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131

抑制剂 & 化合物

67

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Cat. No. Product Name Target Signaling Pathways
T5451 Eph inhibitor 2

Ehp-inhibitor-1

Ephrin Receptor Tyrosine Kinase/Adaptors
Eph inhibitor 2 是一种 Eph 家族酪氨酸激酶抑制剂。
T28773 SI-2

SI2,EPH 116,EPH116,EPH-116

Others Others
SI-2是类固醇受体辅激活因子-3(SRC-3或 AIB1)的抑制剂(SMI)。SI-2可选择性降低细胞中 SRC-3的转录活性和蛋白浓度,并选择性诱导低纳摩尔范围(3-20 nM)内的乳腺癌症细胞死亡,但不影响正常细胞存活率。
T12906 SI-2 hydrochloride

EPH 116 hydrochloride

Src Angiogenesis; Tyrosine Kinase/Adaptors
SI-2 hydrochloride (EPH 116 hydrochloride) 是 SRC-3 的抑制剂,诱导乳腺癌细胞死亡的 IC50 值为 3-20 nM。SI-2 hydrochloride 具有良好的药代动力学特征和改善的毒性,以及可接受的口服可用性。
T4344 ALW-II-41-27

Eph receptor tyrosine kinase inhibitor

Ephrin Receptor Tyrosine Kinase/Adaptors
ALW-II-41-27 (Eph receptor tyrosine kinase inhibitor) 是一种 Eph 受体酪氨酸激酶抑制剂,可用于治疗癌症。
TP1113L [Leu5]-Enkephalin, amide acetate

[Leu5]-Enkephalin, amide acetate(60117-24-0 free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
[Leu5]-Enkephalin, amide acetate 是一种 δ 阿片受体激动剂。
T22545 Acephate

acetylphosphoramidothioicacido,s-dimethylester,Ortran,Orthene,Acetamidophos,chevronorthene,乙酰甲胺磷

AChE Neuroscience
Acephate (Orthene) 是能产生胆碱毒性的抗胆碱酯酶杀虫剂。它能够有效抑制蟑螂的 AChE,但对大鼠 AChE 的抑制作用较弱。
T0141 Cephalonium

头孢洛宁,Cefalonium

Others Others
Cephalonium (Cefalonium) 是第一代头孢菌素类抗生素。
T21425 Mephenytoin

Mesantoin,Methoin,Insulton,Phenantoin,美芬妥因,Methylphenetoin

P450 Metabolism
Mephenytoin (Phenantoin) 是 CYP2C19 及 CYP2B6 的底物,是一种抗惊厥剂。
T0199 Cephradine

Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定

TOPK; Antibacterial; Antibiotic MAPK; Microbiology/Virology
Cephradine (Anspor) 是广谱口服活性头孢菌素。它对革兰氏阳性和革兰氏阴性病原体都有活性。它已用于泌尿生殖系统、胃肠道和呼吸道感染以及皮肤和软组织感染的研究。它通过直接抑制TOPK 抑制太阳紫外线诱导的皮肤炎症。
T36839 (R)-Mephenytoin

R-Mephenytoin,(R)-Mephenytoin,(–)-Mephenytoin

Others Others
(R)-Mephenytoin ((–)-Mephenytoin) 是 Mephenytoin 的 R-对映体,Mephenytoin 是一种抗惊厥药。
T1008 Cephalexin

头孢氨苄,Cefalexin,Cephacillin

Antibacterial; Antibiotic Microbiology/Virology
Cephalexin (Cephacillin) 是一种强口服活性的头孢菌素抗生素。它通过破坏细菌细胞壁的生长来杀死革兰氏阳性和一些革兰氏阴性细菌。它可研究肺炎、链球菌性咽喉炎、细菌性心内膜炎等。
T4581 3-hydroxycephem

Others Others
3-hydroxycephem 是各类头孢中间体。
T21824 Sephin1

NSC 65390,IFB-088

Phosphatase Metabolism
Sephin1 (IFB-088) 是 GADD34 (PPP1R15A) 的选择性抑制剂,这是一种应激诱导的蛋白磷酸酶 1 复合物调节亚基,可将 eIF2α 去磷酸化。
T0015 Mephenesin

Cresoxydiol,甲酚甘油醚,Memphenesin,Mephedan,Decontractyl

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Mephenesin (Cresoxydiol) 是 NMDA 受体拮抗剂,也是中枢性肌松弛剂。
T0997 Temephos

双硫磷,Temefos

AChR; Parasite Microbiology/Virology; Neuroscience
Temephos (Temefos) 是一种胆碱酯酶抑制剂,是一种有机硫代磷酸盐杀虫剂,用于治疗被携带疾病的昆虫侵染的水。
T20022 Cephalexin monohydrate

Cephalexin hydrate,Cephacillin hydrate,Cefalexin hydrate

Antibiotic Microbiology/Virology
Cephalexin monohydrate (Cephalexin hydrate) 是一种可口服的半合成头孢菌素类抗生素,具有显著的抗菌活性, 通过靶向青霉素结合蛋白 (PBPs)抑制细菌增殖。
TP1367 [D-Ala2]leucine-enkephalin

