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77

抑制剂 & 化合物

12

天然产物

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Cat. No. Product Name Target Signaling Pathways
T10511 Anti-hypertensive sulfonanilide 1

Others Others
Anti-hypertensive sulfonanilide 1 is an antihypertensive compound.
T3474 RO 46-8443

Endothelin Receptor GPCR/G Protein
Ro 46-844 是选择性非肽内皮素受体拮抗剂。它对ETB(IC50: 34-69 nM) 的选择性比ETA 受体 (IC50: 6800 nM) 高的100倍以上。
T22398 Phenidone

菲尼酮,1-phenyl-3-pyrazolidinone

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenidone (1-phenyl-3-pyrazolidinone) 是可口服发环氧化酶和脂氧合酶双重抑制剂,可改善实验性自身免疫性脑脊髓炎大鼠的瘫痪,降低自发性高血压大鼠的血压,可用作照片显像剂。
T0993 Methoxamine hydrochloride

Methoxamine HCl,盐酸甲氧明

Adrenergic Receptor GPCR/G Protein; Neuroscience
Methoxamine hydrochloride (Methoxamine HCl) 是一种 alpha1 肾上腺素能受体的选择性激动剂。它通过 Prazosin 敏感机制在兔肺动脉显著增加 ATP、ADP 和 AMP 的溢出,但不增加腺苷的溢出。它引起血管收缩和外周血管阻力增加。
T28482 Firibastat

QGC 001,QGC-001,RB-150,RB150,QGC001,RB 150

Aminopeptidase Metabolism
Firibastat (RB150) 是一种具有口服活性的 EC33 前体药物。Firibastat 是一种首创的脑氨基肽酶 A(APA) 抑制剂 (Ki=200 nM),选择性地抑制高血压大鼠脑血管紧张素 II 转化为血管紧张素 III,降低血压。
T5329 Trandolapril

Angiotensin-converting Enzyme (ACE) Metabolism
Trandolapril 是 Trandolaprilat 的前体药物。Trandolapril 是一种口服血管紧张素转换酶抑制剂,在高血压和充血性心力衰竭及心肌梗死领域有研究价值。
T0287 Hexamethonium Bromide

Gangliostat,溴化六甲铵,Simpatoblock,六甲溴铵,Hexamethonium Dibromide

Apoptosis; Dopamine Receptor; AChR Apoptosis; GPCR/G Protein; Neuroscience
Hexamethonium Bromide (Hexamethonium Dibromide) 是神经节中神经元型烟碱型 AChR 的特异性拮抗剂。在自发性高血压动物模型中,它能降低其交感神经活动和血压。
T22236 Alprenolol hydrochloride

阿普洛尔盐酸盐,盐酸阿普洛尔

5-HT Receptor GPCR/G Protein; Neuroscience
Alprenolol hydrochloride 是一种非选择性β受体阻滞剂,也是5-HT1A 受体拮抗剂。
T3046 BMY 7378 dihydrochloride

BMY7378 HCl

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
BMY 7378 dihydrochloride (BMY7378 HCl) 是选择性 α1D 肾上腺素受体拮抗剂,也是5-HT1A 受体部分激动剂。它同表达克隆大鼠 α1D-AR 的膜结合的亲和力 (Ki=2 nM)  是同克隆大鼠 α1A-AR (Ki=800 nM) 或仓鼠 α1B-AR (Ki=600 nM) 结合的亲和力 的100 以上。
T9097 Guanadrel

Others Others
Guanadrel 是一种抗高血压药。
T1615 Irbesartan

厄贝沙坦,SR-47436,BMS-186295

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Irbesartan (SR-47436) 是一种 1 型血管紧张素 II 受体拮抗剂,IC50为1.3 nM。
T23044 N,N'-Dicyclohexylurea

DCU,1,3-Dicyclohexylurea,NSC 17013,Dicyclohexylurea,Dicyclohexylcarbodiamide,AURORA KA-3582,N,N-二环己脲

Epoxide Hydrolase Metabolism
N,N'-Dicyclohexylurea (AURORA KA-3582) 是一种可溶性环氧化物水解酶 (sEH) 抑制剂。
T6835 Fenoldopam mesylate

Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526,非诺多泮甲磺酸盐

Dopamine Receptor GPCR/G Protein; Neuroscience
Fenoldopam mesylate (Corlopam mesylate) 是一种多巴胺受体D1选择性激动剂。
T80661 Antihypertensive sulfonanilide XVII

