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149

抑制剂 & 化合物

15

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T23760	AT-IAP
	AT-IAP is an effective dual antagonist of XIAP and cIAP1.
T5400	Q203 IAP6,Telacebec	Antibacterial; Antibiotic	Microbiology/Virology
	Q203 (Telacebec)是一种中氮杂吡啶酰胺。在培养基中抑制结核分枝杆菌H37Rv 活性的MIC50值为2.7 nM。
TP2292	survivin (baculoviral IAP repeat-containing protein 5) (21-28)	Others	Others
	Survivin (baculoviral inhibitor of apoptosis IAP repeat-containing protein-5) is a member of the IAP gene family, which has been implicated in both inhibitions of apoptosis and mitosis regulation1. Survivin is one of the most uniformly up-regulated genes
T18612	Bestatin-amido-Me PROTAC IAP binding moiety 1	Others	Others
	Bestatin-amido-Me, a derivative of Bestatin, acts as an IAP ligand and interacts with ABL inhibitor through a linker to produce SNIPER[1].
T74847	PROTAC pan-IAP degrader-1
	PROTACpan-IAP degrader-1 (Compound 9) 是一种 pan-IAPPROTAC 降解剂。PROTACpan-IAP degrader-1 在 MM.1S 细胞中降解 XIAP、cIAP1 和 cIAP2 的 DC50分别为 0.7、2.4 和 6.2 nM。
T18613	MV-1-NH-Me PROTAC IAP binding moiety 2	Others	Others
	MV-1-NH-Me, an MV-1-derived IAP ligand, connects to an ABL inhibitor through a linker, resulting in the formation of SNIPER[1].
T6428	BV6	IAP	Apoptosis
	BV6 是 c-IAP1 和 XIAP 的拮抗剂，它们是凋亡抑制剂 (IAP) 家族的成员。
TQ0029	ASTX660	IAP	Apoptosis
	ASTX660 是一种口服生物可利用的 cIAP 和 XIAP 双重拮抗剂。
T12932L	SM-164	Apoptosis; IAP	Apoptosis
	SM-164 是细胞渗透性 Smac 类似物，与含有 BIR2 和 BIR3 结构域的 XIAP 蛋白结合，IC50值为 1.39 nM，它用作XIAP 的强效拮抗剂。
T2080	LCL161	IAP	Apoptosis
	LCL161 是一种 SMAC 模拟物，可有效结合并抑制多种 IAP。它抑制 HEK293 细胞中 XIAP 和 MDA-MB-231细胞中 cIAP1的 IC50分别为 35 和 0.4 nM。
T6299	GDC-0152 GDC0152	IAP	Apoptosis
	GDC-0152 是一种 IAP 抑制剂，可以与 XIAP、cIAP1和cIAP2的 BIR3 结合域，以及ML-IAP 的 BIR 结合域结合，Ki 值分别为 28 nM、17 nM、43 nM 和 14 nM。
T16163	MV1	Apoptosis	Apoptosis
	MV1 是一种 IAP 拮抗剂。当与 HaloTag 配体结合时，它会导致 HaloTag 融合蛋白的蛋白质敲低。
T6007	Birinapant TL32711,比瑞那帕	Apoptosis; IAP; HIV Protease	Apoptosis; Microbiology/Virology; Proteases/Proteasome
	Birinapant (TL32711) 是一种二价 Smac 模拟物，是 XIAP 和 cIAP1的强效拮抗剂，Kd 值分别为 45 nM 和小于 1 nM。它靶向与 TRAF2 相关的 cIAP，并消除 TNF 诱导的 NF-κB 活化。
T3653	MX69	Mdm2; E1/E2/E3 Enzyme; IAP	Apoptosis; Ubiquitination
	MX69 是用于抗癌研究的一种MDM2/XIAP 抑制剂。
T6763	Xevinapant ARRY-334543,SM-406,AT406,Debio-1143	IAP	Apoptosis
	Xevinapant (Debio-1143) 是一种有效的 Smac 模拟物和 IAP 的拮抗剂，能够抑制 XIAP，cIAP1 和 cIAP2 蛋白，Ki 值分别为 66.4，1.9 和 5.1 nM。
T14378	AZD5582	Apoptosis; IAP	Apoptosis
	AZD5582 是一种 IAP 拮抗剂，可诱导凋亡，可与 cIAP1、cIAP2 和 XIAP 的 BIR3 结构域结合，IC50值分别为 15、21和15 nM。
T3299	Xevinapant hydrochloride AT-406 HCl,SM-406	Apoptosis; IAP	Apoptosis
	Xevinapant hydrochloride (AT-406 HCl) 是口服生物可利用的 Smac 模拟物，也是细胞凋亡蛋白抑制剂的拮抗剂。它在无细胞功能测定中有效拮抗 XIAP BIR3 蛋白，诱导细胞 cIAP1 蛋白的快速降解，并抑制各种人类癌细胞系中的癌细胞生长。它在诱导异种移植肿瘤细胞凋亡方面非常有效。
T17870	cIAP1 ligand 1 E3 ligase Ligand 12	Others	Others
