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Search Results for " anti-ulcer "

26

抑制剂 & 化合物

10

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T6928	Pantoprazole SKF96022,泮托拉唑,BY1023	Apoptosis; Proton pump; Autophagy	Apoptosis; Autophagy; Membrane transporter/Ion channel
	Pantoprazole (BY1023) 是一种质子泵抑制剂，用于短期治疗由胃食管反流病引起的食管糜烂和溃疡。它联合阿霉素可显著增加肿瘤生长延迟。它是一种取代的苯并咪唑，是H+/K+-ATPase 抑制剂，可改善 pH 值稳定性，具有抗分泌和抗溃疡的作用。
T0161	Pantoprazole Sodium Hydrate SKF96022 sodium hydrate,泮托拉唑钠水合物,BY1023 (sodium hydrate),SKF96022 (sodium hydrate)	Apoptosis; Potassium Channel; Proton pump; Autophagy	Apoptosis; Autophagy; Membrane transporter/Ion channel
	Pantoprazole Sodium Hydrate (BY1023 (sodium hydrate)) 是一种具有口服活性的质子泵抑制剂。它是取代的苯并咪唑，是H+/K+-ATPase 抑制剂。它可改善 pH 值稳定性，具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T6929	Pantoprazole sodium Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc	Apoptosis; Others; Proton pump; HIF; Autophagy	Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Others
	Pantoprazole sodium (Pantecta) 是一种具有口服活性的质子泵抑制剂，是一种取代的苯并咪唑，是H+/K+-ATPase 抑制剂，IC50为 6.8 μM。它可以改善 pH 值稳定性，具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T4510	Polaprezinc Zinc L-carnosine,聚普瑞锌,L-肌肽锌	Others	Others
	Polaprezinc is an bioavailable chelate comprised of zinc and L-carnosine, known for its gastrointestinal protective properties, as well as its anti-ulcer, antioxidant, and anti-inflammatory effects.
T5008	Teprenone Tetraprenylacetone,Geranylgeranylacetone,替普瑞酮	HSP	Cytoskeletal Signaling; Metabolism
	Teprenone (Geranylgeranylacetone) 是一种热休克蛋白诱导剂，有抗溃疡作用。
T12215	Nexopamil racemate (Rac)-Nexopamil	Calcium Channel; 5-HT Receptor	GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Nexopamil racemate（(Rac)-Nexopamil）是 Nexopamil 的外消旋体。Nexopamil racemate 具有潜在的抗哮喘和抗溃疡活性。
T6548	Irsogladine Dicloguamine,伊索拉定	PDE; AChR	Metabolism; Neuroscience
	Irsogladine (Dicloguamine) 是抗胃溃疡剂，通过 M1 毒蕈碱乙酰胆碱受体结合促进间隙连接细胞间通讯。
T6710	Troxipide 曲昔派特,曲昔匹特,Aplace	Others	Others
	Troxipide (Aplace) 是非分泌型胃保护剂，是口服具有活力的胃炎和胃溃疡的防御因子的增强剂，具有抗溃疡、抗炎和粘液分泌作用。
T77618	COX-2-IN-34	COX	Immunology/Inflammation; Neuroscience
	COX-2-IN-34 是一种选择性的、口服有效的 COX-2 抑制剂，在小鼠实验过程中显示出抗炎活性且无胃溃疡毒性。
T10872L	CP 96021	5-HT Receptor	GPCR/G Protein; Neuroscience
	CP 96021是一组5-HT1受体和5-HT2受体拮抗剂，具有抗炎特性，是治疗胃肠道和呼吸道哮喘的非自身抗溃疡化合物。
T16865	SCH28080	ATPase; Proton pump	Membrane transporter/Ion channel
	SCH28080 是一种可逆且具有 K+ 竞争性的胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂，IC50 值为 20 nM (家兔微粒体膜)。SCH28080 在体内是有效的酸分泌抑制剂，具有抗溃疡活性、抗分泌和细胞保护活性。
T77617	MMP-9-IN-6	MMP	Proteases/Proteasome
