首页 工具
登录
购物车

搜索结果

Search Results for " vesicles "

43

抑制剂 & 化合物

9

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T60043 DPTIP

Phospholipase Metabolism
DPTIP 是一种有效的中性鞘磷脂酶 2 抑制剂,IC50 值为 30 nM。
T77579 JC2-11

IL Receptor; Dehydrogenase; ROS; Caspase; NOD-like Receptor (NLR); AIM2 Apoptosis; Immunology/Inflammation; Metabolism; Proteases/Proteasome
JC2-11 是一种对炎症有抑制作用的化合物。JC2-11 对含有募集结构域的蛋白质 NLRC 4、黑色素瘤 2 中缺失 (AIM 2) 和非典型 (NC) 炎症小体有抑制作用,通过破坏活性氧的产生和 caspase-1 的活性来抑制炎症小体的活化。JC2-11 减少了炎症小体中 caspase-1 (p20) 的分泌、gasdermin D (GSDMD) 的裂解、IL-1β 和乳酸脱氢酶 (LDH) 的释放。
T0719 Tetrabenazine

Xenazine,丁苯那嗪,Ro 1-9569

Others; Dopamine Receptor; Monoamine Transporter GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience; Others
Tetrabenazine (Ro 1-9569) 是 VMAT 抑制剂,用作抗精神病药和治疗各种运动障碍。
T6887 MCC950 sodium

CRID3 sodium salt,CP-456773,CP-456773 sodium,MCC950

NOD-like Receptor (NLR); NOD Immunology/Inflammation; NF-κB
MCC950 sodium (CP-456773 sodium) 是一种炎症小体 NLRP3 的抑制剂 (IC50=7.5 nM in BMDMs; IC50=8.1 nM in HMDMs),具有高效选择性。MCC950 sodium 对其他炎症小体,如 AIM2、 NLRC4 或 NLRP1 没有作用。
T3534 Tetrabenazine Racemate

Nitoman,丁苯那嗪外消旋体,丁苯那嗪,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE

Monoamine Transporter Membrane transporter/Ion channel
Tetrabenazine Racemate (Rubigen) 是一种选择性和可逆的囊泡单胺转运蛋白 2(VMAT-2) 抑制剂。它阻断神经递质吸收到肾上腺素能储存囊泡中,并已被用作囊泡运输系统的高亲和力标记。
TF0112 DPPS

12-Dipalmitoyl-sn-glycero-3-PS sodium salt,DPPS-Na

Others Others
DPPS (12-Dipalmitoyl-sn-glycero-3-PS sodium salt) 是一种阴离子二酰基磷脂,是磷脂酰丝氨酸(PS)的一种形式,是一种位于细胞膜内小叶的带负电荷的磷脂。DPPS 被用来制作阳离子囊泡和脂质体。
T13133 Tetrabenazine Metabolite

(-)-β-Dihydrotetrabenazine,(-)-β-HTBZ

Monoamine Transporter Membrane transporter/Ion channel
Tetrabenazine Metabolite ((-)-β-HTBZ) 是一种囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,是 Tetrabenazine 的一种活性代谢物。Tetrabenazine Metabolite 对 VMAT2 具有高亲和力,其Ki 为13.4 nM。Tetrabenazine Metabolite 常常被用于研究与亨廷顿氏病和其他多动障碍相关的舞蹈病。
T2556 Nandrolone decanoate

癸酸诺龙,19-Nortestosterone decanoate

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Nandrolone decanoate (19-Nortestosterone decanoate) 是一种合成代谢雄激素,通过涉及谷氨酸诱导的 N-甲基-D-天冬氨酸受体过度兴奋的机制诱导攻击性行为表征。
T5850 Benzamil

Benzamil (hydrochloride)

Na+/Ca2+ Exchanger; Sodium Channel Membrane transporter/Ion channel
Benzamil 是 Amiloride 类似物,是 Na+/Ca2+交换体抑制剂,抑制 TRPP3 介导的 Ca2+激活电流,IC50为 1.1 μM。它也是一种非选择性上皮钠通道 (ENaC) 阻滞剂,能增强肌源性血管收缩。
T3230 NLRP3-IN-2

5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide,4-[2-(5-氯-2-甲氧基苯甲酰氨基)乙基]苯磺酰胺,NLRP3 Inflammasome Inhibitor I

