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89

抑制剂 & 化合物

18

天然产物

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Cat. No. Product Name Target Signaling Pathways
T10380 AS19

5-HT Receptor GPCR/G Protein; Neuroscience
AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM). AS19 is selective for 5-HT7 over 5-HT1A, 5-HT1B, 5-HT1D, and 5-HT5A receptors (Kis: 89.7 nM, 490 nM, 6.6 nM and 98.5 nM, respectively).
T12205 Ned 19

Calcium Channel Membrane transporter/Ion channel; Metabolism
Ned 19 is a selective membrane-permeant non competitive antagonist of NAADP and strongly inhibits tumor growth and vascularization as well as lung metastases in mice.
T60095 CCF0058981

SARS-CoV Microbiology/Virology
CCF0058981 (CCF981) 是3-氯苯基类似物,是一种非共价 SARS-CoV-2 3CLpro(SC2)抑制剂,IC50为 68 nM。CCF0058981 抑制 SC1 (SARS-CoV-1 3CLpro),IC50为 19 nM。CCF0058981 具有抗病毒功效,具有用于 COVID-19 研究的潜力。
TP1053L Protein Kinase C 19-31 acetate

Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Protein Kinase C 19-31 acetate(121545-65-1 free base) 是一种蛋白激酶 C (PKC) 的肽抑制剂,源自 PKCa 的假底物调节结构域(残基 19-31),在 25 位用丝氨酸取代野生型丙氨酸作为蛋白激酶 C 底物肽,用于测试蛋白激酶 C 活性。
T76781 Itolizumab

EQ-001

Others Others
Itolizumab (Anti-Human CD6 Recombinant Antibody) 是一种人源化针对 CD6 的细胞外 SRCR 远端结构域 1的重组 抗 CD6 单克隆抗体。Itolizumab 可减缓 T 细胞增殖并抑制促炎细胞因子的产生。Itolizumab 可用于研究银屑病、类风湿性关节炎 (RA)和 COVID-19 疾病等多种疾病。
T14366 AZ10606120 dihydrochloride

P2X Receptor Membrane transporter/Ion channel; Neuroscience
AZ10606120 dihydrochloride 是一种可选择的、有效的、高亲和力的受体拮抗剂,在人和大鼠 P2X 7 受体上的 K D 值分别为 1.4 和 19 nM。AZ10606120 dihydrochloride 抑制肿瘤生长,具有抗血管生成活性 。AZ 10606120在与 ATP 结合位点偶联的位点结合时充当负变构调节剂。
T9287 Hydroxychloroquine

2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol,羟氯喹

SARS-CoV; TLR; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology
Hydroxychloroquine (2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol) 是一种合成抗疟疾剂,有效抑制SARS-CoV-2感染,也抑制 Toll 样受体 7/9 信号传导。
T60165 VB124

Monocarboxylate transporter Membrane transporter/Ion channel
VB124 是一种具有口服活性的、有效且选择性的MCT4抑制剂。VB124 可特异性抑制 MDA-MB-231 细胞中乳酸的涌入和流出,IC50分别为 8.6 nM 和 19 nM。VB124 对 MCT4 的选择性高于 MCT1。VB124可用于心脏肥大、心力衰竭和代谢的研究。
T67747 CB2R/FAAH modulator-3

Cannabinoid Receptor; FAAH GPCR/G Protein; Metabolism; Neuroscience
CB2R/FAAH modulator-3 (compound 27) 是一种双重靶点的调节剂,是 CB2R 的激动剂, 也是FAAH 的抑制剂, 作用于 CB2R 和 CB1R 的 Ki 值分别是 20.1 和 67.6 nM,作用于 FAAH 的IC50值为 3.4 μM。CB2R/FAAH modulator-3 可用于癌症、神经退行性疾病中发生的有害炎症级联反应以及 COVID-19 感染相关研究。
T0134 Imiquimod

咪喹莫特,R 837,S-26308

SARS-CoV; TLR; Autophagy; HSV Autophagy; Immunology/Inflammation; Microbiology/Virology
Imiquimod (R 837) 是一种免疫反应修饰剂,可作为 toll 样受体7 激动剂。它有抗病毒和抗肿瘤作用,可研究外生殖器、肛周疣、癌症和 COVID-19
T67745 CB2R/FAAH modulator-2

