75
28
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1144L |
Lidocaine Hydrochloride hydrate
|
EGFR; Sodium Channel | Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors |
Lidocaine Hydrochloride hydrate 是一种酰胺类局部麻醉剂,具有抗炎作用。 | |||
T0929 |
Docusate sodium
Aerosol OT,多库脂钠,Dioctyl sulfosuccinate sodium salt,Bis(2-ethylhexyl) sulfosuccinate sodium salt,Constonate |
Opioid Receptor; HSV | Endocrinology/Hormones; GPCR/G Protein; Microbiology/Virology; Neuroscience |
Docusate sodium (Aerosol OT) 是一种口服的非处方泻药和大便软化剂,可用于研究便秘。 | |||
T68079 |
Gedocarnil
ZK 113315,SH 530 |
Others | Others |
Gedocarnil(ZK 113315) 可用于研究中枢神经系统疾病。 | |||
T31716 |
Etidocaine Hydrochloride
W-19053,Duranest,W19053,W 19053 |
Sodium Channel | Membrane transporter/Ion channel |
Etidocaine Hydrochloride (W19053) 是一种长效麻醉剂和电压门控钠通道阻滞剂。 | |||
T10431 |
Golidocitinib
AZD4205 |
JAK | Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells |
Golidocitinib (AZD4205) 是一种选择性 JAK1抑制剂,IC50值为 73 nM。 | |||
T16280 |
Nedocromil
FPL 59002,尼多克罗 |
Leukotriene Receptor; Prostaglandin Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Nedocromil (FPL 59002) 对多种介质的作用或形成有抑制作用,包括组胺,前列腺素 D2和白三烯 C4。 | |||
T8146 |
Imidocarb dipropionate
二丙酸咪唑苯脲,二丙酸双咪苯脲 |
Antibiotic; Parasite | Microbiology/Virology |
Imidocarb dipropionate 是一种抗原虫剂,对寄生虫 B. bovis 的 IC50为 87 μg/mL。 | |||
T16558 |
Polidocanol
Polyoxyethylene lauryl ether,Polyoxyethyleneglycol Dodecyl Ether |
Others | Others |
Polidocanol (Polyoxyethylene lauryl ether) 是月桂醇的烷基聚乙二醇醚,是天然矿物油 中天然脂肪醇或烷基醇的衍生物,是一种硬化剂。Polidocanol 可用做局部麻醉,但与 其他麻醉药物合用时有增强麻醉药物对心血管系统作用的风险。 | |||
T40475 |
Ceftobiprole medocaril
BAL5788,头孢比普酯 |
Antibacterial | Microbiology/Virology |
Ceftobiprole medocaril (BAL5788) 是 Ceftobiprole 的前药。Ceftobiprole 是一种广谱的头孢菌素,对耐甲氧西林金黄色葡萄球菌具有活性。 | |||
T19319 |
Ethyl docosa-4,7,10,13,16,19-hexaenoate
|
Others | Others |
Ethyl cis-4,7,10,13,16,19-Docosahexaenoate, the ethyl ester of Docosahexaenoate (DHA), is selectively enriched in the ethyl ester fraction through the alcoholysis process involving fatty acid ethyl esters from tuna oil and lauryl alcohol. | |||
T14875 |
Indocyanine green
Cardiogreen,IC Green,Foxgreen,吲哚菁绿 |
Others | Others |
Indocyanine green (Cardiogreen) 是低毒性荧光剂,普遍用于医学诊断,包括确定心输出量,肝功能和肝血流量,以及用于眼科血管造影。 | |||
T0468 |
Lidocaine
Lignocaine,Alphacaine,Xylocaine,利多卡因 |
Apoptosis; ERK; NF-κB; MEK; Sodium Channel; Histamine Receptor | Apoptosis; GPCR/G Protein; Immunology/Inflammation; MAPK; Membrane transporter/Ion channel; Neuroscience; NF-κB |
Lidocaine (Alphacaine) 是一种酰胺衍生物,抑制涉及复杂电压和依赖性的钠通道,可用于研究室性心律失常。它通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。 | |||
T14060 |
6-Maleimidocapronic acid
|
PROTAC Linker | PROTAC |
6-Maleimidocapronic acid 是一种属于 alkyl chain 类的 PROTAC linker,可用于 PROTAC 分子的合成。 | |||
T19294 |
Docosahexaenoic Acid methyl ester
二十二六烯酸甲酯,Methyl docosahexaenoate,all cis-DHA methyl ester |
Others | Others |
Docosahexaenoic Acid methyl ester (all cis-DHA methyl ester) 是甲基化的二十二碳六烯酸类似物,能够插入膜磷脂中而不被氧化或水解。 | |||
T31716L |
Etidocaine
|
Others | Others |
Etidocaine 是一种氨基酸酰胺,用作局部麻醉剂,具有快速起效和长效特性。 | |||
T1144 |
Lidocaine hydrochloride
Lidocaine HCL,盐酸利多卡因,Lignocaine hydrochloride,Xyloneural,Lidothesin |
Apoptosis; ERK; NF-κB; MEK; Sodium Channel | Apoptosis; MAPK; Membrane transporter/Ion channel; NF-κB |
