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99

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T6422 Brimonidine Tartrate

AGN190342 tartrate,304 tartrate,酒石酸溴莫尼定,AGN190342 (tartrate),UK 14304 (tartrate),UK14304 tartrate

Adrenergic Receptor GPCR/G Protein; Neuroscience
Brimonidine Tartrate (AGN190342 tartrate) 是一种 alpha2 Adrenergic Receptor (alpha2-AR) 受体激动剂。
T0363 Morantel tartrate

CP-12009-18 tartrate,UK 296418 tartrate,酒石酸甲噻嘧啶

Parasite Microbiology/Virology
Morantel tartrate (CP-12009-18 tartrate) 是一种主要用于牲畜的杀虫剂。
T1066L Ketanserin tartrate

KJK 945 tartrate,KJK-945 tartrate,KJK945 tartrate

5-HT Receptor; Serotonin Transporter; Adrenergic Receptor GPCR/G Protein; Neuroscience
Ketanserin tartrate (KJK-945 tartrate) 是 5-HT2A 受体和α1-肾上腺素能受体拮抗剂,具有抗高血压活性,抑制血清素诱导的血管收缩和血小板活化,可用于研究系统性硬化症。
T16989 Tarafenacin D-tartrate

SVT-40776 D-tartrate

Others Others
Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.
T1657 Varenicline Tartrate

Champix tartrate,酒石酸伐尼克兰,Chantix tartrate,CP 526555-18,酒石酸伐仑克林

AChR Neuroscience
Varenicline Tartrate (CP 526555-18) 是α4β2 烟碱乙酰胆碱受体的部分激动剂,EC50为 2.3 μM。它是 α3β4 和 α7 乙酰胆碱受体完全激动剂,EC50值分别为 55 和 18 μM,用于戒烟方面的研究。
T0279 Metaraminol tartrate

重酒石酸间羟胺,Metaradrine tartrate,Metaraminol bitartrate

Adrenergic Receptor GPCR/G Protein; Neuroscience
Metaraminol tartrate (Metaradrine tartrate) 是一种 α-肾上腺素能 (α-adrenergic) 激动剂,是一种直接或间接影响肾上腺素受体的拟交感神经胺,其中 α 效应占主导地位,可作为血管加压剂。
T7164 Levalbuterol tartrate

左旋沙丁胺醇酒石酸盐,Levosalbutamol tartrate

Adrenergic Receptor GPCR/G Protein; Neuroscience
Levalbuterol tartrate (Levosalbutamol tartrate) 是一种短效的β2肾上腺素受体激动剂,是一种 salbutamol 的 R 型对映体。
T22228 Tylvalosin tartrate

酒石酸乙酰异戊酰泰乐菌素,Acetylisovaleryltylosin Tartrate

Antibacterial; Antibiotic Microbiology/Virology
Tylvalosin tartrate (Acetylisovaleryltylosin Tartrate) 是一种对革兰氏阳性细菌具有抗性的大环内酯类抗生素。
T22245 Arformoterol Tartrate

(R,R)-Formoterol tartrate,酒石酸福莫特罗

Adrenergic Receptor GPCR/G Protein; Neuroscience
Arformoterol Tartrate ((R,R)-Formoterol tartrate) 是一种长效 β2-肾上腺素能受体 (β2-AR) 激动剂,Kd=2.9 nM。它是一种 Formoterol 的 (R,R)-对映异构体,可用于慢性阻塞性肺疾病 (COPD) 的研究。
T6946 Pimavanserin tartrate

ACP-103,ACP-103 tartrate,Nuplazid,Pimavanserin,匹莫范色林

5-HT Receptor GPCR/G Protein; Neuroscience
Pimavanserin tartrate (Nuplazid) 是一种有效的5-HT 2A 受体反向激动剂,pIC50和 pKi 值分别为8.73和9.3,用于治疗与帕金森病相关的精神病。
T5203 Sodium Tartrate

Others Others
Sodium Tartrate 是一种的 pH 调节剂,具有抗氧化活性,能够有效延缓高温加热时的水解,使植物油的酸值增加。
T7369L Gemigliptin Tartrate(911637-19-9 free base)