Cannabinoid Receptor; FAAH GPCR/G Protein; Metabolism; Neuroscience
CB2R/FAAH modulator-2 (compound 26) 是一种双重靶点的调节剂,是 CB2R 的激动剂,也是 FAAH 的抑制剂,作用于 CB2R 和 CB1R 的 Ki 值分别是 10.8 和 152.9 nM,作用于FAAH 的 IC50 值为 6.2 μM。CB2R/FAAH modulator-2 可用于癌症、神经退行性疾病中发生的有害炎症级联反应以及 COVID-19 感染相关研究。
T0825 Ebselen

SPI-1005,PZ-51,依布硒,CCG-39161

Phosphatase; Virus Protease; Calcium Channel; COX; HIV Protease Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ebselen (CCG-39161) 是一种谷胱甘肽过氧化物酶模拟物,是电压依赖性钙通道阻断剂。它抑制Mpro 和COVID-19病毒,是HIV-1衣壳 CTD 二聚化的抑制剂,具有抗炎、抗癌和抗氧化活性。
T39581 PI3K-IN-19 hydrochloride

PI3K-IN-19 hydrochloride

PI3K-IN-19 hydrochloride (WO2017153220, step 5) acts as a phosphatidylinositol-3-kinase (PI3K) inhibitor.
T82166 HSP90-IN-27

HSP Cytoskeletal Signaling; Metabolism
HSP90-IN-27(化合物19)是一种HSP90抑制剂。
T81083 STING agonist-19

STINGagonist-19 用于 ISAC(immune-stimulating antibody conjugates)分子的合成。
TP1529 Galanin (1-19), human

Galanin (1-19), human, represents the fragment encompassing amino acids 1 to 19 of the human galanin neuropeptide. Galanin (GAL) is known for its extensive distribution and multifaceted biological roles, such as regulating hormone secretion, providing antinociceptive effects, and altering feeding behavior.
T63660 Anti-inflammatory agent 19

Anti-inflammatory agent 19 能够抑制 NO (IC50: 36.00 μM)。Anti-inflammatory agent 19 对 HMGB1 诱导的后期炎症反应表现出抑制作用。Anti-inflammatory agent 19 能够用于研究后期炎症疾病,如冠状病毒病 (COVID-19)、败血症等。
T34430 RU 24411

RU24411,RU-24411

RU 24411是一种合成的19-nor 类固醇化合物。在没有葡萄糖的情况下,RU 24411 与醛固酮一样能够刺激钠的转运。
T81732 Myosin light chain kinase fragment 11-19 amide

MLCK(11-19) amide

Myosinlight chain kinase fragment 11-19 amide (MLCK(11-19) amide) 为MLCK专一性多肽抑制剂,具抑制低渗透压刺激下Ca2+入细胞的能力,并可应用于人类宫颈癌研究。
T9931 meplazumab

Others Others
meplazumab 是一种人源化抗 CD147 抗体,作为 COVID-19 肺炎患者的附加疗法。
T82126 ICMT-IN-19

ICMT-IN-19 (compound 53)为一种高效ICMT抑制剂,其半抑制浓度(IC50)为0.026 μM。
T61137 VEGFR-2-IN-19

VEGFR-2-IN-19 (Compound 15b) is a highly efficacious inhibitor of VEGFR2, a receptor involved in angiogenesis. Its mechanism of action involves the induction of cellular apoptosis and elevation of intracellular reactive oxygen species. Due to these properties, VEGFR-2-IN-19 holds promise as an effective anticancer agent [1].
T73596 Guanosine triphosphate

Guanosine triphosphate 是一种天然核苷酸。GTP 衍生物可作为抗 COVID-19 的特异性抑制剂。
T74825 TGR5 agonist 2

TGR5 agonist 2 (compound 19) 是一种有效的 TGR5激动剂,EC50值为 0.27 µM。
T38567 STh

STh, also known as Escherichia coli heat-stable toxin, is a 19 amino acid polypeptide containing three disulfide bridges. It serves as an antigen of significance in the quest for a comprehensive enterotoxigenic Escherichia coli (ETEC) vaccine.
TP1053 Protein Kinase C (19-31)

