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49

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T81550 PAP 248–286

Prostatic Acid Phosphatase(248-286)

PAP 248–286是一种精液衍生的生物活性肽,也称为前列腺酸性磷酸酶 (248-286) 或PAP (248-286) 肽,属于精液中的精液衍生病毒感染增强子 (SEVI) 因子。该肽能显著增强HIV病毒颗粒与靶细胞间的附着,从而增加HIV感染率。
T0488 Finasteride

非那雄胺,MK-906

Reductase Endocrinology/Hormones; Metabolism
Finasteride (MK-906) 是 5α-还原酶的竞争性抑制剂,对 II 型 5α-还原酶的IC50为 4.2 nM,对 II 型 5α-还原酶的亲和力是 I 型酶的 100 倍。它可用于研究前列腺增生和雄激素性脱发。
T0696 Naftopidil

KT-611,萘哌地尔,BM-15275

Adrenergic Receptor GPCR/G Protein; Neuroscience
Naftopidil (KT-611) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力Ki 分别为 3.7 nM、20 nM 、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。
T0091 Alfuzosin hydrochloride

SL 77499-10,Alfuzosin HCl,盐酸阿夫唑嗪

Adrenergic Receptor GPCR/G Protein; Neuroscience
Alfuzosin hydrochloride (Alfuzosin HCl) 是一种 α1 肾上腺素受体拮抗剂,可用于良性前列腺增生(BPH)的研究。
T1504 Silodosin

西洛多辛,KAD 3213,KMD 3213

Adrenergic Receptor GPCR/G Protein; Neuroscience
Silodosin (KAD 3213) 是有选择性的、强效的、口服活性的 α1A-adrenergic receptor 阻滞剂,是一种有效且耐受性良好的试剂,可用于研究 LUTS/BPH。它对 α1A-AR 表现出高度的亲和力,是 α1B-AR 和 α1D-AR 亲和力的 162 和 50 倍。
T0197 Terazosin hydrochloride

盐酸特拉唑嗪,Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic

Adrenergic Receptor GPCR/G Protein; Neuroscience
Terazosin hydrochloride (Hytrin) 是一种竞争性和口服活性的 α1-肾上腺素受体拮抗剂,是一种喹唑啉衍生物。它通过舒张血管和打开膀胱来起作用。它可用于良性前列腺增生和高血压的研究。
T6600 Naftopidil dihydrochloride

KT-611,KT-611 2HCl,盐酸萘哌地尔,Naftopidil DiHCl

5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Naftopidil dihydrochloride (KT-611 2HCl) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力Ki 分别为 3.7 nM、20 nM、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。
T6701 Terazosin hydrochloride dihydrate

Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate,盐酸特拉唑嗪(二水合物)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Terazosin hydrochloride dihydrate (Heitrin dihydrate) 是一种竞争性和口服活性的 α1-肾上腺素受体(α1-adrenoceptor) 拮抗剂,是一种喹唑啉衍生物,通过舒张血管和打开膀胱的方式起作用。它可用于研究良性前列腺增生 (BPH) 和高血压。
T9220 Naftopidil hydrochloride

1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,萘哌地尔盐酸盐,KT-611 hydrochloride,BM-15275 hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Naftopidil hydrochloride (BM-15275 hydrochloride) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力 Ki 分别为 3.7 nM、20 nM、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。
T14843 Bifluranol

BX341

Androgen Receptor Endocrinology/Hormones
Bifluranol (BX341) 具有抗雄激素活性,在体内实验中显示出显著的抗前列腺活性,可用于治疗良性前列腺增生 (BPH)。
T11220L UK 227786

hydrochloride(150452-18-9 Free base),1-[4-(1,3-Benzodioxol-5a-ylmethylamino)-6-chloroquinazolin-2-yl]piperidine-4-carboxylic acid;hydrochloride(150452-18-9 Free base),1-[4-(1,3-Benzodioxol-5a-ylmethylamino)-6-chloroquinazolin-2-yl]piperidine-4-carboxylic acid

PDE Metabolism
UK 227786是磷酸二酯酶5(PDE5)抑制剂,可用于前列腺疾病治疗的研究。
T13703 Gestonorone Capronate

