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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T10789 Chitosan oligosaccharide

COS,壳聚糖低聚乳酸酯

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Chitosan oligosaccharide (COS) 是 β-(1→4)-连接的 D-氨基葡萄糖的寡聚体,Chitosan oligosaccharide可激活 AMPK ,抑制NF-κB 和 MAPK在内的炎症信号通路。
T30155 Ascorbyl nicotinate

COS-CB3

Ascorbyl nicotinate is a bioactive chemical.
T10979 DCPIB

Potassium Channel; Chloride channel Membrane transporter/Ion channel
DCPIB 是选择性可逆体积调节性阴离子通道抑制剂,抑制肿胀激活氯电流,在 CPAE 细胞中,IC50值为 4.1 μM。它能够电压依赖性激活钾离子通道 TREK1 和 TRAAK,抑制 TRESK、TASK1 和 TASK3的 IC50值分别为 0.14、0.95 和 50.72 μM。
T8851 I3MT-3

HMPSNE

Hippo pathway Stem Cells
I3MT-3 (HMPSNE) 是一种有效的、具有细胞膜渗透性的、选择性的 3-巯基丙酮酸硫转移酶 (3MST)的抑制剂,IC50值为2.7 μM,对其他硫化氢/磺胺制硫酶没有活性。它靶向位于 3MST 活性位点的过硫半胱氨酸残基。
T16420 P-1075

Potassium Channel Membrane transporter/Ion channel
P-1075 是磺酰脲受体2相关的 ATP 敏感性的钾通道(SUR2-KIR6)的激活剂,EC50为 45 nM。它在兔子中通过打开线粒体 K (ATP) 通道产生活性氧,产生保护心脏的功效。
TP1889 MCL0020

MCL 0020

Melanocortin Receptor GPCR/G Protein; Neuroscience
MCL0020 是一种有效的选择性黑素皮质素MC4受体拮抗剂,IC50为 11.63 nM。它剂量依赖性减轻束缚应激诱发的厌食症,在体内表现出抗焦虑样活性。
T19840 GSK-F1

PI4KA inhibitor-F1

PI4K PI3K/Akt/mTOR signaling
GSK-F1 (PI4KA inhibitor-F1) 是一种新型强效 PI4KA 抑制剂。
T35664 Tetracosactide acetate

Others Others
Tetracosactide acetate 是一种合成的多肽,可刺激肾上腺释放皮质类固醇 ,如皮质醇。Tetracosactide acetate 在溃疡性结肠炎和克罗恩病、青少年和成人类风湿性关节炎和骨关节病方面有研究的价值。
T8915 Glycylsarcosine

GLYCYL-SARCOSINE,甘氨酰肌氨酸

Others Others
Glycylsarcosine (GLYCYL-SARCOSINE) 是由甘氨酸的羧基与肌氨酸的氨基缩合而成的二肽
T19294 Docosahexaenoic Acid methyl ester

二十二六烯酸甲酯,Methyl docosahexaenoate,all cis-DHA methyl ester

Others Others
Docosahexaenoic Acid methyl ester (all cis-DHA methyl ester) 是甲基化的二十二碳六烯酸类似物,能够插入膜磷脂中而不被氧化或水解。
T61037 Glycosyltransferase-IN-1

Others Others
Glycosyltransferase-IN-1 是一种糖基转移酶 (glycosyltransferase) 抑制剂,具有抑菌活性,抑制 MSSA、MRSA 、枯草杆菌和肠杆菌。
T19232 CMC-Na (Viscosity:800-1200 mPa.s)

羧甲基纤维素钠,CMC-Na (Viscosity:800-1200 mPa.s)

Others Others
Sodium carboxymethyl cellulose (CMC-Na) (Viscosity:800-1200 mPa.s) 是一种水溶性纤维素,常用作动物实验的助溶剂,对动物基本没有毒性。
T7184 Firsocostat

ND-630,NDI-010976,GS-0976

Acetyl-CoA Carboxylase Metabolism
Firsocostat (GS-0976) 是有效的乙酰辅酶A 羧化酶 (ACC) 抑制剂,抑制人类 ACC1 和 ACC2 的IC50分别为2.1和6.1 nM。
T3286 Sodium picosulfate monohydrate

Sodium picosulfate hydrate,匹可硫酸钠一水合物,Laxoberal

Others Others
Sodium picosulfate monohydrate (Sodium picosulfate hydrate) 增加水和电解质的分泌并抑制它们的吸收。
T124663 Sericoside

Immunology/Inflammation related Immunology/Inflammation
Sericoside,一种从Terminalia提取的三萜类化合物,具备显著的抗炎特性。此外,sericoside展现出强效的解脂活性,有助于减少皮肤皱纹及改善肤质。
T19712 Levoglucosenone

Others Others
Levoglucosenone 具有细胞毒性。它对抗人肝癌细胞系。
T38089 2F-Peracetyl-Fucose

1,3,4-Tri-O-acetyl-2-deoxy-2-fluoro-L-fucopyranos

Others Others
2F-Peracetyl-Fucose (1,3,4-Tri-O-acetyl-2-deoxy-2-fluoro-L-fucopyranos) 是一种有效的岩藻糖基转移酶 (FUT)抑制剂,在体外炎症模型中抑制唾液酸化和岩藻糖基化。
T15549 Icosabutate

Others Others
Icosabutate is a structurally engineered and orally active ω-3 polyunsaturated fatty acid. Icosabutate is well tolerated, and efficacious in lowering non-high-density lipoprotein cholesterol (non-HDL-C) levels in persistent hypertriglyceridemia.
T67898 α-Glucosidase-IN-22

Glucosidase Metabolism
α-Glucosidase-IN-22是一种α-葡萄糖苷酶选择性抑制剂(IC50=0.64 μM)。α-Glucosidase-IN-22有抗糖尿病的活性,在2型糖尿病(T2DM)研究中具有潜力。
T69467 Azacosterol