吉格列汀酒石酸盐,LC15-0444 tartrate

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Gemigliptin Tartrate (LC15-0444 tartrate) 是一种选择性的,可逆的,竞争性的二肽基肽酶 4 (DPP-4) 抑制剂,对于人重组 DPP-4 的IC50=10.3 nM。Gemigliptin tartrate 具有很强的抗糖基化活性,能够用于晚期糖基化终产物相关的糖尿病并发症的研究。
T11236 Giredestrant tartrate

Estrogen receptor antagonist 1

Estrogen Receptor/ERR; Others Endocrinology/Hormones; Others
Giredestrant tartrate (Estrogen receptor antagonist 1) 是一种新型的、具有口服活性的、有选择性的、有效的的非甾体雌激素受体拮抗剂。Giredestrant tartrate 与 ER 强效结合,导致 ER 无法激活靶向基因的转录,并促使 ER 蛋白降解。Giredestrant tartrate 可用于治疗肿瘤疾病。
T7839 Lasofoxifene Tartrate

CP-336156,酒石酸拉索昔芬

Estrogen Receptor/ERR Endocrinology/Hormones
Lasofoxifene Tartrate (CP-336156) 是一种非甾体类的雌激素受体选择性调节剂 (SERM)。
T0395 Pyrantel tartrate

Banminth,酒石酸噻吩嘧啶

Antibiotic; Parasite Microbiology/Virology
Pyrantel tartrate (Banminth) 是一种四氢嘧啶类广谱牲畜驱虫剂,是烟碱乙酰胆碱受体激动剂。它能引起寄生虫的痉挛性肌肉麻痹。它可研究胃肠道线虫感染。
TQ0022 Capromorelin Tartrate

卡普瑞林酒石酸盐,CP 424391-18

GHSR GPCR/G Protein
Capromorelin Tartrate (CP 424391-18) 是口服有活性的 growth hormone secretagogue receptor 有效激动剂,能够作用于 hGHS-R1a(Ki:7 nM)。
T1628 Rivastigmine tartrate

SDZ-ENA 713,ENA 713,酒石酸卡巴拉汀

AChR; AChE Neuroscience
Rivastigmine tartrate (SDZ-ENA 713) 是一种具有口服活性的、可透过血脑屏障的胆碱酯酶抑制剂,能够抑制丁酰胆碱酯酶和乙酰胆碱酯酶。它是一种拟副交感神经剂或胆碱能剂,用于研究轻度至中度阿尔茨海默氏型痴呆和帕金森氏病引起的痴呆。
T0099 Tolterodine tartrate

Detrol LA,PNU-200583E,Kabi-2234,酒石酸托特罗定

AChR Neuroscience
Tolterodine tartrate (PNU-200583E) 是毒蕈碱受体的有效拮抗剂。 它在体内显示出对膀胱和唾液腺的选择性。
T39010 Xanomeline tartrate

LY 246708 tartrate,Xanomeline tartrate

Xanomeline (LY 246708), a potent agonist of muscarinic M1/M4 receptors, exhibits antipsychotic-like activity and enhances neuronal excitability. It is a valuable compound for studying schizophrenia.
T72431 Theliatinib tartrate

Xiliertinib tartrate,HMPL-309 tartrate,Xiliertinib tartrate ; HMPL-309 tartrate

Theliatinib (Xiliertinib) tartrate 是一种有效、ATP 竞争性、口服活性和高度选择性的EGFR 抑制剂,Ki 为 0.05 nM,IC50为 3 nM。Theliatinib 对EGFRT790M/L858R 突变体的IC50值为 22 nM。Theliatinib 对EGFR 的选择性是其他激酶的 50 倍以上。
T3282 Alimemazine hemitartrate

Alimemazine Tartrate,Methylpromazine Tartrate,酒石酸异丁嗪,Trimeprazine tartrate,Trimeprazine hemitartrate

Others Others
Alimemazine hemitartrate (Trimeprazine hemitartrate) 是血凝素 (HA)-受体的拮抗剂,也是一种吩噻嗪衍生物,常用作止痒剂。
T38913 Furaltadone L-tartrate