	cIAP1 ligand 1 (E3 ligase Ligand 12) 是基于 LCL161 衍生物的细胞凋亡蛋白配体，可募集 IAP 泛素连接酶以降解靶蛋白，可用于和雄激素受体配体偶联开发蛋白降解剂，可用于研究前列腺癌。
T12405	Pentiapine 喷硫平,CGS 10746	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Pentiapine (CGS 10746) 是一种新型的多巴胺释放抑制剂。
T9519	Eliapixant BAY 1817080	P2X Receptor	Membrane transporter/Ion channel; Neuroscience
	Eliapixant (BAY 1817080) 是一种选择性的P2X3受体拮抗剂，IC50值为 8 nM，可用于难治性慢性咳嗽的研究。
T13154	Tiapamil hydrochloride Ro 11-1781 hydrochloride,ORE 5002 hydrochloride	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Tiapamil hydrochloride (Ro 11-1781 hydrochloride) 是一种钙通道阻滞剂，具有抗高血压活性，可用于研究心绞痛和心血管疾病。
T36949	Niaprazine	5-HT Receptor; Adrenergic Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Niaprazine 是有效的组胺 H1 受体拮抗剂，具有抗组胺和抗血清素活性。Niaprazine 在睡眠障碍方面有研究的价值。
T6411	Biapenem CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627	Antibacterial; Antibiotic	Microbiology/Virology
	Biapenem (CLI 86815) 是不经肠道的广谱碳青霉烯抗生素。
T16731	Rentiapril racemate (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril	Angiotensin-converting Enzyme (ACE)	Metabolism
	Rentiapril racemate (SA-446 racemate) 是 Rentiapril 的外消旋体。Rentiapril racemate 具有抗炎活性，可用于研究青光眼。
T11506	Guaiapate Mg 5454,Klamar	Others	Others
	Guaiapate 具有止咳镇静作用。
T6241	Quetiapine hemifumarate Quetiapine Fumarate,ICI-204636,富马酸喹硫平	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Quetiapine hemifumarate (ICI-204636) 是5-HT 受体激动剂和多巴胺受体拮抗剂，对人5-HT1A 和人D2的pEC50值分别为 4.77 和 6.33，具有抗抑郁和抗焦虑作用。
T0162	Quetiapine ICI204636,Quetiapin,喹硫平	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Quetiapine (ICI204636) 是5-HT 受体激动剂和多巴胺受体拮抗剂，对人5-HT1A 的 pEC50值为 4.77，对人 D2的 pIC50值为 6.33。它用于治疗精神分裂症，以及治疗与 I 型双相情感障碍相关的急性躁狂发作。它对人 D2、HT1、5-HT2A、5-HT2C 受体具有中高等亲和力，pKi 值为 7.25、5.74、7.54和5.55。
T4561	Tiaprofenic acid Tiaprofensaeure,噻洛芬酸,Acido tiaprofenico,Surgam	Others; COX	Immunology/Inflammation; Neuroscience; Others
	Tiaprofenic acid (Acido tiaprofenico) 是可口服的非甾体抗炎药，通过抑制环氧化酶抑制前列腺素合成，可用于风湿性疾病的研究。
T1292	Tiapride hydrochloride	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Tiapride 是一种大脑中 D2/3 多巴胺受体的选择性阻滞剂。它用于治疗各种精神和神经系统疾病，包括运动障碍、酒精戒断综合征、精神病的阴性症状以及老年人的攻击和激动。
T17894	cIAP1 Ligand-Linker Conjugates 3 E3 ligase Ligand-Linker Conjugates 40	Others	Others
	cIAP1 Ligand-Linker Conjugates 3 are chemical compounds comprising an IAP ligand designed specifically for the E3 ubiquitin ligase and a PROTAC linker. These conjugates, denoted as cIAP1 Ligand-Linker Conjugates 3, find utility in the design of SNIPERs, short for Specific and Non-genetic IAP-dependent Protein Erasers [1].
T17888	cIAP1 Ligand-Linker Conjugates 6 hydrochloride E3 ligase Ligand-Linker Conjugates 35 hydrochloride	Others	Others
	cIAP1 Ligand-Linker Conjugates 6 hydrochloride is a compound that combines an IAP ligand for the E3 ubiquitin ligase and a PROTAC linker. It is utilized for the purpose of designing SNIPERs[1].