NOD-like Receptor (NLR); NOD Immunology/Inflammation; NF-κB
NLRP3-IN-2 (5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide) 是一种能够合成格列本脲的中间物,对心肌细胞中NLRP3炎症小体的形成具有抑制作用,在小鼠心肌缺血/再灌注后限制梗死面积,且对代谢无影响。
TP1902L1 G-Protein antagonist peptide acetate

Adrenergic Receptor GPCR/G Protein; Neuroscience
G-Protein antagonist peptide acetate 是一种 substance P 相关肽,可抑制 G 蛋白与其受体的结合。G-Protein antagonist peptide acetate 竞争性和可逆性地抑制毒蕈碱型乙酰胆碱受体 M2 (M2 muscarinic receptor) 对 Gi 或 Go 的激活,并通过 β-肾上腺素受体抑制 Gs 的激活。
T35606 1,2-Dioleoyl-sn-glycero-3-phospho-L-serine sodium

1,2-Dioleoyl-sn-glycero-3-PS (sodium salt)

1,2-Dioleoyl-sn-glycero-3-phospho-L-serine sodium (1,2-Dioleoyl-sn-glycero-3-PS (sodium salt)) 可与 DOPC 和 DOPE 一起用于脂质混合物中,作为有效的无毒和非病毒 DNA 载体。 1,2-Dioleoyl-sn-glycero-3-phospho-L-serine sodium 已用于单层囊泡的形成,以研究曲率对膜结构的影响,并用于支持脂质双层的形成,以研究各种支持膜小叶之间脂质重新分布的材料。
T23709 alphaSYN-IN-NAB2

alphaSYN inhibitor NAB2,alphaSYNINNAB2,alphaSYN-IN-NAB2,NAB2,alphaSYN inhibitor-NAB2

alphaSYN-IN-NAB2 是一种神经元保护剂,是一种由 NAB2基因编码的蛋白质。NAB2 高效且具有选择性地保护多种细胞免受 α-syn 毒性。NAB2 对依赖于 E3 泛素连接酶 Rsp5/Nedd4 的内体转运具有促进作用。NAB2 确定 α-syn 生物学中的一个可活性分子节点,该节点可以纠正其潜在病理学的多个方面,包括功能失调的内体和内质网到高尔基体囊泡的运输。NAB2参与细胞分化、凋亡和应激反应等细胞过程,可用来研究癌症、神经发育和神经元活动。
T30290 Bam 1745

Bam1745,Pyroglutamyl peptide bam-1745,Bam-1745

Bam 1745 is a significant adrenomedullary secretory vesicles component.
T24934 Vesamicol

AH-5183,AH 5183,AH5183

Vesamicol is an experimental drug. It acting presynaptically by inhibiting acetylcholine uptake into synaptic vesicles and reducing its release.
TP2460 Lys-phe-phe-phe-ile-ile-trp-och3

Lys-phe-phe-phe-ile-ile-trp-och3 is a hydrophobic peptide which reacts with lipid vesicles.
T68886 FLA-365

FLA-365 is a biochemical that has been shown to inhibit ryanodine-enhanced calcium release from skeletal SR vesicles in a dose-dependent manner.
T26260 Tetrabenazine methanesulfonate

NSC169886,NSC 169886,NSC-169886

Tetrabenazine methanesulfonate is a medicine formerly utilized as an antipsychotic and therapy for various movement disorders. Tetrabenazine methanesulfonate blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high-affin
T74242 (Rac)-POPC

(Rac)-POPC 是制备巨囊泡 (GV) 的模型磷脂。
T68260 Calmidazolium (cation)

Calmidazolium (cation) is a powerful inhibitor of or red blood cell Ca -ATPase & Ca transport into inside-out red blood cell vesicles; an antagonist of calmodulin.
T74759 18:0,18:1 PS sodium

18:0,18:1 PS sodium 是突触囊泡和胆固醇的脂质组成成分,可用于代谢研究。
T74290 16:0 TAP

16:0 TAP 是一种脂质产品。16:0 TAP 可用于制备巨大的单层囊泡运送活性分子。
T40438 PEG-8 laurate

PEG-8 laurate is a monofunctional surfactant and skin penetration enhancer. It disrupts the skin barrier and facilitates the formation of elastic vesicles when synthesized.
T75360 Oxonol VI

Oxonol VI 是一种膜电位的光学指示剂,在脂质囊泡中发挥作用。它能用于监测重组囊泡中与 (Na++K+)-ATPase 活性相关的膜电位变化。
T37309 Diadenosine pentaphosphate pentaammonium

