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抑制剂 & 化合物

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重组蛋白

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Cat. No. Product Name
L3500 组蛋白修饰化合物库

469 compounds
469 个组蛋白修饰相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
L2140 癌细胞分化化合物库

406 compounds
406 个诱导肿瘤细胞分化化合物的独特集合,可用于高通量筛选和高内涵筛选;
L2630 神经元分化化合物库

672 compounds
672 种与神经元分化相关的化合物,可以用于神经系统疾病药物研发
L8000 干细胞分化化合物库

1197 compounds
1197 种干细胞分化信号通路相关的生物活性小分子化合物的特有集合,可用于高通量、高内涵筛选;
L8300 染色质修饰分子库

250 compounds
250 种染色质化学修饰相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;

化合物库

组蛋白修饰化合物库
Cat.No: L3500
Compounds: 469
癌细胞分化化合物库
Cat.No: L2140
Compounds: 406
神经元分化化合物库
Cat.No: L2630
Compounds: 672
干细胞分化化合物库
Cat.No: L8000
Compounds: 1197
染色质修饰分子库
Cat.No: L8300
Compounds: 250
Cat. No. Product Name Target Signaling Pathways
T60485 DIF-3

DIF-3 is a chemical compound that acts by activating GSK-3β to facilitate the degradation of cyclin D1 and c-Myc, resulting in reduced expression levels of these proteins. In addition, DIF-3 inhibits Wnt/β-catenin signaling pathway-related proteins in DLD-1 cells. This compound exerts a potent antiproliferative effect on the HeLa human cervical cancer cell line by inducing cyclin D1 degradation and inhibiting cyclin D1 mRNA expression [1].
T65468 Boc-Phe(3,4-DiF)-OH

Boc-Phe(3,4-DiF)-OH 是一种氨基酸衍生物,在生命科学相关研究中具有广泛的应用。
T65836 Fmoc-Phe(3,4-DiF)-OH

Fmoc-Phe(3,4-DiF)-OH 是一种氨基酸衍生物,在生命科学相关研究中具有广泛的应用。
T65467 Boc-D-Phe(3,4-DiF)-OH

Boc-D-Phe(3,4-DiF)-OH 是一种氨基酸衍生物,在生命科学相关研究中具有广泛的应用。
TP2485 difelikefalin acetate(1024828-77-0 Free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
difelikefalin acetate 是酮体和砌块。
TP2501 Difelikefalin acetate

Difelikefalin acetate(1024828-77-0 free base),CR 845 acetate,Difelikefalin醋酸盐,FE 202845 acetate

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Difelikefalin acetate (CR 845 acetate) 是一种外周受限的 kappa 阿片受体激动剂。CR845 表现出低 P450 CYP 抑制和对大脑的低渗透性。
T9049 Difurazon hydrochloride

Others Others
Difurazon hydrochloride 是一种致突变药物。它可能已用于治疗细菌性痢疾。它是动物饲料中的抗菌促生长剂。
T7088 Diflubenzuron

Dimilin,氟脲杀,Difubenzuron,Larvakil,Difluron

P450 Metabolism
Diflubenzuron (Larvakil) 是杀虫剂 Dimilin 的有效成分,具有杀幼虫和杀卵作用。
TNU0187 2',5-Difluoro-2'-deoxy-1-arabinosyluracil

2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
2',5-Difluoro-2'-deoxy-1-arabinosyluracil (2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine) 是一种尿嘧啶核苷类似物,具有潜在的抗癫痫活性和降压活性,可用于研究抗惊厥和焦虑症。
T3532 5S rRNA modificator

FAI,Furoyl Acylimidazole

Others Others
5S rRNA modificator (FAI) 是一种结构化 RNA 分子上 2'-羟基酰化的合适亲电试剂,产生与现有探针相当的精确结构信息。它可用于 5S rRNA RNA 修饰。
T8844 Diflapolin

Others; FLAP; Epoxide Hydrolase Immunology/Inflammation; Metabolism; Others
Diflapolin 是高活性的双 5-脂氧合酶激活蛋白(FLAP)/可溶性环氧化物水解酶抑制剂,具有显著的抗炎作用和较高的靶向选择性。它抑制分离的 sEH 的活性,IC50为20 nM。它还抑制完整人单核细胞和中性粒细胞中 5-LOX 产物的形成,IC50分别为 30 和 170 nM。
T13111 Tegadifur

40497S,FD 1

Others Others
Tegadifur (40497S) 是一种可口服的抗肿瘤化合物,具有抗新陈代谢作用,常与尿嘧啶林和治疗直肠腺癌。
T64789 ((3S,5R)-5-((1H-1,2,4-Triazol-1-yl)methyl)-5-(2,4-difluorophenyl)tetrahydrofuran-3-yl)methyl 4-methylbenzenesulfonate