(D-ALA2)-亮氨酸脑啡肽

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
[D-Ala2]leucine-enkephalin 是 δ 阿片类激动剂,是能长效抗降解的亮氨酸脑非肽,可用于研究 δ 阿片受体的信号通路。
T21529 (S)-Mephenytoin

Others Others
(S)-Mephenytoin 是一种抗惊厥剂。(S)-Mephenytoin 作为细胞色素 P450 (CYP) 同种型 CYP2C19 的底物,可用于分析细胞色素 P450 代谢。
T7173L [Leu5]-Enkephalin acetate(58822-25-6 free base)

亮氨酸脑啡肽,Leucine enkephalin,Leu-enkephalin,Leucyl-enkephalin

Opioid Receptor; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
[Leu5]-Enkephalin acetate(58822-25-6 free base) 是一种参与伤害感受的内源性神经肽,是 δ-opioid 和 μ-opioid 受体的激动剂(Kis 分别为 4.0 和 3.4 nM)
T7665 [Leu5]-Enkephalin TFA(58822-25-6(free bas))

Leu-enkephalin,Leucine enkephalin,Leucyl-enkephalin

Opioid Receptor; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) 是最有效的 δ 受体。
T7173 [Leu5]-Enkephalin

亮氨酸脑啡肽,Leucine enkephalin,Leucyl-enkephalin,Leu-enkephalin

Opioid Receptor; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
[Leu5]-Enkephalin (Leu-enkephalin) 是一种参与伤害感受的内源性神经肽,是 δ-阿片和 μ-阿片受体的激动剂,Ki 值分别为 4.0 和 3.4 nM
T0286 Bephenium (hydroxynaphthoate)

羟萘酸苄酚宁,Bephenium Hydroxynaphthoate

Parasite Microbiology/Virology
Bephenium hydroxynaphthoate 是一种灭虫剂,可研究蛔虫感染,也是B 型AChR 激动剂。
T1122 Cephalothin sodium

头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin

Antibacterial; Antibiotic Microbiology/Virology
Cephalothin sodium (Cefalotin) 是一种头孢类抗生素, 具有广泛的抗菌活性,抑制革兰氏阳性和阴性菌。
TP1254 [Met5]-Enkephalin, amide TFA

5-Methionine-enkephalin amide (TFA)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) (60117-17-1 free base) 是一种 δ 阿片受体激动剂以及推定的 ζ (zeta) opioid 受体。
T22752L (D-Ser2)-Leu-Enkephalin-Thr

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
(D-Ser2)-Leu-Enkephalin-Thr 是阿片受体的 delta 选择性药物,具有镇痛作用。
T12896L Shepherdin 79-87 acetate

Shepherdin 79-87 acetate (861224-28-4 free base)

HSP; Survivin Apoptosis; Cytoskeletal Signaling; Metabolism
Shepherdin 79-87 acetate 是 Hsp90 和 survivin 之间复合物的拟肽拮抗剂,survivin 是肿瘤细胞活力的另一个关键调节剂。
T8557 N-terminally acetylated Leu-enkephalin

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
N-terminally acetylated Leu-enkephalin 是一种五氨基酸内源性肽,可作为阿片受体激动剂。N-末端乙酰化 Leu-脑啡肽是 Leu-脑啡肽的 N-末端乙酰化形式。
T5570 Cephalothin

头孢噻吩,Cephalotin acid

Antibacterial; Antibiotic Microbiology/Virology
Cephalothin 是一种 β-内酰胺抗生素,抑制 C 类 β-内酰胺酶活性的 Ki 值为 0.32 µM。
T5038 Cephapirin Sodium

Antibacterial; Antibiotic Microbiology/Virology
Cephapirin sodium 是一种半合成头孢菌素类抗生素,对革兰氏阳性菌和革兰氏阴性菌有杀菌作用。
T1364 7-Aminodeacetoxycephalosporanic acid

7-ADCA,Cephalexin Impurity B,Cefalexine EP IMpurity B,Deacetoxycephalosporanic Acid,头孢氨苄杂质B,7-Aminodesacetoxycephalosporanic acid

Antibiotic Microbiology/Virology
7-Aminodeacetoxycephalosporanic acid (Cefalexine EP IMpurity B) 是一种头孢菌素合成中的关键中间体。
T7142 Cephalosporin C zinc salt

Others Others
Cephalosporin C zinc salt 是 SAMHD1的有效抑制剂,IC50值为 1.1 μM。
T31631 Enkephalin-leu, ala(2)-ser(6)-

DALES,2-Ala-6-ser-leu-enkephalin

Enkephalin-leu, ala(2)-ser(6)- is an active compound at the delta (non-complexed) opioid receptor.
T70232 3,4-Dephostatin

3,4-Dephostatin is an inhibitor of the interactions of CFTR-associated ligand (CAL) and PSD-95/Dlg1/ZO-1 (PDZ) domain.
T31242 Deacetylcephaloglycin

