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75

抑制剂 & 化合物

28

天然产物

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Cat. No. Product Name Target Signaling Pathways
T1144L Lidocaine Hydrochloride hydrate

EGFR; Sodium Channel Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
Lidocaine Hydrochloride hydrate 是一种酰胺类局部麻醉剂,具有抗炎作用。
T0929 Docusate sodium

Aerosol OT,多库脂钠,Dioctyl sulfosuccinate sodium salt,Bis(2-ethylhexyl) sulfosuccinate sodium salt,Constonate

Opioid Receptor; HSV Endocrinology/Hormones; GPCR/G Protein; Microbiology/Virology; Neuroscience
Docusate sodium (Aerosol OT) 是一种口服的非处方泻药和大便软化剂,可用于研究便秘。
T68079 Gedocarnil

ZK 113315,SH 530

Others Others
Gedocarnil(ZK 113315) 可用于研究中枢神经系统疾病。
T31716 Etidocaine Hydrochloride

W-19053,Duranest,W19053,W 19053

Sodium Channel Membrane transporter/Ion channel
Etidocaine Hydrochloride (W19053) 是一种长效麻醉剂和电压门控钠通道阻滞剂。
T10431 Golidocitinib

AZD4205

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Golidocitinib (AZD4205) 是一种选择性 JAK1抑制剂,IC50值为 73 nM。
T16280 Nedocromil

FPL 59002,尼多克罗

Leukotriene Receptor; Prostaglandin Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Nedocromil (FPL 59002) 对多种介质的作用或形成有抑制作用,包括组胺,前列腺素 D2和白三烯 C4。
T8146 Imidocarb dipropionate

二丙酸咪唑苯脲,二丙酸双咪苯脲

Antibiotic; Parasite Microbiology/Virology
Imidocarb dipropionate 是一种抗原虫剂,对寄生虫 B. bovis 的 IC50为 87 μg/mL。
T16558 Polidocanol

Polyoxyethylene lauryl ether,Polyoxyethyleneglycol Dodecyl Ether

Others Others
Polidocanol (Polyoxyethylene lauryl ether) 是月桂醇的烷基聚乙二醇醚,是天然矿物油 中天然脂肪醇或烷基醇的衍生物,是一种硬化剂。Polidocanol 可用做局部麻醉,但与 其他麻醉药物合用时有增强麻醉药物对心血管系统作用的风险。
T40475 Ceftobiprole medocaril

BAL5788,头孢比普酯

Antibacterial Microbiology/Virology
Ceftobiprole medocaril (BAL5788) 是 Ceftobiprole 的前药。Ceftobiprole 是一种广谱的头孢菌素,对耐甲氧西林金黄色葡萄球菌具有活性。
T19319 Ethyl docosa-4,7,10,13,16,19-hexaenoate

Others Others
Ethyl cis-4,7,10,13,16,19-Docosahexaenoate, the ethyl ester of Docosahexaenoate (DHA), is selectively enriched in the ethyl ester fraction through the alcoholysis process involving fatty acid ethyl esters from tuna oil and lauryl alcohol.
T14875 Indocyanine green

Cardiogreen,IC Green,Foxgreen,吲哚菁绿

Others Others
Indocyanine green (Cardiogreen) 是低毒性荧光剂,普遍用于医学诊断,包括确定心输出量,肝功能和肝血流量,以及用于眼科血管造影。
T0468 Lidocaine

Lignocaine,Alphacaine,Xylocaine,利多卡因

Apoptosis; ERK; NF-κB; MEK; Sodium Channel; Histamine Receptor Apoptosis; GPCR/G Protein; Immunology/Inflammation; MAPK; Membrane transporter/Ion channel; Neuroscience; NF-κB
Lidocaine (Alphacaine) 是一种酰胺衍生物,抑制涉及复杂电压和依赖性的钠通道,可用于研究室性心律失常。它通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。
T14060 6-Maleimidocapronic acid

PROTAC Linker PROTAC
6-Maleimidocapronic acid 是一种属于 alkyl chain 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T19294 Docosahexaenoic Acid methyl ester

二十二六烯酸甲酯,Methyl docosahexaenoate,all cis-DHA methyl ester

Others Others
Docosahexaenoic Acid methyl ester (all cis-DHA methyl ester) 是甲基化的二十二碳六烯酸类似物,能够插入膜磷脂中而不被氧化或水解。
T31716L Etidocaine