IMD760,Diazasterol

Others Others
Azacosterol (Diazasterol) 是一种DHCR24抑制剂。Azacosterol 口服或腹腔注射后会在皮质神经元中发生一系列反应。
T6675 Sodium Picosulfate

Evacuol,Picolax,匹克硫酸钠,Sodium Picosulphate,匹可硫酸钠,Laxoberal

Others Others
Sodium Picosulfate (Laxoberal) 可以抑制水和电解质的吸收,促进它们的分泌。
TP1031 Tetracosactide

Tetracosactrin,替可克肽

Others Others
Tetracosactide (Tetracosactrin) 是一种肾上腺皮质激素 (ACTH) 的类似物,能够刺激肾上腺皮质激素分泌。
T60715 α-Glucosidase-IN-4

Glucosidase Metabolism
α-Glucosidase-IN-4 是一种有效的α- 葡萄糖苷酶 (α-glucosidase)抑制剂,具有降血压和降糖活性。
T19261 D-Glucose-13C6

D-(+)-Glucose-13C6,Glucose-13C6,Dextrose-13C6

Endogenous Metabolite Metabolism
D-Glucose-13C6 (Dextrose-13C6) 是一种 D-Glucose 的同位素标记物,可作为代谢示踪剂,可用于研究机体代谢相关疾病和部分物质的代谢过程。
T9785 20-(tert-Butoxy)-20-oxoicosanoic acid

PROTAC Linker PROTAC
20-(tert-Butoxy)-20-oxoicosanoic acid 可以作为 ADC linker 或 PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。
T19319 Ethyl docosa-4,7,10,13,16,19-hexaenoate

Others Others
Ethyl cis-4,7,10,13,16,19-Docosahexaenoate, the ethyl ester of Docosahexaenoate (DHA), is selectively enriched in the ethyl ester fraction through the alcoholysis process involving fatty acid ethyl esters from tuna oil and lauryl alcohol.
T4181 Cosan 528

Others Others
Cosan 528 是一种生物活性化学品。
T76148 Glucose oxidase

Endogenous Metabolite Metabolism
Glucose oxidase 是从真菌黑曲霉中提取的酶,是食品工业中一种重要的工业用酶, 广泛用于葡萄酒、啤酒、果汁、奶粉等食品脱氧、面粉改良、防止食品褐变等方面。Glucose oxidase 具有抗氧化和潜在的抗癌活性。
T10035 10,12-Tricosadiynoic acid

TDA,TCDA

Acyltransferase Metabolism
10,12-Tricosadiynoic acid 是一种口服有效的酰基辅酶 A 氧化酶-1 (ACOX1) 抑制剂,具有高特异性,选择性,高亲和力的特点。10,12-Tricosadiynoic acid 可改善线粒体脂质和 ROS 代谢,在高脂饮食或肥胖引起的代谢性疾病中有研究的价值。
T74041 GDP-L-fucose

Endogenous Metabolite Metabolism
GDP-L-fucose 是一种广泛存在与真菌和植物中的核苷酸糖,参与从头代谢途径和次要的补救代谢途径。
T23910 Cosalane

NSC 658586,NSC-658586,NSC 640067

HIV Protease Microbiology/Virology; Proteases/Proteasome
Cosalane (NSC 658586) 是一种 HIV 复制抑制剂,是人和小鼠趋化因子受体 7 (CCR7)信号传导的抑制剂,具有抗病毒活性,可阻断 CCR7 与其天然配体 CCL19 和 CCL21 结合。Cosalane 对多种 HIV-1 株系和 HIV-2 具有活性。
T8823 Locostatin

Raf MAPK
Locostatin 是一种有效的细胞渗透性 Raf 激酶抑制剂蛋白 (RKIP)/Raf1 激酶相互作用抑制剂和细胞迁移抑制剂。
T67728 α-Glucosidase-IN-23

Glucosidase Metabolism
α-Glucosidase-IN-23 是具有口服活性的 α-Glucosidase 抑制剂。α-Glucosidase-IN-23 通过抑制 a-glucosidase 降低血糖 (IC50= 4.48 μM)。α-Glucosidase-IN-23 可用于糖尿病的研究。
T4355 Fuscoside

OPC 21268

Vasopressin Receptor GPCR/G Protein
Fuscoside (OPC 21268) 是一种非肽精氨酸加压素(AVP) 受体 V 拮抗剂,IC50值为0.4 μM。
T3510 Olumacostat Glasaretil

Acetyl-CoA Carboxylase Metabolism
Olumacostat glasaretil 是乙酰辅酶A 羧化酶的有效抑制剂。
T0777 Tilmicosin

LY-177370,替米考星,EL-870

Antibacterial; Antibiotic Microbiology/Virology
Tilmicosin (EL-870) 是一种抗生素,可研究曼氏杆菌和巴氏杆菌相关的牛羊呼吸系统疾病。
T19859 Nicosulfuron

Milagro,Accent,Motivell,烟嘧磺隆

Others Others
Nicosulfuron (Milagro) 是一种磺酰脲类的选择性除草剂,常用作出苗后的除草剂,保护玉米作物免受杂草的侵害。它也能够降低乙酰乳酸合酶的活性。
T20503 Elfacos EHP

2-ethylhexyl palmitate,棕榈酸辛酯

Others Others
Elfacos EHP (2-ethylhexyl palmitate) 是一种衍生自 2-乙基己醇和棕榈酸的脂肪酸酯,可用作化妆品配方。
T22439 Tilmicosin phosphate

磷酸替米考星,替米考星磷酸盐

Antibacterial; Antibiotic Microbiology/Virology
Tilmicosin phosphate 是一种抗生素,可研究曼氏杆菌和巴氏杆菌相关的牛羊呼吸系统疾病。
T27828 Licostinel