Deacetylcephaloglycin is an active metabolite of cephaloglycin, excreted in human urine.
T63218 Encephalitic alphavirus-IN-1

Encephalitic alphavirus-IN-1 能够抑制委内瑞拉马脑炎病毒 (VEEV) (EC50: 0.24 μM)和东部马脑炎病毒 (EEEV) (EC50: 0.16 μM)的活性。Encephalitic alphavirus-IN-1 没有明显的细胞毒性,而且表现出较强的小鼠血浆稳定性。
T41038 Sephadex G 50

Sephadex G 50 is a gel filtration medium commonly utilized in gel permeation chromatography for effective fractionation of glycopeptide mixtures.
T125321 Polycephalin C

Polycephalin C 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125321。
T64401 2,3,5,6-Tetra(9H-carbazol-9-yl)terephthalonitrile

2,3,5,6-Tetra(9H-carbazol-9-yl)terephthalonitrile 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64401。
T24032 Ephedrine levulinate

L-Ephedrine levulinate

Ephedrine levulinate is an alkaloid. Ephedrine acts as an agonist at alpha- and beta-adrenergic receptors and indirectly causes the release of norepinephrine from sympathetic neurons.
T77591 N-[5-[[[3-(6-Amino-4-methylpyridin-3-yl)-1-methyl-1H-indazol-5-yl]carbonyl]amino]-2-methylphenyl]-N′-methylterephthalamide

N-[5-[[[3-(6-Amino-4-methylpyridin-3-yl)-1-methyl-1H-indazol-5-yl]carbonyl]amino]-2-methylphenyl]-N′-methylterephthalamide在BD2 DEC-Tec实验中的IC50值为22nM。
T75281 Cephalexin hydrochloride monohydrate

Cephalexin (Cefalexin) hydrochloride monohydrate 是一种口服有效的半合成头孢菌素类抗生素(antibiotic),对广泛的革兰氏阳性及革兰氏阴性细菌展现出抗菌活性。该化合物通过靶向青霉素结合蛋白(PBPs)抑制细菌细胞壁的组装,应用于包括肺炎、链球菌性咽喉炎、细菌性心内膜炎在内的疾病研究。
T83504 [D-Ala2] Leu-Enkephalinamide

[D-Ala2] Leu-Enkephalinamide,一种脑啡肽类似物,展现出优异的角膜通透性及镇痛效果,适用于眼部疾病研究。
TP1255 [Met5]-Enkephalin, amide

5-Methionine-enkephalin amide

[Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.Met-enkephalin circulates in several forms, some of which may be derived from proteins other than proenkephalin A, and plasma levels of both free n
T31634 [Des-Tyr1]-Met-Enkephalin

Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-

Enkephalin-met, des-tyr(1)- ccauses retrograde amnesia in rats.
T37888 Desacetylcephapirin sodium

Desacetyl cefapirin is an active metabolite of the cephalosporin antibiotic cefapirin .1 Desacetyl cefapirin is active against E. coli, K. pneumoniae, P. mirabilis, and S. aureus with MIC values of 120, 24, 34, and 0.42 μg/ml, respectively.References1. Jones, R.N., and Packer, R.R. Cefotaxime, cephalothin, and cephapirin: Antimicrobial activity and synergy studies of cephalosporins with significant in vivo desacetyl metabolite concentrations. Diagn. Microbiol. Infect. Dis. 2(1), 65-68 (1984). De...
T73773 Metanephrine

Metanephrine 是肾上腺素的 O-甲基化代谢物,可用于嗜铬细胞瘤的研究。
T25804L Metkephamid acetate

Lilly 127623,LY127623,LY-127623,LY 127623

Metkephamid acetate is a synthetic opioid pentapeptide and derivative of [Met]enkephalin. It shows as a potent agonist of the δ- and μ-opioid receptors with roughly equipotent affinity, and also has similarly high affinity as well as subtype-selectivity f
T29410 3-Hydroxymephenytoin

3-Hydroxymephenytoin is a bioactive chemical.
T69070 Cephradine sodium

Cephradine sodium is the salt form of Cephradine (free base), a semi-synthetic cephalosporin antibiotic. Cefradin inhibits the last stage of bacterial cell wall synthesis by binding to certain penicillin-binding proteins which results in cell lysis. Cell lysis is mediated by bacterial cell wall autolytic enzymes. Cefradin may interfere with autolysin inhibitors.
T14929 Cephradine monohydrate

头孢拉定一水合物,Cefradine monohydrate

Antibacterial Microbiology/Virology
Cephradine monohydrate, a first-generation cephalosporin, is active against a wide range of Gram-positive and Gram-negative bacteria.