Furaltadone L-tartrate,Altafur L-tartrate

Furaltadone L-tartrate (Altafur L-tartrate), a nitrofuran antimicrobial agent, is potentially useful for researching Salmonella enteritidis infections in chickens. It demonstrates both inhibitory and bactericidal properties against Staphylococci in vitro.
T11248 Evogliptin tartrate

DA-1229 tartrate

DPP-4 Proteases/Proteasome
Evogliptin tartrate has potential for anti-atherosclerosis therapy that targets arterial inflammation. Evogliptin tartrate is a potent, orally bioavailable and selective dipeptidyl peptidase-4 (DPP-4) inhibitor, with antidiabetic activity.
T20193 L-Carnitine tartrate

L-Carnitine L-tartrate,Carnipure tartrate

L-Carnitine tartrate is a Carnitine/ Constituent of striated muscle and liver. It is used to treatment of hyperlipoproteinemias.
T19182 Afegostat D-Tartrate

Isofagomine D-Tartrate,D-Isofagomine D-Tartrate

Others Others
Afegostat D-Tartrate is a pharmacological chaperone that specifically and reversibly binds acid-β-glucosidase (GCase) in the endoplasmic reticulum with high affinity.
T32510 L-771688 tartrate

L771688 tartrate,L 771688 tartrate

L-771688 tartrate is a bioactive chemical.
T24001 Diisopropyl tartrate

Diisopropyl (+)-L-tartrate,L-DIPT,BRN 1727863

Diisopropyl tartrate is a reagent for kinetic resolution of racemic allylic alcohols and α-furfuryl amides. It acts by enantioselective epoxidation.
T27939 LY2940094 tartrate

LY2940094,LY 2940094,LY-2940094 tartrate,LY-2940094

LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.
T0293L Metyrapone Tartrate

SU 4885,Metopirone tartrate,SU-4885,SU4885

Metyrapone Tartrate is an inhibitor of the STEROID 11-beta-monooxygenase enzyme which is used as a test for feedback hypothalamic-pituitary mechanism in the diagnosis of Cushing SYNDROME.
T4560L2 Alprenolol tartrate, (S)-

(S)-Alprenolol tartrate,l-Alprenolol bitartrate

Alprenolol tartrate, (S)- is an 5-HT1A antagonist.
T2358L ENMD-2076 tartrate

ENMD-2076,L-(+) Tartrate salt of ENMD-981693,ENMD2076,ENMD 2076

ENMD-2076 is an orally active kinase inhibitor. It also has antiangiogenic and antiproliferative mechanisms of action.
T11832 Ledipasvir D-tartrate

GS-5885 D-tartrate,雷迪帕韦 D-酒石酸

Others Others
Ledipasvir D-tartrate with EC50 values of 34 pM against GT1a and 4 pM against GT1b replicon. is an inhibitor of the hepatitis C virus NS5A.
T36811 uPSEM 817 tartrate

Selective ultrapotent PSEM (uPSEM) agonist for α7L131G,Q139L,Y217F-GlyR (PSAM4-GlyR) and PSAM4-5-HT3 chimeric ion channel agonist (EC50 values are 0.3 and 0.5 nM, respectively). Suppresses firing of layer 2/3 cortical neurons expressing PSAM4-GlyR in brain slices. Increases contralateral rotation in mice expressing PSAM4-GlyR unilaterally in the substantia nigra reticulata (LED 0.1 mg/kg). Magnus et al (2019) Ultrapotent chemogenetics for research and potential clinical applications. Science 3...
T69516 Thenalidine tartrate

Thenalidine is an antihistamine with anticholinergic properties used as an antipruritic drug. It was withdrawn from the US, Canadian, and UK markets due to a risk of neutropenia. Thenalidine is an antagonist of the H1-receptor.
T68311 Ritanserin tartrate

Ritanserin tartrateis is a selective and potent serotonin-2 antagonist.
T69109 Ellipticine tartrate

Ellipticine tartrate is a DNA intercalating agent and a DNA topoisomerase II inhibitor.
T21385 Cinitapride

西尼必利,Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove

5-HT Receptor GPCR/G Protein; Neuroscience
Cinitapride (Blaston) 是一种促胃药。它减缓肌肉的活动,以减轻诸如胃酸反流、胃排空延迟和溃疡性消化不良等病症的症状。 Cinitapride 作为 5-HT2 受体的拮抗剂和 5-HT1 和 5-HT4 受体的激动剂。
T69120 Pempidine tartrate