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Gestonorone Capronate 是一种孕激素,在良性前列腺肥大和子宫内膜癌领域有研究价值。
T35182 Xinidamine

BRN 0891979,Xinidaminum,Xinidamino

Xinidamine (BRN 0891979) 具有抗肿瘤活性,可用于研究良性前列腺增生、黄斑变性和前列腺上皮内瘤 。Xinidamine 对PWR-1E 细胞的增殖具有抑制作用,IC50为4μM。
T22316 Doxazosin

UK 33274,多沙唑嗪

Adrenergic Receptor GPCR/G Protein; Neuroscience
Doxazosin (UK 33274) 是选择性的拮抗突触后的α1肾上腺素受体。
T27798 Lapisteride

CS891B,CS-891,CS-891B,CS891

Others Others
Lapisteride (CS-891) 一种类固醇5α-还原酶抑制剂,可用于治疗良性前列腺增生(BPH)和雄激素性脱发,可有效预防或治疗AGA 。
T15688 L-771688

SNAP 6383

Adrenergic Receptor GPCR/G Protein; Neuroscience
L-771688(SNAP 6383) 是一种新型有效和选择性的 α1A-肾上腺素受体拮抗剂, Ki 值为 0.43±0.02 nM。L-771688 KE 用于治疗良性前列腺增生。
T83965 Tamsolusin Hydrochloride

YM 12617,LY-253352

Adrenergic Receptor GPCR/G Protein; Neuroscience
Tamsolusin Hydrochloride (YM 12617) 是一种高选择性α-1A肾上腺素受体拮抗剂,可用于治疗良性前列腺肥大。
T28922 Taprizosin

Taprizosin Mesylate,UK-338003,UK-338,003,UK338003,UK 338003

Adrenergic Receptor GPCR/G Protein; Neuroscience
Taprizosin(UK-338003)是一种具有选择性和口服活性的 α1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,可用于舒张血管,用于治疗良性前列腺增生症。
T1499 Dutasteride

GG 745,Avodart,度他雄胺,GI 198745

Apoptosis; Reductase Apoptosis; Endocrinology/Hormones; Metabolism
Dutasteride (GI 198745) 是一种 5α 还原酶同工酶抑制剂,还可能因其结构域 DHT 相似对雄激素受体产生脱靶效应。
T22232 Alfuzosin

Alfuzosin 是选择性和竞争性的α1肾上腺素受体拮抗剂,可用于良性前列腺增生(BPH)的研究。
T11286 Fiduxosin

A 185980.1,ABT 980

Adrenergic Receptor GPCR/G Protein; Neuroscience
Fiduxosin 是一种具有选择性和有效性的 α1-adrenoceptor 拮抗剂,对 α1a-adrenoceptor,α1b-adrenoceptor 和 α1d-adrenoceptor 有抑制作用,Ki 值分别为 0.160 nM,24.9 nM 和 0.920 nM。Fiduxosin 可用于治疗良性前列腺增生。
T0272 Nilutamide

尼鲁米特,RU23908

Androgen Receptor Endocrinology/Hormones
Nilutamide (RU23908) 是一种非甾体抗雄激素药物,有用于转移性前列腺癌的潜力。
T0210L Tamsulosin

LY253351 free base,HSDB7744,(R)-(-)-YM12617 free base,Harnal-D,Flowmax,HSDB 7744,HSDB-7744

Adrenergic Receptor GPCR/G Protein; Neuroscience
Tamsulosin ((R)-(-)-YM12617 free base) 是一种肾上腺素能受体α 1A 拮抗剂,用于良性前列腺增生(BPH)的治疗。Tansulosin 用于治疗排尿困难,这是前列腺肥大的一种常见症状。Tansulosin 和其他被称为α受体阻滞剂的药物通过放松膀胱颈部肌肉和前列腺本身的肌肉纤维来发挥作用,使其更容易排尿。
T20681 Estramustine