Protein Kinase C 19-31,PKC (19-31)

Protein Kinase C (19-31), a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate pepti
T36217 19-hydroxy Cholesterol

19-hydroxy Cholesterol is formed during metabolic oxidation of cholesterol. It has been used as an internal standard for the quantitative determination of sterols by mass spectroscopic analysis.[1]
T70601 MDK03855

MDK03855, also known as A2AR antagonist 19, is an adenosine A2A receptor (A2AR) antagonist. MDK03855 has CAS#1454903-85-5. The last five digit of CAS# was used for name.
T82306 Glucagon (22-29)

Glucagon (22-29) 作为Glucagon (19–29)的部分激动剂,能特异性抑制肝质膜 Ca2+泵,其作用机制与腺苷酸环化酶激活无关。
T39412 ACAT-IN-5

ACAT-IN-5 (example 19) is a compound that functions as an inhibitor of acyl-Coenzyme A: cholesterol acyltransferase (ACAT). By inhibiting ACAT, this compound effectively suppresses the transcription mediated by NF-κB.
T76456 Protein Kinase C (19-35) Peptide

Protein Kinase C (19-35) Peptide 是PKC 假底物抑制剂/区域。Protein Kinase C (19-35) Peptide 阻断PKC 激酶结构域的底物结合位点,使PKC 的细胞质形式失活。
TP1052 Protein Kinase C (19-31) (TFA)(121545-65-1,free)

PKC (19-31) (TFA),Protein Kinase C (19-31) (TFA)

Protein Kinase C (19-31) TFA, a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate p
T78770 Garcinone B

Angiotensin-converting Enzyme (ACE) Metabolism
Garcinone B,一种氧杂蒽酮衍生物,为山竹果皮中分离的天然产物,有效抑制ACE2和Mpro,适用于COVID-19研究。
T80691 β-Herpesvirus protease-IN-1

Virus Protease Microbiology/Virology
β-Herpesvirus protease-IN-1 (compound 19)为一种针对β-herpesvirus蛋白酶的抑制剂,其对HCMVPro的IC50值为2.5 μM,而对HHV6Pro的IC50值则为0.33 μM。
T79010 Lp-PLA2-IN-12

Phospholipase Metabolism
Lp-PLA2-IN-12(compound 19)为一种Lp-PLA2抑制剂,主要应用于神经退行性疾病(如AD、青光眼、AMD)及心血管疾病(诸如动脉粥样硬化)的研究。
T82199 HIF-1 alpha (556-574) (TFA)

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
HIF-1 alpha (556-574) TFA 是一种由19个氨基酸组成的缺氧诱导因子-1 (HIF-1) 短肽段,起着调控氧稳态响应的关键作用。
T73372 GNE-2256

GNE-2256 (molecule 19) 是一种具有口服活性的IRAK4(白介素 1 受体关联激酶 4) 抑制剂 (IRAK4Ki=1.4 nM ; IL-6IC50=190 nM)。
T63023 PTP1B-IN-19

PTP1B-IN-19 (Compound 43) 是一种有潜力的选择性苯并咪唑衍生物,能够作为蛋白质酪氨酸磷酸酶 1B (PTP1B) 抑制剂 (Ki: 23.3 μM)。PTP1B-IN-17 能够用于研究 2 型糖尿病。
T76767 Daxdilimab

Daxdilimab 是一种 anti-ILT7单克隆抗体,ILT7 是 pDC 型树突状细胞特有的细胞表面分子。Daxdilimab 可用于 COVID-19 感染的急性肺损伤 (ALI) 的研究。
T76067 Dabcyl-KTSAVLQSGFRKME-Edans TFA

Dabcyl-KTSAVLQSGFRKME-Edans TFA 是一种用于测量蛋白酶酶促活性的荧光肽,具有研究2019-nCoV (COVID-19) 感染潜力的特性。该化合物作为底物,用于相关蛋白酶活性的测定。
T40893 Estrogen receptor modulator 6

Estrogen receptor modulator 6 (compound 3a) is a highly specific and potent agonist of the estrogen receptor (ER) β with a remarkable affinity (K i = 0.44 nM). This compound exhibits an impressive 19-fold selectivity for ERβ over ERα, as evidenced by its affinity (K i = 8.4 nM).
T75116 COVID-19 Spike Protein mRNA-LNP

