86
19
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6479 |
Dovitinib lactate hydrate
Dovitinib (TKI258) Lactate,多韦替尼,Dovitinib Lactate,TKI258 |
VEGFR; FGFR; FLT; PDGFR; c-Kit | Angiogenesis; Tyrosine Kinase/Adaptors |
Dovitinib lactate hydrate (TKI258) 是一种多靶点的酪氨酸激酶抑制剂,抑制 FLT3,c-Kit,FGFR1/3,VEGFR1/2/3和 PDGFRα/β的 IC50值分别为 1,2,8/9,10/13/8,27/210 nM。 | |||
T7104 |
Dovitinib lactate
CHIR-258 lactate,多韦替尼乳酸盐,TKI-258 lactate |
VEGFR; FGFR; FLT; PDGFR; c-Kit | Angiogenesis; Tyrosine Kinase/Adaptors |
Dovitinib lactate (TKI-258 lactate) 是一种多靶点的酪氨酸激酶抑制剂,抑制FLT3,c-Kit,FGFR1/3,VEGFR1/2/3和PDGFRα/β的IC50值分别为 1,2,8/9,10/13/8,27/210 nM。 | |||
T40923 |
Calcium lactate
Lactic acid calcium,Hemicalcium L-lactate,Lactate calcium,乳酸钙,Conclyte calcium |
Others | Others |
Calcium lactate (Conclyte calcium) 被饮料工业用作强化果汁的钙源。Calcium lactate 促进豆芽生长和植酸降解。 | |||
T5967 |
Ethacridine lactate
乳酸依沙吖啶,Acrinol,6,9-DIAMINO-2-ETHOXYACRIDINE LACTATE |
Others; Antibacterial | Microbiology/Virology; Others |
Ethacridine lactate (Acrinol) 是一种聚 (ADP-核糖) 糖水解酶 (PARG) 抑制剂,也是一种抗菌剂和流产剂。它有抗金黄色葡萄球菌和其他革兰氏阳性球菌的活性。 | |||
T4103 |
(L)-Sodium lactate
L-乳酸钠,Sodium L-Lactate |
Others | Others |
(L)-Sodium lactate (Sodium L-Lactate) 是由乳酸脱氢酶从丙酮酸中产生的。它在无氧糖酵解过程中或增殖活跃的细胞中产生。 它在人和动物的血液和肌肉液中少量存在。剧烈运动后,肌肉和血液中的乳酸浓度会增加。 它也存在于肝脏、肾脏、胸腺、人羊水以及其他器官和体液中。 | |||
T8785 |
HALOFUGINONE LACTATE
|
DNA/RNA Synthesis; TGF-beta/Smad | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Stem Cells |
HALOFUGINONE LACTATE 是 febrifugine 的卤化衍生物,它是一种天然的含有喹唑啉酮的化合物,存在于中草药 D. febrifuga 中。Halofuginone 以 ATP 依赖性方式抑制脯氨酰-tRNA 合成酶,Ki 为 18.3 nM。 Halofuginone 是 I 型胶原合成的特异性抑制剂,通过抑制 TGF-β 活性来减轻骨关节炎 (OA) | |||
T1440 |
Ethacridine lactate monohydrate
乳酸依沙吖啶一水物,利凡诺 |
Antibacterial; Antibiotic | Microbiology/Virology |
Ethacridine lactate monohydrate 是一种聚 (ADP-核糖) 糖基水解酶 (PARG) 抑制剂,有抗金黄色葡萄球菌和其他革兰氏阳性球菌的活性。它也是抗菌剂和流产剂。 | |||
T32809 |
L-Lactate ion
L-Lactate,Lactate ion, L- |
||
L-Lactate ion is the conjugate base of lactic acid. | |||
T26300 |
Tylosin, lactate
lactate (1:1),Tylosin |
||
Tylosin, lactate is a bacteriostat feed additive used in veterinary medicine. It is a macrolide antibiotic that has a broad spectrum of activity against Gram-positive organisms but a limited range of Gram-negative organisms. It is found naturally as a fer | |||
T12117 |
MSI-1436 lactate
Trodusquemine lactate,Aminosterol-1436 lactate |
Others | Others |