Others Others
Antihypertensive sulfonanilide XVII 是一种可口服的抗高血压磺酰苯胺类小分子化合物,可用于研究高血压。
T79267 Antihypertensive agent 3

Antihypertensive agent 3 (compound 4a) 是一种针对血管紧张素 II 受体 1(AT1) 的拮抗剂,其在自发性高血压大鼠(SHRs)的模型中表现出显著的降压效果。
T79266 Antihypertensive agent 2

Antihypertensive agent 2 (Compound 4g) 为一种有效的血管紧张素 II 受体 1 拮抗剂,其降血压效能可与Losartan媲美或更胜一筹。
T16329 Nitroflurbiprofen

NO-flurbiprofen,Nitroxybutyl flurbiprofen,硝基氟比洛芬,HCT 1206

COX Immunology/Inflammation; Neuroscience
Nitroflurbiprofen (Nitroxybutyl flurbiprofen) 是一种释放 NO 的环氧合酶抑制剂,可调节门脉高压性肝硬化大鼠肝内血管张力的增加。
T17111 Todralazine hydrochloride

Ecarazine hydrochloride,盐酸托屈嗪

Adrenergic Receptor GPCR/G Protein; Neuroscience
Todralazine hydrochloride (Ecarazine hydrochloride) 是一种 β2AR 阻滞剂,具有抗氧化和自由基清除活性。 Todralazine hydrochloride 可用于抗高血压的研究。
T14942 CGP48369

RAAS Endocrinology/Hormones
CGP48369 是一种有效的血管紧张素 II 受体 (angiotensin II receptor) 拮抗剂,具有降血压作用,可增强自发性高血压大鼠冠状动脉的内皮依赖性松弛。
T2528 Latanoprost

Xalatan,PHXA41,拉坦前列腺素,拉坦前列素

GPR; Prostaglandin Receptor; RAR/RXR  Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism
Latanoprost (Xalatan) 是前列腺素 F2α 类似物,是一种前列腺素受体激动剂,能够降低眼内压。
T0126 Diazoxide

氯甲苯噻嗪,二氮嗪,SRG-95213,Sch-6783,Proglycem

ATPase; Potassium Channel; Autophagy Autophagy; Membrane transporter/Ion channel
Diazoxide (Proglycem) 是一种 ATP 敏感性的钾离子通道激活剂,是一种苯并噻二嗪衍生物,是一种用于高血压急症的外周血管扩张剂。
T36506 Tempone

4-Oxo-tempo

Tempone 是一种氨基氧烷,具有自由基清除剂的作用,会与活性氧(ROS)发生反应。静脉注射 Tempone 可降低自发性高血压大鼠的平均动脉。
T10595 BQ-788

BQ788

Endothelin Receptor GPCR/G Protein
BQ-788 是一种具有选择性和有效性的 ETB 受体拮抗剂,具有潜在的高血压活性,抑制 ET-1 与 ETB 受体结合,抑制外源性 ET-1 诱导的冠状动脉灌注压升高。
T37496L Alamandine TFA

RAAS Endocrinology/Hormones
Alamandine TFA 是肾素-血管紧张素系统 (RAS) 的成员,是一种血管活性肽,是 G 蛋白偶联受体 MrgD 的内源性配体。它通过抗高血压作用来保护肾脏和心脏。
T24932 Vatanidipine

AE-0047,AE 0047,AE0047

Calcium Channel Membrane transporter/Ion channel; Metabolism
Vatanidipine (AE0047) 是一种新型的双氢吡啶(DHP)型钙通道阻滞剂,具有缓慢起效的药理作用。在各种实验性高血压模型中观察到缓慢起效和持久的降压作用。
T1275 Phentolamine mesylate

Phentolamine methanesulfonate,甲磺酸酚妥拉明,Phentolamine mesilate

Adrenergic Receptor GPCR/G Protein; Neuroscience
Phentolamine mesylate (Phentolamine methanesulfonate) 是一种非选择性的、可逆的,具有口服活性的 α1 和 α2 肾上腺素能受体阻滞剂,能够扩张使血管,降低周围血管阻力。它可用于研究嗜铬细胞瘤相关的高血压,心力衰竭和勃起功能障碍。
T12596 (4E)-SUN9221

5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
(4E)-SUN9221 是一种有效的 α1-adrenergic 受体和 5-HT2 受体双重拮抗剂,在高血压大鼠中显示出抗高血压和抗血小板聚集活性。
T20570 Labetalol