T17891	cIAP1 Ligand-Linker Conjugates 2 E3 ligase Ligand-Linker Conjugates 37	Others	Others
	cIAP1 Ligand-Linker Conjugates 2 is a chemical compound that combines an IAP ligand for the E3 ubiquitin ligase with a PROTAC linker. This compound is particularly useful in the design of SNIPERs [1].
T17889	cIAP1 Ligand-Linker Conjugates 14 E3 ligase Ligand-Linker Conjugates 36	Others	Others
	cIAP1 Ligand-Linker Conjugates 14 consist of an IAP ligand that targets the E3 ubiquitin ligase and a PROTAC linker. These conjugates, known as cIAP1 Ligand-Linker Conjugates 14, are used in the development of SNIPERs[1].
T17901	cIAP1 Ligand-Linker Conjugates 10 E3 ligase Ligand-Linker Conjugates 47	Others	Others
	cIAP1 Ligand-Linker Conjugates 10 comprise of an IAP ligand and a PROTAC linker, which facilitates the design of SNIPERs. These conjugates incorporate an IAP ligand that interacts with the E3 ubiquitin ligase, and a PROTAC linker. SNIPERs can be developed using cIAP1 Ligand-Linker Conjugates 10.
T17899	cIAP1 Ligand-Linker Conjugates 9 E3 ligase Ligand-Linker Conjugates 45	Others	Others
	cIAP1 Ligand-Linker Conjugates 9 feature an IAP ligand specifically targeting the E3 ubiquitin ligase, along with a PROTAC linker. It is valuable tools for developing SNIPERs[1].
T17869	cIAP1 ligand 2 E3 ligase Ligand 11	Others	Others
	cIAP1 ligand 2, a derivative of LCL161, is an IAP ligand that can be connected to the ABL ligand for protein via a linker, resulting in the formation of SNIPER.
T17898	cIAP1 Ligand-Linker Conjugates 7 E3 ligase Ligand-Linker Conjugates 44	Others	Others
	cIAP1 Ligand-Linker Conjugates 7 is a chemical compound that combines an IAP ligand for the E3 ubiquitin ligase with a PROTAC linker. It is utilized in the design of SNIPERs[1].
T17896	cIAP1 Ligand-Linker Conjugates 4 E3 ligase Ligand-Linker Conjugates 42	Others	Others
	cIAP1 Ligand-Linker Conjugates 4 is a chemical compound that comprises an IAP ligand specifically designed for the E3 ubiquitin ligase and a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 4, has the potential to be utilized in the development of SNIPERs[1].
T17886	cIAP1 Ligand-Linker Conjugates 15 hydrochloride E3 ligase Ligand-Linker Conjugates 34 hydrochloride	Others	Others
	cIAP1 Ligand-Linker Conjugates 15 hydrochloride is a chemical compound that combines an IAP ligand for the E3 ubiquitin ligase and a PROTAC linker. This compound is useful in the development of SNIPERs[1].
T17897	cIAP1 Ligand-Linker Conjugates 13 E3 ligase Ligand-Linker Conjugates 43	Others	Others
	cIAP1 Ligand-Linker Conjugates 13, containing an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker, are utilized in the development of SNIPERs[1].
T17885	cIAP1 Ligand-Linker Conjugates 11 E3 ligase Ligand-Linker Conjugates 33	Others	Others