COVID-19 Spike Protein mRNA-LNP 是一种RNA传递系统,利用脂质纳米粒(LNP)封装COVID-19 Spike Protein mRNA,提高翻译效率与细胞活性。COVID-19 Spike Protein,位于新冠病毒膜表面,负责与宿主细胞受体结合和膜融合,是病毒进入细胞的关键因素,同时也是疫苗设计与宿主中和抗体生成的核心靶点。
T70256 L-163491

L-163491 is a drug which acts as a partial agonist of angiotensin II receptor type 1, and with lower affinity as an agonist of angiotensin II receptor type 2, mimicking the action of angiotensin II. Its practical applications to date have been limited to scientific research into the function of the angiotensin receptor system, but it has been suggested as a potential therapeutic agent for the treatment of inflammation of the lungs associated with certain viral diseases such as COVID-19.
T22091 Imiquimod hydrochloride

Imiquimod hydrochloride (R 837 hydrochloride)是一种免疫反应调节剂,是一种选择性的 toll 样受体 7 (TLR7) 激动剂。Imiquimod hydrochloride 在体内表现出抗病毒和抗肿瘤作用。Imiquimod hydrochloride 可用于外生殖器、肛周疣、癌症和 COVID-19 的研究。
T75102 COVID-19 Spike Protein mRNA(N1-Me-Pseudo UTP)

COVID-19 Spike Protein mRNA 用于表达新型冠状病毒肺炎刺突蛋白,关键于 RNA 传递、翻译效率与细胞活力的检测。该蛋白定位于病毒膜表面,主导病毒与宿主细胞膜受体的结合及膜融合,促使 COVID-19 病毒入侵细胞。同时,它是宿主中和抗体作用的主要位点与疫苗开发的核心靶标。
T63473 Anti-inflammatory agent 18

Anti-inflammatory agent 18 能够抑制NO 的活性 (IC50: 15.94 μM),对 HMGB1 诱导的后期炎症反应具有抑制作用,能够用于研究后期炎症疾病,如冠状病毒病 (COVID-19)、败血症等。
T64273 Nampt-IN-10 TFA

Nampt-IN-10 TFA (compound 4) 是一种磷酸核糖转移酶 (NAMPT) 抑制剂。Nampt-IN-10 TFA 对 A2780 (IC50: 5 nM) 和 CORL23 (IC50: 19 nM) 具有细胞效能。Nampt-IN-10 TFA 能够用做 ADCs 的非抗有丝分裂有效载荷。
T22633 CCT251545 analogue, Compound 51

Others Others
CCT251545 analog is a potent and selective CDK8/19 inhibitor (IC50: 5.1 nM and 5.6 nM, respectively). Mediator complex-associated kinases CDK8 and CDK19 are involved in the regulation of multiple transcription pathways. CDK8 plays as an oncogene in gastri
T36885 BMSpep-57 hydrochloride

BMSpep-57 hydrochloride, a potent macrocyclic peptide, competitively inhibits PD-1/PD-L1 interaction, exhibiting an IC50 value of 7.68 nM. It binds to PD-L1 with dissociation constants (Kds) of 19 nM and 19.88 nM as determined by MST and SPR assays, respectively. This compound enhances T cell functionality by promoting IL-2 production in PBMCs[1].
T76008 Protein Kinase C (19-31) (TFA)

Protein Kinase C (19-31) TFA 是蛋白激酶 C (PKC)的抑制剂,是由 PKCa (残基 19-31) 伪底物调控域衍生而来,25 位丝氨酸取代野生型丙氨酸作为蛋白激酶 C 底物肽,用于检测蛋白激酶 C 的活性。Protein kinase C (PKC) TFA 通过磷酸化丝氨酸和苏氨酸氨基酸残基上的羟基来调控其它蛋白的功能。