Pempidine tartrate is a nicotinic antagonist most commonly used as an experimental tool. It has been used as a ganglionic blocker in the treatment of hypertension but has largely been supplanted for that purpose by more specific drugs.
T69939 Hexamethonium tartrate

Hexamethonium tartrate is a nicotinic cholinergic antagonist often referred to as the prototypical ganglionic blocker. It is poorly absorbed from the gastrointestinal tract and does not cross the blood-brain barrier. It has been used for a variety of therapeutic purposes including hypertension but, like the other ganglionic blockers, it has been replaced by more specific drugs for most purposes, although it is widely used a research tool.
T70224 Bupivacaine tartrate

Bupivacaine is a BK/SK, Kv1, Kv3, TASK-2 K Channel and voltage-gated Na channel blocker used as an anesthetic. It maybe neurotoxic at high does, inducing apoptosis in neuroblastoma cells. It acts by binding to the intracellular portion of voltage-gated sodium channels and blocking sodium influx into nerve cells.
T22294 Cinitapride Hydrogen Tartrate

5-HT Receptor GPCR/G Protein; Neuroscience
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors
T70379 PF-04479745 tartrate

PF-04479745, also known as PF-4479745, is a potent and selective 5-HT2C agonist (EC50 = 10 nM). PF-4479745 displayed robust pharmacology in a preclinical canine model of stress urinary incontinence (SUI) and no measurable functional agonism at the key selectivity targets 5-HT2A and 5-HT2B in relevant tissue-based assay systems.
T11176 Eliglustat hemitartrate

Genz-112638,依利格鲁司特酒石酸盐,Eliglustat tartrate

Others Others
Eliglustat hemitartrate (Genz-112638) 是一种高效的、特异性的、有口服活性的葡糖脑苷脂合成酶抑制剂(IC50:24 nM)。
T6722 Vinflunine Tartrate

Microtubule Associated Cytoskeletal Signaling
Vinflunine Tartrate 是一种独特的新型长春花生物碱,具有抑制有丝分裂和微管蛋白相互作用活性的特性。
T27021 Cinitapride Tartrate

Cinitapride Tartrate is an agonist of the 5-HT1 and 5-HT4 receptors and is also an antagonist of the 5-HT2 receptors.
T71636 Golvatinib tartrate

Golvatinib tartrate is an orally bioavailable dual kinase inhibitor of c-Met (hepatocyte growth factor receptor) and VEGFR-2 (vascular endothelial growth factor receptor-2) tyrosine kinases with potential antineoplastic activity.
T34923 TRH tartrate

TRH tartrate is a thyrotropin-releasing hormone.
T8149L Dobutamine tartrate

Dobutamine tartrate is a cardiotonic.
T29102 Vedaclidine tartrate

Vedaclidine tartrate is a muscarinic analgesic.
T29913L Altanserin tartrate

R-53,200

Altanserin tartrate is a compound that binds to the 5-HT2A receptor. Labeled with the isotope fluorine-18 it is used as a radioligand in positron emission tomography (PET) studies of the brain.