	cIAP1 Ligand-Linker Conjugates 11 is a chemical compound that combines an IAP ligand specifically designed for the E3 ubiquitin ligase with a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 11, is useful in the development of SNIPERs[1], allowing for the targeted degradation of proteins.
T17895	cIAP1 Ligand-Linker Conjugates 1 E3 ligase Ligand-Linker Conjugates 41	Others	Others
	cIAP1 Ligand-Linker Conjugates 1 is composed of an IAP ligand for the E3 ubiquitin ligase and a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 1, is particularly useful in the development of SNIPERs[1].
T17893	cIAP1 Ligand-Linker Conjugates 5 E3 ligase Ligand-Linker Conjugates 39	Others	Others
	cIAP1 Ligand-Linker Conjugates 5 is a chemical compound consisting of an IAP ligand that targets the E3 ubiquitin ligase, and a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 5, is specifically designed for the development of SNIPERs[1].
T17900	cIAP1 Ligand-Linker Conjugates 8 E3 ligase Ligand-Linker Conjugates 46	Others	Others
	cIAP1 Ligand-Linker Conjugates 8 comprises an IAP ligand for the E3 ubiquitin ligase and a PROTAC linker. This compound is specifically utilized for the purpose of SNIPER design[1].
T17884	cIAP1 Ligand-Linker Conjugates 11 Hydrochloride E3 ligase Ligand-Linker Conjugates 33 Hydrochloride	Others	Others
	cIAP1 Ligand-Linker Conjugates 11 Hydrochloride is a chemical compound consisting of an IAP ligand that targets the E3 ubiquitin ligase, along with a PROTAC linker. It is primarily utilized in the development of SNIPERs, a molecular tool for targeted protein degradation[1].
T17890	cIAP1 Ligand-Linker Conjugates 2 Hydrochloride E3 ligase Ligand-Linker Conjugates 37 Hydrochloride,cIAP1 Ligand-Linker Conjugates 2 Hydrochloride (1312302-14-9 free base)	Others	Others
	cIAP1 Ligand-Linker Conjugates 2 Hydrochloride is a chemical compound that combines an IAP ligand, which targets the E3 ubiquitin ligase, with a PROTAC linker. It is utilized in the creation of SNIPERs[1].
T17892	cIAP1 Ligand-Linker Conjugates 12 E3 ligase Ligand-Linker Conjugates 38	Others	Others
	cIAP1 Ligand-Linker Conjugates 12 is a chemical compound that combines an IAP ligand, which targets the E3 ubiquitin ligase, with a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 12, is valuable for creating SNIPERs[1].
T17887	cIAP1 Ligand-Linker Conjugates 15 E3 ligase Ligand-Linker Conjugates 34	Others	Others
	cIAP1 Ligand-Linker Conjugates 15 consists of an IAP ligand that targets the E3 ubiquitin ligase, along with a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 15, is suitable for the development of SNIPERs[1].
T68160	tiapirinol
	tiapirinol 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T68160，CAS号为 14785-50-3。
T79483	MDM2/XIAP-IN-3
	MDM2/XIAP-IN-3（化合物 3e）为MDM2/XIAP双重抑制剂，能够下调MDM2与XIAP蛋白水平，提升p53表达，进而抑制癌细胞增殖并诱导细胞凋亡。