化合物

AS19
Cat.No: T10380
Synonym:
Target: 5-HT Receptor
Ned 19
Cat.No: T12205
Synonym:
Target: Calcium Channel
CCF0058981
Cat.No: T60095
Synonym:
Target: SARS-CoV
Protein Kinase C 19-31 acetate
Cat.No: TP1053L
Synonym: Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate
Target: PKC
Itolizumab
Cat.No: T76781
Synonym: EQ-001
Target: Others
AZ10606120 dihydrochloride
Cat.No: T14366
Synonym:
Target: P2X Receptor
Hydroxychloroquine
Cat.No: T9287
Synonym: 2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol,羟氯喹
Target: SARS-CoV, TLR, Parasite, Autophagy
VB124
Cat.No: T60165
Synonym:
Target: Monocarboxylate transporter
CB2R/FAAH modulator-3
Cat.No: T67747
Synonym:
Target: Cannabinoid Receptor, FAAH
Imiquimod
Cat.No: T0134
Synonym: 咪喹莫特,R 837,S-26308
Target: SARS-CoV, TLR, Autophagy, HSV
CB2R/FAAH modulator-2
Cat.No: T67745
Synonym:
Target: Cannabinoid Receptor, FAAH
Ebselen
Cat.No: T0825
Synonym: SPI-1005,PZ-51,依布硒,CCG-39161
Target: Phosphatase, Virus Protease, Calcium Channel, COX, HIV Protease
PI3K-IN-19 hydrochloride
Cat.No: T39581
Synonym: PI3K-IN-19 hydrochloride
Target:
HSP90-IN-27
Cat.No: T82166
Synonym:
Target: HSP
STING agonist-19
Cat.No: T81083
Synonym:
Target:
Galanin (1-19), human
Cat.No: TP1529
Synonym:
Target:
Anti-inflammatory agent 19
Cat.No: T63660
Synonym:
Target:
RU 24411
Cat.No: T34430
Synonym: RU24411,RU-24411
Target:
Myosin light chain kinase fragment 11-19 amide
Cat.No: T81732
Synonym: MLCK(11-19) amide
Target:
meplazumab
Cat.No: T9931
Synonym:
Target: Others
ICMT-IN-19
Cat.No: T82126
Synonym:
Target:
VEGFR-2-IN-19
Cat.No: T61137
Synonym:
Target:
Guanosine triphosphate
Cat.No: T73596
Synonym:
Target:
TGR5 agonist 2
Cat.No: T74825
Synonym:
Target:
STh
Cat.No: T38567
Synonym:
Target:
Protein Kinase C (19-31)
Cat.No: TP1053
Synonym: Protein Kinase C 19-31,PKC (19-31)
Target:
19-hydroxy Cholesterol
Cat.No: T36217
Synonym:
Target:
MDK03855
Cat.No: T70601
Synonym:
Target:
Glucagon (22-29)
Cat.No: T82306
Synonym:
Target:
ACAT-IN-5
Cat.No: T39412
Synonym:
Target:
Protein Kinase C (19-35) Peptide
Cat.No: T76456
Synonym:
Target:
Protein Kinase C (19-31) (TFA)(121545-65-1,free)
Cat.No: TP1052
Synonym: PKC (19-31) (TFA),Protein Kinase C (19-31) (TFA)
Target:
Garcinone B
Cat.No: T78770
Synonym:
Target: Angiotensin-converting Enzyme (ACE)
β-Herpesvirus protease-IN-1
Cat.No: T80691
Synonym:
Target: Virus Protease
Lp-PLA2-IN-12
Cat.No: T79010
Synonym:
Target: Phospholipase
HIF-1 alpha (556-574) (TFA)
Cat.No: T82199
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase
GNE-2256
Cat.No: T73372
Synonym:
Target:
PTP1B-IN-19
Cat.No: T63023
Synonym:
Target:
Daxdilimab
Cat.No: T76767
Synonym:
Target:
Dabcyl-KTSAVLQSGFRKME-Edans TFA
Cat.No: T76067
Synonym:
Target:
Estrogen receptor modulator 6
Cat.No: T40893
Synonym:
Target:
COVID-19 Spike Protein mRNA-LNP
Cat.No: T75116
Synonym:
Target:
L-163491
Cat.No: T70256
Synonym:
Target:
Imiquimod hydrochloride
Cat.No: T22091
Synonym:
Target:
COVID-19 Spike Protein mRNA(N1-Me-Pseudo UTP)
Cat.No: T75102
Synonym:
Target:
Anti-inflammatory agent 18
Cat.No: T63473
Synonym:
Target:
Nampt-IN-10 TFA
Cat.No: T64273
Synonym:
Target:
CCT251545 analogue, Compound 51
Cat.No: T22633
Synonym:
Target: Others
BMSpep-57 hydrochloride
Cat.No: T36885
Synonym:
Target:
Protein Kinase C (19-31) (TFA)
Cat.No: T76008
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN3651 Cichoriin