化合物

Brimonidine Tartrate
Cat.No: T6422
Synonym: AGN190342 tartrate,304 tartrate,酒石酸溴莫尼定,AGN190342 (tartrate),UK 14304 (tartrate),UK14304 tartrate
Target: Adrenergic Receptor
Morantel tartrate
Cat.No: T0363
Synonym: CP-12009-18 tartrate,UK 296418 tartrate,酒石酸甲噻嘧啶
Target: Parasite
Ketanserin tartrate
Cat.No: T1066L
Synonym: KJK 945 tartrate,KJK-945 tartrate,KJK945 tartrate
Target: 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor
Tarafenacin D-tartrate
Cat.No: T16989
Synonym: SVT-40776 D-tartrate
Target: Others
Varenicline Tartrate
Cat.No: T1657
Synonym: Champix tartrate,酒石酸伐尼克兰,Chantix tartrate,CP 526555-18,酒石酸伐仑克林
Target: AChR
Metaraminol tartrate
Cat.No: T0279
Synonym: 重酒石酸间羟胺,Metaradrine tartrate,Metaraminol bitartrate
Target: Adrenergic Receptor
Levalbuterol tartrate
Cat.No: T7164
Synonym: 左旋沙丁胺醇酒石酸盐,Levosalbutamol tartrate
Target: Adrenergic Receptor
Tylvalosin tartrate
Cat.No: T22228
Synonym: 酒石酸乙酰异戊酰泰乐菌素,Acetylisovaleryltylosin Tartrate
Target: Antibacterial, Antibiotic
Arformoterol Tartrate
Cat.No: T22245
Synonym: (R,R)-Formoterol tartrate,酒石酸福莫特罗
Target: Adrenergic Receptor
Pimavanserin tartrate
Cat.No: T6946
Synonym: ACP-103,ACP-103 tartrate,Nuplazid,Pimavanserin,匹莫范色林
Target: 5-HT Receptor
Sodium Tartrate
Cat.No: T5203
Synonym:
Target: Others
Gemigliptin Tartrate(911637-19-9 free base)
Cat.No: T7369L
Synonym: 吉格列汀酒石酸盐,LC15-0444 tartrate
Target: Proteasome, DPP-4
Giredestrant tartrate
Cat.No: T11236
Synonym: Estrogen receptor antagonist 1
Target: Estrogen Receptor/ERR, Others
Lasofoxifene Tartrate
Cat.No: T7839
Synonym: CP-336156,酒石酸拉索昔芬
Target: Estrogen Receptor/ERR
Pyrantel tartrate
Cat.No: T0395
Synonym: Banminth,酒石酸噻吩嘧啶
Target: Antibiotic, Parasite
Capromorelin Tartrate
Cat.No: TQ0022
Synonym: 卡普瑞林酒石酸盐,CP 424391-18
Target: GHSR
Rivastigmine tartrate
Cat.No: T1628
Synonym: SDZ-ENA 713,ENA 713,酒石酸卡巴拉汀
Target: AChR, AChE
Tolterodine tartrate
Cat.No: T0099
Synonym: Detrol LA,PNU-200583E,Kabi-2234,酒石酸托特罗定
Target: AChR
Xanomeline tartrate
Cat.No: T39010
Synonym: LY 246708 tartrate,Xanomeline tartrate
Target:
Theliatinib tartrate
Cat.No: T72431
Synonym: Xiliertinib tartrate,HMPL-309 tartrate,Xiliertinib tartrate ; HMPL-309 tartrate
Target:
Alimemazine hemitartrate
Cat.No: T3282
Synonym: Alimemazine Tartrate,Methylpromazine Tartrate,酒石酸异丁嗪,Trimeprazine tartrate,Trimeprazine hemitartrate
Target: Others
Furaltadone L-tartrate
Cat.No: T38913
Synonym: Furaltadone L-tartrate,Altafur L-tartrate
Target:
Evogliptin tartrate
Cat.No: T11248
Synonym: DA-1229 tartrate
Target: DPP-4
L-Carnitine tartrate
Cat.No: T20193
Synonym: L-Carnitine L-tartrate,Carnipure tartrate
Target:
Afegostat D-Tartrate
Cat.No: T19182
Synonym: Isofagomine D-Tartrate,D-Isofagomine D-Tartrate
Target: Others
L-771688 tartrate
Cat.No: T32510
Synonym: L771688 tartrate,L 771688 tartrate
Target:
Diisopropyl tartrate
Cat.No: T24001
Synonym: Diisopropyl (+)-L-tartrate,L-DIPT,BRN 1727863
Target:
LY2940094 tartrate
Cat.No: T27939
Synonym: LY2940094,LY 2940094,LY-2940094 tartrate,LY-2940094
Target:
Metyrapone Tartrate
Cat.No: T0293L
Synonym: SU 4885,Metopirone tartrate,SU-4885,SU4885
Target:
Alprenolol tartrate, (S)-
Cat.No: T4560L2
Synonym: (S)-Alprenolol tartrate,l-Alprenolol bitartrate
Target:
ENMD-2076 tartrate
Cat.No: T2358L
Synonym: ENMD-2076,L-(+) Tartrate salt of ENMD-981693,ENMD2076,ENMD 2076
Target:
Ledipasvir D-tartrate
Cat.No: T11832
Synonym: GS-5885 D-tartrate,雷迪帕韦 D-酒石酸
Target: Others
uPSEM 817 tartrate
Cat.No: T36811
Synonym:
Target:
Thenalidine tartrate
Cat.No: T69516
Synonym:
Target:
Ritanserin tartrate
Cat.No: T68311
Synonym:
Target:
Ellipticine tartrate
Cat.No: T69109
Synonym:
Target:
Cinitapride
Cat.No: T21385
Synonym: 西尼必利,Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove
Target: 5-HT Receptor
Pempidine tartrate
Cat.No: T69120
Synonym:
Target:
Hexamethonium tartrate
Cat.No: T69939
Synonym:
Target:
Bupivacaine tartrate
Cat.No: T70224
Synonym:
Target:
Cinitapride Hydrogen Tartrate
Cat.No: T22294
Synonym:
Target: 5-HT Receptor
PF-04479745 tartrate
Cat.No: T70379
Synonym:
Target:
Eliglustat hemitartrate
Cat.No: T11176
Synonym: Genz-112638,依利格鲁司特酒石酸盐,Eliglustat tartrate
Target: Others
Vinflunine Tartrate
Cat.No: T6722
Synonym:
Target: Microtubule Associated
Cinitapride Tartrate
Cat.No: T27021
Synonym:
Target:
Golvatinib tartrate
Cat.No: T71636
Synonym:
Target:
TRH tartrate
Cat.No: T34923
Synonym:
Target:
Dobutamine tartrate
Cat.No: T8149L
Synonym:
Target:
Vedaclidine tartrate
Cat.No: T29102
Synonym:
Target:
Altanserin tartrate
Cat.No: T29913L
Synonym: R-53,200
Target:
Cat. No. Product Name Target Signaling Pathways
T2782L Catharanthine Tartrate(2468-21-5(free base))