Others Others
((3S,5R)-5-((1H-1,2,4-Triazol-1-yl)methyl)-5-(2,4-difluorophenyl)tetrahydrofuran-3-yl)methyl 4-methylbenzenesulfonate 是一种医药中间体,可用于合成具有抗癌活性的泊沙康唑。
T31458 DiFMUP

6,8-Difluoro-4-methylumbelliferyl phosphate

DiFMUP (6,8-Difluoro-4-methylumbelliferyl phosphate) 是一种荧光底物,抑制蛋白酪氨酸磷酸酶(PTPs),可用于检测苏氨酸磷酸酶的活性。
T1466 Nadifloxacin

OPC7251,那氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Nadifloxacin (OPC7251) 是一种对粉刺有效的广谱氟喹诺酮类抗生素。
T6472 Difluprednate

Myser,Epitopic,二氟孕甾丁酯,CM 9155

Others Others
Difluprednate (Myser) 是一种可用于术后眼睛疼痛和炎症的皮质类固醇。
T2548 Diflorasone

Glucocorticoid Receptor Endocrinology/Hormones
Diflorasone 是一种皮质类固醇激素受体激动剂,具有抗炎和免疫抑制作用。它可通过细胞膜扩散进入细胞,并与细胞质中的糖皮质激素受体结合。它用于研究湿疹、牛皮癣等皮肤病。
T9354 2,4-Difluorobenzaldehyde

2,4-Difluoro-benzaldehyde,2,4-二氟苯甲醛

Others Others
2,4-Difluorobenzaldehyde 靶点-A 型肉毒杆菌神经毒素(肉毒杆菌)。
T60162 1H-Pyrazole-5-carboxamide, 4-(5-chloro-2-furanyl)-1,3-bis(2,4-difluorophenyl)-4,5-dihydro-5-methyl-N-[(4-methyl-2-morpholinyl)methyl]

Others Others
1H-Pyrazole-5-carboxamide, 4-(5-chloro-2-furanyl)-1,3-bis(2,4-difluorophenyl)-4,5-dihydro-5-methyl-N-[(4-methyl-2-morpholinyl)methyl]是一种抗纤维化的化合物。
T8751 AZD8931 diFuMaric acid

4-[[4-[(3-氯-2-氟苯基)氨基]-7-甲氧基-6-喹唑啉基]氧基]-N-甲基-1-哌啶乙酰胺二富马酸盐

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
AZD8931 diFuMaric acid 是一种可逆的 ATP 竞争性 EGFR、ErbB2 和 ErbB3 抑制剂(IC50 分别为 4 nM、3 nM 和 4 nM)。
T20103 Isoxadifen-ethyl

Isoxadifen-ethyl

Others Others
Isoxadifen-ethyl 是除草剂安全剂和农用化学品。 Isoxadifen-ethyl 可有效减轻烟嘧磺隆对玉米的损伤。
T20833 Diflufenzopyr

SAN-835H,SAN835H,SAN 835H

Others Others
Diflufenzopyr (SAN 835H) 是一种生长素转运抑制剂,属于缩氨基脲类。
T0808 Diflunisal

Flovacil,二氟尼柳,Dolobid,MK-647,Fluniget,Dolobis

Epigenetic Reader Domain; COX Chromatin/Epigenetic; Immunology/Inflammation; Neuroscience
Diflunisal (Dolobid) 是一种水杨酸盐衍生物,是环氧合酶的抑制剂,具有非甾体抗炎和尿酸舒缓性能,可单独用作止痛剂和类风湿关节炎患者。
T67291 2′,2′-Difluorodeoxyuridine

dFdU,2',2'-Difluoro-2'-deoxyuridine

Drug Metabolite Metabolism
2′,2′-Difluorodeoxyuridine (dFdU) 是 Gemcitabine 的主要代谢产物。2′,2′-Difluorodeoxyuridine 具有抗癌和抗肿瘤活性,在低氧条件下的显示出放射增敏作用,可用于研究胰腺癌。
T21012 Diflufenican

M&B 38544,吡氟草胺

Others Others
Diflufenican (M&B 38544) 是一种选择性除草剂,用于专门防治某些阔叶杂草。
T1597 Proadifen hydrochloride

U-5446,RP-5171,SKF-525A,盐酸丙基解痉素

P450 Metabolism
Proadifen hydrochloride (RP-5171) 是细胞色素 P450抑制剂,它的 IC50值为19μM。
T67826 Alalevonadifloxacin

