) 抑制剂(IC50: 1.1 μM)。GRK5-IN-4 对 GRK5 的选择性是 GRK2 的90倍。GRK5-IN-4 能够用于研究心力衰竭。
T82991 AP-C3

AP-C3为cGMP依赖性蛋白激酶II (cGKII) 的有效抑制剂,其pIC50值为6.3。该化合物仅对cGKII依赖性阴离子分泌表现出微弱的抑制作用。
T61693 AAK1-IN-5

AAK1-IN-5 is a potent and specific inhibitor of adaptor protein-2-associated kinase 1 (AAK1), characterized by its ability to penetrate the central nervous system and its oral bioavailability. It displays high selectivity, with an AAK1 inhibitory potency (IC 50) of 1.2 nM, a binding affinity (K i) of 0.05 nM, and an inhibitory potency against cellular AAK1 activity (cell IC 50) of 0.5 nM. AAK1-IN-5 holds promise for investigating neuropathic pain in scientific research [1].
T63057 LRRK2-IN-5

LRRK2-IN-5 (compound 25) 是一种口服具有活力的、能透过血脑屏障的、选择性富含亮氨酸重复蛋白激酶 2 基因 (LRRK2) 抑制剂,对 GS LRRK2 (IC50: 1.2 μM) 和 WT LRRK2 (IC50: 16 μM) 具有抑制作用。LRRK2-IN-5 能够抑制 LRRK2 Ser1292 和 Ser925 的自磷酸化。
T63923 ATR-IN-5

ATR-IN-5 是 ATR 的有效抑制剂。其中 ATR 是 PIKK 家族的成员,是一类参与基因组稳定性和 DNA 损伤修复的蛋白激酶。ATR-IN-5 对 ATR 激酶介导的疾病如增殖性疾病和癌症表现出研究潜力。
T82989 AP-C6

AP-C6 是一种有效的 cGMP 依赖性蛋白激酶 II (cGKII) 抑制剂,其 pIC50 值为 6.5。该化合物能够在体外浓度依赖性地抑制人 cGKII 的活性,并能够通过抑制 PDE 来增强 cAMP 信号传导。
T83670 F1 TFA

Tat-IKIP (46-60),Tat-Inhibitor of NF-κB Kinase-interacting Peptide

F1是一种抗炎肽,由HIV-1 Tat蛋白质转导域与对应于抑制因子NF-κB激酶-相互作用肽(IKIP)46-60残基的15氨基酸肽链接而成。在5 µM浓度下,F1抑制了小鼠腹腔巨噬细胞中LPS诱导的IκB激酶α(IKKα)和IKKβ的磷酸化以及NF-κB(p65)的核内转移。在体内,F1(5 mg/kg)降低了LPS诱导的脓毒症小鼠模型中IL-6、TNF-α和IL-1β的血清水平,并增加了生存率。
T64266 KR-39038

KR-39038 是一种口服具有活力的 GRK5 (G 蛋白偶联受体激酶 5) 抑制剂 (IC50: 0.02 μM)。KR-39038 能够抑制新生儿心肌细胞的 HDAC5 通路,明显抑制血管紧张素 II 诱导的细胞肥大,具有显著的抗心肌肥厚和改善心功能作用。KR-39038 能够用于进行心力衰竭的研究。
T82243 hAChE-IN-5

GSK-3 PI3K/Akt/mTOR signaling; Stem Cells
hAChE-IN-5(化合物49)是一种同时针对hAChE和hBuChE的有效抑制剂,其IC50值均为0.17 μM。此外,hAChE-IN-5对GSK3β同样展现出良好的抑制活性,IC50值为0.21 μM。作为tau蛋白聚集和Aβ1-42自聚集的抑制剂,hAChE-IN-5能够结合PAS,进而阻止Aβ依赖的神经毒性。其能穿透血脑屏障(BBB),显示出成为多靶点抗阿尔茨海默病药物研究的潜力。
T36650 Ansatrienin B