Apo-Labetalol,Albetol,Trandate,Dilevalol,拉贝洛尔,Normodyne

Adrenergic Receptor GPCR/G Protein; Neuroscience
Labetalol (Apo-Labetalol) 是一种抗高血压药物,可用于心血管疾病的研究,如妊娠期高血压。它是一种口服具有活性的选择性 α1- 和非选择性 β-肾上腺素能受体 (adrenergic receptor) 竞争性拮抗剂。
T31598 Ecadotril

S.049,BAY-y 7432,BAY y 7432,BP 1.02,S049

Ecadotril is a neutral endopeptidase (NEP) inhibitor, which plays an anti hypertensive role.
T24478 MK-8141

MK 8141,ACT 077825,ACT077825,ACT-077825

MK-8141 is a renin inhibitor. It displays some antihypertensive efficacy in hypertensive patients.
T34945 Trimazosin hydrochloride

CP19106-1,CP 19106-1,Trimazosin HCl,CP-19106-1

Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.
T28039 Milfasartan

LR-B081,LRB-081,LR-B-081,LRB 081,LR-B 081

Milfasartan is a potent, selective antagonist of AT1 receptor with oral activity. It markedly lowers the blood-pressure in conscious renal and spontaneously hypertensive rats.
T17112 Todralazine

Ecarazine

Others Others
Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.
T71396 FCE-24379

FCE-24379 is a selective antagonist of vascular serotonin receptors that has been shown to lowers blood pressure in hypertensive rats.
T38424 (R)-Fadrozole

FAD286,(R)-CGS 16949A free base,(R)-Fadrozole

(R)-Fadrozole ((R)-CGS 16949A; FAD286) is a potent nonsteroidal inhibitor. (R)-Fadrozole also inhibits human placental aromatase (pIC 50 = 6.17) and aldosterone biosynthesis. (R)-Fadrozole reverses cardiac fibrosis in spontaneously hypertensive heart failure rats..
T40688 Fulvine

Fulvine, a pyrrolizidine alkaloid extracted from Crotalaria fulva seeds, exhibits hepatotoxic properties and can be employed for inducing hypertensive pulmonary vascular disease in vivo.
T21416 Hydroflumethiazide

Diurometon,Glomerulin,Diuredemina,Flutizide,Hidroflumetiazid

Hydroflumethiazide is a thiazide diuretic. It has also shown the activity of anti-hypertensive.
T27743 KRH-594 free acid

WK14922K,WK-1492,WK-14922K,WK1492

KRH-594 is a potent, specific and insurmountable AT1 receptor antagonist. KRH-594 ameliorates hyperlipidaemia and nephropathy in diabetic spontaneously hypertensive rats. KRH-594 prevents end-organ damage in stroke-prone spontaneously hypertensive/Izm ra
T13328 AE0047 Hydrochloride

Calcium Channel Membrane transporter/Ion channel; Metabolism
AE0047 Hydrochloride is a blocker of calcium, and used in the research of the hypertensive disease.
T27306 Fasidotril

BP 1137,BP1137,BP-1.137,BP1.137,BP-1137,BP 1.137

Fasidotril is a NEP/ACE inhibitor. Fasidotril was an effective oral antihypertensive agent during chronic treatment in high-renin renovascular rats, normal-renin SHR, and low-renin DOCA-salt hypertensive rats and in patients with essential hypertension.
T11642 Imidaprilate

Imidaprilat,6366A

RAAS Endocrinology/Hormones
Imidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin-converting enzyme (ACE) inhibitor (IC50: 2.6 nM). It is used in the research of the hypertensive disease.
T78063 Endothelin-1 (1-31) (Human) TFA

ERK MAPK
Endothelin-1 (1-31) (Human) TFA 是源自chymase对大ET-1选择性水解的一种有效血管收缩剂和血压升高剂。
TP2126 R 892

Potent and selective bradykinin B1 receptor antagonist (ID50 values are 2.8 and > 600 nM at B1 and B2 receptors respectively). Exhibits no intrinsic agonist activity and is resistant to aminopeptidase and kininase II (ACE) cleavage. Displays hypertensive
T26802 BIBS-222

BIBS 222

BIBS-222, a nonpeptide angiotensin II (Ang II) receptor antagonist, appears to be an effective antihypertensive in the model of the renal hypertensive rat.
T15680 L-159282

MK 996

Others Others
L-159282 is an orally active and nonpeptide angiotensin II receptor antagonist. It also has anti-hypertensive activity.
T81681 Neuromedin U-25 (porcine)

