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92

抑制剂 & 化合物

46

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0578 Erythrosin B

Iodeosin,Tetraiodofluorescein,藻红B

Others Others
Erythrosin B (Iodeosin) 是一种四碘荧光素,在某些食物(樱桃、鱼)中用作红色色素,用作某些细胞类型的染色剂,以及用作牙菌斑的披露物。其分子结构与甲状腺素相似。
T0305 Erythrosine B

Erythrosine I,Erythrosin extra bluish,Erythrosin B,赤藓红B

Others Others
Erythrosine B (Erythrosine I) 是一种已被用于开发动物模型的新型光敏剂,在食品和纺织工业的人造染料中具有广泛的应用。
T20556L Tyrosyltyrosine acetate

Others Others
Tyrosyltyrosine acetate 是一种肽。
T20700 Racemetirosine

Others Others
Racemetirosine 是一种酪氨酸 3-单加氧酶抑制剂,因此会抑制儿茶酚胺的合成。
T60278 Tyrosinase-IN-2

Tyrosinase Proteases/Proteasome
Tyrosinase-IN-2 (compound 67) 是一种有效的酪氨酸酶抑制剂。酪氨酸酶是一种含铜金属酶,负责黑色素生物合成和酶促褐变中的限速催化步骤。Tyrosinase-IN-2 具有研究皮肤美白剂和食品防腐剂的潜力。
T67939 Tyrosinase-IN-16

Tyrosinase-IN-16对酪氨酸酶具有抑制作用。
T5466 Tyrosine kinase-IN-1

VEGFR; FGFR; FLT; PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
Tyrosine kinase-IN-1是一种多靶点酪氨酸激酶抑制剂,能够抑制KDR (IC50:4 nM),Flt-1 (IC50:20 nM),FGFR1 (IC50:4 nM) 和 PDGFRα (IC50:2 nM)。
T60108 PDGFR Tyrosine Kinase Inhibitor III

PDGF Receptor Tyrosine Kinase Inhibitor III

PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
PDGFR Tyrosine Kinase Inhibitor III (PDGF Receptor Tyrosine Kinase Inhibitor III) (PDGF Receptor Tyrosine Kinase Inhibitor III)是一种多激酶抑制剂,可抑制 PDGFR、EGFR、FGFR、PKA 和 PKC 等。PDGFR Tyrosine Kinase Inhibitor III 可用于肌萎缩侧索硬化症的研究。
T77746 Tyrosine kinase-IN-7

EGFR; Antiviral Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Tyrosine kinase-IN-7 是一种有效的酪氨酸激酶 EGFR 抑制剂,抑制 EGFR(WT) 和 EGFR(T790M) ,在多种癌细胞系中显示出抗癌和抗肿瘤活性。Tyrosine kinase-IN-7 具有潜在的抗炎和抗病毒活性。
T9492 3-METHOXY-DL-TYROSINE

Others Others
3-METHOXY-DL-TYROSINE 是一种在人体和许多其他生物体中发现的天然氨基酸,是一种非必需氨基酸。它是神经递质多巴胺的前体,参与大脑中多巴胺水平的调节,在多种疾病中有潜在治疗应用,包括帕金森病、抑郁症和肥胖症。
T7096 Tildipirosin

Antibacterial; Antibiotic Microbiology/Virology
Tildipirosin 是一种具有长效抗菌作用的大环内酯抗生素。
T20698L Leucyltyrosine acetate

Others Others
Leucyltyrosine acetate 是一种肽。
T22368 Metyrosine

甲酪氨酸,α-Methyltyrosine

COX Immunology/Inflammation; Neuroscience
Metyrosine (α-Methyltyrosine) 是一种选择性酪氨酸羟化酶抑制剂,可显著抑制高 COX-2 活性和有效控制血压,具有抗炎和抗溃疡作用。
T31931L Gizzerosine HCl

Gizzerosine HCl(89238-78-8 Free base)

Others Others
Gizzerosine HCl 是鱼粉热处理过程中产生的一种物质,可诱导的肉鸡雏鸡组织病理学病变,可提高离体鸡原产鸡的细胞内环腺苷-3',5'-单磷酸水平。
T19922 L-m-Tyrosine

L(-)mTyrosine,3-羟基-L-苯基丙氨酸,L (-) m Tyrosine,LmTyrosine,3-Hydroxy-L-Phenylalanine,L-(-)-m-Tyrosine

Others Others
L-m-Tyrosine (3-Hydroxy-L-Phenylalanine) 是一种非天然氨基酸。L-m-Tyrosine 在治疗帕金森病、关节炎和阿尔茨海默病方面显示出潜力。
T78554 Tyrosinase-IN-12

Tyrosinase Proteases/Proteasome
Tyrosinase-IN-12(Non-competitive tyrosinase inhibitor) 是一种有效的非竞争性酪氨酸酶抑制剂,IC50 值为 49.33 ± 2.64 µM,Ki 值为31.25 ± 0.25 µM。Tyrosinase-IN-12 具有显著的抗氧化和自由基清除活性,减少活性氧 (ROS) 的产生(IC50:25.39 ± 0.77 µM)。Tyrosinase-IN-12 可用于研究食品和水果中物质的褐变。
T31162 Cysteinyltyrosine