MSI-1436 lactate is a selective, non-competitive the enzyme protein-tyrosine phosphatase 1B (PTB1B)inhibitor(IC50 of appr 1 μM) | |||
T28236 |
Onalespib lactate
AT-13387 lactate,ATI-13387AU,ATI-13387,ATI 13387,ATI-13387A |
||
Onalespib lactate is a second-generation, potent and selective HSP90 Inhibitor with antitumor activity. | |||
T33057 |
Lysine lactate
|
||
Lysine lactate is a bioactive chemical. | |||
T68415 |
Tozasertib lactate
|
||
Tozasertib lactate is a potent and selective small-molecule inhibitor of the Aurora kinases which suppresses tumor growth by inducing apoptosis in tumor cells in which Aurora kinases are overexpressed. | |||
T39862 | Trimethoprim lactate | ||
Trimethoprim lactic is a bacteriostatic antibiotic and an orally active dihydrofolate reductase inhibitor. Trimethoprim lactic is active against a wide range of Gram-positive and Gram-negative aerobic bacteria . Trimethoprim lactic has the potential for urinary tract infections, Shigellosis and Pneumocystis pneumonia treatment. | |||
T30456 |
Biperiden lactate
|
||
Biperiden lactate is a biochemical. | |||
T24659 |
Prenylamine lactate
Agozol,Angormin |
||
Prenylamine lactate is a drug formerly used in the treatment of angina pectoris. Prenylamine depletes myocardial catecholamine stores and has some calcium channel blocking activity. | |||
T30453 |
Bimethoxycaine lactate
U 0045,U-0045,NSC 9108,NSC9108,NSC-9108 |
||
Bimethoxycaine lactate is a bioactive chemical. | |||
T33054 |
Lysine DL-lactate
|
||
Lysine DL-lactate is a bioactive chemical. | |||
T20440 |
Benzyl lactate
AI3 15720,AI3-15720,AI315720 |
||
Benzyl Lactate is an agent of biochemical. | |||
T4310L |
Prexasertib lactate hydrate
Prexasertib monolactate monohydrate,LY-2606368,LY 2606368,LY2606368,Prexasertib monolactate monohydrate salt |
||
Prexasertib is an effective and selective Chk1/Chk2 inhibitor. Prexasertib causes Replication Catastrophe and Antitumor Effects through CHK1-Dependent Mechanisms. | |||
T6702L |
Terbinafine lactate
DRG-0286,Terbinafine hydrochloride,Lamisil Krem,SF 86-327 hydrochloride,Lamisil,Lamisil AT |
||
Terbinafine, a synthetic allylamine antifungal, inhibits ergosterol synthesis by inhibiting squalene epoxidase, an enzyme that is part of the fungal cell membrane synthesis pathway. | |||
T21151 |
AT-9283 L-lactate
AT-9283,AT 9283,AT9283 |
||