Lidocaine hydrochloride (Lignocaine hydrochloride) 抑制涉及复杂电压和依赖性的钠通道。它通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。Lidocaine 是一种酰胺衍生物,是一种研究室性心律失常的药物和有效的肿瘤抑制剂。 | |||
T35009 |
Vadocaine
Vadocaina,Vadocainum |
Others | Others |
Vadocaine (Vadocaina) 是一种新型的镇咳化合物,可用于局部麻醉,可用于研究中枢神经系统和心血管系统。 | |||
T124800 | Endocrocin | ||
Endocrocin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124800,CAS号为 481-70-9。 | |||
T30271 |
Azidocillin sodium salt
Nalpen,Globacillin,Longatren |
||
Azidocillin sodium salt is a type of penicillin. | |||
TQ0247 |
7-Epi-docetaxel
7-Epidocetaxel,7-表多西他赛,4-epi-Docetaxel,7-Epitaxotere |
Others | Others |
7-Epi-10-oxo-docetaxel (7-Epitaxotere) is a impurity of docetaxel. | |||
T77174 | Efmarodocokin alfa | ||
Efmarodocokin alfa为人IL-22与IgG4可结晶片段的融合蛋白,具有激活IL-22信号的功能。该化学物质主要用于重症COVID-19肺炎的研究。 | |||
T77173 | Eflepedocokin alfa | ||
Eflepedocokin alfa 是一种具有潜在细胞保护活性的重组融合蛋白。Eflepedocokin alfa 由人的IL-22与人的IgG2-Fc 结构域融合组成。Eflepedocokin alfa 可激活IL-22/IL-22R 介导的信号转导通路以及STAT3。Eflepedocokin alfa 在免疫反应和细菌感染、增强肠道屏障功能、肠道免疫和组织修复方面发挥作用。 | |||
T37532 |
Docosahexaenoyl Glycine
|
||
The ω-3 polyunsaturated fatty acids (PUFAs) found in fish oils provide cardiovascular benefits. Docosahexaenoic acid (DHA), a C22:6 PUFA, is the most abundant ω-3 fatty acid in neural tissues, especially in the retina and brain. It can be synthesized from other dietary ω-3 PUFAs or taken as a nutritional supplement. Docosahexaenoyl glycine consists of DHA with glycine attached at its carboxy terminus. | |||
T77230 |
1-O-Hexadecyl-2-O-docosahexaenoyl-sn-glycero-3-phosphorylcholine
|
||
1-O-Hexadecyl-2-O-docosahexaenoyl-sn-glycero-3-phosphorylcholine为存在于尿中的内源性代谢物,用于肥胖研究。 | |||
T19520 |
Piridocaine hydrochloride
Lucaine hydrochloride |
Others | Others |
Piridocaine hydrochloride is a piperidyl propanol ester of orthoaminobenzoic acid. | |||
T73194 |
DOCK2-IN-1
|
||
DOCK2-IN-1 是 CPYPP 类似物,也是DOCK2的抑制剂 (IC50=19.1 μM)。DOCK2-IN-1 以可逆方式结合DOCK2DHR-2 结构域以抑制其催化活性。DOCK2-IN-1 阻断淋巴细胞中趋化因子受体和抗原受体介导的 Rac 的激活。DOCK2-IN-1 显着抑制趋化反应和 T 细胞活化。 | |||
TD0084 |
DiI triflate [1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine triflate]
|
||
DiI triflate is one of lipophilic fluorescent stains for labeling membranes and other hydrophobic structures. The fluorescence of these environment-sensitive dyes is greatly enhanced when incorporated into membranes or bound to lipophilic biomolecules such as proteins although they are weakly fluorescent in water. | |||
TQ0142 |
10-Oxo Docetaxel
Docetaxel Impurity 1,10-氧多西他赛 |
Others | Others |
10-Oxo Docetaxel is a Docetaxel intermediate having remarkable antitumor properties. | |||
T62520 | Imidocarb dihydrochloride monohydrate | ||
Imidocarb dihydrochloride monohydrate 是一种有效的抗原虫剂,能够作用于寄生虫 B. bovis (IC50: 87 μg/ml)。 | |||
T25720 |
Lidocaine methiodide
Methyllidocaine iodide,N-Methyllidocaine |
||
Lidocaine methiodide is an antiarrythmic. It is also exhibiting arrythmogenic effects in subjects. | |||
T72141 |
Ceftobiprole medocaril sodium
头孢比普酯钠盐,BAL5788 sodium |
||
Ceftobiprole medocaril (BAL5788) sodium 是 Ceftobiprole 的胃肠外前药。Ceftobiprole 是一种非肠道吡咯烷酮头孢菌素。Ceftobiprole 是一种广谱头孢菌素,对甲氧西林 (MRSA) 和耐万古霉素葡萄球菌 (VRSA) 和耐青霉素链球菌具有高水平的体外活性。Ceftobiprole 也抑制革兰氏阳性和革兰氏阴性病原体。 | |||
