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113

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T20549 Neutral red

Others Others
Neutral Red 是含氮 pH 指示剂(pKi=6.8),是类囊体内部酸化的指示剂。它能够将溶酶体染成红色。
T31012 Coriphosphine

Neutral Yellow

Coriphosphine is a bioactive chemical.
T30970 Clivorine

J1.344.443I,Clivorine (neutral)

Clivorine is an otonecine pyrrolizidine alkaloid from the genus Ligularia.
T7693 Thiorphan

Neprilysin Metabolism
Thiorphan 是选择性neprilysin 抑制剂 (IC50:6.9 nM) 。
T22711 DCB

3,3'-dichlorobenzaldazine

Others; GluR Neuroscience; Others
DCB (3,3'-dichlorobenzaldazine) 是 mGluR5 的变构配体,显示出 3,3'-二甲氧基苯扎嗪 (DMeOB) 的负调节作用。 DCB 在 3,3'-二氟苯扎嗪 (DFB) 的帮助下阻断 mGluR 的正变构调节。
TQ0106 Sacubitrilat

LBQ-657

Neprilysin Metabolism
Sacubitrilat (LBQ-657) 是活性的脑啡肽酶 (NEP) 抑制剂。
TNU1631 N6-Methyladenosine 5’-monophos phate triethylammonium salt (neutral 4229-50-9)

N6-Methyladenosine 5’-monophos phate triethylammonium salt (neutral 4229-50-9) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TNU1631。
T0413 Cinromide

醒隆酰胺,trans-3-Bromo-N-ethylcinnamamide

Others Others
Cinromide (trans-3-Bromo-N-ethylcinnamamide) 是抗惊厥药,能够抑制上皮中性氨基酸转运蛋白 B0AT1 (SLC6A19),其 IC50=0.5 μM。
TNU1630 2’-O-Methyl-N6-methyladenosine 5’-monophosphate triethylammonium salt (60091-05-6 neutral molecule)

2’-O-Methyl-N6-methyladenosine 5’-monophosphate triethylammonium salt (60091-05-6 neutral molecule) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TNU1630。
T19033 Nile Red

Phenoxazone 9,尼罗红,Nile Blue A oxazone

Others Others
Nile Red (Nile Blue A oxazone) 是一种选择性疏水性荧光染料,针对细胞内脂质小滴和中性脂质。它在所有有机溶剂中均具有强烈的荧光性,其荧光颜色范围从金黄色到深红色。
T4574 Sacubitril

AHU 377,AHU377,沙库必曲,AHU-377

Neprilysin Metabolism
Sacubitril (AHU-377) 是一种有效的NEP 抑制剂,IC50=5 nM。它是研究心力衰竭药物 LCZ696 的组分之一。
T4200 Sacubitril hemicalcium salt

AHU-377 (hemicalcium salt),LCZ696中间体,AHU377 calcium salt

Neprilysin Metabolism
Sacubitril hemicalcium salt (AHU377 calcium salt) 是一种有效的 NEP 抑制剂,IC50=5 nM。它是研究心力衰竭药物 LCZ696 的组分之一。
T1176 Racecadotril

Acetorphan,消旋卡多曲

Neprilysin; Proteasome Metabolism; Proteases/Proteasome; Ubiquitination
Racecadotril (Acetorphan) 是一种中性内肽酶 (NEP) 抑制剂,具有止泻作用。Racecadotril 及其活性代谢物 Thiorphan 抑制小鼠脑中纯化的NEP 活性,Ki 分别为 4500 和 6.1 nM。
T2318 Sacubitril/Valsartan