Others Others
Etidocaine 是一种氨基酸酰胺,用作局部麻醉剂,具有快速起效和长效特性。
T1144 Lidocaine hydrochloride

Lidocaine HCL,盐酸利多卡因,Lignocaine hydrochloride,Xyloneural,Lidothesin

Apoptosis; ERK; NF-κB; MEK; Sodium Channel Apoptosis; MAPK; Membrane transporter/Ion channel; NF-κB
Lidocaine hydrochloride (Lignocaine hydrochloride) 抑制涉及复杂电压和依赖性的钠通道。它通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。Lidocaine 是一种酰胺衍生物,是一种研究室性心律失常的药物和有效的肿瘤抑制剂。
T35009 Vadocaine

Vadocaina,Vadocainum

Others Others
Vadocaine (Vadocaina) 是一种新型的镇咳化合物,可用于局部麻醉,可用于研究中枢神经系统和心血管系统。
T124800 Endocrocin

Endocrocin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124800,CAS号为 481-70-9。
T30271 Azidocillin sodium salt

Nalpen,Globacillin,Longatren

Azidocillin sodium salt is a type of penicillin.
TQ0247 7-Epi-docetaxel

7-Epidocetaxel,7-表多西他赛,4-epi-Docetaxel,7-Epitaxotere

Others Others
7-Epi-10-oxo-docetaxel (7-Epitaxotere) is a impurity of docetaxel.
T77174 Efmarodocokin alfa

Efmarodocokin alfa为人IL-22与IgG4可结晶片段的融合蛋白,具有激活IL-22信号的功能。该化学物质主要用于重症COVID-19肺炎的研究。
T77173 Eflepedocokin alfa

Eflepedocokin alfa 是一种具有潜在细胞保护活性的重组融合蛋白。Eflepedocokin alfa 由人的IL-22与人的IgG2-Fc 结构域融合组成。Eflepedocokin alfa 可激活IL-22/IL-22R 介导的信号转导通路以及STAT3。Eflepedocokin alfa 在免疫反应和细菌感染、增强肠道屏障功能、肠道免疫和组织修复方面发挥作用。
T37532 Docosahexaenoyl Glycine

The ω-3 polyunsaturated fatty acids (PUFAs) found in fish oils provide cardiovascular benefits. Docosahexaenoic acid (DHA), a C22:6 PUFA, is the most abundant ω-3 fatty acid in neural tissues, especially in the retina and brain. It can be synthesized from other dietary ω-3 PUFAs or taken as a nutritional supplement. Docosahexaenoyl glycine consists of DHA with glycine attached at its carboxy terminus.
T77230 1-O-Hexadecyl-2-O-docosahexaenoyl-sn-glycero-3-phosphorylcholine

1-O-Hexadecyl-2-O-docosahexaenoyl-sn-glycero-3-phosphorylcholine为存在于尿中的内源性代谢物,用于肥胖研究。
T19520 Piridocaine hydrochloride

Lucaine hydrochloride

Others Others
Piridocaine hydrochloride is a piperidyl propanol ester of orthoaminobenzoic acid.
T73194 DOCK2-IN-1

DOCK2-IN-1 是 CPYPP 类似物,也是DOCK2的抑制剂 (IC50=19.1 μM)。DOCK2-IN-1 以可逆方式结合DOCK2DHR-2 结构域以抑制其催化活性。DOCK2-IN-1 阻断淋巴细胞中趋化因子受体和抗原受体介导的 Rac 的激活。DOCK2-IN-1 显着抑制趋化反应和 T 细胞活化。
TD0084 DiI triflate [1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine triflate]

DiI triflate is one of lipophilic fluorescent stains for labeling membranes and other hydrophobic structures. The fluorescence of these environment-sensitive dyes is greatly enhanced when incorporated into membranes or bound to lipophilic biomolecules such as proteins although they are weakly fluorescent in water.
TQ0142 10-Oxo Docetaxel

Docetaxel Impurity 1,10-氧多西他赛

Others Others
10-Oxo Docetaxel is a Docetaxel intermediate having remarkable antitumor properties.
T62520 Imidocarb dihydrochloride monohydrate

Imidocarb dihydrochloride monohydrate 是一种有效的抗原虫剂,能够作用于寄生虫 B. bovis (IC50: 87 μg/ml)。
T25720 Lidocaine methiodide