CGP 63446,ACEA1021,ACEA 1021,ACEA-1021,CGP-63446

GluR Neuroscience
Licostinel (CGP 63446) 是一种谷氨酸受体拮抗剂。 Licostinel 可防止永久性局灶性脑缺血。
T125751 Eriodictyol-8-glucoside

Eriodictyol-8-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125751。
T130743 6-Glucosyl-3,4',5,7-tetrahydroxyflavanone

6-Glucosyl-3,4',5,7-tetrahydroxyflavanone 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T130743。
T14452 Azido-PEG4-tetra-Ac-beta-D-glucose

Others Others
Azido-PEG4-tetra-Ac-beta-D-glucose is a polyethylene glycol (PEG) based PROTAC linker utilized for the synthesis of PROTACs[1].
T21121 Henicosafluoro-10-iododecane

Perfluorodecyl iodide,1-Iodoperfluorodecane,Henicosafluorodecyl Iodide,Perfluoro-1-iododecane,Decane, heneicosafluoro-1-iodo-

Henicosafluoro-10-iododecane is a biochemical.
T124963 Phloretin 3',5'-Di-C-glucoside

Phloretin 3',5'-Di-C-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124963。
T126275 Prenyl glucoside

Prenyl glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126275,CAS号为 117861-55-9。
T63361 α-Glucosidase-IN-13

α-Glucosidase-IN-13 是 α-glucosidase 抑制剂 (IC50: 5.69 μM)。
T75420 alpha-1,3/4-Fucosyltransferase (α1,3/4FucT)

alpha-1,3/4-Fucosyltransferase (α1,3/4FucT) (Hp3/4FT) 存在于幽门螺杆菌中。alpha-1,3/4-Fucosyltransferase (α1,3/4FucT) 催化岩藻糖从供体 GDP-β-l-岩藻糖转移到 GlcNAc。
T125936 Sibiricose A3

Sibiricose A3 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125936,CAS号为 139726-39-9。
T124583 26-Desglucoavenacoside A

26-Desglucoavenacoside A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124583,CAS号为 59795-21-0。

化合物

Chitosan oligosaccharide
Cat.No: T10789
Synonym: COS,壳聚糖低聚乳酸酯
Target: AMPK
Ascorbyl nicotinate
Cat.No: T30155
Synonym: COS-CB3
Target:
DCPIB
Cat.No: T10979
Synonym:
Target: Potassium Channel, Chloride channel
I3MT-3
Cat.No: T8851
Synonym: HMPSNE
Target: Hippo pathway
P-1075
Cat.No: T16420
Synonym:
Target: Potassium Channel
MCL0020
Cat.No: TP1889
Synonym: MCL 0020
Target: Melanocortin Receptor
GSK-F1
Cat.No: T19840
Synonym: PI4KA inhibitor-F1
Target: PI4K
Tetracosactide acetate
Cat.No: T35664
Synonym:
Target: Others
Glycylsarcosine
Cat.No: T8915
Synonym: GLYCYL-SARCOSINE,甘氨酰肌氨酸
Target: Others
Docosahexaenoic Acid methyl ester
Cat.No: T19294
Synonym: 二十二六烯酸甲酯,Methyl docosahexaenoate,all cis-DHA methyl ester
Target: Others
Glycosyltransferase-IN-1
Cat.No: T61037
Synonym:
Target: Others
CMC-Na (Viscosity:800-1200 mPa.s)
Cat.No: T19232
Synonym: 羧甲基纤维素钠,CMC-Na (Viscosity:800-1200 mPa.s)
Target: Others
Firsocostat
Cat.No: T7184
Synonym: ND-630,NDI-010976,GS-0976
Target: Acetyl-CoA Carboxylase
Sodium picosulfate monohydrate
Cat.No: T3286
Synonym: Sodium picosulfate hydrate,匹可硫酸钠一水合物,Laxoberal
Target: Others
Sericoside
Cat.No: T124663
Synonym:
Target: Immunology/Inflammation related
Levoglucosenone
Cat.No: T19712
Synonym:
Target: Others
2F-Peracetyl-Fucose
Cat.No: T38089
Synonym: 1,3,4-Tri-O-acetyl-2-deoxy-2-fluoro-L-fucopyranos
Target: Others
Icosabutate
Cat.No: T15549
Synonym:
Target: Others
α-Glucosidase-IN-22
Cat.No: T67898
Synonym:
Target: Glucosidase
Azacosterol
Cat.No: T69467
Synonym: IMD760,Diazasterol
Target: Others
Sodium Picosulfate
Cat.No: T6675
Synonym: Evacuol,Picolax,匹克硫酸钠,Sodium Picosulphate,匹可硫酸钠,Laxoberal
Target: Others
Tetracosactide
Cat.No: TP1031
Synonym: Tetracosactrin,替可克肽
Target: Others
α-Glucosidase-IN-4
Cat.No: T60715
Synonym:
Target: Glucosidase
D-Glucose-13C6
Cat.No: T19261
Synonym: D-(+)-Glucose-13C6,Glucose-13C6,Dextrose-13C6
Target: Endogenous Metabolite
20-(tert-Butoxy)-20-oxoicosanoic acid
Cat.No: T9785
Synonym:
Target: PROTAC Linker
Ethyl docosa-4,7,10,13,16,19-hexaenoate
Cat.No: T19319
Synonym:
Target: Others
Cosan 528
Cat.No: T4181
Synonym:
Target: Others
Glucose oxidase
Cat.No: T76148
Synonym:
Target: Endogenous Metabolite
10,12-Tricosadiynoic acid
Cat.No: T10035
Synonym: TDA,TCDA
Target: Acyltransferase
GDP-L-fucose
Cat.No: T74041
Synonym:
Target: Endogenous Metabolite
Cosalane
Cat.No: T23910
Synonym: NSC 658586,NSC-658586,NSC 640067
Target: HIV Protease
Locostatin
Cat.No: T8823
Synonym:
Target: Raf
α-Glucosidase-IN-23
Cat.No: T67728
Synonym:
Target: Glucosidase
Fuscoside
Cat.No: T4355
Synonym: OPC 21268
Target: Vasopressin Receptor
Olumacostat Glasaretil
Cat.No: T3510
Synonym:
Target: Acetyl-CoA Carboxylase
Tilmicosin
Cat.No: T0777
Synonym: LY-177370,替米考星,EL-870
Target: Antibacterial, Antibiotic
Nicosulfuron
Cat.No: T19859
Synonym: Milagro,Accent,Motivell,烟嘧磺隆
Target: Others
Elfacos EHP
Cat.No: T20503
Synonym: 2-ethylhexyl palmitate,棕榈酸辛酯
Target: Others
Tilmicosin phosphate
Cat.No: T22439
Synonym: 磷酸替米考星,替米考星磷酸盐
Target: Antibacterial, Antibiotic
Licostinel
Cat.No: T27828
Synonym: CGP 63446,ACEA1021,ACEA 1021,ACEA-1021,CGP-63446
Target: GluR
Eriodictyol-8-glucoside
Cat.No: T125751
Synonym:
Target:
6-Glucosyl-3,4',5,7-tetrahydroxyflavanone
Cat.No: T130743
Synonym:
Target:
Azido-PEG4-tetra-Ac-beta-D-glucose
Cat.No: T14452
Synonym:
Target: Others
Henicosafluoro-10-iododecane
Cat.No: T21121
Synonym: Perfluorodecyl iodide,1-Iodoperfluorodecane,Henicosafluorodecyl Iodide,Perfluoro-1-iododecane,Decane, heneicosafluoro-1-iodo-
Target:
Phloretin 3',5'-Di-C-glucoside
Cat.No: T124963
Synonym:
Target:
Prenyl glucoside
Cat.No: T126275
Synonym:
Target:
α-Glucosidase-IN-13
Cat.No: T63361
Synonym:
Target:
alpha-1,3/4-Fucosyltransferase (α1,3/4FucT)
Cat.No: T75420
Synonym:
Target:
Sibiricose A3
Cat.No: T125936
Synonym:
Target:
26-Desglucoavenacoside A
Cat.No: T124583
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T19117 3-Deoxyglucosone