NSC-89201,NSC 89201,LEO 275,LEO275,雌莫司汀,NSC89201,LEO-275

Microtubule Associated Cytoskeletal Signaling
Estramustine (LEO-275) 是一种与雌二醇相连的氮芥,通常为磷酸盐。它已被用于治疗前列腺肿瘤;还具有防辐射功能。它被前列腺细胞选择性吸收,并通过干扰微管动力学和降低血浆睾酮水平发挥抗肿瘤作用。
T1050 Prazosin hydrochloride

Prazosin hydrochloride,哌唑嗪盐酸盐,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,盐酸哌唑嗪,Minipress

Potassium Channel; MRP; Adrenergic Receptor; ABC; Autophagy Autophagy; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Prazosin hydrochloride (Vasoflex) 是一种选择性肾上腺素能 α-1 拮抗剂,可降低外周阻力并放松血管平滑肌。 它可用于研究高血压和酒精使用障碍。 它是一种合成哌嗪衍生物,具有降压抗肾上腺素能特性。它抑制有机阳离子转运蛋白 OCT-1 和 OCT-3,IC50分别为 1.8 和 13 μM 。
T70396 Fexapotide triflutate

Fexapotide triflutate is a caspase and TNF signaling pathway activator used to treat benign prostatic hyperplasia (BPH).
T11220 ER21355

Others Others
ER21355, utilized for the treatment of prostatic diseases, acts as a phosphodiesterase 5 (PDE5) inhibitor.
T28956 TF-505

FR-146687,FK-687,TF 505,FK687

TF-505, a steroid 5α-reductase inhibitor, is used potentially for the treatment of benign prostatic hyperplasia.
T32029 GYKI-16084

GYKI 16084

GYKI-16084 is a postsynaptic alpha2 receptor blocker with potential efficacy in the treatment of benign prostatic hyperplasia.
T20024 Tadalafil, (6R ,12aS)-

Tadalafil (6R ,12aS)- Lilly,Tadalafil specified impurity A,(-)-Tadalafil (6R ,12aS) diastereomer

Tadalafil is a carboline derivative and Phosphodiesterase 5 Inhibitor. It is used primarily to treat Erectile dysfunction, Benign Prostatic Hyperplasia, and Primary Pulmonary Hypertension.
T33826 Osaterone

Osaterone is effective against prostatic hyperplasia in dogs.
T31681 Estradiol undecylate

AI352642,AI3-52642,AI3 52642

Estradiol undecylate can be used in the treatment of prostatic cancer.
T4451L Estramustine phosphate

LS 299,NSC 89199,NSC-89199,LS-299,LS299

Estramustine phosphate can be used to treat prostatic neoplasms; also has radiation protective properties.
T24378 L-771688 dihydrochloride

L 771688 dihydrochloride

L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.
T10780 CGP-53153

Others Others
CGP-53153 is a steroidal inhibitor of 5 alpha-reductase (IC50s: 36 and 262 nM in rat and human prostatic tissue).
T3290L Pikamilone Sodium

GABA-NG,Nicotinoyl-GABA sodium salt,GABA NG,GABANG,Pikamilone Na

Pikamilone Sodium is a prodrug of GABA used for therapy of neurogenic bladder in spinal and benign prostatic hyperplasia.
T69927 Fiduxosin hydrochloride

Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.
T21016 Cyproterone

BAY 94-8367,Ciproterone,Androcur,SH 80881

Cyproterone, an anti-androgen, is used in combination with estrogen for the therapy of hirsutism and severe acne in females and as a palliative in prostatic carcinoma.
T10273 AhR modulator-1

Others Others
AhR modulator-1 is a selective and orally active aryl hydrocarbon receptor (AhR) modulator. It inhibits metastasis, in part, by inhibiting prostatic VEGF production prior to tumor formation. It also possesses anti-estrogenic properties in rat uterus.
T61729 Terazosin

Terazosin, a quinazoline derivative, is an orally active and competitive antagonist of α1-adrenoceptors. Its mechanism of action involves relaxing blood vessels and promoting bladder opening. Terazosin exhibits therapeutic potential for treating benign prostatic hyperplasia (BPH) and high blood pressure [1][2][3].
T78945 WCA-814