化合物

Eph inhibitor 2
Cat.No: T5451
Synonym: Ehp-inhibitor-1
Target: Ephrin Receptor
SI-2
Cat.No: T28773
Synonym: SI2,EPH 116,EPH116,EPH-116
Target: Others
SI-2 hydrochloride
Cat.No: T12906
Synonym: EPH 116 hydrochloride
Target: Src
ALW-II-41-27
Cat.No: T4344
Synonym: Eph receptor tyrosine kinase inhibitor
Target: Ephrin Receptor
[Leu5]-Enkephalin, amide acetate
Cat.No: TP1113L
Synonym: [Leu5]-Enkephalin, amide acetate(60117-24-0 free base)
Target: Opioid Receptor
Acephate
Cat.No: T22545
Synonym: acetylphosphoramidothioicacido,s-dimethylester,Ortran,Orthene,Acetamidophos,chevronorthene,乙酰甲胺磷
Target: AChE
Cephalonium
Cat.No: T0141
Synonym: 头孢洛宁,Cefalonium
Target: Others
Mephenytoin
Cat.No: T21425
Synonym: Mesantoin,Methoin,Insulton,Phenantoin,美芬妥因,Methylphenetoin
Target: P450
Cephradine
Cat.No: T0199
Synonym: Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定
Target: TOPK, Antibacterial, Antibiotic
(R)-Mephenytoin
Cat.No: T36839
Synonym: R-Mephenytoin,(R)-Mephenytoin,(–)-Mephenytoin
Target: Others
Cephalexin
Cat.No: T1008
Synonym: 头孢氨苄,Cefalexin,Cephacillin
Target: Antibacterial, Antibiotic
3-hydroxycephem
Cat.No: T4581
Synonym:
Target: Others
Sephin1
Cat.No: T21824
Synonym: NSC 65390,IFB-088
Target: Phosphatase
Mephenesin
Cat.No: T0015
Synonym: Cresoxydiol,甲酚甘油醚,Memphenesin,Mephedan,Decontractyl
Target: NMDAR, iGluR
Temephos
Cat.No: T0997
Synonym: 双硫磷,Temefos
Target: AChR, Parasite
Cephalexin monohydrate
Cat.No: T20022
Synonym: Cephalexin hydrate,Cephacillin hydrate,Cefalexin hydrate
Target: Antibiotic
[D-Ala2]leucine-enkephalin
Cat.No: TP1367
Synonym: (D-ALA2)-亮氨酸脑啡肽
Target: Opioid Receptor
(S)-Mephenytoin
Cat.No: T21529
Synonym:
Target: Others
[Leu5]-Enkephalin acetate(58822-25-6 free base)
Cat.No: T7173L
Synonym: 亮氨酸脑啡肽,Leucine enkephalin,Leu-enkephalin,Leucyl-enkephalin
Target: Opioid Receptor, Endogenous Metabolite
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
Cat.No: T7665
Synonym: Leu-enkephalin,Leucine enkephalin,Leucyl-enkephalin
Target: Opioid Receptor, Endogenous Metabolite
[Leu5]-Enkephalin
Cat.No: T7173
Synonym: 亮氨酸脑啡肽,Leucine enkephalin,Leucyl-enkephalin,Leu-enkephalin
Target: Opioid Receptor, Endogenous Metabolite
Bephenium (hydroxynaphthoate)
Cat.No: T0286
Synonym: 羟萘酸苄酚宁,Bephenium Hydroxynaphthoate
Target: Parasite
Cephalothin sodium
Cat.No: T1122
Synonym: 头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin
Target: Antibacterial, Antibiotic
[Met5]-Enkephalin, amide TFA
Cat.No: TP1254
Synonym: 5-Methionine-enkephalin amide (TFA)
Target: Opioid Receptor
(D-Ser2)-Leu-Enkephalin-Thr
Cat.No: T22752L
Synonym:
Target: Opioid Receptor
Shepherdin 79-87 acetate
Cat.No: T12896L
Synonym: Shepherdin 79-87 acetate (861224-28-4 free base)
Target: HSP, Survivin
N-terminally acetylated Leu-enkephalin
Cat.No: T8557
Synonym:
Target: Opioid Receptor
Cephalothin
Cat.No: T5570
Synonym: 头孢噻吩,Cephalotin acid
Target: Antibacterial, Antibiotic
Cephapirin Sodium
Cat.No: T5038
Synonym:
Target: Antibacterial, Antibiotic
7-Aminodeacetoxycephalosporanic acid
Cat.No: T1364
Synonym: 7-ADCA,Cephalexin Impurity B,Cefalexine EP IMpurity B,Deacetoxycephalosporanic Acid,头孢氨苄杂质B,7-Aminodesacetoxycephalosporanic acid
Target: Antibiotic
Cephalosporin C zinc salt
Cat.No: T7142
Synonym:
Target: Others
Enkephalin-leu, ala(2)-ser(6)-
Cat.No: T31631
Synonym: DALES,2-Ala-6-ser-leu-enkephalin
Target:
3,4-Dephostatin
Cat.No: T70232
Synonym:
Target:
Deacetylcephaloglycin
Cat.No: T31242
Synonym:
Target:
Encephalitic alphavirus-IN-1
Cat.No: T63218
Synonym:
Target:
Sephadex G 50
Cat.No: T41038
Synonym:
Target:
Polycephalin C
Cat.No: T125321
Synonym:
Target:
2,3,5,6-Tetra(9H-carbazol-9-yl)terephthalonitrile
Cat.No: T64401
Synonym:
Target:
Ephedrine levulinate
Cat.No: T24032
Synonym: L-Ephedrine levulinate
Target:
N-[5-[[[3-(6-Amino-4-methylpyridin-3-yl)-1-methyl-1H-indazol-5-yl]carbonyl]amino]-2-methylphenyl]-N′-methylterephthalamide
Cat.No: T77591
Synonym:
Target:
Cephalexin hydrochloride monohydrate
Cat.No: T75281
Synonym:
Target:
[D-Ala2] Leu-Enkephalinamide
Cat.No: T83504
Synonym:
Target:
[Met5]-Enkephalin, amide
Cat.No: TP1255
Synonym: 5-Methionine-enkephalin amide
Target:
[Des-Tyr1]-Met-Enkephalin
Cat.No: T31634
Synonym: Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-
Target:
Desacetylcephapirin sodium
Cat.No: T37888
Synonym:
Target:
Metanephrine
Cat.No: T73773
Synonym:
Target:
Metkephamid acetate
Cat.No: T25804L
Synonym: Lilly 127623,LY127623,LY-127623,LY 127623
Target:
3-Hydroxymephenytoin
Cat.No: T29410
Synonym:
Target:
Cephradine sodium
Cat.No: T69070
Synonym:
Target:
Cephradine monohydrate
Cat.No: T14929
Synonym: 头孢拉定一水合物,Cefradine monohydrate
Target: Antibacterial
Cat. No. Product Name Target Signaling Pathways
TN1480 Cephaeline