T37634 |
17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic Acid
|
||
Docosapentaenoic acid (DPA) is a ω-3 fatty acid found in fish oils. 17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-docosapentaenoic acid is a metabolite of lipoxygenase-mediated oxidation of DPA that is produced endogenously by aspirin-enhanced COX-2 activity. It has been shown to activate Nrf2-dependent antioxidant gene expression, to act as a PPARγ agonist (EC50 = ~200 nM), and to inhibit pro-inflammatory cytokine and nitric oxide production at biological concentration ranges (5-25 μM). | |||
T38527 |
2',3'-Dideoxy-5-iodocytidine
|
||
2',3'-Dideoxy-5-iodocytidine, a chemical compound, is employed in gene sequencing and functions as an antibiotic. It exhibits significant efficacy specifically against Mycobacterium. | |||
T19163 |
7-Epi-10-oxo-docetaxel
Docetaxel Impurity 2 |
Others | Others |
7-Epi-10-oxo-docetaxel (Docetaxel Impurity 2) is an impurity of docetaxel detected by HPLC. | |||
T36868 |
4-oxo Docosahexaenoic Acid
|
||
4-oxo Docosahexaenoic acid (4-oxo DHA) is a putative metabolite of DHA with antiproliferative and PPARγ agonist activity. It inhibits the growth of several triple negative breast cancer cell lines (MCF-10F, trMCF, bsMCF, MDA-MB-231, and BT549) at 50-100 μM, however it increased proliferation of MCF-7 cells. 4-oxo DHA binds covalently to PPARγ and activates gene transcription in luciferase reporter assays and in dendritic cells with EC50 values of approximately 8-16 μM. | |||
T29981 |
Amidochlor
Caswell No. 005B,EPA Pesticide Chemical Code 128001,MON 4620,MON 4621,Limit |
||
Amidochlor is a growth regulator. | |||
TNU0763 |
2’-Deoxy-2’-fluoro-N3-(n-docecyl)uridine
|
||
2'-Deoxy-2'-fluoro-N3-(n-docecyl)uridine is a Nucleoside Derivative - Fluoro-modified nucleoside, 2'-Modified nucleoside. | |||
TD0083 |
DiIiodide1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine iodide]
DiI碘化物 |
||
DiI iodide1 is one of lipophilic fluorescent stains for labeling membranes and other hydrophobic structures. The fluorescence of these environment-sensitive dyes is greatly enhanced when incorporated into membranes or bound to lipophilic biomolecules such as proteins although they are weakly fluorescent in water. | |||
T34382 |
Rodocaine
R-19317,R 19317,R19317 |
||
Rodocaine is a biochemical. | |||
T16694 |
Pyridoclax
MR-29072 |
BCL | Apoptosis |
Pyridoclax is an inhibitor of potential Mcl-1. | |||
T24171 |
Iodoclorgyline
6-Iodoclorgyline |
||
Iodoclorgyline is an inhibitor of monoamine oxidase A. | |||
T77161 | Docaravimab | ||
Docaravimab为针对ERA (Evelyn-Rockitniki-Abelseth) 糖蛋白胞外域表位G-III的抗体,适用于狂犬病研究。 | |||
T38644 |
Docetaxal
PNU-101383,10-Acetyl docetaxel |
||
Docetaxal, also known as 10-Acetyl docetaxel, is an analog of Docetaxel exhibiting potent anticancer properties. It acts as a microtubule disassembly inhibitor, effectively inhibiting mitosis. | |||
T71805 |
DOCK5-IN-C21
|
||
DOCK5-IN-C21 is an allosteric inhibitor of the guanine nucleotide exchange factor DOCK5. | |||
T37633 |
17-oxo-4(Z),7(Z),10(Z),13(Z),15(E),19(Z)-Docosahexaenoic Acid
|
||