Others Others
Cichoriin 对SARS-CoV-2有明显活性,是治疗重症COVID-19的潜在候选物质。
T8070 Nonadecanoic acid

Others Others
Nonadecanoic acid 是19 C 长的饱和脂肪酸,是白蚁防御时分泌的主要物质。
T0194 Chloroquine phosphate

Chloroquine diphosphate,Aralen phosphate,磷酸氯喹,Chingamin phosphate

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine phosphate (Aralen phosphate) 是广泛用于疟疾和类风湿性关节炎的抗疟疾和抗炎剂。它是autophagy 和toll-like receptors 抑制剂,有效抑制SARS-CoV-2(COVID-19) 感染 (EC50=1.13 μM)。
T3921 Punicalagin

安石榴甙,安石榴苷

SARS-CoV; HBV Microbiology/Virology
Punicalagin 是一种在石榴中发现的主要鞣花单宁,是可逆且非竞争性的3CLpro 抑制剂,有抗氧化、抗炎和抗癌作用。它有潜力研究 COVID-19
TN3948 ent-3Beta-Angeloyloxykaur-16-en-19-oic acid

Others Others
ent-3Beta-Angeloyloxykaur-16-en-19-oic acid是一种天然产物,属于菊科蟛蜞菊属,其产品编号为 TN3948,CAS号为 74635-61-3。ent-3Beta-Angeloyloxykaur-16-en-19-oic acid可用作对照参考。
TN3939 ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid

Others Others
ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid是一种天然产物,属于菊科苍耳属,其产品编号为 TN3939,CAS号为 55483-24-4。ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid可用作对照参考。
TN6493 19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene

19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene是一种天然产物,属于松科松属,其产品编号为 TN6493,CAS号为 1011714-20-7。19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene可用作对照参考。
TN2757 2-Epitormentic acid

Others Others
2-Epitormentic acid是一种天然产物,属于蔷薇科委陵菜属,其产品编号为 TN2757,CAS号为 119725-19-8。2-Epitormentic acid可用作对照参考。
TN2700 2,3-dihydrosciadopitysin

Others Others
2,3-dihydrosciadopitysin是一种天然产物,属于罗汉松科罗汉松属,其产品编号为 TN2700,CAS号为 34421-19-7。2,3-dihydrosciadopitysin可用作对照参考。
TN2486 1-(3,4-Dimethoxyphenyl)propane-1,2-diol

Others Others
β-Aflatrem是一种天然产物,属于金粟兰科金粟兰属,其产品编号为 TN2486,CAS号为 20133-19-1。β-Aflatrem可用作对照参考。
TN3254 7alpha-Hydroxystigmasterol

Others Others
7alpha-Hydroxystigmasterol是一种天然产物,属于菊科苍耳属,其产品编号为 TN3254,CAS号为 64998-19-2。7alpha-Hydroxystigmasterol可用作对照参考。
T75670 Lacto-N-fucopentaose II

Lacto-N-fucopentaose II (LNFP II)作为人Lewis血型决定因子的半抗原,其单唾液神经节苷/糖脂以及唾液酰衍生物CA 19-9,都是胆胰恶性肿瘤中的分子肿瘤标记物(TM)。
TN3269 8,9-Didehydro-7-hydroxydolichodial

Others Others
8,9-Didehydro-7-hydroxydolichodial是一种天然产物,属于败酱科败酱属,其产品编号为 TN3269,CAS号为 97856-19-4。8,9-Didehydro-7-hydroxydolichodial可用作对照参考。
TN1194 16beta,17-Dihydroxy-ent-kaurane-19-oic acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
16beta,17-Dihydroxy-ent-kaurane-19-oic acid as an anti-HIV principle, it showed significant activity against HIV replication in H9 lymphocyte cells with an EC50 value of 0.8 microgram/mL. It also possesses the activities of decompression and blood viscosi
TN5637 5-(Z-Heptadec-8-enyl)resorcinol