Ansatrienin B is an ansamycin antibiotic and antifungal agent first isolated from S. collinus and S. rishiriensis., In fetal rat long bones, it is an inhibitor of parathyroid hormone-induced calcium release (IC50 = 21 nM), which is a measure of bone resorption, and pp60c-src kinase (IC50 = 50 nM). It is an inhibitor of translation at the protein synthesis stage by specific inhibition of L-leucine incorporation (IC50 = 58 nM in A549 cells). It also inhibits TNF-α-induced expression of intercellul...
T38269 Purfalcamine

Purfalcamine is an orally active, selective Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1) inhibitor with an IC50 of 17 nM and an EC50 of 230 nM. Purfalcamine has antimalarial activity and causes malaria parasites developmental arrest at the schizont stage[1][2]. Purfalcamine has low activity against Toxoplasma gondii calcium-dependent protein kinase 3 (TgCDPK3)[1]. Purfalcamine (225, 450 nM) has no effect on the parasitemia in the first 32 hours. After about 40 hours, paras...
T37590 ML 3403

p38 MAPK inhibitor (IC50 = 0.38 μM). Inhibits the release of IL-1β and TNF-α in a peripheral blood mononuclear cell (PBMC) assay (IC50 values are 0.039 and 0.16 μM respectively). Laufer et al (2003) Novel substituted pyridinyl imidazoles as potent anticytokine agents with low activity against hepatic cytochrome P450 enzymes. J.Med.Chem. 46 3230 PMID:12852754 |Kammerer et al (2007) Pharmacokinetics of ML3403 ({4-[5-(4-fluorophenyl)-2-methylsulfanyl-3H-imidazol-4-yl]-pyridin-2-yl}-(1-phenylethyl)-...