17-oxo-4(Z),7(Z),10(Z),13(Z),15(E),19(Z)-Docosahexaenoic acid is a metabolite of lipoxygenase-mediated oxidation of DHA that is produced endogenously by aspirin-enhanced COX-2 activity. It has been shown to activate Nrf2-dependent antioxidant gene expression, to act as a PPARγ agonist (EC50 = ~200 nM), and to inhibit pro-inflammatory cytokine and nitric oxide production at biological concentration ranges (5-25 μM). | |||
T64415 |
22-(tert-Butoxy)-22-oxodocosanoic acid
|
||
22-(tert-Butoxy)-22-oxodocosanoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64415,CAS号为 1642333-05-8。 | |||
TNU0629 |
5-Iodocytosine
|
||
5-Iodocytosine is a Heterocyclic compound-pyrimidine, intermediate and building block, halo-. | |||
T25308 | Deoxymulundocandin | ||
Deoxymulundocandin is an echinocandin type antifungal antibiotic from Aspergillus sydowii. | |||
T14059 | 6-Maleimidocaproic acid-PFP ester | Others | Others |
6-Maleimidocaproic acid-PFP ester is a hydrocarbon-based PROTAC linker, suitable for the synthesis of PROTACs[1]. | |||
T15155 |
Docebenone
AA 861 |
Others | Others |
Docebenone is a selective and orally active inhibitor of 5-LO. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3033 |
Deoxycorticosterone acetate
醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮 |
Glucocorticoid Receptor; Endogenous Metabolite; Adrenergic Receptor | Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience |
Deoxycorticosterone acetate (Cortexone acetate) 是肾上腺产生的类固醇激素,具有盐皮质激素活性,并作为醛固酮的前体。 | |||
T19295 |
Docosapentaenoic acid 22n-3
|
Endogenous Metabolite | Metabolism |
Docosapentaenoic acid 22n-3 是在所有动物细胞膜中发现的磷脂组成成分。 | |||
T9862 |
Pseudocoptisine chloride
盐酸异黄连碱,Isocoptisine chloride |
AChE | Neuroscience |
Pseudocoptisine chloride (Isocoptisine chloride) 是从 Corydalis Tuber 中分离出来的,具有抗炎和抗健忘的作用。 Pseudocoptisine chloride 抑制乙酰胆碱酯酶 (AChE) 活性 (IC50 = 12.8 μM)。 | |||
T12514 |
Podocarpic acid
|
Others; TRP/TRPV Channel | Membrane transporter/Ion channel; Others |
Podocarpic acid 是一种天然产物,是一种新型 TRPA1 激活剂。 | |||
T9784 |
Docosanedioic acid
|
PROTAC Linker | PROTAC |
Docosanedioic acid 可以作为ADC linker 或PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。 | |||
TQ0134 |
Podocarpusflavone A
|
Topoisomerase | DNA Damage/DNA Repair |
Podocarpusflavone A is a DNA topoisomerase I inhibitor. It has moderated anti-proliferative activity induce cell apoptosis in MCF-7. | |||
T5942 |
Docosanoic acid
Behenic Acid,山嵛酸 |
DNA/RNA Synthesis; Endogenous Metabolite | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
Docosanoic acid (Behenic Acid) 是一种较难吸收的饱和脂肪酸,能提高人类胆固醇水平。 | |||
T5369 |
Docosahexaenoic Acid
Cervonic acid,DHA |
Others; Endogenous Metabolite | Metabolism; Others |
Docosahexaenoic Acid 是一种ω-3脂肪酸,在脑和视网膜中较为丰富,且能够直接从鱼油和母乳中获得。 | |||
T0884 |
1-Docosanol
Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol |
Antifection; HSV | Microbiology/Virology |
1-Docosanol (Behenic alcohol) 是一种具有抗病毒活性的饱和 22 碳脂肪醇,局部用于治疗复发性单纯性唇疱疹发作并缓解相关疼痛并可能有助于更快地治愈疮。 | |||
TN6962 |
Docosane
|
Others | Others |
Docosane 是一种直链烷烃,可用于合成具有热能储存/释放能力的结构复合材料。 | |||
T0186 |
Docetaxel trihydrate
RP-56976 (Trihydrate),RP56976 (NSC 628503) Trihydrate,多西他赛三水合物 |
Apoptosis; BCL; Microtubule Associated | Apoptosis; Cytoskeletal Signaling |
Docetaxel trihydrate (RP-56976 Trihydrate) 是一种抗肿瘤试剂,抑制微管解聚的IC50值为 0.2 μM。它是紫杉醇的半合成类似物,能减弱 bcl-2 和 bcl-xL 基因表达的影响。它阻滞G2/M 细胞周期,导致细胞凋亡。 | |||
T1034 |