Methyllidocaine iodide,N-Methyllidocaine

Lidocaine methiodide is an antiarrythmic. It is also exhibiting arrythmogenic effects in subjects.
T72141 Ceftobiprole medocaril sodium

头孢比普酯钠盐,BAL5788 sodium

Ceftobiprole medocaril (BAL5788) sodium 是 Ceftobiprole 的胃肠外前药。Ceftobiprole 是一种非肠道吡咯烷酮头孢菌素。Ceftobiprole 是一种广谱头孢菌素,对甲氧西林 (MRSA) 和耐万古霉素葡萄球菌 (VRSA) 和耐青霉素链球菌具有高水平的体外活性。Ceftobiprole 也抑制革兰氏阳性和革兰氏阴性病原体。
T37634 17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic Acid

Docosapentaenoic acid (DPA) is a ω-3 fatty acid found in fish oils. 17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-docosapentaenoic acid is a metabolite of lipoxygenase-mediated oxidation of DPA that is produced endogenously by aspirin-enhanced COX-2 activity. It has been shown to activate Nrf2-dependent antioxidant gene expression, to act as a PPARγ agonist (EC50 = ~200 nM), and to inhibit pro-inflammatory cytokine and nitric oxide production at biological concentration ranges (5-25 μM).
T38527 2',3'-Dideoxy-5-iodocytidine

2',3'-Dideoxy-5-iodocytidine, a chemical compound, is employed in gene sequencing and functions as an antibiotic. It exhibits significant efficacy specifically against Mycobacterium.
T19163 7-Epi-10-oxo-docetaxel

Docetaxel Impurity 2

Others Others
7-Epi-10-oxo-docetaxel (Docetaxel Impurity 2) is an impurity of docetaxel detected by HPLC.
T36868 4-oxo Docosahexaenoic Acid

4-oxo Docosahexaenoic acid (4-oxo DHA) is a putative metabolite of DHA with antiproliferative and PPARγ agonist activity. It inhibits the growth of several triple negative breast cancer cell lines (MCF-10F, trMCF, bsMCF, MDA-MB-231, and BT549) at 50-100 μM, however it increased proliferation of MCF-7 cells. 4-oxo DHA binds covalently to PPARγ and activates gene transcription in luciferase reporter assays and in dendritic cells with EC50 values of approximately 8-16 μM.
T29981 Amidochlor

Caswell No. 005B,EPA Pesticide Chemical Code 128001,MON 4620,MON 4621,Limit

Amidochlor is a growth regulator.
TNU0763 2’-Deoxy-2’-fluoro-N3-(n-docecyl)uridine

2'-Deoxy-2'-fluoro-N3-(n-docecyl)uridine is a Nucleoside Derivative - Fluoro-modified nucleoside, 2'-Modified nucleoside.
TD0083 DiIiodide1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine iodide]

DiI碘化物

DiI iodide1 is one of lipophilic fluorescent stains for labeling membranes and other hydrophobic structures. The fluorescence of these environment-sensitive dyes is greatly enhanced when incorporated into membranes or bound to lipophilic biomolecules such as proteins although they are weakly fluorescent in water.
T34382 Rodocaine

R-19317,R 19317,R19317

Rodocaine is a biochemical.
T16694 Pyridoclax

MR-29072

BCL Apoptosis
Pyridoclax is an inhibitor of potential Mcl-1.
T24171 Iodoclorgyline

6-Iodoclorgyline

Iodoclorgyline is an inhibitor of monoamine oxidase A.
T77161 Docaravimab

Docaravimab为针对ERA (Evelyn-Rockitniki-Abelseth) 糖蛋白胞外域表位G-III的抗体,适用于狂犬病研究。
T38644 Docetaxal

PNU-101383,10-Acetyl docetaxel

Docetaxal, also known as 10-Acetyl docetaxel, is an analog of Docetaxel exhibiting potent anticancer properties. It acts as a microtubule disassembly inhibitor, effectively inhibiting mitosis.
T71805 DOCK5-IN-C21

DOCK5-IN-C21 is an allosteric inhibitor of the guanine nucleotide exchange factor DOCK5.
T37633 17-oxo-4(Z),7(Z),10(Z),13(Z),15(E),19(Z)-Docosahexaenoic Acid