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Alalevonadifloxacin 是一种DNA 回旋酶和DNA 拓扑异构酶抑制剂,是一种喹诺酮类针对Mrsa 的新型抗菌化合物。Alalevonadifloxacin 对治疗细菌性革兰氏阳性、革兰氏阴性和厌氧性感染有潜在作用。
T24444 Medifoxamine

LG 152,Medifoxamina,LG-152,LG152

Dopamine Receptor; Monoamine Oxidase GPCR/G Protein; Neuroscience
Medifoxamine (LG 152) 是一种选择性非单胺氧化酶抑制剂,通过对5 HT 再摄取的抑制展现其抗抑郁活性。Medifoxamine 优先抑制多巴胺再摄取 (dopamine reuptake)。
T50062 2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide

PDE Metabolism
2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide 是一种 PDE 抑制剂。
T50030 1-(2,4-difluorophenyl)guanidine hydrochloride

Others Others
1-(2,4-difluorophenyl)guanidine hydrochloride 是一种化合物,是电压门控钠通道Nav1.7的强效选择性抑制剂,Nav1.7是疼痛信号传输的关键参与者,因此它能够减少疼痛信号的传递,从而产生镇痛作用。
T35449 α-(difluoromethyl)-DL-Arginine

DFMA,RMI 71897,α-(difluoromethyl)-DL-Arginine

Others Others
α-(difluoromethyl)-DL-Arginine (RMI 71897) 是一种酶激活的、不可逆的大肠杆菌(Ki = 800 μM)、铜绿假单胞菌和肺炎克雷伯菌精氨酸脱羧酶抑制剂。在0.01 mM 时,它已被证明可以防止渗透胁迫诱导的燕麦叶片细胞精氨酸脱羧酶活性和腐胺合成的增加。当α-(difluoromethyl)-DL-Arginine 与多种多胺类似物联用时,能在10 mM 的最低浓度下抑制克氏锥虫在哺乳动物宿主细胞中的生长,并在T 细胞受体α缺陷小鼠模型中阻止小锥虫的生长。
T27172 Difamilast

PDE Metabolism
Difamilast 是局部的、选择性的非甾体磷酸二酯酶 4 抑制剂,对 B 亚型抑制作用较好 (IC50=11.2 nM)。它在研究轻度至中度特应性皮炎方面有研究的价值。
T8142 Difloxacin hydrochloride

Difloxacin HCl,盐酸二氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Difloxacin hydrochloride (Difloxacin HCl) 是一种广谱抗菌药物。它干扰 DNA 促旋酶和拓扑异构酶 IV 的活性,抑制细菌 DNA 促旋酶并显示出浓度依赖性的杀菌作用。
T5000 Diflucortolone valerate

Afusona,戊酸双氟可龙,Diflucortolone 21-valerate

Others; Antibacterial; Antifungal Microbiology/Virology; Others
Diflucortolone valerate (Diflucortolone 21-valerate) 是一种强效皮质类固醇,可研究各种皮肤疾病。
T21192 Diflorasone Diacetate

Apexicon E,Psorcon,Maxiflor,醋酸双氟拉松,Florone E

Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.
T66604 4-(Difluoromethoxy)-2-nitroaniline

4-(Difluoromethoxy)-2-nitroaniline 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66604,CAS号为 97963-76-3。
T30064 Aniline, m-chloro-N-(2,2-difluoroethyl)-

Aniline, m-chloro-N-(2,2-difluoroethyl)- is a bioactive chemical.
T66553 2-(((3aR,4S,6R,6aS)-6-(7-(((1R,2S)-2-(3,4-Difluorophenyl)cyclopropyl)amino)-5-(propylthio)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl)oxy)ethanol

2-(((3aR,4S,6R,6aS)-6-(7-(((1R,2S)-2-(3,4-Difluorophenyl)cyclopropyl)amino)-5-(propylthio)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl)oxy)ethanol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66553,CAS号为 274693-26-4。
T65424 (S)-(-)-9,10-Difluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyrido-[1,2,3-de]-1,4-benzoxazine-6-carboxylic acid

(S)-(-)-9,10-Difluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyrido-[1,2,3-de]-1,4-benzoxazine-6-carboxylic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65424,CAS号为 100986-89-8。
TNU0305 5-Difluoromethyluridine

Nucleoside Derivatives - 5-Modified pyrimidine nucleosides; Fluoro-modified nucleosides
T66603 4-(Difluoromethoxy)benzene-1,2-diamine

4-(Difluoromethoxy)benzene-1,2-diamine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66603,CAS号为 172282-50-7。
T67102 1-(4-(2,4-Difluorobenzoyl)piperidin-1-yl)ethanone