吐根鹼,吐根酚碱

Virus Protease; Influenza Virus; HIF Angiogenesis; Chromatin/Epigenetic; Microbiology/Virology
Cephaeline 对受保护的原代 CLL 细胞具有高度活性(相对 IC50 为 35nM),并通过抑制 HIF-1α± 和扰乱细胞内氧化还原稳态发挥作用。
T8031 Terephthalic acid

Others; Endogenous Metabolite Metabolism; Others
Terephthalic acid 是一种三种酞酸盐的异构体,是聚酯 PET 的前体,能够用于制作服装和塑料。
T0453 Phenylephrine hydrochloride

NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Phenylephrine hydrochloride (NCI-c55641) 是选择性的α1-肾上腺素能受体激动剂,对α1A,α1B 和α1D 受体的pKis 分为4.70,4.87和5.86。
T1287 Synephrine

辛弗林,Oxedrine

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Synephrine (Oxedrine) 是来自 Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂,是一种生物碱。它也是一种拟交感神经化合物,能够用于减肥。
T4945 Normetanephrine hydrochloride

DL-Normetanephrine hydrochloride,DL-去甲变肾上腺素盐酸盐

Endogenous Metabolite Metabolism
Normetanephrine hydrochloride (DL-Normetanephrine hydrochloride) 是肾上腺素的代谢物。它与肾上腺素一起存在于尿液和某些组织中。
T13655 DL-Norepinephrine hydrochloride

去甲肾上腺素盐酸盐,Lys,DL-lysine

Adrenergic Receptor GPCR/G Protein; Neuroscience
DL-Norepinephrine hydrochloride (DL-lysine) 是一种靶向α1 adrenoceptor 和β1 adrenoceptor 的神经递质,可降低心内膜下氧分压。它是一种模拟内源性去甲肾上腺素的拟交感神经作用的合成苯乙胺。
TN2326 (Z)-Butylidenephthalide

(Z)-3-Butylidenephthalide

Glucosidase Metabolism
(Z)-Butylidenephthalide ((Z)-3-Butylidenephthalide) 具有抗肿瘤和降血糖作用,能有效抑制胶质瘤的肿瘤生长,抑制 R-葡萄糖苷酶活性。
T3366 Cephalotaxine

ZINC19795976,三尖杉碱,(-)-Cephalotaxine,Cephalotaxlen

Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Cephalotaxine (ZINC19795976) 是从头孢紫杉中分离得到的一种生物碱,具有抗白血病和抗病毒活性,如抗 Zika 病毒。
T2217 Cephalomannine

Baccatin III,三尖杉宁碱

Microtubule Associated Cytoskeletal Signaling
Cephalomannine (Baccatin III) 是一种从云南红豆杉中提取的紫杉醇衍生物,具有抗肿瘤活性,可用于癌症研究。
T8063 Cephapirin Benzathine

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cephapirin Benzathine 是头孢哌啶的苄硫醚盐形式,是一种广谱抗生素。
T0131 Cepharanthine

NSC-623442,千金藤碱,千金藤素

Apoptosis; TNF; HIV Protease; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Cepharanthine (NSC-623442) 是从Stephania cepharanthaHayata 中提取的一种生物碱,具有抗炎、抗氧化作用。它可抑制肿瘤坏死因子 (TNF)-α 介导的 NFκB 刺激、质膜脂质过氧化和血小板聚集,并抑制细胞因子的产生。
T7044 Norepinephrine