Docetaxel
多西他赛,NSC 628503,RP-56976,多烯紫杉醇 |
Apoptosis; Microtubule Associated; Endogenous Metabolite | Apoptosis; Cytoskeletal Signaling; Metabolism |
Docetaxel (RP-56976) 是紫杉醇的半合成类似物,是一种微管解聚抑制剂 (IC50=0.2 μM)。Docetaxel 可以减弱 bcl-2 和 bcl-xL 基因表达的影响,具有诱导凋亡、抗肿瘤活性。 | |||
TN2619 |
13-Oxopodocarp-8(14)-en-18-oic acid
|
Others | Others |
13-Oxopodocarp-8(14)-en-18-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2619,CAS号为 63976-69-2。 | |||
TN5604 |
Isodocarpin
Macrocalin A |
||
Isodocarpin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5604,CAS号为 10391-08-9。 | |||
TN3879 | Docosyl caffeate | ||
Docosyl caffeate shows moderate antioxidant activity in DPPH and ABTS scavenging assays, it also has significant anti-inflammation activity. Docosyl caffeate exhibits potent elastase inhibitory activity, with the IC50 value of 1.4 microg/mL. | |||
T61296 |
2-Hydroxydocosanoic acid
|
||
2-Hydroxydocosanoic acid exhibits antioxidant, cholinesterase inhibitory, and antimicrobial properties [1]. | |||
T12357 |
Palmitoyldocosahexaenoyl phosphatidylcholine
|
Others | Others |
Palmitoyldocosahexaenoyl phosphatidylcholine, an endogenous metabolite. | |||
TN6896 |
Methyl cis-13-docosenoate
|
||
Methyl cis-13-docosenoate is a natural product. | |||
TN2612 |
13-Hydroxy-8,11,13-podocarpatrien-18-oic acid
|
Others | Others |
13-Hydroxy-8,11,13-podocarpatrien-18-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2612,CAS号为 61597-83-9。 | |||
TN3828 |
Dendocarbin A
|
Others | Others |
Dendocarbin A是一种天然产物,属于蓼科蓼属,其产品编号为 TN3828,CAS号为 350986-74-2。Dendocarbin A可用作对照参考。 | |||
TN3206 | 7,15-Dihydroxypodocarp-8(14)-en-13-one | Others | Others |
7,15-Dihydroxypodocarp-8(14)-en-13-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3206,CAS号为 262355-96-4。 | |||
T12570 |
Pseudocoptisine acetate
Isocoptisine acetate,异黄连碱乙酸盐 |
Others | Others |
Pseudocoptisine acetate is a quaternary alkaloid isolated from the tubers of Corydalis turtschaninovii,with anti-inflammatory properties. | |||
T36797 | 1-Alaninechlamydocin | ||
1-Alaninechalmydocin is a fungal metabolite originally isolated from a Great Lakes-derived Tolypocladium sp. and an inhibitor of histone deacetylases (HDACs). It reduces total HDAC activity in HeLa cell lysates in a concentration-dependent manner. 1-Alaninechlamydocin reduces proliferation of MIA PaCa-2, PANC-1, and hTERT-HPNE cells (GI50s = 5.3, 14, and 2.0 nM, respectively). | |||
T80949 |
Tridocosahexaenoin
|
||
Tridocosahexaenoin 是一种具有抗氧化特性的三酰基甘油。 | |||
TN2613 |
13-Methyl-8,11,13-podocarpatriene-3,12-diol
|
Others | Others |
13-Methyl-8,11,13-podocarpatriene-3,12-diol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2613,CAS号为 769140-74-1。 | |||
T13661 |
Docosatrienoic Acid
cis-13,16,19-docosatrienoic acid,(13Z,16Z,19Z)-13,16,19-Docosatrienoic acid |
Others | Others |
Docosatrienoic acid is a rare omega-3 fatty acid; Ki value is 5×M, which inhibits the binding of LTB4 to porcine neutrophil membrane. | |||
TN6098 |
Pseudocolumbamine
|
||
Pseudocolumbamine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6098,CAS号为 64191-04-4。 | |||
TN2699 |
2,3-Dihydropodocarpusflavone A
|
Others | Others |
2,3-Dihydropodocarpusflavone A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2699,CAS号为 852875-96-8。 |