1-(4-(2,4-Difluorobenzoyl)piperidin-1-yl)ethanone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67102,CAS号为 84162-82-3。
T38419 Difelikefalin

CR-845,FE-202845

Difelikefalin (CR-845; FE-202845) is a peripherally restricted, selective agonist of the kappa opioid receptor (KOR). It exhibits anti-inflammatory properties and holds promise for modulating pruritus in conditions associated with chronic kidney disease.
T65469 N-Boc-3,5-difluoro-L-phenylalanine

N-Boc-3,5-difluoro-L-phenylalanine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65469,CAS号为 205445-52-9。
T71543 Difethialone

Difethialone is an anticoagulant rodenticide and a vitamin K antagonist.
T36822 Benzovindiflupyr

Benzovindiflupyr is a fungicide.1It inhibits mitochondrial complex II, also known as succinate dehydrogenase (SDH; IC50= 5.2 nM), and mycelial growth ofS. sclerotiorum(EC50= 0.011 μg/ml). Benzovindiflupyr (60 μg/ml) completely protects eggplant leaves fromS. sclerotioruminfection. Formulations containing benzovindiflupyr have been used to control various fungal diseases in agriculture. 1.Gao, Y., He, L., Zhu, J., et al.The relationship between features enabling SDHI fungicide binding to the Sc-S...
T33289 Meproadifen

Meproadifen enhances activation and desensitization of the acetylcholine receptor-ionic channel complex (AChR).
T66337 1-Cyclopropyl-6,8-difluoro-7-((4aS,7aS)-hexahydro-1H-pyrrolo[3,4-b]pyridin-6(2H)-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid

1-Cyclopropyl-6,8-difluoro-7-((4aS,7aS)-hexahydro-1H-pyrrolo[3,4-b]pyridin-6(2H)-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66337,CAS号为 151213-15-9。
T39363 2,4-Difluororesorcinol

2,4-Difluororesorcinol is a fluorinated building block.
T66697 (R)-3-((tert-Butoxycarbonyl)amino)-4-(2,4-difluorophenyl)butanoic acid

(R)-3-((tert-Butoxycarbonyl)amino)-4-(2,4-difluorophenyl)butanoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66697,CAS号为 851307-12-5。