化合物

Cat.No: T23760

Cat.No: T5400

Synonym: IAP6,Telacebec

Target: Antibacterial, Antibiotic

survivin (baculoviral IAP repeat-containing protein 5) (21-28)

Cat.No: TP2292

Target: Others

Bestatin-amido-Me

Cat.No: T18612

Synonym: PROTAC IAP binding moiety 1

Target: Others

PROTAC pan-IAP degrader-1

Cat.No: T74847

Cat.No: T18613

Synonym: PROTAC IAP binding moiety 2

Target: Others

Cat.No: T6428

Target: IAP

Cat.No: TQ0029

Target: IAP

Cat.No: T12932L

Target: Apoptosis, IAP

Cat.No: T2080

Target: IAP

Cat.No: T6299

Synonym: GDC0152

Target: IAP

Cat.No: T16163

Target: Apoptosis

Cat.No: T6007

Synonym: TL32711,比瑞那帕

Target: Apoptosis, IAP, HIV Protease

Cat.No: T3653

Target: Mdm2, E1/E2/E3 Enzyme, IAP

Cat.No: T6763

Synonym: ARRY-334543,SM-406,AT406,Debio-1143

Target: IAP

Cat.No: T14378

Target: Apoptosis, IAP

Xevinapant hydrochloride

Cat.No: T3299

Synonym: AT-406 HCl,SM-406

Target: Apoptosis, IAP

Cat.No: T17870

Synonym: E3 ligase Ligand 12

Target: Others

Cat.No: T12405

Synonym: 喷硫平,CGS 10746

Target: Dopamine Receptor

Cat.No: T9519

Synonym: BAY 1817080

Target: P2X Receptor

Tiapamil hydrochloride

Cat.No: T13154

Synonym: Ro 11-1781 hydrochloride,ORE 5002 hydrochloride

Target: Calcium Channel

Cat.No: T36949

Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor

Cat.No: T6411

Synonym: CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627

Target: Antibacterial, Antibiotic

Rentiapril racemate

Cat.No: T16731

Synonym: (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril

Target: Angiotensin-converting Enzyme (ACE)