Sacubitril mixture with Valsartan,沙库必曲/缬沙坦,Valsartan,Sacubitril,LCZ696

Apoptosis; RAAS; Neprilysin Apoptosis; Endocrinology/Hormones; Metabolism
Sacubitril/Valsartan (LCZ696),以1:1摩尔比由Valsartan(一种ARB)和Sacubitril(AHU377)组成,为创新口服血管紧张素受体-脑啡肽酶(ARN)双重抑制剂,旨在治疗高血压与心力衰竭。其作用机制包括抑制炎症、氧化应激及细胞凋亡,有助于改善糖尿病心肌病。
T21102 L-4FPG

L-4-氟苯甘氨酸,L4FPG,L 4FPG

Others Others
L-4FPG 是甘氨酸衍生物,抑制中性氨基酸转运蛋白 ASCT1 和 ASCT2。
T60043 DPTIP

Phospholipase Metabolism
DPTIP 是一种有效的中性鞘磷脂酶 2 抑制剂,IC50 值为 30 nM。
T10918 NEP-IN-1

Neprilysin Metabolism
NEP-IN-1 是中性肽链内切酶 (NEP) 的抑制剂 (IC50 = 2 nM)。
T19626 LHW090-A7

(ALPHAS)-3'-氯-ALPHA-[[(1S)-2-乙氧基-1-甲基-2-氧代乙基]氨基][1,1'-联苯]-4-丙酸

Neprilysin Metabolism
LHW090-A7 是一种中性肽链内切酶 (NEP) 抑制剂,是一种负责脑啡肽代谢失活的酶。
T8549 HEPES

Others Others
HEPES 是两性离子化学缓冲剂,在 pH 值为 6.8 至 8.2 时为有效的缓冲液,广泛应用于细胞培养。它是溶酶体生物发生的有效诱导剂。
T0757 Omeprazole

Losec,Prilosec,奥美拉唑,奥美拉挫,H 16868,Antra

Proton pump; Phospholipase; Antibacterial; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Omeprazole (Losec) 是一种质子泵抑制剂,有研究胃肠道疾病的潜力。它竞争性抑制 CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阳性菌和革兰氏阴性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。
T7449 o-Phenanthroline monohydrate

Phenanthroline monohydrate,1, 10-Phenanthroline monohydrate,邻菲罗啉

MMP Proteases/Proteasome
o-Phenanthroline monohydrate (1, 10-Phenanthroline monohydrate) 是一种金属螯合剂,能够与 Fe2+形成红色螯合物,λmax为 510 nm,可防止链脲佐菌素诱导染色体畸变。它也是一种 MMP 的抑制剂。
T8617 GMQ hydrochloride

NSC 403387 hydrochloride

Others Others
GMQ hydrochloride (NSC-403387 hydrochloride) 是一种有效的选择性酸感应离子通道 (ASIC) 调节剂。它在中性 pH 值下激活 ASIC3 通道并阻止酸引起的最大峰值电流。
T19080 DOPE

1,2-二油酰-SN-甘油-3-磷酰乙醇胺

Others Others
DOPE (DOPE) 是一种阳离子脂质体的中性辅助脂质 (helper lipid),能够与阳离子磷脂结合,增强裸 siRNA 的转染效率。
T27119L (Rac)-Daglutril

SLV 306 acetic acid,2-((3S)-3-(1-(2-(ethoxycarbonyl)-4-phenylbutyl)cyclopentane-1-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)acetic acid

Others Others
(Rac)-Daglutril (SLV 306 acetic acid) 是 Daglutril 的消旋体。Daglutril 是一种口服活性的混合中性内肽酶/内皮素转化酶抑制剂,正在开发用于治疗原发性高血压和充血性心力衰竭。
T3640 GW4869

GW554869A,GW 4869,GW69A

Phospholipase Metabolism
GW4869 (GW69A) 是一种中性鞘磷脂酶 N-SMase 的抑制剂 (IC50=1 μM),具有选择性和非竞争性。GW4869 也可以抑制外泌体合成/释放,常用于外泌体相关研究。
T36957 BODIPY 493/503