化合物

DIF-3
Cat.No: T60485
Synonym:
Target:
Boc-Phe(3,4-DiF)-OH
Cat.No: T65468
Synonym:
Target:
Fmoc-Phe(3,4-DiF)-OH
Cat.No: T65836
Synonym:
Target:
Boc-D-Phe(3,4-DiF)-OH
Cat.No: T65467
Synonym:
Target:
difelikefalin acetate(1024828-77-0 Free base)
Cat.No: TP2485
Synonym:
Target: Opioid Receptor
Difelikefalin acetate
Cat.No: TP2501
Synonym: Difelikefalin acetate(1024828-77-0 free base),CR 845 acetate,Difelikefalin醋酸盐,FE 202845 acetate
Target: Opioid Receptor
Difurazon hydrochloride
Cat.No: T9049
Synonym:
Target: Others
Diflubenzuron
Cat.No: T7088
Synonym: Dimilin,氟脲杀,Difubenzuron,Larvakil,Difluron
Target: P450
2',5-Difluoro-2'-deoxy-1-arabinosyluracil
Cat.No: TNU0187
Synonym: 2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine
Target: Nucleoside Antimetabolite/Analog
5S rRNA modificator
Cat.No: T3532
Synonym: FAI,Furoyl Acylimidazole
Target: Others
Diflapolin
Cat.No: T8844
Synonym:
Target: Others, FLAP, Epoxide Hydrolase
Tegadifur
Cat.No: T13111
Synonym: 40497S,FD 1
Target: Others
((3S,5R)-5-((1H-1,2,4-Triazol-1-yl)methyl)-5-(2,4-difluorophenyl)tetrahydrofuran-3-yl)methyl 4-methylbenzenesulfonate
Cat.No: T64789
Synonym:
Target: Others
DiFMUP
Cat.No: T31458
Synonym: 6,8-Difluoro-4-methylumbelliferyl phosphate
Target:
Nadifloxacin
Cat.No: T1466
Synonym: OPC7251,那氟沙星
Target: Antibacterial, Antibiotic
Difluprednate
Cat.No: T6472
Synonym: Myser,Epitopic,二氟孕甾丁酯,CM 9155
Target: Others
Diflorasone
Cat.No: T2548
Synonym:
Target: Glucocorticoid Receptor
2,4-Difluorobenzaldehyde
Cat.No: T9354
Synonym: 2,4-Difluoro-benzaldehyde,2,4-二氟苯甲醛
Target: Others
1H-Pyrazole-5-carboxamide, 4-(5-chloro-2-furanyl)-1,3-bis(2,4-difluorophenyl)-4,5-dihydro-5-methyl-N-[(4-methyl-2-morpholinyl)methyl]
Cat.No: T60162
Synonym:
Target: Others
AZD8931 diFuMaric acid
Cat.No: T8751
Synonym: 4-[[4-[(3-氯-2-氟苯基)氨基]-7-甲氧基-6-喹唑啉基]氧基]-N-甲基-1-哌啶乙酰胺二富马酸盐
Target: EGFR
Isoxadifen-ethyl
Cat.No: T20103
Synonym: Isoxadifen-ethyl
Target: Others
Diflufenzopyr
Cat.No: T20833
Synonym: SAN-835H,SAN835H,SAN 835H
Target: Others
Diflunisal
Cat.No: T0808
Synonym: Flovacil,二氟尼柳,Dolobid,MK-647,Fluniget,Dolobis
Target: Epigenetic Reader Domain, COX
2′,2′-Difluorodeoxyuridine
Cat.No: T67291
Synonym: dFdU,2',2'-Difluoro-2'-deoxyuridine
Target: Drug Metabolite
Diflufenican
Cat.No: T21012
Synonym: M&B 38544,吡氟草胺
Target: Others
Proadifen hydrochloride
Cat.No: T1597
Synonym: U-5446,RP-5171,SKF-525A,盐酸丙基解痉素
Target: P450
Alalevonadifloxacin
Cat.No: T67826
Synonym:
Target: DNA gyrase, Topoisomerase, Antibacterial
Medifoxamine
Cat.No: T24444
Synonym: LG 152,Medifoxamina,LG-152,LG152
Target: Dopamine Receptor, Monoamine Oxidase
2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide
Cat.No: T50062
Synonym:
Target: PDE
1-(2,4-difluorophenyl)guanidine hydrochloride
Cat.No: T50030
Synonym:
Target: Others
α-(difluoromethyl)-DL-Arginine
Cat.No: T35449
Synonym: DFMA,RMI 71897,α-(difluoromethyl)-DL-Arginine
Target: Others
Difamilast
Cat.No: T27172
Synonym:
Target: PDE
Difloxacin hydrochloride
Cat.No: T8142
Synonym: Difloxacin HCl,盐酸二氟沙星
Target: Antibacterial, Antibiotic
Diflucortolone valerate
Cat.No: T5000
Synonym: Afusona,戊酸双氟可龙,Diflucortolone 21-valerate
Target: Others, Antibacterial, Antifungal
Diflorasone Diacetate
Cat.No: T21192
Synonym: Apexicon E,Psorcon,Maxiflor,醋酸双氟拉松,Florone E
Target:
4-(Difluoromethoxy)-2-nitroaniline
Cat.No: T66604
Synonym:
Target:
Aniline, m-chloro-N-(2,2-difluoroethyl)-
Cat.No: T30064
Synonym:
Target:
2-(((3aR,4S,6R,6aS)-6-(7-(((1R,2S)-2-(3,4-Difluorophenyl)cyclopropyl)amino)-5-(propylthio)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl)oxy)ethanol
Cat.No: T66553
Synonym:
Target:
(S)-(-)-9,10-Difluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyrido-[1,2,3-de]-1,4-benzoxazine-6-carboxylic acid
Cat.No: T65424
Synonym:
Target:
5-Difluoromethyluridine
Cat.No: TNU0305
Synonym:
Target:
4-(Difluoromethoxy)benzene-1,2-diamine
Cat.No: T66603
Synonym:
Target:
1-(4-(2,4-Difluorobenzoyl)piperidin-1-yl)ethanone
Cat.No: T67102
Synonym:
Target:
Difelikefalin
Cat.No: T38419
Synonym: CR-845,FE-202845
Target:
N-Boc-3,5-difluoro-L-phenylalanine
Cat.No: T65469
Synonym:
Target:
Difethialone
Cat.No: T71543
Synonym:
Target:
Benzovindiflupyr
Cat.No: T36822
Synonym:
Target:
Meproadifen
Cat.No: T33289
Synonym:
Target:
1-Cyclopropyl-6,8-difluoro-7-((4aS,7aS)-hexahydro-1H-pyrrolo[3,4-b]pyridin-6(2H)-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
Cat.No: T66337
Synonym:
Target:
2,4-Difluororesorcinol
Cat.No: T39363
Synonym:
Target:
(R)-3-((tert-Butoxycarbonyl)amino)-4-(2,4-difluorophenyl)butanoic acid
Cat.No: T66697
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8150 Nudifloramide