去甲肾上腺素,Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol

MMP; Endogenous Metabolite; Adrenergic Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Neuroscience; Proteases/Proteasome
Norepinephrine (Levophed) 是β1选择性的肾上腺素能受体激动剂,EC50值为 5.37 μM。它可上调鼻咽癌肿瘤细胞中血管内皮生长因子、基质金属蛋白酶MMP-2和MMP-9的表达。
TN7236 Cephalandole B

IL Receptor Immunology/Inflammation
cephalandole B 是一种从青黛中分离出两种吲哚生物碱,能明显地抑制了IL-17A 基因的表达,以剂量依赖的方式抑制了Jukat 细胞的IL-17A 荧光素酶报告。
T6688 Synephrine hydrochloride

辛弗林盐酸盐,Oxedrine hydrochloride,Synephrine HCl

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Synephrine hydrochloride (Oxedrine hydrochloride) 是一种来自Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂的生物碱,也是一种拟交感神经化合物,能够用于减肥。
T38141 Glycerophospholipids, cephalins

Phosphatidylethanolamines (egg)

Glycerophospholipids, cephalins (Phosphatidylethanolamines (egg)) 是一种从鸡蛋中分离出来的磷脂酰乙醇胺的混合物,在 sn-1和 sn-2位置有各种脂肪酰基。Glycerophospholipids, cephalins 完全水解可得到1mol 的甘油、磷酸、乙醇胺和2mol 的脂肪酸。Phosphatidylethanolamines 在膜融合和细胞分裂过程中收缩环的拆卸中起作用,可调节膜的弯曲度。Phosphatidylethanolamines 能够在没有任何蛋白质或核酸的帮助下传播传染性朊病毒。Phosphatidylethanolamines 在细菌膜中的主要作用之一是分散由阴离子膜磷脂引起的负电荷。
T0989 7-Aminocephalosporanic acid

7-氨基头孢烷酸,7-ACA

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
7-Aminocephalosporanic acid (7-ACA) 用于合成头孢菌素类抗生素及其中间体。
TN1141 Isodeoxyelephantopin

异去氧苦地胆素,异去氧苦地胆苦素

NF-κB; Reactive Oxygen Species; Autophagy Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Isodeoxyelephantopin 是从地胆草中分离得到的一种倍半萜烯内酯,能调节 LncRNA 的表达,有抗乳腺癌的作用。它可诱导活性氧的生成,抑制 NF-κB 的激活。
T1064 Norepinephrine bitartrate monohydrate

酒石酸去甲肾上腺素,Levophed,Noradrenaline bitartrate monohydrate,降肾上腺素

Endogenous Metabolite; Adrenergic Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Neuroscience
Norepinephrine bitartrate monohydrate (Levophed) 是一种β1-选择性的肾上腺素能受体激动剂,EC50为 5.37 μM。
T10147 4-Hydroxymephenytoin

(+/-)-4'-Hydroxymephenytoin

Others; Drug Metabolite Metabolism; Others
4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) 是抗癫痫药 mephenytoin 的代谢产物。Mephenytoin 是 CYP2C19的配体。
T3S2072 3-Butylidenephthalide

Butylidene phthalide,n-Butylidenephthalide,丁烯基苯酞,丁烯基苯酞;丁烯基酞内酯

Parasite; Glucosidase Metabolism; Microbiology/Virology
3-Butylidenephthalide (Butylidene phthalide) 是从 Ligusticum chuanxiongHort 鉴定出的一种邻苯二甲酸酐衍生物,有杀虫活性。
TN1079 Deoxyelephantopin

NF-κB NF-κB
Deoxyelephantopin 是来自Elephantopus scaber 的,具有生物活性的天然倍半萜烯内酯,能够抑制NF-κB,MAPK,PI3K/Akt 和β-catenin 信号传导。它可广泛用于癌症方面的研究。
T21066 Norepinephrine bitartrate salt

Adrenergic Receptor GPCR/G Protein; Neuroscience
Norepinephrine bitartrate salt 是一种肾上腺素能神经递质。
T3S1852 Cephaeline hydrochloride

Others; Virus Protease; Influenza Virus Microbiology/Virology; Others
Cephaeline hydrochloride 是 Indian Ipecac 中的一种酚类生物碱。它有效抑制病毒 ZIKV 和 EBOV 感染。
T17310 Phenylephrine

去氧肾上腺素,L-Phenylephrine,去氧肾上腺素碱,(R)-(-)-Phenylephrine

Adrenergic Receptor GPCR/G Protein; Neuroscience
Phenylephrine ((R)-(-)-Phenylephrine) 是一种选择性的α1-肾上腺素受体激动剂,常用作减充血剂。
TN6014 Norcepharadione B

鱼腥草

Norcepharadione B shows good inhibitory activity against the replication of HSV-1, it also shows antimalarial activity with EC50 values of 7.5mug/ml. Norcepharadione B exhibits significant cytotoxicity against five human tumor cell lines (A-549, SK-OV-3,
TN6283 Stepharine