	MMP-9-IN-6 是一种 MMP-9 抑制剂，其 IC50 值为50 μM, 具有较好的抗溃疡功效。MMP-9-IN-6 具有潜在的抗肿瘤活性，可用于研究组织重塑、伤口修复和动脉粥样硬化。
T1639	Amlexanox 氨来呫诺,CHX3673,Amoxanox,氨来诺,AA673	IL Receptor; FGFR; Others; IκB/IKK	Angiogenesis; Immunology/Inflammation; NF-κB; Others; Tyrosine Kinase/Adaptors
	Amlexanox (AA673) 是一种特异性的 IKKε和 TBK1抑制剂，其 IC50=1-2 μM。
T62396	KB-5492 free base
	KB-5492 free base 是一种有效的和选择性的sigma 受体抑制剂，抑制 [3H]1,3-di(2-tolyl)guanidine (DTG) 与sigma 受体结合，IC50值为 3.15 μM。KB-5492 free base 是一种抗溃疡剂。
T1562	Rebamipide Proamipide,OPC12759,瑞巴派特	Free radical scavengers; COX; Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience; oxidation-reduction
	Rebamipide (OPC12759) 是一种粘膜保护剂，可诱导COX-2表达，增加PGE2水平，并以 COX-2 依赖性方式增强胃粘膜防御。
T19763	Cetraxate hydrochloride DV-1006,DV 1006,Cetraxate HCl,盐酸西曲酸酯,DV1006	Serine/threonin kinase	Cell Cycle/Checkpoint; Metabolism
	Cetraxate hydrochloride (DV10062) 是一种有效的顶体蛋白酶 (acrosomal proteinase acrosin) 抑制剂，Ki 和 IC50分别为 0.94 μM 和 3.3 μM。它是一种口服有活性的抗溃疡试剂 (anti-ulcer)，具有粘膜保护作用，可用于研究胃溃疡。
T24728	Rosaprostol C 83
	Rosaprostol is an agent of the anti-ulcer drug.
T10008	BTM-1086	Others	Others
	BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.
T69801	AU-461
	AU-461 is a gastric H(+)/K(+) ATPase inhibitor which acts as an anti-ulcer agent.
T28613	RP73870 RP 73870,RP-73870
	RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.
T24254	KB-5492 anhydrous KB-5492,KB5492,KB 5492
	KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.
T68200	Roxatidine hydrochloride
	Roxatidine hydrochloride is an anti-ulcer agent and histamine antagonist that suppresses gastric acid secretion. It effectively heals duodenal and gastric ulcers and reduces ulcer pain. Roxatidine acetate has an improved safety profile compared to other similar drugs, in part because lower doses of roxatidine acetate are therapeutically effective.
T69805	AU-006
	AU-006 is an anti-ulcer drug which is effective in the treatment of gastric ulcers by inhibiting gastric acid secretion.
T0157L	Roxatidine acetate
	Roxatidine acetate is an anti-ulcer agent and histamine antagonist that inhibits gastric acid secretion. Compared to other similar drugs, Roxatidine acetate has an improved safety profile, in part because lower doses of roxatidine acetate are therapeutica
T81074	Sucrose octasulfate sodium
	Sucrose octasulfate为硫糖铝组分，能直接刺激胃粘膜D细胞以促进生长抑素样免疫反应(SLI)的释放，进而发挥内源性胃生长抑素的溃疡愈合功能，适用于抗胃溃疡研究。
T74118	Roxatidine
	Roxatidine 是 Roxatidine acetate 的活性代谢产物，是组胺 H2受体拮抗剂。Roxatidine 是抗溃疡药，抑制组胺释放（从而抑制质子分泌）并抑制炎症和血管生成的重要标志物 VEGF-1 的产生。具有抗过敏性炎症作用。