1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide,1-甲基-6-氧代吡啶-3-甲酰胺

PARP; Endogenous Metabolite Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Nudifloramide (1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide) 是烟酰胺-腺嘌呤二核苷酸(NAD) 降解的一种最终产物,可显著抑制PARP-1活性。
TN7218 Diformylphloroglucinol

2,4,6-Trihydroxyisophthalaldehyde

Antioxidant oxidation-reduction
Diformylphloroglucinol (2,4,6-Trihydroxyisophthalaldehyde) 是从蓝桉树的叶子中分离出的酰基间苯三酚,是合成具有抗氧化和抗溃疡活性间苯三酚化合物的原料。
T34398 Rotundifuran

Others Others
Rotundifuran 是从 Vitex rotundifolia 的果实中提取的。 Rotundifuran 抑制细胞周期进程并诱导人髓性白血病细胞凋亡。
T3822 Bellidifolin

Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Bellidifolin (Bellidifoline) 是从獐牙菜的茎中提取的一种呫吨酮,它能作为病毒蛋白 R 的抑制剂,具有保肝、降血糖、抗炎、抗氧化、抗肿瘤作用。
TN4163 Grandifloric acid

Others Others
Grandifloric acid是一种天然产物,属于菊科豨莶属,其产品编号为 TN4163,CAS号为 22338-69-8。Grandifloric acid可用作对照参考。
TN4164 Grandifloroside

TNF Apoptosis
Grandifloroside shows good antioxidative and potent anti-inflammatory activities, it also exhibits potent inhibitory activity against TNF-α and 5α-reductase, suggests that it might be developed as a source of potent anti-oxidative and anti-inflammatory ag
T72806 Isobellidifolin

异雏菊叶龙胆酮

Isobellidifolin,一种蒽酮类化合物,同时兼具自由基清除剂和抗氧化功能,亦显示出有效的抗真菌活性。
T79996 N,N′-Diferuloylputrescine

Melanocortin Receptor GPCR/G Protein; Neuroscience
N,N′-Diferuloylputrescine 作为pigmentation的抑制剂,有效减少了57%的色素沉着,并显著降低了MITF蛋白水平。同时,该化合物对活性氧表现出强大的抗氧化活性。
T81961 Lacto-N-difucohexaose I

LDFH I

LNDFH I是一种连接子,它能够将含Lewis b糖链的寡糖有效结合形成水不溶性多糖。
TN4678 Nudifloside D

Others Others
Nudifloside D is a natural product from Jasminum nudiflorum.
TN2605 12alpha-Hydroxygrandiflorenic acid

Others Others
12alpha-Hydroxygrandiflorenic acid是一种天然产物,属于菊科蟛蜞菊属,其产品编号为 TN2605,CAS号为 63768-17-2。12alpha-Hydroxygrandiflorenic acid可用作对照参考。
T82559 Difucosyllacto-N-neohexaose

Difucosyllacto-N-neohexaose 是人乳中分离得到的低聚糖。
T78481 Lactodifucotetraose

2′,3-Difucosyllactose,Difucosyllactose

Lactodifucotetraose (Difucosyllactose),一种四糖,源自人乳。该分子包括D-葡萄糖,D-半乳糖及L-fucose。
T20217 Grandiflorenic acid

Grandiflorenic acid can reproduce the uterine responses induced by aqueous extract of zoapatle leaves. It is suggested that grandiflorenic acid may have an antifertility effect.
T4114 Diffractaic Acid

NSC 5901,地弗地衣酸,NSC 685595

Apoptosis; LTR Apoptosis; Immunology/Inflammation
Diffractaic Acid (NSC 685595) 是松萝的主要成分,具有止痛和解热效果,在各种疾病研究中可作为有效的促凋亡剂。
TN6510 Cordifolioside A

Cordifolioside A possesses immunomodulatory activity, it has a potential in vivo radioprotective effect as well as in vitro cytoprotective activity.
TN4676 Nudifloside B

Others Others
Nudifloside B is a natural product from Jasminum nudiflorum.
TN4677 Nudifloside C

Others Others
Nudifloside C is a natural product from Jasminum nudiflorum.
T81960 Lacto-N-difucohexaose II

LNDFH II,Lacto-N-fucohexaose

Lacto-N-difucohexaose II (LNDFH II) 为人乳中的一种重要低聚糖,对婴儿健康具有显著作用。
TN2602 12-Oxograndiflorenic acid

Others Others
12-Oxograndiflorenic acid 是一种可从凤仙花和土茯苓中提取得到的天然产物,对部分细胞具有细胞毒性。
TN4923 Rubicordifolin