Neuromedin U-25 (porcine) 是一类具有子宫刺激和升高血压作用的肽。
T14672 BMS-248360

Others Others
BMS-248360 is a potent and orally active dual antagonist of both angiotensin II receptor (AT1) and endothelin A (ETA) receptor. With Kis of 10 nM and 1.9 nM for hAT1 and hETA receptor, respectively. BMS-248360 shows hypertensive effects[1].
T71065 Quinapril-d5

Quinapril-d5 is intended for use as an internal standard for the quantification of quinapril by GC- or LC-MS. Quinapril is a prodrug form of the angiotensin converting enzyme (ACE) inhibitor quinaprilat. In vivo, quinapril reduces mean arterial pressure in renal hypertensive and spontaneously hypertensive rats. It inhibits angiotensin I-induced pressor responses in normotensive rats and dogs. Quinapril prevents left ventricular heart failure in CHF 14.6 cardiomyopathic hamsters. Formulations con...
T62288 AD013

AD013 是一种双重的 cACE 和 NEP 抑制剂。AD013 是通过 C 域选择性 ACE 抑制剂赖诺普利-色氨酸合成。AD013 具有潜力提供强效抗高血压和心脏保护作用。
TP1892 γ1-MSH

Endogenous melanocortin MC3 receptor agonist (pKi = 7.46) that displays ~ 40-fold selectivity over MC4. Increases the release of extracellular dopamine, which induces grooming and vertical activity (rearing) in rats. Exhibits hypertensive, tachycardic and