Androgen Receptor Endocrinology/Hormones
WCA-814是雄激素受体(AR)拮抗剂与Hsp90抑制剂的融合化合物,能够诱导全长AR及AR-V7降解,并展现出对前列腺癌细胞的细胞毒性(IC50: LNCaP细胞为171.2 nM,22Rv1细胞为26.5 nM)。
TP1094 TAK-448

MVT-602

TAK-448 (MVT-602) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM.TAK-448 has been used in trials studying the treatment of Prostate Cancer, Low Testosterone, Prostatic Neoplasms, and Hypogonadotropic Hypogonadism.
T28245 ONO-0300302

ONO 0300302

ONO-0300302 is a slow tight binding LPA1 antagonist (IC50: 0.16 nM) used to treat Benign Prostatic Hyperplasia. ONO-0300302 inhibits significantly an LPA-induced increase of intraurethral pressure (IUP) in rat (3 mg/kg, p.o.) and dog (1 mg/kg, p.o.) over
T76430 GR 87389

GR 87389 是一种有效的NK2受体拮抗剂。GR 87389 以竞争性方式拮抗 GA 64349 诱导的人类逼尿肌、前列腺和前列腺尿道平滑肌条收缩。
T9660 Bexlosteride

Bexlosteride (LY300502) 是一种苯并喹啉酮类人 I 型 5α-还原酶抑制剂。Bexlosteride 在 LNCaP 细胞培养物中显示出代谢抑制、抗增殖和抗分泌作用。Bexlosteride 可用于前列腺癌的研究。
T76275 Fexapotide

Fexapotide (NX-1207 free acid) 在细胞水平上通过选择性诱导细胞凋亡,降低前列腺体积。它主要用于研究下尿路症状(LUTS)与良性前列腺增生(BPH)。
T75377 Thymolphthalein monophosphate disodium hydrate

Thymolphthalein monophosphate disodium hydrate 是用于测定酸性及碱性磷酸酶显色底物。反应过程中释放的百里酚酞可增加介质pH,促使颜色产生并终止水解作用,特别适合于血清中前列腺磷酸酶的特异性检测。
T69618 XR3054

XR3054 is a novel inhibitor of farnesyl protein transferase (FPTase). XR3054 inhibited the proliferation of the prostatic cancer cell lines LnCAP and PC3 and the colon carcinoma SW480 and HT1080 (IC50 values of 12.4, 12.2, 21.4 and 8.8 microM, respectively) but was relatively inactive when tested against a panel of breast carcinoma cell lines. The activity did not relate to the presence of mutant or wild-type ras in the cell lines tested. In conclusion XR3054 inhibits ras farnesylation, MAP kina...
T21668 Finasteride acetate

Finasteride (MK-906) acetate 是一种高效的5α-还原酶 (5α-reductase) 竞争性抑制剂,其对 II 型 5α-还原酶的IC50值仅为 4.2 nM,其对该型酶的亲和力是对 I 型酶亲和力的约100倍。因此,Finasteride acetate 主要在良性前列腺增生症 (BPH) 和雄激素性脱发研究领域中应用。