Topoisomerase DNA Damage/DNA Repair
Rubicordifolin exhibits potent cytotoxic and antitumor activities.
T81958 Lacto-N-neodifucohexaose II

LNnDFH II

Lacto-N-neodifucohexaose II(Compd 9),一种关键的人乳四糖衍生物,为点击化学反应试剂。该化合物含 Azide 基团,适用于铜催化叠氮-炔环加成反应(CuAAc),与含 Alkyne 基团的分子反应。同时,它也能与含 DBCO 或 BCN 基团的分子,进行菌株促进的炔-叠氮环加成反应(SPAAC)。
TN2606 12alpha-Methoxygrandiflorenic acid

Others Others
12alpha-Methoxygrandiflorenic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2606,CAS号为 135383-94-7。

天然产物

Nudifloramide
Cat.No: T8150
Synonym: 1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide,1-甲基-6-氧代吡啶-3-甲酰胺
Target: PARP, Endogenous Metabolite
Diformylphloroglucinol
Cat.No: TN7218
Synonym: 2,4,6-Trihydroxyisophthalaldehyde
Target: Antioxidant
Rotundifuran
Cat.No: T34398
Synonym:
Target: Others
Bellidifolin
Cat.No: T3822
Synonym: Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮
Target: Others, HIV Protease
Grandifloric acid
Cat.No: TN4163
Synonym:
Target: Others
Grandifloroside
Cat.No: TN4164
Synonym:
Target: TNF
Isobellidifolin
Cat.No: T72806
Synonym: 异雏菊叶龙胆酮
Target:
N,N′-Diferuloylputrescine
Cat.No: T79996
Synonym:
Target: Melanocortin Receptor
Lacto-N-difucohexaose I
Cat.No: T81961
Synonym: LDFH I
Target:
Nudifloside D
Cat.No: TN4678
Synonym:
Target: Others
12alpha-Hydroxygrandiflorenic acid
Cat.No: TN2605
Synonym:
Target: Others
Difucosyllacto-N-neohexaose
Cat.No: T82559
Synonym:
Target:
Lactodifucotetraose
Cat.No: T78481
Synonym: 2′,3-Difucosyllactose,Difucosyllactose
Target:
Grandiflorenic acid
Cat.No: T20217
Synonym:
Target:
Diffractaic Acid
Cat.No: T4114
Synonym: NSC 5901,地弗地衣酸,NSC 685595
Target: Apoptosis, LTR
Cordifolioside A
Cat.No: TN6510
Synonym:
Target:
Nudifloside B
Cat.No: TN4676
Synonym:
Target: Others
Nudifloside C
Cat.No: TN4677
Synonym:
Target: Others
Lacto-N-difucohexaose II
Cat.No: T81960
Synonym: LNDFH II,Lacto-N-fucohexaose
Target:
12-Oxograndiflorenic acid
Cat.No: TN2602
Synonym:
Target: Others
Rubicordifolin
Cat.No: TN4923
Synonym:
Target: Topoisomerase
Lacto-N-neodifucohexaose II
Cat.No: T81958
Synonym: LNnDFH II
Target:
12alpha-Methoxygrandiflorenic acid
Cat.No: TN2606
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-04146 TNF alpha Protein, Human, Recombinant (hFc)

DIF,TNFA,tumor necrosis factor,TNFSF2,TNF-α,TNF-alp...

Human HEK293 Cells
TNF alpha Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 45.8 kDa and the accession number is P01375.
TMPY-00936 TNF alpha Protein, Human, Recombinant

TNFA,TNFSF2,TNF-alpha,TNF-α,DIF,肿瘤坏死因子,tumor necros...

Human E. coli
TNF alpha Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.5 kDa and the accession number is P01375.
TMPY-01294 TNF alpha Protein, Mouse, Recombinant

TNF-α,Tnfsf1a,TNF-alpha,TNF-a,Tnfa,tumor necrosis factor,TNF...

Mouse E. coli
TNF alpha Protein, Mouse, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.39 kDa and the accession number is P06804.
TMPK-00583 TNF alpha Protein, Ferret, Recombinant (His)

TNF-α,DIF,TNFα,TNF-alpha,TNF α,Cachectin,APC1 prote...

Ferret E. coli
TNF alpha Protein, Ferret, Recombinant (His) is expressed in E. coli expression system with C-His tag. The predicted molecular weight is 18.88 kDa and the accession number is A3FBF1.
TMPY-05237 TNF alpha Protein, Human, Recombinant, Biotinylated

TNFSF2,DIF,TNF-α,tumor necrosis factor,肿瘤坏死因子,TNF-a...