Diadenosine pentaphosphate pentaammonium, an endogenous vasoactive purine dinucleotide isolated from thrombocytes, is one component of the diadenosine polyphosphates (ApnA, n=2-7) family. These compounds are found in secretory vesicles, including those in platelets, chromaffin cells, Torpedo synaptic terminals, and brain synaptosomes[1][2].
T41088 Diadenosine pentaphosphate pentalithium

Diadenosine pentaphosphate pentalithium is an endogenous vasoactive purine dinucleotide, isolated from thrombocytes. It is a member of the diadenosine polyphosphates (ApnA, n=2–7) and is found in secretory vesicles of platelets, chromaffin cells, Torpedo synaptic terminals, and brain synaptosomes.
T81654 NorA-IN-1

NorA-IN-1 (Compound 16) 为NorA抑制剂,能够抑制外翻膜囊泡中NorA外排泵的活性,适用于多药耐药性研究。
T10191 7-Chlorokynurenic acid sodium salt

7-CKA sodium salt

Others Others
7-Chlorokynurenic acid sodium salt (7-CKA sodium salt) is a potent and selective antagonist of the glycine B coagonist site of the NMDA receptor (IC50: 0.56 μM). It is also a potent inhibitor of the reuptake of glutamate into synaptic vesicles (Ki: 0.59 μ
T61663 SBI-581

SBI-581 is an orally active, potent selective inhibitor of serine-threonine kinase TAO3, with an IC 50 of 42 nM. It effectively promotes the accumulation of TKS5α at RAB11-positive vesicles and inhibits the formation of invadopodia. Additionally, SBI-581 exhibits reasonable pharmacokinetics in mice when administered via IP injection, demonstrating significant antitumor activity [1].
T74306 Chol-PEG

Chol-PEG 是一种非离子表面活性剂囊泡,可用于血液持续给药系统。
T37310 Diadenosine pentaphosphate pentasodium

Diadenosine pentaphosphate pentasodium, an endogenous vasoactive purine dinucleotide isolated from thrombocytes, serves as a key component of secretory vesicles in platelets, chromaffin cells, Torpedo synaptic terminals, and brain synaptosomes. This compound, along with other diadenosine polyphosphates (ApnA, n=2-7), plays a crucial role in physiological processes[1][2].
T74875 1,5-Dihexadecyl N-(3-carboxy-1-oxopropyl)-L-glutamate

1,5-Dihexadecyl N-(3-carboxy-1-oxopropyl)-L-glutamate 是脂质化合物,主要用于提高磷脂囊泡包封蛋白质的效率。
T74758 18:0,22:6 PS sodium

18:0,22:6 PS sodium 是突触囊泡和胆固醇的脂质组成成分,可用于代谢研究。
T80685 γ-Bag cell peptide

γ-袋细胞肽,一种肽类化合物,靠近卵激素原N末端区域定位,能在胰岛素促进下释放其囊泡内容。该肽在中枢及周围神经系统研究中具有应用价值。
T23983 Deutetrabenazine metabolite M4

SD-1018,Deuterated monohydroxy tetrabenazine,D6-tetrabenazine metabolite M4

Deutetrabenazine metabolite M4 is believed to be related to its effect as a reversible depletion of monoamines from nerve terminals. The major circulating metabolites of Deutetrabenazine, are reversible inhibitors of VMAT2, resulting in decreased uptake
T41193 FFN 270

FFN 270 is a fluorescent false neurotransmitter (FFN). Fluorescent substrate for NET and VMAT2. Labels noradrenergic neurons and their synaptic vesicles, and enables imaging of synaptic vesicle content release from specific axonal sitesin vivo. Selectively labels NA neurons over other monoamine and CNS targets. Exhibits two resolved absorption/excitation maxima depending on solvent pH (excitation maxima: 320 nm or 365 nm, emission maxima: 475 nm).
T81286 RG33 Peptide

"RG33 Peptide 是抗 2 型糖尿病 (T2D) 的化合物,它显著增强了胰岛素抵抗小鼠的葡萄糖清除效率。此外,该肽还能高效溶解脂质囊泡,并在培养的巨噬细胞中促进胆固醇排泄。RG33 Peptide 主要用于 2 型糖尿病的研究领域。"
T76315 HKPao

HKPao (Hunter-killer peptide ao) 是一种具有抗肥胖和抗肿瘤促凋亡活性的生物活性肽,能够促使细胞释放囊泡中的细胞色素 c。
T77276 DOPE-mPEG (MW 2000)