BDP 493/503 lipid stain,Pyrromethene 546

Others Others
BODIPY 493/503 (Pyrromethene 546) 是一种亲脂性荧光探针,Ex/Em 为 493/503 nm。 BODIPY 493/503 定位于极性脂质,可用于标记细胞中性脂质含量以及活细胞和固定细胞应用。
T11820 LAT1-IN-1

2-氨基-2-去甲菠烷羧酸,BCH

Apoptosis; Others Apoptosis; Others
LAT1-IN-1 (BCH) 是 L 型氨基酸转运蛋白 1 的选择性竞争性抑制剂,显着抑制细胞对氨基酸的摄取和 mTOR 磷酸化,从而诱导抑制癌症生长和细胞凋亡。
T0674 Lansoprazole

兰索拉唑,A-65006,AG-1749

Proton pump; Phospholipase; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Lansoprazole (A-65006) 是一种可抑制胃酸生成的质子泵抑制剂。它是中性鞘磷脂酶的外泌体抑制剂。
T1021 (R)-Lansoprazole

Dexlansoprazole,右旋兰索拉唑,T 168390,TAK 390,R-(+)-Lansoprazole

Proton pump Membrane transporter/Ion channel
(R)-Lansoprazole (T 168390) 是Lansoprazole 的R 型异构体。Lansoprazole 是口服有效的质子泵抑制剂,能抑制胃酸生成。Lansoprazole 是中性鞘磷脂酶(N-SMase)的抑制剂(外泌体抑制剂),能透过血脑屏障。
T22391 Omeprazole Sodium

P450; Proton pump; Antibacterial; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Omeprazole 是有效的质子泵抑制剂,在胃肠道疾病的研究中具有价值。它竞争性抑制CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阴性菌和革兰氏阳性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。
T2086 ELN-441958

ELN 441958

Bradykinin Receptor GPCR/G Protein
ELN-441958是一种B1受体拮抗剂,能够抑制B1激动剂配体[3H] DAKD 与IMR-90细胞结合(Ki:0.26 nM),相较于B2受体,它对B1受体的抑制作用具有更高的选择性,且比抑制μ阿片受体选择性高500多倍,比抑制δ阿片受体选择性高2000多倍。
T40194 MeAIB

α-(Methylamino)isobutyric acid

Others Others
MeAIB 是一种n -乙酰转移酶抑制剂,抑制SNAT2相关信号通路。MeAIB 是氨基酸转运系统a (ATA1)的特异性底物。氨基酸转运系统a (ATA1)以Na+流动调控短链中性氨基酸的摄取。
TP1917L1 Sar-[D-Phe8]-des-Arg9-Bradykinin acetate

Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base)

Bradykinin Receptor GPCR/G Protein
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) 是一种有效的选择性缓激肽 B1 受体激动剂(兔主动脉中的 EC50 = 9.02 nM),对氨肽酶、激肽酶 I 和 II (ACE) 以及中性内肽酶切割具有抗性。在体内表现出降血压和血管生成活性。
T3627 IQ-1S free acid

IQ-1,IQ-1S,IQ-1S (free acid)

NF-κB; JNK MAPK; NF-κB
IQ-1S free acid (IQ-1S) 是 NF-κB/激活蛋白1 (AP-1) 抑制剂(IC50:2.3±0.41 μM)。它对 JNK1(Kd:240 nM)、JNK2(Kd:360 nM) 和 JNK3(Kd:100 nM)的都具有高的结合亲和力 。
T4019 Cambinol

SIRT1/2 Inhibitor IV,NSC 112546

Apoptosis; Phospholipase; Sirtuin Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Cambinol (SIRT1/2 Inhibitor IV) 是一种SIRT1和SIRT2的抑制剂,IC50值分别为 56 μM 和 59 μM。它是中性鞘磷脂酶的外泌体抑制剂。
T10491 Galidesivir