17-oxo-4(Z),7(Z),10(Z),13(Z),15(E),19(Z)-Docosahexaenoic acid is a metabolite of lipoxygenase-mediated oxidation of DHA that is produced endogenously by aspirin-enhanced COX-2 activity. It has been shown to activate Nrf2-dependent antioxidant gene expression, to act as a PPARγ agonist (EC50 = ~200 nM), and to inhibit pro-inflammatory cytokine and nitric oxide production at biological concentration ranges (5-25 μM).
T64415 22-(tert-Butoxy)-22-oxodocosanoic acid

22-(tert-Butoxy)-22-oxodocosanoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64415,CAS号为 1642333-05-8。
TNU0629 5-Iodocytosine

5-Iodocytosine is a Heterocyclic compound-pyrimidine, intermediate and building block, halo-.
T25308 Deoxymulundocandin

Deoxymulundocandin is an echinocandin type antifungal antibiotic from Aspergillus sydowii.
T14059 6-Maleimidocaproic acid-PFP ester

Others Others
6-Maleimidocaproic acid-PFP ester is a hydrocarbon-based PROTAC linker, suitable for the synthesis of PROTACs[1].
T15155 Docebenone

AA 861

Others Others
Docebenone is a selective and orally active inhibitor of 5-LO.

化合物

Lidocaine Hydrochloride hydrate
Cat.No: T1144L
Synonym:
Target: EGFR, Sodium Channel
Docusate sodium
Cat.No: T0929
Synonym: Aerosol OT,多库脂钠,Dioctyl sulfosuccinate sodium salt,Bis(2-ethylhexyl) sulfosuccinate sodium salt,Constonate
Target: Opioid Receptor, HSV
Gedocarnil
Cat.No: T68079
Synonym: ZK 113315,SH 530
Target: Others
Etidocaine Hydrochloride
Cat.No: T31716
Synonym: W-19053,Duranest,W19053,W 19053
Target: Sodium Channel
Golidocitinib
Cat.No: T10431
Synonym: AZD4205
Target: JAK
Nedocromil
Cat.No: T16280
Synonym: FPL 59002,尼多克罗
Target: Leukotriene Receptor, Prostaglandin Receptor, Histamine Receptor
Imidocarb dipropionate
Cat.No: T8146
Synonym: 二丙酸咪唑苯脲,二丙酸双咪苯脲
Target: Antibiotic, Parasite
Polidocanol
Cat.No: T16558
Synonym: Polyoxyethylene lauryl ether,Polyoxyethyleneglycol Dodecyl Ether
Target: Others
Ceftobiprole medocaril
Cat.No: T40475
Synonym: BAL5788,头孢比普酯
Target: Antibacterial
Ethyl docosa-4,7,10,13,16,19-hexaenoate
Cat.No: T19319
Synonym:
Target: Others
Indocyanine green
Cat.No: T14875
Synonym: Cardiogreen,IC Green,Foxgreen,吲哚菁绿
Target: Others
Lidocaine
Cat.No: T0468
Synonym: Lignocaine,Alphacaine,Xylocaine,利多卡因
Target: Apoptosis, ERK, NF-κB, MEK, Sodium Channel, Histamine Receptor
6-Maleimidocapronic acid
Cat.No: T14060
Synonym:
Target: PROTAC Linker
Docosahexaenoic Acid methyl ester
Cat.No: T19294
Synonym: 二十二六烯酸甲酯,Methyl docosahexaenoate,all cis-DHA methyl ester
Target: Others
Etidocaine
Cat.No: T31716L
Synonym:
Target: Others
Lidocaine hydrochloride
Cat.No: T1144
Synonym: Lidocaine HCL,盐酸利多卡因,Lignocaine hydrochloride,Xyloneural,Lidothesin
Target: Apoptosis, ERK, NF-κB, MEK, Sodium Channel
Vadocaine
Cat.No: T35009
Synonym: Vadocaina,Vadocainum
Target: Others
Endocrocin
Cat.No: T124800
Synonym:
Target:
Azidocillin sodium salt
Cat.No: T30271
Synonym: Nalpen,Globacillin,Longatren
Target:
7-Epi-docetaxel
Cat.No: TQ0247
Synonym: 7-Epidocetaxel,7-表多西他赛,4-epi-Docetaxel,7-Epitaxotere
Target: Others
Efmarodocokin alfa
Cat.No: T77174
Synonym:
Target:
Eflepedocokin alfa
Cat.No: T77173
Synonym:
Target:
Docosahexaenoyl Glycine
Cat.No: T37532
Synonym:
Target:
1-O-Hexadecyl-2-O-docosahexaenoyl-sn-glycero-3-phosphorylcholine
Cat.No: T77230
Synonym:
Target:
Piridocaine hydrochloride
Cat.No: T19520
Synonym: Lucaine hydrochloride
Target: Others
DOCK2-IN-1
Cat.No: T73194
Synonym:
Target:
DiI triflate [1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine triflate]
Cat.No: TD0084
Synonym:
Target:
10-Oxo Docetaxel
Cat.No: TQ0142
Synonym: Docetaxel Impurity 1,10-氧多西他赛
Target: Others
Imidocarb dihydrochloride monohydrate
Cat.No: T62520
Synonym:
Target:
Lidocaine methiodide
Cat.No: T25720
Synonym: Methyllidocaine iodide,N-Methyllidocaine
Target:
Ceftobiprole medocaril sodium
Cat.No: T72141
Synonym: 头孢比普酯钠盐,BAL5788 sodium
Target:
17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic Acid
Cat.No: T37634
Synonym:
Target:
2',3'-Dideoxy-5-iodocytidine
Cat.No: T38527
Synonym:
Target:
7-Epi-10-oxo-docetaxel
Cat.No: T19163
Synonym: Docetaxel Impurity 2
Target: Others
4-oxo Docosahexaenoic Acid
Cat.No: T36868
Synonym:
Target:
Amidochlor
Cat.No: T29981
Synonym: Caswell No. 005B,EPA Pesticide Chemical Code 128001,MON 4620,MON 4621,Limit
Target:
2’-Deoxy-2’-fluoro-N3-(n-docecyl)uridine
Cat.No: TNU0763
Synonym:
Target:
DiIiodide1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine iodide]
Cat.No: TD0083
Synonym: DiI碘化物
Target:
Rodocaine
Cat.No: T34382
Synonym: R-19317,R 19317,R19317
Target:
Pyridoclax
Cat.No: T16694
Synonym: MR-29072
Target: BCL
Iodoclorgyline
Cat.No: T24171
Synonym: 6-Iodoclorgyline
Target:
Docaravimab
Cat.No: T77161
Synonym:
Target:
Docetaxal
Cat.No: T38644
Synonym: PNU-101383,10-Acetyl docetaxel
Target:
DOCK5-IN-C21
Cat.No: T71805
Synonym:
Target:
17-oxo-4(Z),7(Z),10(Z),13(Z),15(E),19(Z)-Docosahexaenoic Acid
Cat.No: T37633
Synonym:
Target:
22-(tert-Butoxy)-22-oxodocosanoic acid
Cat.No: T64415
Synonym:
Target:
5-Iodocytosine
Cat.No: TNU0629
Synonym:
Target:
Deoxymulundocandin
Cat.No: T25308
Synonym:
Target:
6-Maleimidocaproic acid-PFP ester
Cat.No: T14059
Synonym:
Target: Others
Docebenone
Cat.No: T15155
Synonym: AA 861
Target: Others
Cat. No. Product Name Target Signaling Pathways
T3033 Deoxycorticosterone acetate

醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮

Glucocorticoid Receptor; Endogenous Metabolite; Adrenergic Receptor Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
Deoxycorticosterone acetate (Cortexone acetate) 是肾上腺产生的类固醇激素,具有盐皮质激素活性,并作为醛固酮的前体。
T19295 Docosapentaenoic acid 22n-3

Endogenous Metabolite Metabolism
Docosapentaenoic acid 22n-3 是在所有动物细胞膜中发现的磷脂组成成分。
T9862 Pseudocoptisine chloride

盐酸异黄连碱,Isocoptisine chloride

AChE Neuroscience
Pseudocoptisine chloride (Isocoptisine chloride) 是从 Corydalis Tuber 中分离出来的,具有抗炎和抗健忘的作用。 Pseudocoptisine chloride 抑制乙酰胆碱酯酶 (AChE) 活性 (IC50 = 12.8 μM)。
T12514 Podocarpic acid

Others; TRP/TRPV Channel Membrane transporter/Ion channel; Others
Podocarpic acid 是一种天然产物,是一种新型 TRPA1 激活剂。
T9784 Docosanedioic acid 

PROTAC Linker PROTAC
Docosanedioic acid 可以作为ADC linker 或PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。
TQ0134 Podocarpusflavone A

Topoisomerase DNA Damage/DNA Repair
Podocarpusflavone A is a DNA topoisomerase I inhibitor. It has moderated anti-proliferative activity induce cell apoptosis in MCF-7.
T5942 Docosanoic acid