3-Deoxy-D-glucosone,2-keto-3-Deoxyglucose

GPX; Glucagon Receptor GPCR/G Protein; oxidation-reduction
3-Deoxyglucosone(3-Deoxy-D-glucosone) 是美拉德反应和多元醇反应的中间体途径合成。3-Deoxyglucosone 与蛋白质氨基快速反应形成晚期糖基化末端蛋白 (AGEs)。3-Deoxyglucosone 可使谷胱甘肽过氧化物酶失活,可与低葡萄糖协同作用以增强 GLP-1 分泌,可以作为糖尿病生物学检测的标志物。
TN2430 Glucodigifucoside

洋地黄毒苷元葡萄糖基岩藻糖苷,洋地黄

Glucodigifucoside 是可从洋地黄种子中分离得到的强心苷,对人肾腺癌细胞有特异性细胞毒性。
TN4368 Kaempferol-3,7-di-O-β-glucoside

Kaempferol 3,7-di-O-glucoside

Glucosidase; Amylase Metabolism
Kaempferol-3,7-di-O-β-glucoside (Kaempferol 3,7-diglucoside) 是一种来自 Morettia philaena 的黄酮醇,对 α-淀粉酶 (α-amylase)、α-葡萄糖苷酶 (α-glucosidase) 和乙酰胆碱酯酶 (Acetylcholinesterase) 具有抑制作用。Kaempferol-3,7-di-O-β-glucoside 具有神经保护活性,可减缓分化神经元细胞 SH-SY5Y 免受 Amyloid β 肽诱导的损伤。Kaempferol-3,7-di-O-β-glucoside 可用于研究阿尔茨海默氏症类的神经系统疾病。
T2S1682 Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside

Pinocembrin 7-O-(3''-galloyl-4'',6''-(S)-hexahydroxydiphenoyl)-beta-D-glucose,pinocembrin-7-o-3-o-galloyl-4-6-hexahydroxydiphenoyl-beta-d-glucoside

Amylase Metabolism
Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside 可抑制 α-淀粉酶活性,IC50值为0.03 umol/ml。
T9784 Docosanedioic acid 

PROTAC Linker PROTAC
Docosanedioic acid 可以作为ADC linker 或PROTAC linker,用于合成抗体偶联药物或合成 PROTAC。
T2771 Orcinol glucoside

Sakakin,苔黑酚葡萄糖苷

Antioxidant oxidation-reduction
Orcinol glucoside (Sakakin) 是一种提取自莪术中的活性成分,具有抗抑郁活性。它能诱导 MSC 转化为成骨细胞,并通过 Wnt/β-catenin 信号通路阻断脂肪形成。
T3S1628 Vitexin-4''-O-glucoside

Vitexin -4''-O-glucoside,牡荆素-4''-O-葡萄糖苷

Others Others
Vitexin-4''-O-glucoside (Vitexin -4''-O-glucoside) 是一种从Crataegus pinnatifida 叶片中得到的类黄酮成分。
TN7040 Taxifolin 7-O-β-D-glucoside

花旗松素7-O-葡萄糖苷,Taxifolin 7-Glucoside

Others Others
Taxifolin 7-O-β-D-glucoside 是一种 Scutellaria baicalensis 种子萌发阶段的主要代谢产物。它是一种主要存在于胚乳中的类黄酮,能够防御病原体和紫外线损伤。
TN1961 Myricetin 3-O-glucoside