BCX4430,Immucillin-A

Others Others
Galidesivir (BCX4430) 是一种广谱抗病毒化合物,是一种腺苷类似物,能抑制病毒 RNA 依赖的 RNA 聚合酶 (RdRp) 活性。Galidesivir 在体外对多种 RNA 病毒病原体有抑制作用,可减少受感染动物的肺部感染。
T10671 Candoxatril

UK 79300

Others Others
Candoxatril is an inhibitor neutral endopeptidase (NEP).
T28721 Sch 47896

Sch47896,Sch-47896

Sch 47896 is an inhibitor of neutral metalloendopeptidase (NEP).
T28715 Sch 34826

Sch34826,Sch-34826

Sch 34826 is a potent, selective neutral endopeptidase inhibitor.
T23698 Aladotril

BP1137,BP 1137,BP-1137

Aladotril is an inhibitor of neutral endopeptidase. Its prodrug is aladotrilat.
T12994 SQ28603

Squibb 28603,SQ28,603

Others Others
SQ28603 is a potent and selective neutral endopeptidase 3.4.24.11 (NEP) inhibitor.
T22563 AM6545

Others Others
CB1 selective neutral antagonist
T12936 SMP-028

Others Others
SMP-028 is a neutral cholesterol esterase (CEase) inhibitor(IC50 : 1.01 μM).
T70567 CGS 25462

CGS 25462 is a neutral endopeptidase (NEP) inhibitor.
T39124 BAY 1217224

BAY 1217224 is a neutral, non-prodrug Thrombin inhibitor with good oral pharmacokinetics.
T29053 UK-447841

UK 447841

UK-447841, a neutral endopeptidase (NEP) inhibitor, is used potentially for the treatment of female sexual dysfunction.
T28726 SCH-39370

SCH 39370

SCH-39370 is a potent and specific neutral metalloendopeptidase (NEP) inhibitor.
T21219 Isatin-O

Isatin-3-oxime

Isatin-O acts as a neutral BBB crossing reactivator for acetylcholinesterase inhibited by paraoxon and is also an anticonvulsant.
T31598 Ecadotril

S.049,BAY-y 7432,BAY y 7432,BP 1.02,S049

Ecadotril is a neutral endopeptidase (NEP) inhibitor, which plays an anti hypertensive role.
T23699 Aladotrilat

Fasidotrilat

Aladotrilat is an inhibitor of neutral endopeptidase. Its prodrug is aladrotril.