Calcium Channel Membrane transporter/Ion channel; Metabolism
Catharanthine Tartrate(2468-21-5(free base)) 是从马达加斯加长春花中分离得到的天然产物,Catharanthine Tartrate 抑制电压操作的L 型Ca2+通道,具有抗癌和降血压活性。
T0861 Tylosin tartrate

酒石酸泰洛星,酒石酸泰乐菌素

Antibacterial; Antibiotic Microbiology/Virology
Tylosin tartrate 是一种大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高效的抗菌活性。它作为饲料添加剂可促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
T1186 Ifenprodil Tartrate

Potassium Channel; NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Ifenprodil tartrate 是典型的非竞争性 NMDA 受体拮抗剂,抑制 GIRK (Kir3),通过基底 GIRK 活性减少内向电流,有用做脑血管舒张试剂的潜力。它对 NR1A/NR2B 受体亲和力是 NR1A/NR2A 受体的 400 倍。
T3013 Catharanthine tartrate

Catharanthine hemitartrate,酒石酸长春质碱

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Catharanthine tartrate (Catharanthine hemitartrate) 是长春花中的一种生物碱,可抑制电压门控 L 型钙离子通道,具有抗肿瘤和降血压活性。
T65128 Tartaric acid disodium dihydrate

Disodium L-(+)-Tartrate Dihydrate

Phosphatase; Endogenous Metabolite Metabolism
Tartaric acid disodium dihydrate (Disodium L-(+)-Tartrate Dihydrate) 常用来制作分子生物学和细胞培养中的缓冲液,。Tartaric acid disodium dihydrate 是酸性磷酸酶抑制剂, 可增加秋水仙碱结合 tubulin1的概率。
T20779 Kitasamycin tartrate

Leucomycin tartrate

Kitasamycin tartrate, a macrolide antibiotic produced by Streptomyces kitasatoensis, has a wide spectrum of antimicrobial activity.
T6213 Vinorelbine ditartrate

Vinorelbine Tartrate,Nor-5'-anhydrovinblastine ditartrate,KW-2307,Navelbine tartrate,长春瑞滨酒石酸盐,酒石酸长春瑞滨

Microtubule Associated; Autophagy Autophagy; Cytoskeletal Signaling
Vinorelbine ditartrate (KW-2307)是一种抗有丝分裂剂,能够抑制 Hela 细胞的增殖,IC50值为 1.25 nM。
T20173 Noradrenaline tartrate