AT-9283 L-lactate is an inhibitor of aurora kinase. | |||
T62524 | Panobinostat lactate | ||
Panobinostat lactate 是一种有效的、口服具有活力的、非选择性 HDAC 抑制剂,具有抗肿瘤作用。Panobinostat lactate 诱导细胞凋亡 (apoptosis) 和自噬 (autophagy)。Panobinostat lactate 能够有效干扰 HIV 潜伏期。Panobinostat lactate 能够用于研究难治性或复发性多发性骨髓瘤。 | |||
T78348 |
Lactate oxidase
|
||
Lactate oxidase是一种FMN依赖性酶,能催化乳酸转化为丙酮酸并同时释放过氧化氢,常用于乳酸的检测。 | |||
T68672 | Amsacrine lactate | ||
Amsacrine lactate is an aminoacridine derivative with potential antineoplastic activity. Although its mechanism of action is incompletely defined, amsacrine may intercalate into DNA and inhibit topoisomerase II, resulting in DNA double-strand breaks, arrest of the S/G2 phase of the cell cycle, and cell death. | |||
T81962 | Lactate transportor 1 | Monocarboxylate transporter | Membrane transporter/Ion channel |
Lactate transporter 1 (compound 1) 作为一种活性乳酸运输蛋白,主要在活细胞内发挥作用。在Hela、CAL27、MCF7和MCF10A细胞系中,Lactate transporter 1 均显示出了明显的毒性,其半抑制浓度(IC50)值依次为3.36、3.27、5.58和7.66 μM。此外,在HeLa细胞中,Lactate transporter 1 与Cisplatin表现出了协同抑制的作用。 | |||
T62975 |
Haloperidol lactate
|
||
Haloperidol lactate 是一种有效的抗精神病药。Haloperidol lactate 具有潜力进行精神障碍的研究。Haloperidol lactate 能够用于急性和慢性精神分裂症和多发性秽语综合征。 | |||
T68742 | Inamrinone lactate | ||
Inamrinone lactate is a positive inotropic cardiotonic with vasodilator properties, phosphodiesterase inhibitory activity, and the ability to stimulate calcium ion influx into the cardiac cell. | |||
T64542 |
Lactate potassium
|
||
Lactate potassium 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64542,CAS号为 996-31-6。 | |||
T66299 |
Ciprofloxacin lactate
|
||
Ciprofloxacin lactate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66299,CAS号为 97867-33-9。 | |||
T70625 |
Nicotine lactate
|
||
Nicotine is a naturally produced alkaloid in the nightshade family of plants (most predominantly in tobacco and Duboisia hopwoodii) and is widely used recreationally as a stimulant and anxiolytic. As a pharmaceutical drug, it is used for smoking cessation to relieve withdrawal symptoms. Nicotine acts as a receptor agonist at most nicotinic acetylcholine receptors (nAChRs), except at two nicotinic receptor subunits (nAChRα9 and nAChRα10) where it acts as a receptor antagonist. | |||
T76116 | L-Lactate dehydrogenase | ||
L-Lactate dehydrogenase (L-乳酸脱氢酶) 是一种氧化还原酶。L-Lactate dehydrogenase 在体内催化 NADH 将丙酮酸还原为 L-乳酸。 | |||
T76146 | D-Lactate dehydrogenase | ||