Myricetin 3-O-beta-D-glucopyranoside

Immunology/Inflammation related Immunology/Inflammation
Myricetin 3-O-glucoside (Myricetin 3-O-beta-D-glucopyranoside) 是一种从Tibouchina paratropica 提取 的黄酮醇。Myricetin 3-O-glucoside 具有很多活性,包括抗利什曼原虫、抗炎和抗菌活性。
TN7217 4,6-Benzilidine-D-Glucose

4,6-Benzilidine-D-Glucose 是一种临床抗肿瘤化合物,在化学诱导肝细胞癌大鼠中显示出抗肿瘤活性。
T5250 Levoglucosan

1,6-anhydro-b-D-Glucose,1,6-脱水-β-D-葡萄糖

Others; Endogenous Metabolite Metabolism; Others
Levoglucosan (1,6-anhydro-b-D-Glucose) 是一种无水己糖,是 β -D-葡萄糖的 1,6-无水衍生物。它是由碳水化合物,如淀粉和纤维素的热解形成的。左旋葡聚糖还可用于手性聚合物如不可水解葡萄糖聚合物的合成。左旋葡聚糖也可以通过糖的焦糖化产生。食用焦糖或含焦糖的甜食可导致尿中左旋葡聚糖水平短期增加5倍(从20 μm /mM肌酐增加到100 μm /mM肌酐)。
T3874 Diosgenin glucoside

延龄草苷,地索苷,Disogluside,Trillin

Apoptosis; Others; Autophagy Apoptosis; Autophagy; Others
Diosgenin glucoside (Trillin) 是一种来自蒺藜的皂苷元类天然产物,可通过调节自噬和减轻细胞凋亡来保护脊髓免受损伤。它通过调节小胶质细胞 M1 极化提供神经保护,和其他具有类似活性的合成糖苷可用于治疗高胆固醇血症和动脉粥样硬化。
T4S1439 6'-O-beta-D-Glucosylgentiopicroside

6'-O-β-D-葡萄糖基龙胆苦苷,6'-O-Glucosylgentiopicroside

Antifungal Microbiology/Virology
6'-O-beta-D-Glucosylgentiopicroside (6'-O-Glucosylgentiopicroside) 是一种环烯醚萜,分离自G. straminea 根中。它能显著抑制 fMLP 诱导的超氧化物生成。
T4514 N-Acetyl-D-Glucosamine

N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc

Endogenous Metabolite Metabolism
N-Acetyl-D-Glucosamine (NAG) 是葡萄糖的单糖衍生物。
T3761 1-Octacosanol

n-Octacosanol,二十八烷醇,Montanyl alcohol,Cluytyl alcohol,Octacosanol,Octacosyl alcohol,Octanosol

Others Others
1-Octacosanol (Octanosol) 是直链脂肪族 28 碳脂肪醇,具有抗疲劳作用。
TN6964 Tricosane

Others Others
Tricosane 是来自 Vernonia amygdalina 的天然产物。
T6S2038 Ziyuglycoside II

Apoptosis; Antioxidant; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Ziyuglycoside II 是从地榆中提取的一种三萜皂苷,可诱导活性氧 产生和凋亡,具有抗炎和抗癌作用。
TN2213 Imperialine 3-β-D-glucoside

Sipeimine-3-beta-D-glucoside,西贝母碱苷

Others Others
Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) 是 Imperialine 的糖苷。它对多重耐药肿瘤细胞表现出抗肿瘤特性。
T36115 Colchicoside

3-Demethylcolchicine glucoside

Others Others
Colchicoside (3-Demethylcolchicine glucoside) 提取自嘉兰,在胰腺癌小鼠模型中显示出疗效。
T4S0758 Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden

槲皮素-3-O-Β-D-葡萄糖-7-O-Β-D-龙胆双糖苷,Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside

Others Others
Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden (Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside) 是一种黄酮,来源于 Quercetin 中。
T4726 D-Glucose 6-phosphate sodium

G6P sodium salt,D-Glucose 6-phosphate sodium salt,D-葡萄糖-6-磷酸钠盐,Sodium Glucose-6-Phosphate

Others; Endogenous Metabolite Metabolism; Others
D-Glucose 6-phosphate sodium (G6P sodium salt) 是内源性代谢产物的一种。
T7647 Eicosadienoic acid

二十碳二烯酸,11,14-二十碳二烯酸C20:2

Endogenous Metabolite Metabolism
Eicosadienoic acid 是天然存在的 n-6 多不饱和脂肪酸,主要再动物组织中获得。
T5369 Docosahexaenoic Acid

Cervonic acid,DHA

Others; Endogenous Metabolite Metabolism; Others
Docosahexaenoic Acid 是一种ω-3脂肪酸,在脑和视网膜中较为丰富,且能够直接从鱼油和母乳中获得。
T5711 Methylnissolin-3-O-glucoside

(6aR, 11 aR)-3-hydroxy-9,l0-diMethoxy pt,美迪紫檀苷,黄芪异黄烷苷,7,2'-二羟基-3',4'-二甲氧基异黄烷

Others Others
Methylnissolin-3-O-glucoside ((6aR, 11 aR)-3-hydroxy-9,l0-diMethoxy pt) 是一种类黄酮,从黄芪的根中获得,具有抗炎活性。
T5748 Ipecoside

AIDS031406

Others Others
Ipecoside (AIDS031406) 是一种生物碱,分离自Psychotria。
T2S1464 Thiocolchicoside

硫秋水仙苷;噻可撒可,Thiocolchicine 2-glucoside analog,硫秋水仙苷,Coltramyl

Others; GABA Receptor Membrane transporter/Ion channel; Neuroscience; Others
Thiocolchicoside (Thiocolchicine 2-glucoside analog) 是秋水仙碱的半合成硫衍生物,是竞争性 GABAA 受体拮抗剂和甘氨酸受体拮抗剂。它是肌肉松弛剂,具有抗炎作用,可用于缓解疼痛的研究。
T4956 Tetrahydroxystilbene-2-O-β-D-glucoside

tetrahydroxyl diphenylethylene-2-o-gluco,何首乌苷,EH-201

Others Others
Tetrahydroxystilbene-2-O-β-D-glucoside (EH-201) 是一种低分子量的促红细胞生成素诱导剂。
T4855 Tricosanoic acid