Cat.No: T11506

Synonym: Mg 5454,Klamar

Target: Others

Quetiapine hemifumarate

Cat.No: T6241

Synonym: Quetiapine Fumarate,ICI-204636,富马酸喹硫平

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Cat.No: T0162

Synonym: ICI204636,Quetiapin,喹硫平

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR, Histamine Receptor

Tiaprofenic acid

Cat.No: T4561

Synonym: Tiaprofensaeure,噻洛芬酸,Acido tiaprofenico,Surgam

Target: Others, COX

Tiapride hydrochloride

Cat.No: T1292

Target: Dopamine Receptor

cIAP1 Ligand-Linker Conjugates 3

Cat.No: T17894

Synonym: E3 ligase Ligand-Linker Conjugates 40

Target: Others

cIAP1 Ligand-Linker Conjugates 6 hydrochloride

Cat.No: T17888

Synonym: E3 ligase Ligand-Linker Conjugates 35 hydrochloride

Target: Others

cIAP1 Ligand-Linker Conjugates 2

Cat.No: T17891

Synonym: E3 ligase Ligand-Linker Conjugates 37

Target: Others

cIAP1 Ligand-Linker Conjugates 14

Cat.No: T17889

Synonym: E3 ligase Ligand-Linker Conjugates 36

Target: Others

cIAP1 Ligand-Linker Conjugates 10

Cat.No: T17901

Synonym: E3 ligase Ligand-Linker Conjugates 47

Target: Others

cIAP1 Ligand-Linker Conjugates 9

Cat.No: T17899

Synonym: E3 ligase Ligand-Linker Conjugates 45

Target: Others

Cat.No: T17869

Synonym: E3 ligase Ligand 11

Target: Others

cIAP1 Ligand-Linker Conjugates 7

Cat.No: T17898

Synonym: E3 ligase Ligand-Linker Conjugates 44

Target: Others

cIAP1 Ligand-Linker Conjugates 4

Cat.No: T17896

Synonym: E3 ligase Ligand-Linker Conjugates 42

Target: Others

cIAP1 Ligand-Linker Conjugates 15 hydrochloride

Cat.No: T17886

Synonym: E3 ligase Ligand-Linker Conjugates 34 hydrochloride

Target: Others

cIAP1 Ligand-Linker Conjugates 13

Cat.No: T17897

Synonym: E3 ligase Ligand-Linker Conjugates 43

Target: Others

cIAP1 Ligand-Linker Conjugates 11

Cat.No: T17885

Synonym: E3 ligase Ligand-Linker Conjugates 33

Target: Others

cIAP1 Ligand-Linker Conjugates 1

Cat.No: T17895

Synonym: E3 ligase Ligand-Linker Conjugates 41

Target: Others

cIAP1 Ligand-Linker Conjugates 5

Cat.No: T17893

Synonym: E3 ligase Ligand-Linker Conjugates 39

Target: Others

cIAP1 Ligand-Linker Conjugates 8

Cat.No: T17900

Synonym: E3 ligase Ligand-Linker Conjugates 46

Target: Others

cIAP1 Ligand-Linker Conjugates 11 Hydrochloride

Cat.No: T17884

Synonym: E3 ligase Ligand-Linker Conjugates 33 Hydrochloride

Target: Others

cIAP1 Ligand-Linker Conjugates 2 Hydrochloride

Cat.No: T17890

Synonym: E3 ligase Ligand-Linker Conjugates 37 Hydrochloride,cIAP1 Ligand-Linker Conjugates 2 Hydrochloride (1312302-14-9 free base)