Stepharine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6283,CAS号为 2810-21-1。
TN6252 Isostephodeline

Isostephodeline 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6252,CAS号为 56648-85-2。
TN3850 Dihydroepistephamiersine 6-acetate

Others Others
Dihydroepistephamiersine 6-acetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3850,CAS号为 57361-74-7。
T8265 p-Synephrine

Others Others
p-Synephrine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T8265,CAS号为 614-35-7。
TN6261 Stephodeline

Stephodeline 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6261,CAS号为 56596-12-4。
TN4833 Prostephanaberrine

Others Others
Prostephanaberrine is a natural product from Stephania japonica.
TN3857 Dihydrooxoepistephamiersine

Others Others
Dihydrooxoepistephamiersine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3857,CAS号为 51804-69-4。
T75425 Synephrine hemitartrate

Synephrine (Oxedrine) hemitartrate,一种生物碱,是一种来自Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂。Synephrine hemitartrate 是一种拟交感神经化合物,可用于减肥。
TN6293 Stephalonine M

Stephalonine M 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6293,CAS号为 2376321-05-8。
TN6020 4-Hydroxycephalotaxine

4-Hydroxycephalotaxine is a natural product from Cephalotaxus fortunei.
T20473 Bis(2-ethylhexyl) terephthalate

Bis(2-ethylhexyl) terephthalate is an agent of biochemical.
TN3622 Cephalocyclidin A

Others Others
Cephalocyclidin A是一种天然产物,属于三尖杉科三尖杉属,其产品编号为 TN3622,CAS号为 421583-14-4。Cephalocyclidin A可用作对照参考。
TN6018 Epistephamiersine

Epistephamiersine是一种天然产物,属于防己科千金藤属,其产品编号为 TN6018,CAS号为 52389-15-8。Epistephamiersine可用作对照参考。
T81816 Met-Enkephalin-Arg-Phe

Met-Enkephalin-Arg-Phe 是一种天然七肽,具有镇痛活性。
TN6291 Stephalonine N

Stephalonine N 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6291,CAS号为 2376321-20-7。
T31429 Dibutyl terephthalate

Dibutyl terephthalate is a biochemical.
T82859 Blepharotriol

Blepharotriol为Maytenus blepharodes中发现的一种酚类三萜化合物。该化合物具有抗菌特性,对Bacillus subtilis的最小抑菌浓度(MIC)为8-4 µg/ml。此外,Blepharotriol在HeLa、Hep-2、Vero细胞上的半数抑制浓度(IC50)分别为12.2、>20、>20 µM,表明其具有一定的细胞毒性。
TN2588 11-Hydroxytephrosin

TNF; NF-κB Apoptosis; NF-κB
11-Hydroxytephrosin inhibits NF-kappaB activity.
T82639 Cyclocephaloside II

Cyclocephaloside II,一种从Astragalus brachypterus和Astragalus microcephalus的根部提取的天然产物。
TN5605 7-Epi-10-deacetylcephalomannine

7-Epi-10-deacetylcephalomannine is a natural product from Taxus sumatrana.
T81235 S-(-)-N-trans-Feruloyl normetanephrine

S-(-)-N-trans-Feruloyl normetanephrine为天然产物,呈现弱抗乙酰胆碱酯酶活性,可从Bassia indica Wight地上部分提取。
TN6290 Stephalonine L

Stephalonine L 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6290,CAS号为 2379277-60-6。
TN6022 Stephavanine

Stephavanine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6022,CAS号为 33116-33-5。
T83525 (Rac)-Tephrosin

(Rac)-Tephrosin为存在于Tephrosia purpurea中的天然产物。
T83234 8-Demethoxycephatonine

8-Demethoxycephatonine是从Menispermaceae科植物Sinomenium acutum中分离出的一种异喹啉生物碱。
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天然产物