Tricosan-1-oic acid,二十三烷酸

Endogenous Metabolite Metabolism
Tricosanoic acid (Tricosan-1-oic acid) 是毛发生长激活剂,是长链脂肪酸。
T5942 Docosanoic acid

Behenic Acid,山嵛酸

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Docosanoic acid (Behenic Acid) 是一种较难吸收的饱和脂肪酸,能提高人类胆固醇水平。
T3S0488 Syringaresinol diglucoside

Syringaresinol-di-O-glucoside,丁香树脂醇双葡萄糖苷

Others Others
Syringaresinol diglucoside (Syringaresinol-di-O-glucoside) 是一种提取自竹叶中的天然化合物。
T3025 Asiaticoside

BRN0078195,CCRIS8995,Emdecassol,Ba 2742,Madecassol,积雪草皂苷,NSC166062,积雪草苷

Apoptosis; p38 MAPK; Reactive Oxygen Species; Endogenous Metabolite; TGF-beta/Smad Apoptosis; Immunology/Inflammation; MAPK; Metabolism; NF-κB; Stem Cells
Asiaticoside (Emdecassol) 是一种从积雪草中分离得到的三萜皂苷化合物,具有抗氧化、抗炎、抗溃疡等作用。在瘢痕疙瘩成纤维细胞中,它通过活化 Smad7,抑制 TGF-βRI 和 TGF-βRII,抑制 TGF-β/Smad 信号通路。
T2902 Costunolide

Costus lactone,NSC 106404,Costunolid,(+)-Costunolide,木香烃内酯

Apoptosis; Endogenous Metabolite; Telomerase Apoptosis; DNA Damage/DNA Repair; Metabolism
Costunolide (Costus lactone) 是一种天然的倍半萜内酯,具有抗氧化、抗炎、抗过敏、骨重塑、神经保护、促进毛发生长、抗癌和抗糖尿病的特性,可诱导乳腺癌细胞周期阻滞和凋亡。
T5S0581 Sec-O-Glucosylhamaudol

亥茅酚苷,Hamaudol 3-glucoside

Others; Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience; Others
Sec-O-Glucosylhamaudol (Hamaudol 3-glucoside) 是从滨海前胡中分离得到的一种天然产物,能够降低 μ 阿片受体的蛋白水平,可用于缓解疼痛的研究。它通过调节脂多糖刺激的 RAW264.7 细胞系中的 p38 丝裂原活化蛋白激酶具有抗炎作用。
TN6753 1-TETRACOSANOL

二十四醇,Tetracosanol,LIGNOCERYL ALCOHOL

Others Others
1-Tetracosanol (LIGNOCERYL ALCOHOL) 是从多根火龙果 Hylocereus polyrhizus 中提取的天然成分。
TN2237 Steviol-19-O-glucoside

Steviol-19-O-Glucoside,甜菊醇-19-葡萄糖苷

Others Others
Steviol-19-O-glucoside 是甜叶菊 Stevia rebuadiana 中甜菊糖苷生物合成途径的天然产物。
T124477 Resveratrol 4'-(6-galloylglucoside)

Resveratrol-4'-O-(6"-galloyl)glucoside

Others Others
Resveratrol 4'-(6-galloylglucoside) (Resveratrol-4'-O-(6"-galloyl)glucoside)是一种天然产物,存在于植物掌叶大黄 rhubarb (Rheum palmatum L.)的根中。
TN7250 Torachrysone Triglucoside

1-[8-[(O-β-D-Glucopyranosyl-(1→3)-O-β-D-glucopyranosyl-(1→6)-β-D-glucopyranosyl)oxy]-1-hydroxy-6-methoxy-3-methyl-2-naphthalenyl]ethanone

Others Others
Torachrysone Triglucoside 是从决明子种子中分离出来的葡萄糖苷 具有潜在的抗肿瘤活性。
T3426 Bacoside A

MMP; Others; TNF; Dopamine Receptor; NOS; ROS Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience; Others; Proteases/Proteasome
Bacoside A has a possible anticancer activity that could be inducing cell cycle arrest and apoptosis through Notch pathway in GBM in vitro. It exerts cytoprotective efficacy by attenuation of ROS generated through oxidative stress by an increase in the concentration of antioxidant enzymes and sustain membrane integrity which leads to restoring the damage caused by tBHP. Bacoside A can able to inhibit the progression of Experimental Autoimmune Encephalomyelitis (EAE) may be by the inhibition of i...
TN7248 Torachrysone tetraglucoside

Antioxidant; Antifungal Microbiology/Virology; oxidation-reduction
Torachrysone tetraglucoside 是从豆科植物决明子中分离得到的酚苷,具有抗氧化和抗菌活性。
TN6760 1-Eicosanol

Others Others
1-Eicosanol 是从金丝桃分离得到的天然产物,具有抗氧化作用。
T7997 β-D-Glucose pentaacetate

β-D-葡萄糖五乙酸酯,Penta-O-acetyl-β-D-glucopyranose,1,2,3,4,6-beta-D-葡萄糖五乙酸酯

Others Others
β-D-Glucose pentaacetate (Penta-O-acetyl-β-D-glucopyranose) 一种能够用于生化反应的物质。
T4924 α-D-Glucose-1-phosphate disodium

A-D-葡萄糖-1-磷酸-二钠盐,α-D-Glucose 1-phosphate disodium salt hy,α-D-Glucopyranose 1-phosphate