化合物

Neutral red
Cat.No: T20549
Synonym:
Target: Others
Coriphosphine
Cat.No: T31012
Synonym: Neutral Yellow
Target:
Clivorine
Cat.No: T30970
Synonym: J1.344.443I,Clivorine (neutral)
Target:
Thiorphan
Cat.No: T7693
Synonym:
Target: Neprilysin
DCB
Cat.No: T22711
Synonym: 3,3'-dichlorobenzaldazine
Target: Others, GluR
Sacubitrilat
Cat.No: TQ0106
Synonym: LBQ-657
Target: Neprilysin
N6-Methyladenosine 5’-monophos phate triethylammonium salt (neutral 4229-50-9)
Cat.No: TNU1631
Synonym:
Target:
Cinromide
Cat.No: T0413
Synonym: 醒隆酰胺,trans-3-Bromo-N-ethylcinnamamide
Target: Others
2’-O-Methyl-N6-methyladenosine 5’-monophosphate triethylammonium salt (60091-05-6 neutral molecule)
Cat.No: TNU1630
Synonym:
Target:
Nile Red
Cat.No: T19033
Synonym: Phenoxazone 9,尼罗红,Nile Blue A oxazone
Target: Others
Sacubitril
Cat.No: T4574
Synonym: AHU 377,AHU377,沙库必曲,AHU-377
Target: Neprilysin
Sacubitril hemicalcium salt
Cat.No: T4200
Synonym: AHU-377 (hemicalcium salt),LCZ696中间体,AHU377 calcium salt
Target: Neprilysin
Racecadotril
Cat.No: T1176
Synonym: Acetorphan,消旋卡多曲
Target: Neprilysin, Proteasome
Sacubitril/Valsartan
Cat.No: T2318
Synonym: Sacubitril mixture with Valsartan,沙库必曲/缬沙坦,Valsartan,Sacubitril,LCZ696
Target: Apoptosis, RAAS, Neprilysin
L-4FPG
Cat.No: T21102
Synonym: L-4-氟苯甘氨酸,L4FPG,L 4FPG
Target: Others
DPTIP
Cat.No: T60043
Synonym:
Target: Phospholipase
NEP-IN-1
Cat.No: T10918
Synonym:
Target: Neprilysin
LHW090-A7
Cat.No: T19626
Synonym: (ALPHAS)-3'-氯-ALPHA-[[(1S)-2-乙氧基-1-甲基-2-氧代乙基]氨基][1,1'-联苯]-4-丙酸
Target: Neprilysin
HEPES
Cat.No: T8549
Synonym:
Target: Others
Omeprazole
Cat.No: T0757
Synonym: Losec,Prilosec,奥美拉唑,奥美拉挫,H 16868,Antra
Target: Proton pump, Phospholipase, Antibacterial, Autophagy
o-Phenanthroline monohydrate
Cat.No: T7449
Synonym: Phenanthroline monohydrate,1, 10-Phenanthroline monohydrate,邻菲罗啉
Target: MMP
GMQ hydrochloride
Cat.No: T8617
Synonym: NSC 403387 hydrochloride
Target: Others
DOPE
Cat.No: T19080
Synonym: 1,2-二油酰-SN-甘油-3-磷酰乙醇胺
Target: Others
(Rac)-Daglutril
Cat.No: T27119L
Synonym: SLV 306 acetic acid,2-((3S)-3-(1-(2-(ethoxycarbonyl)-4-phenylbutyl)cyclopentane-1-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)acetic acid
Target: Others
GW4869
Cat.No: T3640
Synonym: GW554869A,GW 4869,GW69A
Target: Phospholipase
BODIPY 493/503
Cat.No: T36957
Synonym: BDP 493/503 lipid stain,Pyrromethene 546
Target: Others
LAT1-IN-1
Cat.No: T11820
Synonym: 2-氨基-2-去甲菠烷羧酸,BCH
Target: Apoptosis, Others
Lansoprazole
Cat.No: T0674
Synonym: 兰索拉唑,A-65006,AG-1749
Target: Proton pump, Phospholipase, Antibacterial
(R)-Lansoprazole
Cat.No: T1021
Synonym: Dexlansoprazole,右旋兰索拉唑,T 168390,TAK 390,R-(+)-Lansoprazole
Target: Proton pump
Omeprazole Sodium
Cat.No: T22391
Synonym:
Target: P450, Proton pump, Antibacterial, Autophagy
ELN-441958
Cat.No: T2086
Synonym: ELN 441958
Target: Bradykinin Receptor
MeAIB
Cat.No: T40194
Synonym: α-(Methylamino)isobutyric acid
Target: Others
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Cat.No: TP1917L1
Synonym: Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base)
Target: Bradykinin Receptor
IQ-1S free acid
Cat.No: T3627
Synonym: IQ-1,IQ-1S,IQ-1S (free acid)
Target: NF-κB, JNK
Cambinol
Cat.No: T4019
Synonym: SIRT1/2 Inhibitor IV,NSC 112546
Target: Apoptosis, Phospholipase, Sirtuin
Galidesivir
Cat.No: T10491
Synonym: BCX4430,Immucillin-A
Target: Others
Candoxatril
Cat.No: T10671
Synonym: UK 79300
Target: Others
Sch 47896
Cat.No: T28721
Synonym: Sch47896,Sch-47896
Target:
Sch 34826
Cat.No: T28715
Synonym: Sch34826,Sch-34826
Target:
Aladotril
Cat.No: T23698
Synonym: BP1137,BP 1137,BP-1137
Target:
SQ28603
Cat.No: T12994
Synonym: Squibb 28603,SQ28,603
Target: Others
AM6545
Cat.No: T22563
Synonym:
Target: Others
SMP-028
Cat.No: T12936
Synonym:
Target: Others
CGS 25462
Cat.No: T70567
Synonym:
Target:
BAY 1217224
Cat.No: T39124
Synonym:
Target:
UK-447841
Cat.No: T29053
Synonym: UK 447841
Target:
SCH-39370
Cat.No: T28726
Synonym: SCH 39370
Target:
Isatin-O
Cat.No: T21219
Synonym: Isatin-3-oxime
Target:
Ecadotril
Cat.No: T31598
Synonym: S.049,BAY-y 7432,BAY y 7432,BP 1.02,S049
Target:
Aladotrilat
Cat.No: T23699
Synonym: Fasidotrilat
Target:
Cat. No. Product Name Target Signaling Pathways
T6627 Phosphoramidon Disodium