Cephaeline
Cat.No: TN1480
Synonym: 吐根鹼,吐根酚碱
Target: Virus Protease, Influenza Virus, HIF
Terephthalic acid
Cat.No: T8031
Synonym:
Target: Others, Endogenous Metabolite
Phenylephrine hydrochloride
Cat.No: T0453
Synonym: NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride
Target: Endogenous Metabolite, Adrenergic Receptor
Synephrine
Cat.No: T1287
Synonym: 辛弗林,Oxedrine
Target: Endogenous Metabolite, Adrenergic Receptor
Normetanephrine hydrochloride
Cat.No: T4945
Synonym: DL-Normetanephrine hydrochloride,DL-去甲变肾上腺素盐酸盐
Target: Endogenous Metabolite
DL-Norepinephrine hydrochloride
Cat.No: T13655
Synonym: 去甲肾上腺素盐酸盐,Lys,DL-lysine
Target: Adrenergic Receptor
(Z)-Butylidenephthalide
Cat.No: TN2326
Synonym: (Z)-3-Butylidenephthalide
Target: Glucosidase
Cephalotaxine
Cat.No: T3366
Synonym: ZINC19795976,三尖杉碱,(-)-Cephalotaxine,Cephalotaxlen
Target: Antiviral, Influenza Virus
Cephalomannine
Cat.No: T2217
Synonym: Baccatin III,三尖杉宁碱
Target: Microtubule Associated
Cephapirin Benzathine
Cat.No: T8063
Synonym:
Target: Others, Antibacterial, Antibiotic
Cepharanthine
Cat.No: T0131
Synonym: NSC-623442,千金藤碱,千金藤素
Target: Apoptosis, TNF, HIV Protease, Autophagy
Norepinephrine
Cat.No: T7044
Synonym: 去甲肾上腺素,Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol
Target: MMP, Endogenous Metabolite, Adrenergic Receptor, Autophagy
Cephalandole B
Cat.No: TN7236
Synonym:
Target: IL Receptor
Synephrine hydrochloride
Cat.No: T6688
Synonym: 辛弗林盐酸盐,Oxedrine hydrochloride,Synephrine HCl
Target: Endogenous Metabolite, Adrenergic Receptor
Glycerophospholipids, cephalins
Cat.No: T38141
Synonym: Phosphatidylethanolamines (egg)
Target:
7-Aminocephalosporanic acid
Cat.No: T0989
Synonym: 7-氨基头孢烷酸,7-ACA
Target: Others, Antibacterial, Antibiotic
Isodeoxyelephantopin
Cat.No: TN1141
Synonym: 异去氧苦地胆素,异去氧苦地胆苦素
Target: NF-κB, Reactive Oxygen Species, Autophagy
Norepinephrine bitartrate monohydrate
Cat.No: T1064
Synonym: 酒石酸去甲肾上腺素,Levophed,Noradrenaline bitartrate monohydrate,降肾上腺素
Target: Endogenous Metabolite, Adrenergic Receptor, Autophagy
4-Hydroxymephenytoin
Cat.No: T10147
Synonym: (+/-)-4'-Hydroxymephenytoin
Target: Others, Drug Metabolite
3-Butylidenephthalide
Cat.No: T3S2072
Synonym: Butylidene phthalide,n-Butylidenephthalide,丁烯基苯酞,丁烯基苯酞;丁烯基酞内酯
Target: Parasite, Glucosidase
Deoxyelephantopin
Cat.No: TN1079
Synonym:
Target: NF-κB
Norepinephrine bitartrate salt
Cat.No: T21066
Synonym:
Target: Adrenergic Receptor
Cephaeline hydrochloride
Cat.No: T3S1852
Synonym:
Target: Others, Virus Protease, Influenza Virus
Phenylephrine
Cat.No: T17310
Synonym: 去氧肾上腺素,L-Phenylephrine,去氧肾上腺素碱,(R)-(-)-Phenylephrine
Target: Adrenergic Receptor
Norcepharadione B
Cat.No: TN6014
Synonym: 鱼腥草
Target:
Stepharine
Cat.No: TN6283
Synonym:
Target:
Isostephodeline
Cat.No: TN6252
Synonym:
Target:
Dihydroepistephamiersine 6-acetate
Cat.No: TN3850
Synonym:
Target: Others
p-Synephrine
Cat.No: T8265
Synonym:
Target: Others
Stephodeline
Cat.No: TN6261
Synonym:
Target:
Prostephanaberrine
Cat.No: TN4833
Synonym:
Target: Others
Dihydrooxoepistephamiersine
Cat.No: TN3857
Synonym:
Target: Others
Synephrine hemitartrate
Cat.No: T75425
Synonym:
Target:
Stephalonine M
Cat.No: TN6293
Synonym:
Target:
4-Hydroxycephalotaxine
Cat.No: TN6020
Synonym:
Target:
Bis(2-ethylhexyl) terephthalate
Cat.No: T20473
Synonym:
Target:
Cephalocyclidin A
Cat.No: TN3622
Synonym:
Target: Others
Epistephamiersine
Cat.No: TN6018
Synonym:
Target:
Met-Enkephalin-Arg-Phe
Cat.No: T81816
Synonym:
Target:
Stephalonine N
Cat.No: TN6291
Synonym:
Target:
Dibutyl terephthalate
Cat.No: T31429
Synonym:
Target:
Blepharotriol
Cat.No: T82859
Synonym:
Target:
11-Hydroxytephrosin
Cat.No: TN2588
Synonym:
Target: TNF, NF-κB
Cyclocephaloside II
Cat.No: T82639
Synonym:
Target:
7-Epi-10-deacetylcephalomannine
Cat.No: TN5605
Synonym:
Target:
S-(-)-N-trans-Feruloyl normetanephrine
Cat.No: T81235
Synonym:
Target:
Stephalonine L
Cat.No: TN6290
Synonym:
Target:
Stephavanine
Cat.No: TN6022
Synonym:
Target:
(Rac)-Tephrosin
Cat.No: T83525
Synonym:
Target:
8-Demethoxycephatonine
Cat.No: T83234
Synonym:
Target:
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