化合物

PAP 248–286
Cat.No: T81550
Synonym: Prostatic Acid Phosphatase(248-286)
Target:
Finasteride
Cat.No: T0488
Synonym: 非那雄胺,MK-906
Target: Reductase
Naftopidil
Cat.No: T0696
Synonym: KT-611,萘哌地尔,BM-15275
Target: Adrenergic Receptor
Alfuzosin hydrochloride
Cat.No: T0091
Synonym: SL 77499-10,Alfuzosin HCl,盐酸阿夫唑嗪
Target: Adrenergic Receptor
Silodosin
Cat.No: T1504
Synonym: 西洛多辛,KAD 3213,KMD 3213
Target: Adrenergic Receptor
Terazosin hydrochloride
Cat.No: T0197
Synonym: 盐酸特拉唑嗪,Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic
Target: Adrenergic Receptor
Naftopidil dihydrochloride
Cat.No: T6600
Synonym: KT-611,KT-611 2HCl,盐酸萘哌地尔,Naftopidil DiHCl
Target: 5-HT Receptor, Adrenergic Receptor
Terazosin hydrochloride dihydrate
Cat.No: T6701
Synonym: Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate,盐酸特拉唑嗪(二水合物)
Target: Adrenergic Receptor
Naftopidil hydrochloride
Cat.No: T9220
Synonym: 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,萘哌地尔盐酸盐,KT-611 hydrochloride,BM-15275 hydrochloride
Target: Adrenergic Receptor
Bifluranol
Cat.No: T14843
Synonym: BX341
Target: Androgen Receptor
UK 227786
Cat.No: T11220L
Synonym: hydrochloride(150452-18-9 Free base),1-[4-(1,3-Benzodioxol-5a-ylmethylamino)-6-chloroquinazolin-2-yl]piperidine-4-carboxylic acid;hydrochloride(150452-18-9 Free base),1-[4-(1,3-Benzodioxol-5a-ylmethylamino)-6-chloroquinazolin-2-yl]piperidine-4-carboxylic acid
Target: PDE
Gestonorone Capronate
Cat.No: T13703
Synonym:
Target: Prostaglandin Receptor
Xinidamine
Cat.No: T35182
Synonym: BRN 0891979,Xinidaminum,Xinidamino
Target:
Doxazosin
Cat.No: T22316
Synonym: UK 33274,多沙唑嗪
Target: Adrenergic Receptor
Lapisteride
Cat.No: T27798
Synonym: CS891B,CS-891,CS-891B,CS891
Target: Others
L-771688
Cat.No: T15688
Synonym: SNAP 6383
Target: Adrenergic Receptor
Tamsolusin Hydrochloride
Cat.No: T83965
Synonym: YM 12617,LY-253352
Target: Adrenergic Receptor
Taprizosin
Cat.No: T28922
Synonym: Taprizosin Mesylate,UK-338003,UK-338,003,UK338003,UK 338003
Target: Adrenergic Receptor
Dutasteride
Cat.No: T1499
Synonym: GG 745,Avodart,度他雄胺,GI 198745
Target: Apoptosis, Reductase
Alfuzosin
Cat.No: T22232
Synonym:
Target:
Fiduxosin
Cat.No: T11286
Synonym: A 185980.1,ABT 980
Target: Adrenergic Receptor
Nilutamide
Cat.No: T0272
Synonym: 尼鲁米特,RU23908
Target: Androgen Receptor
Tamsulosin
Cat.No: T0210L
Synonym: LY253351 free base,HSDB7744,(R)-(-)-YM12617 free base,Harnal-D,Flowmax,HSDB 7744,HSDB-7744
Target: Adrenergic Receptor
Estramustine
Cat.No: T20681
Synonym: NSC-89201,NSC 89201,LEO 275,LEO275,雌莫司汀,NSC89201,LEO-275
Target: Microtubule Associated
Prazosin hydrochloride
Cat.No: T1050
Synonym: Prazosin hydrochloride,哌唑嗪盐酸盐,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,盐酸哌唑嗪,Minipress
Target: Potassium Channel, MRP, Adrenergic Receptor, ABC, Autophagy
Fexapotide triflutate
Cat.No: T70396
Synonym:
Target:
ER21355
Cat.No: T11220
Synonym:
Target: Others
TF-505
Cat.No: T28956
Synonym: FR-146687,FK-687,TF 505,FK687
Target:
GYKI-16084
Cat.No: T32029
Synonym: GYKI 16084
Target:
Tadalafil, (6R ,12aS)-
Cat.No: T20024
Synonym: Tadalafil (6R ,12aS)- Lilly,Tadalafil specified impurity A,(-)-Tadalafil (6R ,12aS) diastereomer
Target:
Osaterone
Cat.No: T33826
Synonym:
Target:
Estradiol undecylate
Cat.No: T31681
Synonym: AI352642,AI3-52642,AI3 52642
Target:
Estramustine phosphate
Cat.No: T4451L
Synonym: LS 299,NSC 89199,NSC-89199,LS-299,LS299
Target:
L-771688 dihydrochloride
Cat.No: T24378
Synonym: L 771688 dihydrochloride
Target:
CGP-53153
Cat.No: T10780
Synonym:
Target: Others
Pikamilone Sodium
Cat.No: T3290L
Synonym: GABA-NG,Nicotinoyl-GABA sodium salt,GABA NG,GABANG,Pikamilone Na
Target:
Fiduxosin hydrochloride
Cat.No: T69927
Synonym:
Target:
Cyproterone
Cat.No: T21016
Synonym: BAY 94-8367,Ciproterone,Androcur,SH 80881
Target:
AhR modulator-1
Cat.No: T10273
Synonym:
Target: Others
Terazosin
Cat.No: T61729
Synonym:
Target:
WCA-814
Cat.No: T78945
Synonym:
Target: Androgen Receptor
TAK-448
Cat.No: TP1094
Synonym: MVT-602
Target:
ONO-0300302
Cat.No: T28245
Synonym: ONO 0300302
Target:
GR 87389
Cat.No: T76430
Synonym:
Target:
Bexlosteride
Cat.No: T9660
Synonym:
Target:
Fexapotide
Cat.No: T76275
Synonym:
Target:
Thymolphthalein monophosphate disodium hydrate
Cat.No: T75377
Synonym:
Target:
XR3054
Cat.No: T69618
Synonym:
Target:
Finasteride acetate
Cat.No: T21668
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T41288 Myristoleic acid