DOPE-mPEG (MW 2000),一种磷脂多分散PEG(亦称DOPE脂质体),广泛应用于制备靶向给药脂质体及巨大单层囊泡(GUVs)。此化合物能显著降低脂质体对pH的敏感性,其作用具浓度依赖性。
T37236 (±)17(18)-DiHETE

Eicosapentaenoic acid is an ω-3 fatty acid abundantly available in marine organisms. (±)17(18)-DiHETE is one of the major metabolites produced when eicosapentaenoic acid (EPA) is incubated with various rat tissue homogenates or cynomolgus monkey seminal vesicles. The route of production of (±)17(18)-DiHETE likely proceeds through cytochrome P450-catalyzed epoxidation at the ω-3 double bond followed by conversion to the vicinal diols by epoxide hydrolase. EPA is also metabolized preferentially by...
T83757 RG33 TFA

RG33是一种33个氨基酸的合成肽,与apolipoprotein A1 (ApoA1)的C-末端域中两个Y类螺旋的209-219和220-241氨基酸相对应。它能溶解含有1,2-dimyristoyl-sn-glycero-3-PC (DMPC)的多层囊泡(MLVs),形成重组HDL。与脂质结合的RG33在J774巨噬细胞中诱导胆固醇外流。RG33 (12 mg/kg)可降低胰岛素抵抗性小鼠的血糖水平。
T37743 N-octadecanoyl-L-Homoserine lactone

Quorum sensing is a regulatory system used by bacteria for controlling gene expression in response to increasing cell density. This regulatory process manifests itself with a variety of phenotypes including biofilm formation and virulence factor production. Coordinated gene expression is achieved by the production, release, and detection of small diffusible signal molecules called autoinducers. The N-acylated homoserine lactones (AHLs) comprise one such class of autoinducers, each of which gener...
T37741 N-hexadecanoyl-L-Homoserine lactone

C16-HSL,N-palmitoyl-L-Homoserine,N-hexadecanoyl-L-Homoserine lactone

Quorum sensing is a regulatory system used by bacteria for controlling gene expression in response to increasing cell density.[1] This regulatory process manifests itself with a variety of phenotypes including biofilm formation and virulence factor production.[2] Coordinated gene expression is achieved by the production, release, and detection of small diffusible signal molecules called autoinducers. The N-acylated homoserine lactones (AHLs) comprise one such class of autoinducers, each of which...