Target: Others

cIAP1 Ligand-Linker Conjugates 12

Cat.No: T17892

Synonym: E3 ligase Ligand-Linker Conjugates 38

Target: Others

cIAP1 Ligand-Linker Conjugates 15

Cat.No: T17887

Synonym: E3 ligase Ligand-Linker Conjugates 34

Target: Others

Cat.No: T68160

Cat.No: T79483

Cat. No.	Product Name	Target	Signaling Pathways
TN2091	Polygalacin D	Apoptosis; IAP	Apoptosis
	Polygalacin D 是从桔梗中分离的一种天然产物，具有抗癌和抗增殖特性。它通过 PI3K/Akt 途径诱导凋亡。它抑制 IAP 蛋白家族的表达，并通过抑制 GSK3β，Akt 的磷酸化和 PI3K 的表达来阻断 PI3K/Akt 途径。
T8213	Isolinderalactone	NOS; STAT	Immunology/Inflammation; JAK/STAT signaling; Stem Cells
	Isolinderalactone 具有抗炎和抗癌能力，具有中等的 iNOS 抑制活性，IC50 值为 0.30 uM。
T6485	Embelin NSC 91874,恩贝酸,恩贝酸/恩贝灵,Emberine,Embelic acid	Apoptosis; NF-κB; Lipoxygenase; IAP; Prostaglandin Receptor; Autophagy	Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Metabolism; NF-κB
	Embelin (Embelic acid) 是从日本 Ardisia 草药中分离出来的一种非肽类细胞渗透性XIAP 抑制剂，诱导口腔鳞癌细胞自噬和凋亡。它阻断 NF-kappaB 信号通路，从而抑制 NF-kappaB 调节的抗凋亡和转移基因产物。在高水平 XIAP 的前列腺癌细胞中抑制细胞生长，诱导凋亡，并激活 caspase-9。
T4292	Thiaproline L-Thioproline,L-Thiaproline,L-硫代脯氨酸	Others	Others
	Thiaproline (L-Thiaproline) 已用于肽偶联反应。
T38250	L-Sepiapterin
	L-Sepiapterin, also known as Sepiapterin, is a precursor compound crucial for the production of tetrahydrobiopterin (BH4), which serves as a coenzyme for endothelial nitric oxide synthase (eNOS). This compound demonstrates its efficacy by improving endothelial dysfunction in small mesenteric arteries from db/db mice and promoting angiogenesis. Moreover, L-Sepiapterin exerts inhibitory effects on cellular proliferation and migration in ovarian cancer cells through the down-regulation of p70S6K-de...
T75650	Rivulariapeptolides 1121
	Rivulariapeptolides 1121，作为一种高效的选择性丝氨酸蛋白酶抑制剂，对胰凝蛋白酶、弹性蛋白酶和蛋白酶K展示出了显著的抑制活性，其IC50值分别为35.52 nM、13.24 nM和48.05 nM。
T75649	Rivulariapeptolides 1185
	Rivulariapeptolides 1185 是一种高效的选择性丝氨酸蛋白酶抑制剂，其对胰凝蛋白酶、弹性蛋白酶和蛋白酶 K 的 IC50分别为 13.17 nM、23.59 nM 和 55.26 nM。
T75648	Rivulariapeptolides 1155
	Rivulariapeptolides 1155 是一种有效的丝氨酸蛋白酶 (serine protease) 抑制剂，对糜蛋白酶、弹性蛋白酶、蛋白蛋白酶 K 的 IC50分别为 41.84、4.94、56.54 nM。
TN1241	3,8''-Biapigenin 3,8'-Biapigenin,3,8″-双芹菜素	ROS	Immunology/Inflammation
	3, 8''-Biapigenin can modulate intracellular ROS production.
TN5496	2'',3''-Dihydro-3',3'''-biapigenin 2,3-Dihydro-3',3'''-biapigenin
	2'',3''-Dihydro-3',3'''-biapigenin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5496，CAS号为 151455-25-3。
TN5500	3',3'''-Biapigenin
	3',3'''-Biapigenin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5500，CAS号为 151455-26-4。
TN6500	Microgrewiapine A
	Microgrewiapine A is a selective cytotoxic agent for colon cancer cells over normal colon cells and to exhibit nicotinic receptor antagonistic activity for both the hα3β4 and hα4β2 receptor subtypes.
T75651	Rivulariapeptolides 988
	Rivulariapeptolides 988作为一种高效选择性丝氨酸蛋白酶抑制剂，对胰凝蛋白酶、弹性蛋白酶和蛋白酶K的IC50分别为95.46 nM、15.29 nM和85.50 nM。
TN4598	Myrciaphenone A	Others	Others
	Myrciaphenone A is a natural product from Limoniastrum feei (Girard) Batt.
TN5678	Salviaplebeiaside
	Salviaplebeiaside is a natural product from Vitex negundo var. cannabifolia.

天然产物

Cat.No: TN2091

Target: Apoptosis, IAP

Isolinderalactone

Cat.No: T8213

Target: NOS, STAT

Cat.No: T6485

Synonym: NSC 91874,恩贝酸,恩贝酸/恩贝灵,Emberine,Embelic acid

Target: Apoptosis, NF-κB, Lipoxygenase, IAP, Prostaglandin Receptor, Autophagy

Cat.No: T4292

Synonym: L-Thioproline,L-Thiaproline,L-硫代脯氨酸

Target: Others

Cat.No: T38250

Rivulariapeptolides 1121

Cat.No: T75650

Rivulariapeptolides 1185

Cat.No: T75649

Rivulariapeptolides 1155

Cat.No: T75648

3,8''-Biapigenin

Cat.No: TN1241

Synonym: 3,8'-Biapigenin,3,8″-双芹菜素

Target: ROS

2'',3''-Dihydro-3',3'''-biapigenin

Cat.No: TN5496

Synonym: 2,3-Dihydro-3',3'''-biapigenin

3',3'''-Biapigenin

Cat.No: TN5500

Microgrewiapine A

Cat.No: TN6500

Rivulariapeptolides 988

Cat.No: T75651

Myrciaphenone A

Cat.No: TN4598

Target: Others

Salviaplebeiaside

Cat.No: TN5678

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