Others; Endogenous Metabolite Metabolism; Others
α-D-Glucose 1-phosphate disodium salt hydrate 是合成葡萄糖醛酸的起始原料。它可用作心脏病研究所必需的细胞抑制剂、抗生素、免疫抑制剂和循环系统研究材料。
TN1824 Kaempferol 3-sophoroside-7-glucoside

Antioxidant oxidation-reduction
Kaempferol 3-sophoroside-7-glucoside 是一种龙脷叶中的生物活性成分,属于黄酮类,具有抗氧化和抗肥胖活性。
T3415 Secoisolariciresinol diglucoside

亚麻木酚素,LGM2605

ROS Immunology/Inflammation
Secoisolariciresinol diglucoside (LGM2605) 在铁过载诱导的氧化还原炎症损伤的体外模型中具有细胞保护作用。 Secoisolariciresinol Diglucoside(25 mg/kg b.w.) 通过抑制 ROS 水平介导的酶和非酶抗氧化剂水平升高来防止肝脏受到过氧化损伤,从而发挥抗高血糖作用。
T8121 Octacosanoic acid

Anti-infection Microbiology/Virology
Octacosanoic acid 具有抗血小板和抗血栓作用。
TN1564 Delphinidin 3-glucoside chloride

Delphinidin-3-O-glucoside chloride,飞燕草素葡萄糖苷,氯化飞燕草素葡萄糖苷

Others Others
Delphinidin-3-O-glucoside chloride has antioxidant activity.
T4884 alpha-D-glucose

α-D-Glucose,α-葡萄糖,alpha-Glucose,α-Dextrose

Others; Endogenous Metabolite Metabolism; Others
alpha-D-glucose (α-Dextrose) 是内源性代谢产物的一种。
TN1414 Aurantio-obtusin β-D-glucoside

橙黄决明素-6-O-葡萄糖苷,Aurantio-obtusin beta-D-glucoside

Others Others
Aurantio-obtusin β-D-glucoside (Aurantio-obtusin beta-D-glucoside) 是分离自决明子的 aurantio-obtusi 的葡糖苷。
TMS0879 Asiaticoside B

积雪草苷 B,积雪草苷B

Others Others
Asiaticoside B 是一种从类叶升麻中分离得到的三萜糖苷,具有抗肿瘤作用。 它对 HepG2 和 MCF-7 癌细胞系具有显著的细胞毒性。
TN1017 Physion 8-O-β-D-glucoside

大黄素甲醚-8-o-β-D-葡萄糖苷,Physcion 1-O-beta-D-glucoside

Others Others
Physion 8-O-β-D-glucoside 是一种 Fallopia multiflora 的活性成分,可用于头晕的研究。
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天然产物