Behenic Acid,山嵛酸

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Docosanoic acid (Behenic Acid) 是一种较难吸收的饱和脂肪酸,能提高人类胆固醇水平。
T5369 Docosahexaenoic Acid

Cervonic acid,DHA

Others; Endogenous Metabolite Metabolism; Others
Docosahexaenoic Acid 是一种ω-3脂肪酸,在脑和视网膜中较为丰富,且能够直接从鱼油和母乳中获得。
T0884 1-Docosanol

Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol

Antifection; HSV Microbiology/Virology
1-Docosanol (Behenic alcohol) 是一种具有抗病毒活性的饱和 22 碳脂肪醇,局部用于治疗复发性单纯性唇疱疹发作并缓解相关疼痛并可能有助于更快地治愈疮。
TN6962 Docosane

Others Others
Docosane 是一种直链烷烃,可用于合成具有热能储存/释放能力的结构复合材料。
T0186 Docetaxel trihydrate

RP-56976 (Trihydrate),RP56976 (NSC 628503) Trihydrate,多西他赛三水合物

Apoptosis; BCL; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Docetaxel trihydrate (RP-56976 Trihydrate) 是一种抗肿瘤试剂,抑制微管解聚的IC50值为 0.2 μM。它是紫杉醇的半合成类似物,能减弱 bcl-2 和 bcl-xL 基因表达的影响。它阻滞G2/M 细胞周期,导致细胞凋亡。
T1034 Docetaxel

多西他赛,NSC 628503,RP-56976,多烯紫杉醇

Apoptosis; Microtubule Associated; Endogenous Metabolite Apoptosis; Cytoskeletal Signaling; Metabolism
Docetaxel (RP-56976) 是紫杉醇的半合成类似物,是一种微管解聚抑制剂 (IC50=0.2 μM)。Docetaxel 可以减弱 bcl-2 和 bcl-xL 基因表达的影响,具有诱导凋亡、抗肿瘤活性。
TN2619 13-Oxopodocarp-8(14)-en-18-oic acid

Others Others
13-Oxopodocarp-8(14)-en-18-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2619,CAS号为 63976-69-2。
TN5604 Isodocarpin

Macrocalin A

Isodocarpin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5604,CAS号为 10391-08-9。
TN3879 Docosyl caffeate

Docosyl caffeate shows moderate antioxidant activity in DPPH and ABTS scavenging assays, it also has significant anti-inflammation activity. Docosyl caffeate exhibits potent elastase inhibitory activity, with the IC50 value of 1.4 microg/mL.
T61296 2-Hydroxydocosanoic acid

2-Hydroxydocosanoic acid exhibits antioxidant, cholinesterase inhibitory, and antimicrobial properties [1].
T12357 Palmitoyldocosahexaenoyl phosphatidylcholine

Others Others
Palmitoyldocosahexaenoyl phosphatidylcholine, an endogenous metabolite.
TN6896 Methyl cis-13-docosenoate

Methyl cis-13-docosenoate is a natural product.
TN2612 13-Hydroxy-8,11,13-podocarpatrien-18-oic acid

Others Others
13-Hydroxy-8,11,13-podocarpatrien-18-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2612,CAS号为 61597-83-9。
TN3828 Dendocarbin A

Others Others
Dendocarbin A是一种天然产物,属于蓼科蓼属,其产品编号为 TN3828,CAS号为 350986-74-2。Dendocarbin A可用作对照参考。
TN3206 7,15-Dihydroxypodocarp-8(14)-en-13-one

Others Others
7,15-Dihydroxypodocarp-8(14)-en-13-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3206,CAS号为 262355-96-4。
T12570 Pseudocoptisine acetate

Isocoptisine acetate,异黄连碱乙酸盐

Others Others
Pseudocoptisine acetate is a quaternary alkaloid isolated from the tubers of Corydalis turtschaninovii,with anti-inflammatory properties.
T36797 1-Alaninechlamydocin

1-Alaninechalmydocin is a fungal metabolite originally isolated from a Great Lakes-derived Tolypocladium sp. and an inhibitor of histone deacetylases (HDACs). It reduces total HDAC activity in HeLa cell lysates in a concentration-dependent manner. 1-Alaninechlamydocin reduces proliferation of MIA PaCa-2, PANC-1, and hTERT-HPNE cells (GI50s = 5.3, 14, and 2.0 nM, respectively).
T80949 Tridocosahexaenoin