化合物

Anti-hypertensive sulfonanilide 1
Cat.No: T10511
Synonym:
Target: Others
RO 46-8443
Cat.No: T3474
Synonym:
Target: Endothelin Receptor
Phenidone
Cat.No: T22398
Synonym: 菲尼酮,1-phenyl-3-pyrazolidinone
Target: Lipoxygenase, COX
Methoxamine hydrochloride
Cat.No: T0993
Synonym: Methoxamine HCl,盐酸甲氧明
Target: Adrenergic Receptor
Firibastat
Cat.No: T28482
Synonym: QGC 001,QGC-001,RB-150,RB150,QGC001,RB 150
Target: Aminopeptidase
Trandolapril
Cat.No: T5329
Synonym:
Target: Angiotensin-converting Enzyme (ACE)
Hexamethonium Bromide
Cat.No: T0287
Synonym: Gangliostat,溴化六甲铵,Simpatoblock,六甲溴铵,Hexamethonium Dibromide
Target: Apoptosis, Dopamine Receptor, AChR
Alprenolol hydrochloride
Cat.No: T22236
Synonym: 阿普洛尔盐酸盐,盐酸阿普洛尔
Target: 5-HT Receptor
BMY 7378 dihydrochloride
Cat.No: T3046
Synonym: BMY7378 HCl
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Guanadrel
Cat.No: T9097
Synonym:
Target: Others
Irbesartan
Cat.No: T1615
Synonym: 厄贝沙坦,SR-47436,BMS-186295
Target: Apoptosis, RAAS
N,N'-Dicyclohexylurea
Cat.No: T23044
Synonym: DCU,1,3-Dicyclohexylurea,NSC 17013,Dicyclohexylurea,Dicyclohexylcarbodiamide,AURORA KA-3582,N,N-二环己脲
Target: Epoxide Hydrolase
Fenoldopam mesylate
Cat.No: T6835
Synonym: Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526,非诺多泮甲磺酸盐
Target: Dopamine Receptor
Antihypertensive sulfonanilide XVII
Cat.No: T80661
Synonym:
Target: Others
Antihypertensive agent 3
Cat.No: T79267
Synonym:
Target:
Antihypertensive agent 2
Cat.No: T79266
Synonym:
Target:
Nitroflurbiprofen
Cat.No: T16329
Synonym: NO-flurbiprofen,Nitroxybutyl flurbiprofen,硝基氟比洛芬,HCT 1206
Target: COX
Todralazine hydrochloride
Cat.No: T17111
Synonym: Ecarazine hydrochloride,盐酸托屈嗪
Target: Adrenergic Receptor
CGP48369
Cat.No: T14942
Synonym:
Target: RAAS
Latanoprost
Cat.No: T2528
Synonym: Xalatan,PHXA41,拉坦前列腺素,拉坦前列素
Target: GPR, Prostaglandin Receptor, RAR/RXR 
Diazoxide
Cat.No: T0126
Synonym: 氯甲苯噻嗪,二氮嗪,SRG-95213,Sch-6783,Proglycem
Target: ATPase, Potassium Channel, Autophagy
Tempone
Cat.No: T36506
Synonym: 4-Oxo-tempo
Target:
BQ-788
Cat.No: T10595
Synonym: BQ788
Target: Endothelin Receptor
Alamandine TFA
Cat.No: T37496L
Synonym:
Target: RAAS
Vatanidipine
Cat.No: T24932
Synonym: AE-0047,AE 0047,AE0047
Target: Calcium Channel
Phentolamine mesylate
Cat.No: T1275
Synonym: Phentolamine methanesulfonate,甲磺酸酚妥拉明,Phentolamine mesilate
Target: Adrenergic Receptor
(4E)-SUN9221
Cat.No: T12596
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor
Labetalol
Cat.No: T20570
Synonym: Apo-Labetalol,Albetol,Trandate,Dilevalol,拉贝洛尔,Normodyne
Target: Adrenergic Receptor
Ecadotril
Cat.No: T31598
Synonym: S.049,BAY-y 7432,BAY y 7432,BP 1.02,S049
Target:
MK-8141
Cat.No: T24478
Synonym: MK 8141,ACT 077825,ACT077825,ACT-077825
Target:
Trimazosin hydrochloride
Cat.No: T34945
Synonym: CP19106-1,CP 19106-1,Trimazosin HCl,CP-19106-1
Target:
Milfasartan
Cat.No: T28039
Synonym: LR-B081,LRB-081,LR-B-081,LRB 081,LR-B 081
Target:
Todralazine
Cat.No: T17112
Synonym: Ecarazine
Target: Others
FCE-24379
Cat.No: T71396
Synonym:
Target:
(R)-Fadrozole
Cat.No: T38424
Synonym: FAD286,(R)-CGS 16949A free base,(R)-Fadrozole
Target:
Fulvine
Cat.No: T40688
Synonym:
Target:
Hydroflumethiazide
Cat.No: T21416
Synonym: Diurometon,Glomerulin,Diuredemina,Flutizide,Hidroflumetiazid
Target:
KRH-594 free acid
Cat.No: T27743
Synonym: WK14922K,WK-1492,WK-14922K,WK1492
Target:
AE0047 Hydrochloride
Cat.No: T13328
Synonym:
Target: Calcium Channel
Fasidotril
Cat.No: T27306
Synonym: BP 1137,BP1137,BP-1.137,BP1.137,BP-1137,BP 1.137
Target:
Imidaprilate
Cat.No: T11642
Synonym: Imidaprilat,6366A
Target: RAAS
Endothelin-1 (1-31) (Human) TFA
Cat.No: T78063
Synonym:
Target: ERK
R 892
Cat.No: TP2126
Synonym:
Target:
BIBS-222
Cat.No: T26802
Synonym: BIBS 222
Target:
L-159282
Cat.No: T15680
Synonym: MK 996
Target: Others
Neuromedin U-25 (porcine)
Cat.No: T81681
Synonym:
Target:
BMS-248360
Cat.No: T14672
Synonym:
Target: Others
Quinapril-d5
Cat.No: T71065
Synonym:
Target:
AD013
Cat.No: T62288
Synonym:
Target:
γ1-MSH
Cat.No: TP1892
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8158 Tilianin

香清兰苷,田蓟苷

Others Others
Tilianin 是一种广泛存在于多种药用植物中的活性黄酮类苷,具有降压、保护心肌、降血脂、抗糖尿病、抗炎、抗氧化等作用。
T6S1369 Vitexin

牡荆素,Apigenin-8-C-glucoside

Antioxidant oxidation-reduction
Vitexin 是一种存在于多种药用植物(如榕树、螺旋藻)中的 c-糖基化的黄酮。 它具有广泛的药理作用,包括抗氧化,抗癌,抗炎,抗痛觉过敏和神经保护作用。
T8044 Ajmalicine

阿吗里新,Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin

Adrenergic Receptor GPCR/G Protein; Neuroscience
Ajmalicine (Raubasine) 是一种有效的抗肾上腺素 (adrenolytic) 剂,优先阻断 α1-肾上腺素受体 (α1-adrenoceptor)。Ajmalicine 是一种可逆性但非竞争性尼古丁受体 (nicotine receptor) 完全抑制剂,IC50 为 72.3 μM。Ajmalicine 还可用于降压、蛇毒,具有镇静活性。
T5581 6-(γ,γ-Dimethylallylamino)purine