化合物

Protein kinase inhibitor 5
Cat.No: T79125
Synonym:
Target: Trk receptor
MK2-IN-3
Cat.No: T9034
Synonym: MK2 Inhibitor III
Target: MAPK
PF-AKT400
Cat.No: T5508
Synonym: (S)-N-[[3-氨基-1-(5-乙基-7H-吡咯并[2,3-D]嘧啶-4-基)吡咯烷-3-基]甲基]-2,4-二氟苯甲酰胺,AKT protein kinase inhibitor
Target: Akt
Protein kinase inhibitor 5 sulfate hydrate
Cat.No: T79126
Synonym:
Target: Trk receptor
Protein kinase inhibitor H-7
Cat.No: T60109
Synonym: 5-(2-methylpiperazine-1-sulfonyl)isoquinoline,蛋白激酶抑制剂H-7,1-(5-Isoquinolinylsulfonyl)-2-methylpiperazine
Target: PKC
HG-10-102-01
Cat.No: T7196
Synonym: [4-[[5-氯-4-(甲基氨基)-2-嘧啶基]氨基]-3-甲氧基苯基]-4-吗啉基甲酮
Target: LRRK2
AKT-IN-1
Cat.No: T4489
Synonym: AZD26,AZD-26,6-[4-(1-氨基环丁基)苯基]-5-苯基-3-吡啶甲酰胺,AZD 26
Target: Akt
CAY10404
Cat.No: T8656
Synonym: 3-(4-METHYLSULPHONYLPHENYL)-4-PHENYL-5-T
Target: Apoptosis, Akt, COX
lavendustin C
Cat.No: T4185
Synonym: HDBA,NSC 666251,N-(2,5-二羟基苄基)-5-氨基水杨酸
Target: CaMK, EGFR, Tyrosinase, Src
PIK-75 hydrochloride
Cat.No: T2287
Synonym: PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75
Target: Apoptosis, DNA-PK, PI3K
8-Bromo-cAMP sodium salt
Cat.No: T6747
Synonym: 8-Br-Camp sodium salt,8-溴腺苷-3',5'-环单磷酸钠,8-Bromo-cAMP(sodium salt),8-Bromo-cAMP
Target: PKA
Lartesertib
Cat.No: T62684
Synonym: ATM Inhibitor-5,M4076
Target: ATM/ATR
Cdc7-IN-5
Cat.No: T10727
Synonym:
Target: CDK
AP-C2
Cat.No: T77570
Synonym:
Target: PKA
H-89 dihydrochloride
Cat.No: T6250
Synonym: Protein kinase inhibitor H-89 dihydrochloride,H 89 2HCl,5-Isoquinolinesulfonamide
Target: PKA, S6 Kinase, Autophagy
GRK5-IN-2
Cat.No: T9609
Synonym:
Target: GRK
JIP-1 (153-163) acetate(438567-88-5 free base)
Cat.No: TP1897L1
Synonym:
Target: JNK
R 59-022 hydrochloride
Cat.No: T72322
Synonym: DKGI-I hydrochloride,Diacylglycerol kinase inhibitor I hydrochloride,DKGI-I hydrochloride ; Diacylglycerol kinase inhibitor I hydrochloride
Target: 5-HT Receptor, PKC
GLPG0259
Cat.No: T27416
Synonym: GLPG-0259,GLPG 0259
Target:
GLPG0259 A
Cat.No: T71274
Synonym:
Target:
PKI(5-24) TFA
Cat.No: T75739
Synonym:
Target:
R 59-022
Cat.No: T16709
Synonym: Diacylglycerol kinase inhibitor I,DKGI-I
Target: Others
GRL018-21
Cat.No: T82258
Synonym:
Target:
PKA Inhibitor (5-24) (trifluoroacetate salt)
Cat.No: T36019
Synonym:
Target:
ζ-Stat trisodium
Cat.No: T40395
Synonym: NSC37044 trisodium,ζ-Stat trisodium
Target:
RIPK2-IN-5
Cat.No: T83640
Synonym:
Target: RIP kinase
B-Raf IN 5
Cat.No: T64116
Synonym:
Target:
PKI(5-22)amide
Cat.No: T76399
Synonym:
Target:
GRK5-IN-3
Cat.No: T62599
Synonym:
Target:
PERK-IN-5
Cat.No: T63008
Synonym:
Target:
ERK1/2 inhibitor 4
Cat.No: T74374
Synonym:
Target:
CCG-273220
Cat.No: T63340
Synonym:
Target:
PKI (5-24),amide
Cat.No: T76482
Synonym:
Target:
AP-C4
Cat.No: T82990
Synonym:
Target:
Lipoxygenin
Cat.No: T35541
Synonym:
Target:
Epsilon-V1-2
Cat.No: T35827
Synonym: PKCε Inhibitor Peptide,Protein KinaseInhibitor Peptide,ɛV1-2
Target:
GRK5-IN-4
Cat.No: T63203
Synonym:
Target:
AP-C3
Cat.No: T82991
Synonym:
Target:
AAK1-IN-5
Cat.No: T61693
Synonym:
Target:
LRRK2-IN-5
Cat.No: T63057
Synonym:
Target:
ATR-IN-5
Cat.No: T63923
Synonym:
Target:
AP-C6
Cat.No: T82989
Synonym:
Target:
F1 TFA
Cat.No: T83670
Synonym: Tat-IKIP (46-60),Tat-Inhibitor of NF-κB Kinase-interacting Peptide
Target:
KR-39038
Cat.No: T64266
Synonym:
Target:
hAChE-IN-5
Cat.No: T82243
Synonym:
Target: GSK-3
Ansatrienin B
Cat.No: T36650
Synonym:
Target:
Purfalcamine
Cat.No: T38269
Synonym:
Target:
ML 3403
Cat.No: T37590
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5736 1,3-Dicaffeoylquinic acid

CYNARIN,1,3-二咖啡酰奎宁酸,Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1S,​3R,​4R,​5R)​-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid

Reactive Oxygen Species; Akt; PI3K Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
1,3-Dicaffeoylquinic acid (CYNARIN) 是一种咖啡酰奎宁酸衍生物,具有抗氧化、自由基清除作用。

天然产物

1,3-Dicaffeoylquinic acid
Cat.No: T5736
Synonym: CYNARIN,1,3-二咖啡酰奎宁酸,Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1S,​3R,​4R,​5R)​-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid
Target: Reactive Oxygen Species, Akt, PI3K
TargetMol Loading
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