3-Deoxyglucosone
Cat.No: T19117
Synonym: 3-Deoxy-D-glucosone,2-keto-3-Deoxyglucose
Target: GPX, Glucagon Receptor
Glucodigifucoside
Cat.No: TN2430
Synonym: 洋地黄毒苷元葡萄糖基岩藻糖苷,洋地黄
Target:
Kaempferol-3,7-di-O-β-glucoside
Cat.No: TN4368
Synonym: Kaempferol 3,7-di-O-glucoside
Target: Glucosidase, Amylase
Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside
Cat.No: T2S1682
Synonym: Pinocembrin 7-O-(3''-galloyl-4'',6''-(S)-hexahydroxydiphenoyl)-beta-D-glucose,pinocembrin-7-o-3-o-galloyl-4-6-hexahydroxydiphenoyl-beta-d-glucoside
Target: Amylase
Docosanedioic acid 
Cat.No: T9784
Synonym:
Target: PROTAC Linker
Orcinol glucoside
Cat.No: T2771
Synonym: Sakakin,苔黑酚葡萄糖苷
Target: Antioxidant
Vitexin-4''-O-glucoside
Cat.No: T3S1628
Synonym: Vitexin -4''-O-glucoside,牡荆素-4''-O-葡萄糖苷
Target: Others
Taxifolin 7-O-β-D-glucoside
Cat.No: TN7040
Synonym: 花旗松素7-O-葡萄糖苷,Taxifolin 7-Glucoside
Target: Others
Myricetin 3-O-glucoside
Cat.No: TN1961
Synonym: Myricetin 3-O-beta-D-glucopyranoside
Target: Immunology/Inflammation related
4,6-Benzilidine-D-Glucose
Cat.No: TN7217
Synonym:
Target:
Levoglucosan
Cat.No: T5250
Synonym: 1,6-anhydro-b-D-Glucose,1,6-脱水-β-D-葡萄糖
Target: Others, Endogenous Metabolite
Diosgenin glucoside
Cat.No: T3874
Synonym: 延龄草苷,地索苷,Disogluside,Trillin
Target: Apoptosis, Others, Autophagy
6'-O-beta-D-Glucosylgentiopicroside
Cat.No: T4S1439
Synonym: 6'-O-β-D-葡萄糖基龙胆苦苷,6'-O-Glucosylgentiopicroside
Target: Antifungal
N-Acetyl-D-Glucosamine
Cat.No: T4514
Synonym: N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc
Target: Endogenous Metabolite
1-Octacosanol
Cat.No: T3761
Synonym: n-Octacosanol,二十八烷醇,Montanyl alcohol,Cluytyl alcohol,Octacosanol,Octacosyl alcohol,Octanosol
Target: Others
Tricosane
Cat.No: TN6964
Synonym:
Target: Others
Ziyuglycoside II
Cat.No: T6S2038
Synonym:
Target: Apoptosis, Antioxidant, Reactive Oxygen Species
Imperialine 3-β-D-glucoside
Cat.No: TN2213
Synonym: Sipeimine-3-beta-D-glucoside,西贝母碱苷
Target: Others
Colchicoside
Cat.No: T36115
Synonym: 3-Demethylcolchicine glucoside
Target: Others
Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden
Cat.No: T4S0758
Synonym: 槲皮素-3-O-Β-D-葡萄糖-7-O-Β-D-龙胆双糖苷,Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside
Target: Others
D-Glucose 6-phosphate sodium
Cat.No: T4726
Synonym: G6P sodium salt,D-Glucose 6-phosphate sodium salt,D-葡萄糖-6-磷酸钠盐,Sodium Glucose-6-Phosphate
Target: Others, Endogenous Metabolite
Eicosadienoic acid
Cat.No: T7647
Synonym: 二十碳二烯酸,11,14-二十碳二烯酸C20:2
Target: Endogenous Metabolite
Docosahexaenoic Acid
Cat.No: T5369
Synonym: Cervonic acid,DHA
Target: Others, Endogenous Metabolite
Methylnissolin-3-O-glucoside
Cat.No: T5711
Synonym: (6aR, 11 aR)-3-hydroxy-9,l0-diMethoxy pt,美迪紫檀苷,黄芪异黄烷苷,7,2'-二羟基-3',4'-二甲氧基异黄烷
Target: Others
Ipecoside
Cat.No: T5748
Synonym: AIDS031406
Target: Others
Thiocolchicoside
Cat.No: T2S1464
Synonym: 硫秋水仙苷;噻可撒可,Thiocolchicine 2-glucoside analog,硫秋水仙苷,Coltramyl
Target: Others, GABA Receptor
Tetrahydroxystilbene-2-O-β-D-glucoside
Cat.No: T4956
Synonym: tetrahydroxyl diphenylethylene-2-o-gluco,何首乌苷,EH-201
Target: Others
Tricosanoic acid
Cat.No: T4855
Synonym: Tricosan-1-oic acid,二十三烷酸
Target: Endogenous Metabolite
Docosanoic acid
Cat.No: T5942
Synonym: Behenic Acid,山嵛酸
Target: DNA/RNA Synthesis, Endogenous Metabolite
Syringaresinol diglucoside
Cat.No: T3S0488
Synonym: Syringaresinol-di-O-glucoside,丁香树脂醇双葡萄糖苷
Target: Others
Asiaticoside
Cat.No: T3025
Synonym: BRN0078195,CCRIS8995,Emdecassol,Ba 2742,Madecassol,积雪草皂苷,NSC166062,积雪草苷
Target: Apoptosis, p38 MAPK, Reactive Oxygen Species, Endogenous Metabolite, TGF-beta/Smad
Costunolide
Cat.No: T2902
Synonym: Costus lactone,NSC 106404,Costunolid,(+)-Costunolide,木香烃内酯
Target: Apoptosis, Endogenous Metabolite, Telomerase
Sec-O-Glucosylhamaudol
Cat.No: T5S0581
Synonym: 亥茅酚苷,Hamaudol 3-glucoside
Target: Others, Opioid Receptor
1-TETRACOSANOL
Cat.No: TN6753
Synonym: 二十四醇,Tetracosanol,LIGNOCERYL ALCOHOL
Target: Others
Steviol-19-O-glucoside
Cat.No: TN2237
Synonym: Steviol-19-O-Glucoside,甜菊醇-19-葡萄糖苷
Target: Others
Resveratrol 4'-(6-galloylglucoside)
Cat.No: T124477
Synonym: Resveratrol-4'-O-(6"-galloyl)glucoside
Target: Others
Torachrysone Triglucoside
Cat.No: TN7250
Synonym: 1-[8-[(O-β-D-Glucopyranosyl-(1→3)-O-β-D-glucopyranosyl-(1→6)-β-D-glucopyranosyl)oxy]-1-hydroxy-6-methoxy-3-methyl-2-naphthalenyl]ethanone
Target: Others
Bacoside A
Cat.No: T3426
Synonym:
Target: MMP, Others, TNF, Dopamine Receptor, NOS, ROS
Torachrysone tetraglucoside
Cat.No: TN7248
Synonym:
Target: Antioxidant, Antifungal
1-Eicosanol
Cat.No: TN6760
Synonym:
Target: Others
β-D-Glucose pentaacetate
Cat.No: T7997
Synonym: β-D-葡萄糖五乙酸酯,Penta-O-acetyl-β-D-glucopyranose,1,2,3,4,6-beta-D-葡萄糖五乙酸酯
Target: Others
α-D-Glucose-1-phosphate disodium
Cat.No: T4924
Synonym: A-D-葡萄糖-1-磷酸-二钠盐,α-D-Glucose 1-phosphate disodium salt hy,α-D-Glucopyranose 1-phosphate
Target: Others, Endogenous Metabolite
Kaempferol 3-sophoroside-7-glucoside
Cat.No: TN1824
Synonym:
Target: Antioxidant
Secoisolariciresinol diglucoside
Cat.No: T3415
Synonym: 亚麻木酚素,LGM2605
Target: ROS
Octacosanoic acid
Cat.No: T8121
Synonym:
Target: Anti-infection
Delphinidin 3-glucoside chloride
Cat.No: TN1564
Synonym: Delphinidin-3-O-glucoside chloride,飞燕草素葡萄糖苷,氯化飞燕草素葡萄糖苷
Target: Others
alpha-D-glucose
Cat.No: T4884
Synonym: α-D-Glucose,α-葡萄糖,alpha-Glucose,α-Dextrose
Target: Others, Endogenous Metabolite
Aurantio-obtusin β-D-glucoside
Cat.No: TN1414
Synonym: 橙黄决明素-6-O-葡萄糖苷,Aurantio-obtusin beta-D-glucoside
Target: Others
Asiaticoside B
Cat.No: TMS0879
Synonym: 积雪草苷 B,积雪草苷B
Target: Others
Physion 8-O-β-D-glucoside
Cat.No: TN1017
Synonym: 大黄素甲醚-8-o-β-D-葡萄糖苷,Physcion 1-O-beta-D-glucoside
Target: Others
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