D-Lactate dehydrogenase(D-LDH)为一种氧化还原酶,以NAD+或NADP+作为受体,特异性作用于供体的CH-OH基团,催化D-乳酸氧化成丙酮酸。该酶主要分布于细菌和真菌中,是生化研究中常用的酶。 | |||
T15435 |
GSK2837808A
|
Dehydrogenase | Metabolism |
GSK2837808A 是一种选择性的乳酸脱氢酶A 抑制剂,对 hLDHA (IC50:2.6 nM) 和 hLDHB (IC50:43 nM)。 | |||
T22336 |
Galloflavin
|
Dehydrogenase | Metabolism |
Galloflavin 是乳酸脱氢酶抑制剂。用 Pyruvate 法得到的 Ki 为 5.46 µM (LDH-A) 以及15.06 µM (LDH-B)。它能够阻断 ATP 的生成和糖酵解,从而抑制癌细胞的增殖。 | |||
T11829 |
LDH-IN-1
|
Dehydrogenase | Metabolism |
LDH-IN-1 是新型的基于吡唑的人乳酸脱氢酶抑制剂,对于 LDHA 和 LDHB 的 IC50 分别为32和27 nM。 | |||
T4295 |
(R)-GNE-140
GNE-140 |
Dehydrogenase | Metabolism |
(R)-GNE-140 (GNE-140) 是 LDHA 抑制剂,能够作用于 LDHA (IC50:3 nM) 和 LDHB (IC50:3 nM)。它的活性是 S 型异构体的 18 倍。 | |||
T1768 |
7ACC2
|
Mitochondrial Metabolism; Monocarboxylate transporter | Membrane transporter/Ion channel; Metabolism |
7ACC2 是单羧酸盐转运蛋白抑制剂,IC50为 11 nM。它还是线粒体丙酮酸转运的有效抑制剂,可抑制乳酸涌入,通过抑制乳酸通量来发挥抗癌作用。 | |||
T11546 |
hDHODH-IN-1
|
Dehydrogenase | Metabolism |
hDHODH-IN-1 是有效的人二氢乳清酸脱氢酶抑制剂, 显示出抗炎作用。 | |||
T3105 |
PFK-158
|
Apoptosis; Glucokinase; Autophagy | Apoptosis; Autophagy; Metabolism |
PFK158 是一种选择性的PFKFB3抑制剂,IC50值为 137 nM。它可减少癌细胞中葡萄糖的摄取,ATP 的产生,乳酸的释放,并诱导细胞凋亡和自噬。它还可以增强 Colistin 对细菌的抵抗力,具有广泛的抗肿瘤活性。 | |||
T12438 |
PfDHODH-IN-1
|
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
PfDHODH-IN-1 是 Leflunomide 活性代谢物的类似物,具有抗疟疾活性。它是恶性疟原虫二氢乳清酸脱氢酶抑制剂。 | |||
T7482 |
3-chloro-5-hydroxybenzoic Acid
|
GPR | Endocrinology/Hormones; GPCR/G Protein |
3-Chloro-5-hydroxybenzoic acid 是一种口服具有活力的乳酸受体GPR81选择性激动剂,对人 GPR81 的EC50为 16 μM。肥胖小鼠模型中,它表现出良好的体内脂肪分解作用。 | |||
T3175 |
LDHA-IN-4
AZ 33,AZ-33,LDHA Inhibitor,AZ33 |
Dehydrogenase | Metabolism |
LDHA-IN-4 (AZ33) 是乳酸脱氢酶 A 选择性抑制剂,IC50=0.5 μM,Kd=0.093 μM。 | |||
T5325 |
Nifurtimox
硝呋替莫,BAY-2502,BAY-A-2502 |
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
Nifurtimox (BAY-A-2502) 是一种用于锥虫病的抗虫剂,可影响乳酸脱氢酶活性。它有潜力研究神经母细胞瘤细胞。 | |||
T0239 |
Lonidamine
AF1890,氯尼达明,DICA,Diclondazolic Acid |
Apoptosis; Hexokinase; Mitochondrial Metabolism | Apoptosis; Metabolism |
Lonidamine (Diclondazolic Acid) 是一种抗肿瘤药物,是己糖激酶、线粒体丙酮酸载体和质膜单羧酸转运蛋白抑制剂,同时也抑制线粒体复合物 II。 | |||
T7460 |
α-Cyano-4-hydroxycinnamic acid
α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基 |
Monocarboxylate transporter | Membrane transporter/Ion channel |
α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) 是非竞争性单羧酸盐转运蛋白 (MCTs) 抑制剂,可抑制线粒体丙酮酸转运蛋白,Ki 值为 6.3 μM。它可作为基质辅助激光解吸电离-飞行时间质谱 (MALDI-TOF) 分析的基质,可以促进肽离子化。 | |||