化合物

DPTIP
Cat.No: T60043
Synonym:
Target: Phospholipase
JC2-11
Cat.No: T77579
Synonym:
Target: IL Receptor, Dehydrogenase, ROS, Caspase, NOD-like Receptor (NLR), AIM2
Tetrabenazine
Cat.No: T0719
Synonym: Xenazine,丁苯那嗪,Ro 1-9569
Target: Others, Dopamine Receptor, Monoamine Transporter
MCC950 sodium
Cat.No: T6887
Synonym: CRID3 sodium salt,CP-456773,CP-456773 sodium,MCC950
Target: NOD-like Receptor (NLR), NOD
Tetrabenazine Racemate
Cat.No: T3534
Synonym: Nitoman,丁苯那嗪外消旋体,丁苯那嗪,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE
Target: Monoamine Transporter
DPPS
Cat.No: TF0112
Synonym: 12-Dipalmitoyl-sn-glycero-3-PS sodium salt,DPPS-Na
Target: Others
Tetrabenazine Metabolite
Cat.No: T13133
Synonym: (-)-β-Dihydrotetrabenazine,(-)-β-HTBZ
Target: Monoamine Transporter
Nandrolone decanoate
Cat.No: T2556
Synonym: 癸酸诺龙,19-Nortestosterone decanoate
Target: Others, HIV Protease
Benzamil
Cat.No: T5850
Synonym: Benzamil (hydrochloride)
Target: Na+/Ca2+ Exchanger, Sodium Channel
NLRP3-IN-2
Cat.No: T3230
Synonym: 5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide,4-[2-(5-氯-2-甲氧基苯甲酰氨基)乙基]苯磺酰胺,NLRP3 Inflammasome Inhibitor I
Target: NOD-like Receptor (NLR), NOD
G-Protein antagonist peptide acetate
Cat.No: TP1902L1
Synonym:
Target: Adrenergic Receptor
1,2-Dioleoyl-sn-glycero-3-phospho-L-serine sodium
Cat.No: T35606
Synonym: 1,2-Dioleoyl-sn-glycero-3-PS (sodium salt)
Target:
alphaSYN-IN-NAB2
Cat.No: T23709
Synonym: alphaSYN inhibitor NAB2,alphaSYNINNAB2,alphaSYN-IN-NAB2,NAB2,alphaSYN inhibitor-NAB2
Target:
Bam 1745
Cat.No: T30290
Synonym: Bam1745,Pyroglutamyl peptide bam-1745,Bam-1745
Target:
Vesamicol
Cat.No: T24934
Synonym: AH-5183,AH 5183,AH5183
Target:
Lys-phe-phe-phe-ile-ile-trp-och3
Cat.No: TP2460
Synonym:
Target:
FLA-365
Cat.No: T68886
Synonym:
Target:
Tetrabenazine methanesulfonate
Cat.No: T26260
Synonym: NSC169886,NSC 169886,NSC-169886
Target:
(Rac)-POPC
Cat.No: T74242
Synonym:
Target:
Calmidazolium (cation)
Cat.No: T68260
Synonym:
Target:
18:0,18:1 PS sodium
Cat.No: T74759
Synonym:
Target:
16:0 TAP
Cat.No: T74290
Synonym:
Target:
PEG-8 laurate
Cat.No: T40438
Synonym:
Target:
Oxonol VI
Cat.No: T75360
Synonym:
Target:
Diadenosine pentaphosphate pentaammonium
Cat.No: T37309
Synonym:
Target:
Diadenosine pentaphosphate pentalithium
Cat.No: T41088
Synonym:
Target:
NorA-IN-1
Cat.No: T81654
Synonym:
Target:
7-Chlorokynurenic acid sodium salt
Cat.No: T10191
Synonym: 7-CKA sodium salt
Target: Others
SBI-581
Cat.No: T61663
Synonym:
Target:
Chol-PEG
Cat.No: T74306
Synonym:
Target:
Diadenosine pentaphosphate pentasodium
Cat.No: T37310
Synonym:
Target:
1,5-Dihexadecyl N-(3-carboxy-1-oxopropyl)-L-glutamate
Cat.No: T74875
Synonym:
Target:
18:0,22:6 PS sodium
Cat.No: T74758
Synonym:
Target:
γ-Bag cell peptide
Cat.No: T80685
Synonym:
Target:
Deutetrabenazine metabolite M4
Cat.No: T23983
Synonym: SD-1018,Deuterated monohydroxy tetrabenazine,D6-tetrabenazine metabolite M4
Target:
FFN 270
Cat.No: T41193
Synonym:
Target:
RG33 Peptide
Cat.No: T81286
Synonym:
Target:
HKPao
Cat.No: T76315
Synonym:
Target:
DOPE-mPEG (MW 2000)
Cat.No: T77276
Synonym:
Target:
(±)17(18)-DiHETE
Cat.No: T37236
Synonym:
Target:
RG33 TFA
Cat.No: T83757
Synonym:
Target:
N-octadecanoyl-L-Homoserine lactone
Cat.No: T37743
Synonym:
Target:
N-hexadecanoyl-L-Homoserine lactone
Cat.No: T37741
Synonym: C16-HSL,N-palmitoyl-L-Homoserine,N-hexadecanoyl-L-Homoserine lactone
Target:
Cat. No. Product Name Target Signaling Pathways
T7917 4'-Hydroxychalcone

4-羟基查耳酮,4′-羟基查耳酮,2-Benzal-4-Hydroxyacetophenone

Proteasome Proteases/Proteasome; Ubiquitination
4'-Hydroxychalcone (2-Benzal-4-Hydroxyacetophenone) 是从甘草根中分离的一种查尔酮,具有保护肝脏的作用。它能诱导大鼠离体肝线粒体囊泡快速释放钾,并引起其线粒体呼吸控制和氧化磷酸化衰退。它能通过抑制蛋白酶体 (proteasome),抑制TNFα 诱导的 NF-κB 活性。
T19554 L-Aspartic aicd sodium

L-Aspartic acid sodium,Sodium L-aspartate

Others; Sodium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
L-Aspartic aicd sodium (Sodium L-aspartate) 是一种氨基酸,是一种结肠特异性活性分子输送的前体活性分子,可促进大鼠前脑膜囊泡的 Na+外排。
T10191L 7-Chlorokynurenic acid