5-(8-Heptadecenyl)-1,3-benzenediol

5-(Z-Heptadec-8-enyl)resorcinol是一种天然产物,属于紫金牛科紫金牛属,其产品编号为 TN5637,CAS号为 52483-19-9。5-(Z-Heptadec-8-enyl)resorcinol可用作对照参考。
T38262 Sphingosine (d14:1)

Sphingosine (d14:1) is a bioactive sphingolipid that has been found in B. mori (silkworm), P. clarkii (crayfish), and A. aurita (jellyfish) extracts. It increases the germination rate of N. rileyi, an entomopathogenic fungus, with an EC50 value of 10.2 nM. Sphingosine (d14:1) inhibits protein kinase C (PKC) in vitro (IC50 = 7.3 mol%) as well as superoxide generation induced by phorbol 12-myristate 13-acetate in neutrophils and reduces growth of CHO cells (IC50s = 19 and 8 μM, respectively).
T72581 SARS-CoV MPro-IN-2

SARS-CoVMPro-IN-2 是一种有效的SARS-CoV-2 Mpro 抑制剂,IC50sub>值为 72.07 nM。病毒的主要蛋白酶 Mpro 作为加工病毒多蛋白的主要酶,有助于 SARS-CoV-2 在宿主细胞中的复制和转录,并已被定性为药物发现的有吸引力的靶点。SARS-CoVMPro-IN-2 具有研究 COVID-19 的潜力。
T38069 Aquastatin A

Aquastatin A is a fungal metabolite originally isolated fromF. aquaeductuumthat has diverse biological activities.1It is active againstS. aureus(MIC = 32 μg/ml) and inhibits enoyl-acyl carrier protein reductase (Fabl; IC50= 3.2 μM) andS. aureusfatty acid synthesis (IC50= 3.5 μM).2Aquastatin A also inhibits the Na+/K+-ATPase and H+/K+-ATPase (IC50s = 7.1 and 6.2 μM, respectively), as well as protein tyrosine phosphatase 1B (PTP1B; IC50= 0.19 μM).1,3 1.Hamano, K., Kinoshita-Okami, M., Minagawa, K....

天然产物

Cichoriin
Cat.No: TN3651
Synonym:
Target: Others
Nonadecanoic acid
Cat.No: T8070
Synonym:
Target: Others
Chloroquine phosphate
Cat.No: T0194
Synonym: Chloroquine diphosphate,Aralen phosphate,磷酸氯喹,Chingamin phosphate
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
Punicalagin
Cat.No: T3921
Synonym: 安石榴甙,安石榴苷
Target: SARS-CoV, HBV
ent-3Beta-Angeloyloxykaur-16-en-19-oic acid
Cat.No: TN3948
Synonym:
Target: Others
ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid
Cat.No: TN3939
Synonym:
Target: Others
19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene
Cat.No: TN6493
Synonym:
Target:
2-Epitormentic acid
Cat.No: TN2757
Synonym:
Target: Others
2,3-dihydrosciadopitysin
Cat.No: TN2700
Synonym:
Target: Others
1-(3,4-Dimethoxyphenyl)propane-1,2-diol
Cat.No: TN2486
Synonym:
Target: Others
7alpha-Hydroxystigmasterol
Cat.No: TN3254
Synonym:
Target: Others
Lacto-N-fucopentaose II
Cat.No: T75670
Synonym:
Target:
8,9-Didehydro-7-hydroxydolichodial
Cat.No: TN3269
Synonym:
Target: Others
16beta,17-Dihydroxy-ent-kaurane-19-oic acid
Cat.No: TN1194
Synonym:
Target: HIV Protease
5-(Z-Heptadec-8-enyl)resorcinol
Cat.No: TN5637
Synonym: 5-(8-Heptadecenyl)-1,3-benzenediol
Target:
Sphingosine (d14:1)
Cat.No: T38262
Synonym:
Target:
SARS-CoV MPro-IN-2
Cat.No: T72581
Synonym:
Target:
Aquastatin A
Cat.No: T38069
Synonym:
Target:
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