T72324 | Lagociclovir valactate | ||
Lagociclovir valactate 是 Lagociclovir 的前药。Lagociclovir valactate 是一种具有口服活性的抗HBV 试剂。 | |||
T5845 |
7ACC1
DEAC,香豆素D1421,Coumarin D 1421,7-(二乙胺基)-2-氧代-2-苯并吡喃-3-羧酸,7-(Diethylamino)coumarin-3-carboxylic acid,D 1421 |
Monocarboxylate transporter | Membrane transporter/Ion channel |
7ACC1 (D 142) 抑制表达MCT1和MCT4肿瘤细胞的乳酸涌入,能选择性干扰肿瘤微环境乳酸通量。 | |||
T60165 |
VB124
|
Monocarboxylate transporter | Membrane transporter/Ion channel |
VB124 是一种具有口服活性的、有效且选择性的MCT4抑制剂。VB124 可特异性抑制 MDA-MB-231 细胞中乳酸的涌入和流出,IC50分别为 8.6 nM 和 19 nM。VB124 对 MCT4 的选择性高于 MCT1。VB124可用于心脏肥大、心力衰竭和代谢的研究。 | |||
T64345 |
4-(Dimethylamino)phenol
|
Others | Others |
4-(Dimethylamino)phenol enhances extracellular lactate dehydrogenase (LDH) levels without significant effects on gluconeogenesis. Only when the membrane becomes permeable to LDH does 4-(Dimethylamino)phenol reduce ATP content. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5220 |
D-(-)-Lactic acid sodium
Sodium D-lactate,D-乳酸钠 |
Others; Endogenous Metabolite | Metabolism; Others |
D-(-)-Lactic acid sodium (Sodium D-lactate) 是一种有机酸。它是一种手性分子,由 L-乳酸和 D-乳酸两种光学异构体组成,其中 L-异构体在生物体中最常见。D-(-)-Lactic acid sodium 也是一种微生物代谢产物。 | |||
T20574 |
Magnesium lactate
Bis(lactato)magnesium |
||
Magnesium lactate is a magnesium donor and buffering agent. | |||
T12996 |
Squalamine lactate
MSI-1256F |
Others | Others |
Squalamine lactate is an aminosterol compound discovered in the tissues of the dogfish shark, with antimicrobial activity. | |||
T5705 |
Glomeratose A
|
Dehydrogenase | Metabolism |
Glomeratose A 是分离自远志Polygala tenuifolia 中,是一种乳酸脱氢酶lactate dehydrogenase 抑制剂。 | |||
TN2252 |
Syrosingopine
|
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Syrosingopine 是 MCT1和 MCT4双重抑制剂,对 MCT4 的效力高 60 倍,可防止乳酸和 H+ 流出。它是可口服抗高血压药物,联合二甲双胍具有研究癌症疾病的潜力。 | |||
T7964 |
Isomalt
异麦芽酮糖醇,Palatinitol,Palatinit |
Others; Dehydrogenase | Metabolism; Others |
Isomalt (Palatinitol) 是无毒的、具有良好耐受性的多元醇和蛋白质稳定的赋形剂,在冷冻干燥过程中可适度稳定乳酸脱氢酶(LDH),并在储存期间表现更好。它传统上在食品工业中用作甜味剂,也在制药中用作压片赋形剂。 | |||
T5S0620 |
3-Dehydrotrametenolic acid
Dehydrotrametenolic acid,松苓新酸,3-氢化去氢松苓酸 |
Apoptosis; Others; Dehydrogenase | Apoptosis; Metabolism; Others |
3-Dehydrotrametenolic acid 是从茯苓菌核分离的一种乳酸脱氢酶抑制剂,可诱导细胞凋亡,具有抗癌活性。它促进体外脂肪细胞分化,在体内起胰岛素增敏剂的作用。 | |||
TN4021 | Ethyl p-hydroxyphenyllactate | Others | Others |