7-chloro-4-hydroxy-2-carboxyquinoline,7-氯犬尿酸,7-CKA

GluR; NMDAR Neuroscience
7-Chlorokynurenic acid (7-chloro-4-hydroxy-2-carboxyquinoline) 是一种有效的选择性 NMDA 受体拮抗剂,对甘氨酸 B 激动剂位点的 IC50 为 0.56 μM。 7-Chlorokynurenic acid 抑制谷氨酸再摄取到突触小泡中,Ki 为 0.59 μM,并在神经轴输送后显示出镇痛作用。
T4969 Guanosine 5'-triphosphate trisodium salt

鸟苷-5'-三磷酸三钠盐,GTP Trisodium salt,5'-GTP trisodium salt

Endogenous Metabolite Metabolism
Guanosine 5'-triphosphate trisodium salt (5'-GTP trisodium salt) 为G蛋白(G proteins)信号转导过程中的活化剂。
T0791 Reserpine

利血平,Serpalan,Serpasil,Serpivite

Others; Potassium Channel; MRP; Monoamine Transporter; Autophagy Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Others
Reserpine (Serpalan) 是一种从催吐萝芙木的根中发现的生物碱。它抑制去甲肾上腺素吸收到储存囊泡中,导致中枢和外周轴突末端的儿茶酚胺和血清素耗尽。它可作为抗高血压药和抗精神病药以及研究工具。
T8270 Deserpidine

地舍平,Harmonyl

RAAS Endocrinology/Hormones
Deserpidine (Harmonyl) 是从 Rauwolfia canescens 的根中分离的生物碱。Deserpidine 与 Reserpine 相关。Deserpidine 是竞争性血管紧张素转化酶抑制剂,可以被用作抗高血压药以及镇定剂。Deserpidine 还减少了肾上腺皮质血管紧张素 II 诱导的醛固酮分泌。
T33342L Methyl reserpate

NSC81464,NSC 81464,NSC-81464,Me reserpate

Norepinephrine Neuroscience
Methyl reserpate (NSC 81464) 是一种从 Rauwolfia vomitoria 的根和叶中提取出来的育亨宾 (Yohimbine) 型生物碱,抑制去甲肾上腺素转运到嗜铬囊泡中。
TN4374 Kaerophyllin

(-)-Kaerophylin

Apoptosis Apoptosis
Kaerophyllin ( (-)-Kaerophylin) 是一种从中药柴胡中分离出的木酚素,抑制肝细胞凋亡小体激活肝星状细胞,通过抑制肝脏炎症和抑制 HSC 活化来保护大鼠肝脏免受 TAA 引起的损伤和纤维化。
T21772 Reserpine hydrochloride

Reserpine hydrochloride 是一种从催吐萝芙木的根中发现的生物碱。它抑制去甲肾上腺素吸收到储存囊泡中,导致中枢和外周轴突末端的儿茶酚胺和血清素耗尽。它可作为抗高血压药和抗精神病药以及研究工具。

天然产物

4'-Hydroxychalcone
Cat.No: T7917
Synonym: 4-羟基查耳酮,4′-羟基查耳酮,2-Benzal-4-Hydroxyacetophenone
Target: Proteasome
L-Aspartic aicd sodium
Cat.No: T19554
Synonym: L-Aspartic acid sodium,Sodium L-aspartate
Target: Others, Sodium Channel, Endogenous Metabolite
7-Chlorokynurenic acid
Cat.No: T10191L
Synonym: 7-chloro-4-hydroxy-2-carboxyquinoline,7-氯犬尿酸,7-CKA
Target: GluR, NMDAR
Guanosine 5'-triphosphate trisodium salt
Cat.No: T4969
Synonym: 鸟苷-5'-三磷酸三钠盐,GTP Trisodium salt,5'-GTP trisodium salt
Target: Endogenous Metabolite
Reserpine
Cat.No: T0791
Synonym: 利血平,Serpalan,Serpasil,Serpivite
Target: Others, Potassium Channel, MRP, Monoamine Transporter, Autophagy
Deserpidine
Cat.No: T8270
Synonym: 地舍平,Harmonyl
Target: RAAS
Methyl reserpate
Cat.No: T33342L
Synonym: NSC81464,NSC 81464,NSC-81464,Me reserpate
Target: Norepinephrine
Kaerophyllin
Cat.No: TN4374
Synonym: (-)-Kaerophylin
Target: Apoptosis
Reserpine hydrochloride
Cat.No: T21772
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