化合物

Cat.No: T6928

Synonym: SKF96022,泮托拉唑,BY1023

Target: Apoptosis, Proton pump, Autophagy

Pantoprazole Sodium Hydrate

Cat.No: T0161

Synonym: SKF96022 sodium hydrate,泮托拉唑钠水合物,BY1023 (sodium hydrate),SKF96022 (sodium hydrate)

Target: Apoptosis, Potassium Channel, Proton pump, Autophagy

Pantoprazole sodium

Cat.No: T6929

Synonym: Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc

Target: Apoptosis, Others, Proton pump, HIF, Autophagy

Cat.No: T4510

Synonym: Zinc L-carnosine,聚普瑞锌,L-肌肽锌

Target: Others

Cat.No: T5008

Synonym: Tetraprenylacetone,Geranylgeranylacetone,替普瑞酮

Target: HSP

Nexopamil racemate

Cat.No: T12215

Synonym: (Rac)-Nexopamil

Target: Calcium Channel, 5-HT Receptor

Cat.No: T6548

Synonym: Dicloguamine,伊索拉定

Target: PDE, AChR

Cat.No: T6710

Synonym: 曲昔派特,曲昔匹特,Aplace

Target: Others

Cat.No: T77618

Target: COX

Cat.No: T10872L

Target: 5-HT Receptor

Cat.No: T16865

Target: ATPase, Proton pump

Cat.No: T77617

Target: MMP

Cat.No: T1639

Synonym: 氨来呫诺,CHX3673,Amoxanox,氨来诺,AA673

Target: IL Receptor, FGFR, Others, IκB/IKK

KB-5492 free base

Cat.No: T62396

Cat.No: T1562

Synonym: Proamipide,OPC12759,瑞巴派特

Target: Free radical scavengers, COX, Prostaglandin Receptor

Cetraxate hydrochloride

Cat.No: T19763

Synonym: DV-1006,DV 1006,Cetraxate HCl,盐酸西曲酸酯,DV1006

Target: Serine/threonin kinase

Cat.No: T24728

Synonym: C 83

Cat.No: T10008

Target: Others

Cat.No: T69801

Cat.No: T28613

Synonym: RP 73870,RP-73870

KB-5492 anhydrous

Cat.No: T24254

Synonym: KB-5492,KB5492,KB 5492

Roxatidine hydrochloride

Cat.No: T68200

Cat.No: T69805

Roxatidine acetate

Cat.No: T0157L

Sucrose octasulfate sodium

Cat.No: T81074

Cat.No: T74118

Cat. No.	Product Name	Target	Signaling Pathways
T2833	Dehydrocostus Lactone Epiligulyl oxide,去氢木香内酯,(-)-Dehydrocostus lactone,去氢木香烃内酯	IκB/IKK	NF-κB
	Dehydrocostus Lactone ((-)-Dehydrocostus lactone) 是一种倍半萜内酯，从云木香中分离得到。
TN1568	Deoxyartemisinin 2-deoxyartemisinin
	Deoxyartemisinin (2-deoxyartemisinin) 是一种口服有效的抗炎和抗溃疡化合物，可从青蒿素青蒿中分离得到。
TN6577	Bletilloside A 3-Methoxyshancigusin I	Others	Others
	Bletilloside A（3-Methoxyshancigusin I）是从条纹苜蓿的块茎中分离出一种新型葡萄糖苷，具有抗胃溃疡活性。
TN2233	Spathulenol	Antioxidant; Antifungal	Microbiology/Virology; oxidation-reduction
	Spathulenol 是一种来自 Aristolochia yunnanensis 的天然成分，具有抗炎、抗氧化、抗增殖、抗溃疡和抗分枝杆菌活性。 Spathulenol 在 DPPH 系统中显示出显著的抗氧化活性，IC50 为 85.60 μg/mL。
T12681	(±)-Vasicine (±)-Peganine	Others	Others
	(±)-Vasicine is the racemate of Vasicine. Vasicine isolated from Peganum harmala seeds, with anti-ulcer activity.
TN1893	Luteolin-3',7-di-O-glucoside	Others	Others
	Luteolin-3',7-di-O-glucoside has anti-ulcer and antioxidant activities.
TN3852	Dihydrolicoisoflavone	Antifection	Microbiology/Virology
	Dihydrolicoisoflavone A possesses weaker anti-H. pylori activity, it may be useful chemopreventive agents for peptic ulcer or gastric cancer in H. pylori-infected individuals.
TN3926	Eicosanyl caffeate	Others	Others
	Eicosanyl caffeate has anti-ulcer and moderate antioxidant properties, it exhibits potent elastase inhibitory activity, with the IC(50) value of 0.99 microg/mL.
TN1302	6,8-Diprenylorobol 6,8-二异戊烯基香豌豆苷元	Others; HIV Protease; Antifection	Microbiology/Virology; Others; Proteases/Proteasome
	6,8-Diprenylorobol possesses weaker anti-H. pylori activity, it may be a useful chemopreventive agent for peptic ulcer or gastric cancer in H. pylori-infected individuals.
TN1913	Marmin	Calcium Channel; Antifection; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
	Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and secondarily due to the prevention of the effects of endogenous acetylcholine and histamine.

天然产物

Dehydrocostus Lactone

Cat.No: T2833

Synonym: Epiligulyl oxide,去氢木香内酯,(-)-Dehydrocostus lactone,去氢木香烃内酯

Target: IκB/IKK

Deoxyartemisinin

Cat.No: TN1568

Synonym: 2-deoxyartemisinin

Cat.No: TN6577

Synonym: 3-Methoxyshancigusin I

Target: Others

Cat.No: TN2233

Target: Antioxidant, Antifungal

Cat.No: T12681

Synonym: (±)-Peganine

Target: Others

Luteolin-3',7-di-O-glucoside

Cat.No: TN1893

Target: Others

Dihydrolicoisoflavone

Cat.No: TN3852

Target: Antifection

Eicosanyl caffeate

Cat.No: TN3926

Target: Others

6,8-Diprenylorobol

Cat.No: TN1302

Synonym: 6,8-二异戊烯基香豌豆苷元

Target: Others, HIV Protease, Antifection

Cat.No: TN1913

Target: Calcium Channel, Antifection, Histamine Receptor

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