Ethyl p-hydroxyphenyllactate是一种天然产物,属于菊科还羊参属,其产品编号为 TN4021,CAS号为 62517-34-4。Ethyl p-hydroxyphenyllactate可用作对照参考。 | |||
TN4552 |
Methyl p-hydroxyphenyllactate
|
Others | Others |
Methyl para-hydroxyphenyllactate(MeHPLA) can suppress the cellular proliferation of estrogen-sensitive MCF-7 breast cancer cells in vitro and to suppress the growth of rat uteri in vivo, high affinity of MeHPLA for the type II estrogen binding site (EBS) | |||
TN1829 |
Kakkalide
|
Dehydrogenase | Metabolism |
Kakkalide 是提取自葛根花中的一种异黄酮。它可以抑制活性氧相关炎症,并改善内皮细胞胰岛素抵抗作用。 | |||
T5S2195 |
Sibiricose A5
西伯利亚远志糖A5 |
Dehydrogenase | Metabolism |
Sibiricose A5 是一种寡糖酯,分离自Polygalae Radix,具有抗氧化作用。 | |||
T2S2211 |
Tenuifoliside C
|
Dehydrogenase | Metabolism |
Tenuifoliside C 是从野生的 polygala tenuifolia 中分离得到的。它对 CYP2E1 催化氯唑酮 6-羟基化反应具有抑制作用。 | |||
T4738 |
Sodium 2-hydroxybutanoate
2-Hydroxybutyric acid sodium salt,2-羟基丁酸钠,DL-2-Hydroxybutyric Acid Sodium Salt,alpha-hydroxybutyrate,SODIUM 2-HYDROXYBUTYRATE |
Others; Endogenous Metabolite | Metabolism; Others |
Sodium 2-hydroxybutanoate (alpha-hydroxybutyrate) 是内源性代谢产物的一种。 | |||
T5702 |
Tenuifoliside B
|
Dehydrogenase | Metabolism |
Tenuifoliside B 是一种分离自Polygalae Radix 中的成分,能够抑制氰化钾引起的缺氧和东莨菪碱引起的记忆障碍。它有成为 AD 先导化合物的潜力。它具有潜在的认知改善和脑保护作用。 | |||
TN1182 |
11-Keto-beta-boswellic acid
11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸 |
Leukotriene Receptor; NF-κB; Lipoxygenase | GPCR/G Protein; Metabolism; NF-κB |
11-Keto-beta-boswellic acid 是来自乳香的一种五环三萜酸,具有抗炎活性和剂量依赖性心脏保护作用,主要是由于抑制5-脂氧合酶、白三烯、NF-κB 的激活和肿瘤坏死因子 α 的产生。 | |||
T5290 |
(S)-2-Hydroxy-3-phenylpropanoic acid
L-(−)-3-Phenyllactic acid,L-3-苯乳酸 |
Others; Endogenous Metabolite | Metabolism; Others |
(S)-2-Hydroxy-3-phenylpropanoic acid (L-(−)-3-Phenyllactic acid) 是苯丙氨酸的代谢产物。苯丙酮尿症患者体液中苯丙氨酸的水平升高。 | |||
TN6945 |
Lactic acid
2-hydroxypropanoic acid |
Others | Others |
Lactic acid (2-hydroxypropanoic acid) 是糖酵解的产物,广泛存在与自然界中。Lactate acid 在体内收缩骨骼肌缺氧时会产生,可在完全有氧条件下被去除。Lactic acid 可作为危重病人的血流动力学指标。Lactic acid 具有抗肿瘤活性。 | |||
T13922 |
Thevetiaflavone
2-Genistein-5-methyl ether,Apigenin-5-methyl ether |
BCL; Caspase | Apoptosis; Proteases/Proteasome |
Thevetiaflavone (2-Genistein-5-methyl ether) 是一种来自 Wikstroemia indica 的天然类黄酮,可抑制乳酸脱氢酶从细胞质中泄漏并提高细胞活力。 | |||
T83725 |
Nigerose
Sakebiose |
||
Nigerose,一种在Acremonium中发现的二糖,当与苷类化合物salidroside联合使用,浓度为150 µM时,可阻止HL-60细胞冷冻保存后的丙二醛(MDA)和活性氧物质(ROS)水平上升,并抑制乳酸脱氢酶(LDH)的释放。 |