NSC 169106,NSC-169106,l-Noradrenaline d-bitartrate,NSC169106,Norepinephrine bitartrate

Norepinephrine bitartrate is a precursor of epinephrine. Norepinephrine is the principal transmitter of most postganglionic sympathetic fibers and of the diffuse projection system in the brain arising from the locus ceruleus.
T6805 Choline bitartrate

2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium,酒石酸氢胆碱

Others; AChR Neuroscience; Others
Choline bitartrate (2-hydroxyethyl(trimethyl)azanium) 是一种存在于食物中的营养胆碱,可影响肝脏疾病、动脉粥样硬化和神经系统疾病等疾病。它是神经递质乙酰胆碱的前体,作为甲基供体参与各种代谢过程和脂质代谢。
T1064 Norepinephrine bitartrate monohydrate

酒石酸去甲肾上腺素,Levophed,Noradrenaline bitartrate monohydrate,降肾上腺素

Endogenous Metabolite; Adrenergic Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Neuroscience
Norepinephrine bitartrate monohydrate (Levophed) 是一种β1-选择性的肾上腺素能受体激动剂,EC50为 5.37 μM。
T21066 Norepinephrine bitartrate salt

Adrenergic Receptor GPCR/G Protein; Neuroscience
Norepinephrine bitartrate salt 是一种肾上腺素能神经递质。
T75425 Synephrine hemitartrate

Synephrine (Oxedrine) hemitartrate,一种生物碱,是一种来自Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂。Synephrine hemitartrate 是一种拟交感神经化合物,可用于减肥。
T3804 Neomangiferin

Mangiferin 7-glucoside,新芒果苷

Phosphatase Metabolism
Neomangiferin (Mangiferin 7-glucoside) 是一种天然的 C-glucosyl xanthone,分离自干燥的Anemarrhena asphodeloides 的根茎中。它能够减轻大鼠高脂饮食诱导的非酒精性脂肪性肝病 (NAFLD)。

天然产物

Catharanthine Tartrate(2468-21-5(free base))
Cat.No: T2782L
Synonym:
Target: Calcium Channel
Tylosin tartrate
Cat.No: T0861
Synonym: 酒石酸泰洛星,酒石酸泰乐菌素
Target: Antibacterial, Antibiotic
Ifenprodil Tartrate
Cat.No: T1186
Synonym:
Target: Potassium Channel, NMDAR, iGluR
Catharanthine tartrate
Cat.No: T3013
Synonym: Catharanthine hemitartrate,酒石酸长春质碱
Target: Others, Calcium Channel
Tartaric acid disodium dihydrate
Cat.No: T65128
Synonym: Disodium L-(+)-Tartrate Dihydrate
Target: Phosphatase, Endogenous Metabolite
Kitasamycin tartrate
Cat.No: T20779
Synonym: Leucomycin tartrate
Target:
Vinorelbine ditartrate
Cat.No: T6213
Synonym: Vinorelbine Tartrate,Nor-5'-anhydrovinblastine ditartrate,KW-2307,Navelbine tartrate,长春瑞滨酒石酸盐,酒石酸长春瑞滨
Target: Microtubule Associated, Autophagy
Noradrenaline tartrate
Cat.No: T20173
Synonym: NSC 169106,NSC-169106,l-Noradrenaline d-bitartrate,NSC169106,Norepinephrine bitartrate
Target:
Choline bitartrate
Cat.No: T6805
Synonym: 2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium,酒石酸氢胆碱
Target: Others, AChR
Norepinephrine bitartrate monohydrate
Cat.No: T1064
Synonym: 酒石酸去甲肾上腺素,Levophed,Noradrenaline bitartrate monohydrate,降肾上腺素
Target: Endogenous Metabolite, Adrenergic Receptor, Autophagy
Norepinephrine bitartrate salt
Cat.No: T21066
Synonym:
Target: Adrenergic Receptor
Synephrine hemitartrate
Cat.No: T75425
Synonym:
Target:
Neomangiferin
Cat.No: T3804
Synonym: Mangiferin 7-glucoside,新芒果苷
Target: Phosphatase
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