Tridocosahexaenoin 是一种具有抗氧化特性的三酰基甘油。
TN2613 13-Methyl-8,11,13-podocarpatriene-3,12-diol

Others Others
13-Methyl-8,11,13-podocarpatriene-3,12-diol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2613,CAS号为 769140-74-1。
T13661 Docosatrienoic Acid

cis-13,16,19-docosatrienoic acid,(13Z,16Z,19Z)-13,16,19-Docosatrienoic acid

Others Others
Docosatrienoic acid is a rare omega-3 fatty acid; Ki value is 5×M, which inhibits the binding of LTB4 to porcine neutrophil membrane.
TN6098 Pseudocolumbamine

Pseudocolumbamine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6098,CAS号为 64191-04-4。
TN2699 2,3-Dihydropodocarpusflavone A

Others Others
2,3-Dihydropodocarpusflavone A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2699,CAS号为 852875-96-8。

天然产物

Deoxycorticosterone acetate
Cat.No: T3033
Synonym: 醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮
Target: Glucocorticoid Receptor, Endogenous Metabolite, Adrenergic Receptor
Docosapentaenoic acid 22n-3
Cat.No: T19295
Synonym:
Target: Endogenous Metabolite
Pseudocoptisine chloride
Cat.No: T9862
Synonym: 盐酸异黄连碱,Isocoptisine chloride
Target: AChE
Podocarpic acid
Cat.No: T12514
Synonym:
Target: Others, TRP/TRPV Channel
Docosanedioic acid 
Cat.No: T9784
Synonym:
Target: PROTAC Linker
Podocarpusflavone A
Cat.No: TQ0134
Synonym:
Target: Topoisomerase
Docosanoic acid
Cat.No: T5942
Synonym: Behenic Acid,山嵛酸
Target: DNA/RNA Synthesis, Endogenous Metabolite
Docosahexaenoic Acid
Cat.No: T5369
Synonym: Cervonic acid,DHA
Target: Others, Endogenous Metabolite
1-Docosanol
Cat.No: T0884
Synonym: Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol
Target: Antifection, HSV
Docosane
Cat.No: TN6962
Synonym:
Target: Others
Docetaxel trihydrate
Cat.No: T0186
Synonym: RP-56976 (Trihydrate),RP56976 (NSC 628503) Trihydrate,多西他赛三水合物
Target: Apoptosis, BCL, Microtubule Associated
Docetaxel
Cat.No: T1034
Synonym: 多西他赛,NSC 628503,RP-56976,多烯紫杉醇
Target: Apoptosis, Microtubule Associated, Endogenous Metabolite
13-Oxopodocarp-8(14)-en-18-oic acid
Cat.No: TN2619
Synonym:
Target: Others
Isodocarpin
Cat.No: TN5604
Synonym: Macrocalin A
Target:
Docosyl caffeate
Cat.No: TN3879
Synonym:
Target:
2-Hydroxydocosanoic acid
Cat.No: T61296
Synonym:
Target:
Palmitoyldocosahexaenoyl phosphatidylcholine
Cat.No: T12357
Synonym:
Target: Others
Methyl cis-13-docosenoate
Cat.No: TN6896
Synonym:
Target:
13-Hydroxy-8,11,13-podocarpatrien-18-oic acid
Cat.No: TN2612
Synonym:
Target: Others
Dendocarbin A
Cat.No: TN3828
Synonym:
Target: Others
7,15-Dihydroxypodocarp-8(14)-en-13-one
Cat.No: TN3206
Synonym:
Target: Others
Pseudocoptisine acetate
Cat.No: T12570
Synonym: Isocoptisine acetate,异黄连碱乙酸盐
Target: Others
1-Alaninechlamydocin
Cat.No: T36797
Synonym:
Target:
Tridocosahexaenoin
Cat.No: T80949
Synonym:
Target:
13-Methyl-8,11,13-podocarpatriene-3,12-diol
Cat.No: TN2613
Synonym:
Target: Others
Docosatrienoic Acid
Cat.No: T13661
Synonym: cis-13,16,19-docosatrienoic acid,(13Z,16Z,19Z)-13,16,19-Docosatrienoic acid
Target: Others
Pseudocolumbamine
Cat.No: TN6098
Synonym:
Target:
2,3-Dihydropodocarpusflavone A
Cat.No: TN2699
Synonym:
Target: Others
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