cis-9-tetradecenoic acid,肉豆蔻酸,9-Tetradecenoic acid,(Z)-Tetradec-9-enoic acid

Apoptosis Apoptosis
Myristoleic acid (9-Tetradecenoic acid) 是 Serenoa repens 提取物中的一种细胞毒性成分。Myristoleic acid 诱导人前列腺 LNCaP 细胞凋亡和坏死。
TN5031 Sitostenone

豆甾-4-烯-3-酮

Others Others
Sitostenone 具有抗氧化活性。 Stigmasta-4-en-3-one(Sitostenone)可用于治疗雄激素依赖性疾病,尤其是治疗良性前列腺增生。
T19687 Phenylethyl isothiocyanate

JC 5411,2-苯基乙基异硫代氰酸酯,JC5411,JC-5411

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
Phenylethyl isothiocyanate (JC5411) 是一种 HDAC 抑制剂。它有可能用于治疗良性前列腺肥大。
TCS1372 Atraric acid

Phosphatase; Androgen Receptor Endocrinology/Hormones; Metabolism
Atraric acid 衍生物作为一种新的化学先导结构,用于作为 AR 拮抗剂的新型治疗化合物,可用于预防或治疗前列腺疾病。它以剂量依赖性方式抑制 PTP1B 活性,IC50 值为 51.5 uM,表明阿特拉酸具有治疗糖尿病的潜力。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
TN1061 Ganoderol B

Androgen Receptor Endocrinology/Hormones
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate cancer and benign prostatic hyperplasia (BPH) therapy through suppressing the function of andr
TN4164 Grandifloroside

TNF Apoptosis
Grandifloroside shows good antioxidative and potent anti-inflammatory activities, it also exhibits potent inhibitory activity against TNF-α and 5α-reductase, suggests that it might be developed as a source of potent anti-oxidative and anti-inflammatory ag
TN6198 Mahanine

Mahanine has effects on the activation of the apoptotic pathway in human leukemia U937 cells, causes the mitochondrial membranes to lose their permeability, resulting in caspase-3 activation and apoptosis. Mahanine can reverse an epigenetically silenced g

天然产物

Myristoleic acid
Cat.No: T41288
Synonym: cis-9-tetradecenoic acid,肉豆蔻酸,9-Tetradecenoic acid,(Z)-Tetradec-9-enoic acid
Target: Apoptosis
Sitostenone
Cat.No: TN5031
Synonym: 豆甾-4-烯-3-酮
Target: Others
Phenylethyl isothiocyanate
Cat.No: T19687
Synonym: JC 5411,2-苯基乙基异硫代氰酸酯,JC5411,JC-5411
Target: HDAC
Atraric acid
Cat.No: TCS1372
Synonym:
Target: Phosphatase, Androgen Receptor
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Ganoderol B
Cat.No: TN1061
Synonym:
Target: Androgen Receptor
Grandifloroside
Cat.No: TN4164
Synonym:
Target: TNF
Mahanine
Cat.No: TN6198
Synonym:
Target:
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