Phosphoramidon Disodium Salt,磷酰胺二钠

RAAS; Neprilysin; Others Endocrinology/Hormones; Metabolism; Others
Phosphoramidon Disodium (Phosphoramidon Disodium Salt) Salt 是一种金属蛋白酶 (metalloprotease) 抑制剂 。Phosphoramidon Disodium Salt 抑制内皮素转化酶 (ECE) ,中性肽内切酶 (NEP) 和血管紧张素转换酶 (ACE) 的IC50分别为 3.5 ,0.034 和 78 μM。
T1214 Ribostamycin sulfate

Vistamycin sulfate,硫酸核糖霉素

Antibacterial; Antibiotic Microbiology/Virology
Ribostamycin sulfate (Vistamycin sulfate) 是一种广谱抗菌剂, 在30S 和50S 核糖体亚基结合抑制细菌蛋白质合成, 还抑制蛋白二硫键异构酶分子伴侣活性, 用于药代动力学和肾毒性研究。
T9135 Epirosmanol

Others Others
Epirosmanol 是含有内酯部分的二萜类化合物。 Epirosmanol 是一种极弱碱性(基本中性)的化合物(基于其 pKa)。
TN5131 Tetrahydrocannabivarin

THCV,delta9-Tetrahydrocannabivarin,CRM,Tetrahydrocannavarin

Cannabinoid Receptor GPCR/G Protein
Tetrahydrocannabivarin (CRM) 是 cannabinoid type 1 receptor 的中性拮抗剂,对 2 型糖尿病有潜在治疗价值。
T8032 4-Pentenoic acid

Others; Endogenous Metabolite Metabolism; Others
4-Pentenoic acid 是内源性代谢产物的一种。
T3739 2,6-Dimethoxyquinone

2,6-Dimethoxy-1,4-benzoquinone,2,6-Dimethoxy-p-benzoquinone,2,6-Dimethoxybenzoquinone,2,6-二甲氧基-1,4-苯醌

Others Others
2,6-Dimethoxyquinone (2,6-Dimethoxy-p-benzoquinone) 是一种植物中提取吸脂诱导因子。它具有抗脂肪、抗癌、抗菌、抗疟疾和抗炎的作用。
T1168 Desonide

Tridesilon,地索奈德,Locapred,Prednacinolone

Glucocorticoid Receptor Endocrinology/Hormones
Desonide (Prednacinolone) 是一种非氟化皮质类固醇抗炎剂,能够作用于糖皮质激素受体。
T8105 Indole-3-carboxaldehyde

3-Formylindole,3-吲哚甲醛

Endogenous Metabolite Metabolism
Indole-3-carboxaldehyde (3-Formylindole) 是由黄化豌豆幼苗的粗酶制剂氧化降解IAA 的产物,是一种卷心菜提取物。它可用于制备吲哚类植物抗毒素环芸香素类似物。
T8098 γ-Hexalactone