Human E. coli
TNF alpha Protein, Human, Recombinant, Biotinylated is expressed in E. coli expression system. The predicted molecular weight is 17.5 kDa and the accession number is P01375.
TMPY-05187 TNF alpha Protein, Mouse, Recombinant, Biotinylated

Tnfa,TNFSF2,肿瘤坏死因子,Tnfsf1a,TNF-alpha,TNFalpha,DIF,T...

Mouse E. coli
TNF alpha Protein, Mouse, Recombinant, Biotinylated is expressed in E. coli expression system. The predicted molecular weight is 17.4 kDa and the accession number is P06804.
TMPK-00119 TNF alpha Protein, Cynomolgus, Recombinant (His)

TNF α,TNFα,APC1 protein,TNF-alpha,TNFA,TNF-α,TNFATNF,TNFSF1A...

Cynomolgus HEK293 Cells
TNF alpha Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with N-His tag. The predicted molecular weight is 18.35 kDa and the accession number is P79337.
TMPK-00120 TNF alpha Protein, Human, Recombinant (His & Avi)

TNFα,APC1 protein,肿瘤坏死因子,TNFSF2,TNF,TNF α,TNF-alpha,TNF-α,TN...

Human HEK293 Cells
TNF alpha Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 20.3 kDa and the accession number is P01375.
TMPK-00121 TNF alpha Protein, Human, Recombinant (His & Avi), Biotinylated

TNF,TNF-alpha,TNFATNF,DIF,TNFalpha,TNFα,TNFA,TNF-α,...

Human HEK293 Cells
TNF alpha Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 20.3 kDa and the accession number is P01375.
TMPH-00403 Toxin A Protein, Clostridioides difficile, Recombinant (His)

Clostridioides difficile E. coli
Toxin A Protein, Clostridioides difficile, Recombinant (His) is expressed in E. coli.
TMPH-03159 DODA Protein, Portulaca grandiflora, Recombinant (His & Myc & SUMO)

DOPA 4,5-dioxygenase,DODA

Portulaca grandiflora E. coli
Opens the cyclic ring of dihydroxy-phenylalanine (DOPA) between carbons 4 and 5, thus producing an unstable seco-DOPA that rearranges nonenzymatically to betalamic acid. DODA Protein, Portulaca grandiflora, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 49.9 kDa and the accession number is Q7XA48.
TMPH-00416 NAD-GDH Protein, Clostridium difficile, Recombinant (His)

Peptoclostridium difficile E. coli
NAD-GDH Protein, Clostridium difficile, Recombinant (His) is expressed in E. coli.
TMPY-01467 M.viridifaciens NA Protein, M.viridifaciens, Recombinant (His)

NP Protein

M.viridifaciens E. coli
M.viridifaciens NA Protein, M.viridifaciens, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 39.7 kDa and the accession number is Q02834.

重组蛋白

TNF alpha Protein, Human, Recombinant (hFc)
Cat.No: TMPY-04146
Species: Human
Expression System: HEK293 Cells
TNF alpha Protein, Human, Recombinant
Cat.No: TMPY-00936
Species: Human
Expression System: E. coli
TNF alpha Protein, Mouse, Recombinant
Cat.No: TMPY-01294
Species: Mouse
Expression System: E. coli
TNF alpha Protein, Ferret, Recombinant (His)
Cat.No: TMPK-00583
Species: Ferret
Expression System: E. coli
TNF alpha Protein, Human, Recombinant, Biotinylated
Cat.No: TMPY-05237
Species: Human
Expression System: E. coli
TNF alpha Protein, Mouse, Recombinant, Biotinylated
Cat.No: TMPY-05187
Species: Mouse
Expression System: E. coli
TNF alpha Protein, Cynomolgus, Recombinant (His)
Cat.No: TMPK-00119
Species: Cynomolgus
Expression System: HEK293 Cells
TNF alpha Protein, Human, Recombinant (His & Avi)
Cat.No: TMPK-00120
Species: Human
Expression System: HEK293 Cells
TNF alpha Protein, Human, Recombinant (His & Avi), Biotinylated
Cat.No: TMPK-00121
Species: Human
Expression System: HEK293 Cells
Toxin A Protein, Clostridioides difficile, Recombinant (His)
Cat.No: TMPH-00403
Species: Clostridioides difficile
Expression System: E. coli
DODA Protein, Portulaca grandiflora, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03159
Species: Portulaca grandiflora
Expression System: E. coli
NAD-GDH Protein, Clostridium difficile, Recombinant (His)
Cat.No: TMPH-00416
Species: Peptoclostridium difficile
Expression System: E. coli
M.viridifaciens NA Protein, M.viridifaciens, Recombinant (His)
Cat.No: TMPY-01467
Species: M.viridifaciens
Expression System: E. coli
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