N6-(2-lsopentenyl)adenine,三刺皂荚碱,Triacanthine

Others Others
6-(γ,γ-Dimethylallylamino)purine (Triacanthine) 是植物生长调节剂。
T6S0657 Isorhynchophylline

IsoRhy,异钩藤碱,Isorhyncophylline,Isorhychophylline,7-Isorhyncophylline

Others Others
Isorhynchophylline (7-Isorhyncophylline) 是一种分离自钩藤中的生物碱类化合物,具有舒张血管、降血压、保护神经免于局部缺血造成损伤的作用。
TCS1704 Artemitin

艾黄素,Artemetin,Artemisetin,Erianthin

Antioxidant oxidation-reduction
Artemitin (Erianthin) 是一种存在于翼齿六棱菊中的天然黄酮,具有抗氧化、抗炎、抗病毒活性。
T4S1102 Liensinine diperchlorate

莲心碱高氯酸盐,莲心碱二高氯酸盐,Liensinine-Perchlorate

Mitophagy; Others; Autophagy Autophagy; Others
Liensinine Diperchlorate 是从芙蕖种子胚中提取的一种异喹啉生物碱。它通过阻断自噬小体-溶酶体融合来抑制晚期自噬,具有抗心律不齐、抗高血压、抗肺纤维化和血管平滑肌松弛等生物学活性。
TN1065 Hirsutine

Apoptosis Apoptosis
Hirsutine 是一种来自钩藤的吲哚生物碱,可诱导细胞凋亡,是一种登革热病毒抑制剂,且毒性低。它具有抗癌、心脏保护、抗高血压、抗心律失常和血管舒张活性。
T1035 Hesperidin

橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷

Apoptosis; Reactive Oxygen Species; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Hesperidin (Cirantin) 是一种广泛存在于柑橘类水果中黄烷酮糖苷,具有减少炎症介质并发挥重要的抗氧化作用,还有抗肿瘤和抗过敏活性。
T12789 S-1-Propenyl-L-cysteine

Others Others
S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensive animal models.
TN2990 3alpha-dihydrocadambine

Others Others
3alpha-Dihydrocadambine exhibits dose-dependent hypotensive and anti-hypertensive effects in anesthetized normotensive rats and in conscious spontaneously hypertensive rats.
T69254 Ajmalicine hydrochloride

Raubasine hydrochloride

Ajmalicine (Raubasine) hydrochloride 是一种有效的抗肾上腺素 (adrenolytic) 剂,优先阻断 α1-肾上腺素受体 (α1-adrenoceptor)。Ajmalicine hydrochloride 是一种可逆性但非竞争性尼古丁受体 (nicotine receptor) 完全抑制剂,其 IC50为 72.3 μM。Ajmalicine hydrochloride 还可用于降压、蛇毒,具有镇静活性。

天然产物

Tilianin
Cat.No: T8158
Synonym: 香清兰苷,田蓟苷
Target: Others
Vitexin
Cat.No: T6S1369
Synonym: 牡荆素,Apigenin-8-C-glucoside
Target: Antioxidant
Ajmalicine
Cat.No: T8044
Synonym: 阿吗里新,Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin
Target: Adrenergic Receptor
6-(γ,γ-Dimethylallylamino)purine
Cat.No: T5581
Synonym: N6-(2-lsopentenyl)adenine,三刺皂荚碱,Triacanthine
Target: Others
Isorhynchophylline
Cat.No: T6S0657
Synonym: IsoRhy,异钩藤碱,Isorhyncophylline,Isorhychophylline,7-Isorhyncophylline
Target: Others
Artemitin
Cat.No: TCS1704
Synonym: 艾黄素,Artemetin,Artemisetin,Erianthin
Target: Antioxidant
Liensinine diperchlorate
Cat.No: T4S1102
Synonym: 莲心碱高氯酸盐,莲心碱二高氯酸盐,Liensinine-Perchlorate
Target: Mitophagy, Others, Autophagy
Hirsutine
Cat.No: TN1065
Synonym:
Target: Apoptosis
Hesperidin
Cat.No: T1035
Synonym: 橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷
Target: Apoptosis, Reactive Oxygen Species, Endogenous Metabolite, Autophagy
S-1-Propenyl-L-cysteine
Cat.No: T12789
Synonym:
Target: Others
3alpha-dihydrocadambine
Cat.No: TN2990
Synonym:
Target: Others
Ajmalicine hydrochloride
Cat.No: T69254
Synonym: Raubasine hydrochloride
Target:
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