γ-caprolactone,gamma-己内酯,γ-己内酯

Others Others
γ-Hexalactone (γ-caprolactone) 是一种存在成熟水果中的 gamma 内酯。它会导致 DNA 损伤,可用作对氧磷酶 1 的底物 (PON1)。
T81764 Monofucosyllacto-N-hexaose III

MFLNH III

Monofucosyllacto-N-hexaose III(MFLNH III)是一种具有特定生物学功能的中性人乳寡糖(HMO)。
T19676 Tributyrin

NSC661583,NSC 661583,NSC-661583,甘油三丁酸酯

Apoptosis Apoptosis
Tributyrin (Glyceryl tributyrate) 是一种中性短链脂肪酸甘油三酯,是一种稳定且吸收迅速的丁酸前药。 它通过生物膜扩散并被细胞内脂肪酶代谢,在体内将有效的丁酸直接释放到细胞中,有抗增殖、促凋亡和诱导分化作用。
T79989 Funiculosin

Antibiotic Microbiology/Virology
Funiculosin为一种中性亲脂性抗生素,能够抑制DNA及RNA病毒,并具备抗真菌活性。在初级鸡胚成纤维细胞中,Funiculosin可有效抑制致病真菌引发的感染。
T35577 Phosphatidylserines (bovine)

Phosphatidylserine is a naturally occurring phospholipid that comprises 2-10% of total phospholipids in mammals and is enriched in the central nervous system, particularly the retina. It is anionic and found mainly on the inner leaflet of the cell membrane. It is biosynthesized from phosphatidylcholine or phosphatidylethanolamine by phosphatidyl synthase 1 (PSS1) or PSS2, respectively, in the endoplasmic reticulum and can be reversibly converted back by the same enzymes. It can also be irreversi...

天然产物

Phosphoramidon Disodium
Cat.No: T6627
Synonym: Phosphoramidon Disodium Salt,磷酰胺二钠
Target: RAAS, Neprilysin, Others
Ribostamycin sulfate
Cat.No: T1214
Synonym: Vistamycin sulfate,硫酸核糖霉素
Target: Antibacterial, Antibiotic
Epirosmanol
Cat.No: T9135
Synonym:
Target: Others
Tetrahydrocannabivarin
Cat.No: TN5131
Synonym: THCV,delta9-Tetrahydrocannabivarin,CRM,Tetrahydrocannavarin
Target: Cannabinoid Receptor
4-Pentenoic acid
Cat.No: T8032
Synonym:
Target: Others, Endogenous Metabolite
2,6-Dimethoxyquinone
Cat.No: T3739
Synonym: 2,6-Dimethoxy-1,4-benzoquinone,2,6-Dimethoxy-p-benzoquinone,2,6-Dimethoxybenzoquinone,2,6-二甲氧基-1,4-苯醌
Target: Others
Desonide
Cat.No: T1168
Synonym: Tridesilon,地索奈德,Locapred,Prednacinolone
Target: Glucocorticoid Receptor
Indole-3-carboxaldehyde
Cat.No: T8105
Synonym: 3-Formylindole,3-吲哚甲醛
Target: Endogenous Metabolite
γ-Hexalactone
Cat.No: T8098
Synonym: γ-caprolactone,gamma-己内酯,γ-己内酯
Target: Others
Monofucosyllacto-N-hexaose III
Cat.No: T81764
Synonym: MFLNH III
Target:
Tributyrin
Cat.No: T19676
Synonym: NSC661583,NSC 661583,NSC-661583,甘油三丁酸酯
Target: Apoptosis
Funiculosin
Cat.No: T79989
Synonym:
Target: Antibiotic
Phosphatidylserines (bovine)
Cat.No: T35577
Synonym:
Target:
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