N-L-Cysteinyl-L-tyrosine,Cys-tyr

Cysteinyltyrosine is a dipeptide composed of cysteine and tyrosine. It is an incomplete breakdown product of protein digestion or protein catabolism.
T124961 Pterosin A

Pterosin A 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124961。
T34713 Stearyl tyrosine

Stearyl-tyrosine,Stearyltyrosine

Stearyl tyrosine is an immunoadjuvants, long-chain stearyl ester of amino acids and peptides.
T80909 Tyrosinase-IN-19

Tyrosinase Proteases/Proteasome
Tyrosinase-IN-19 是竞争性酪氨酸酶抑制剂,对ROS、ABTS+ 及DPPH 自由基展现显著的抗氧化活性。该化合物通过剂量依赖性方式有效抑制酪氨酸酶表达。
T80910 Tyrosinase-IN-15

Tyrosinase Proteases/Proteasome
Tyrosinase-IN-15 (Compound 39)为酪氨酸酶抑制剂,具有IC50值为7.12 μM及Ki值为11.8 μM。
T17184 Tyrosine kinase inhibitor

c-Met/HGFR; Tyrosine Kinases Tyrosine Kinase/Adaptors
Tyrosine kinase inhibitor 是酪氨酸激酶的有效抑制剂。
T38222 N-(α-Linolenoyl) Tyrosine

Certain chronic neurologic disorders, such as Parkinson's disease, are caused by an insufficiency of the neurotransmitter dopamine secondary to the degeneration of substantia nigra dopaminergic neurons. N-(α-Linolenoyl) tyrosine (NALT) is a simple α-amide conjugate between the ω-3 essential fatty acid α-linolenate and the amino acid tyrosine. α-Linolenate is an important precursor to docosahexaenoic acid (DHA), a prominent brain polyunsaturated fatty acid, while tyrosine is the metabolic precurs...
T32675 Leucyl-leucyl-tyrosine

L-Leu-L-leu-L-tyr

Leucyl-leucyl-tyrosine is a bioactive chemical.
T124433 3-Nitro-L-tyrosine ethyl ester hydrochloride

3-Nitro-L-tyrosine ethyl ester hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124433。
T25506 Homotyrosine, (+)-

alpha-Homotyrosine, (+)-,L-Homotyrosine

Homotyrosine, (+)- is an amino acid used as a very stable, selective, and renally safe sodium channel blocker.
T60449 Tyrosinase-IN-1

Tyrosinase-IN-1 (compound 90) 是有效的酪氨酸酶抑制剂。酪氨酸酶是一个很前途的靶点,酪氨酸酶抑制剂可用作美白剂和食品防腐剂,因此在食品、化妆品、农业和医药等领域具有广阔的应用前景。
T124236 N-cis-p-Coumaroyltyrosine

N-cis-p-Coumaroyltyrosine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124236,CAS号为 77201-65-1。
TP1623 [Asp371]-Tyrosinase (369-377), human

Tyrosinase (369-377,YMDGTMSQV) is derived from the membrane protein tyrosinase by posttranslational conversion of the sequence YMNGTMSQV. Presentation of YMDGTMSQV in cells expressing full-length tyrosinase is TAP-(transporter associated with antigen proc
T79406 Tyrosinase-IN-14

Tyrosinase Proteases/Proteasome
Tyrosinase-IN-14 (compound 7m) 是一种针对酪氨酸酶的抑制剂, 它通过改变酪氨酸酶的二级结构来降低其催化活性。此化合物的细胞毒性较低, 并且在水果抗褐变方面显示出活性。特别是,Tyrosinase-IN-14 在抑制香蕉储藏期间的褐变方面表现出了有效性。
T39054 Furosine dihydrochloride

Furosine dihydrochloride, an amino acid derivative, is a significant biochemical indicator of initial Maillard reactions. The compound is strongly associated with various diseases, including diabetes.
T20556 Tyrosyltyrosine

Tyr-tyr,Peptide tyrosine-tyrosine,Tyrosyl tyrosine

Tyrosyltyrosine is a dipeptide.
T60484 Tyrosinase-IN-4

Tyrosinase-IN-4 (compound 34) 是一种有效的酪氨酸酶抑制剂。酪氨酸酶是一种有前途的靶点,酪氨酸酶抑制剂可用作皮肤美白剂和食品防腐剂。 Tyrosinase-IN-4 在食品、化妆品、农业和医药等领域具有应用潜力[1]。
T36384 DL-Tyrosine-13C9,15N

L-Tyrosine-13C9,15N

L-Tyrosine-13C9,15N is intended for use as an internal standard for the quantification of L-tyrosine by GC- or LC-MS. L-Tyrosine is a non-essential amino acid.1It is produced by hydroxylation of phenylalanine by phenylalanine hydroxylase but can also be obtained from dietary sources or degradation of endogenous proteins, resulting in L-tyrosine release.1,2L-Tyrosine is a precursor in the biosynthesis of catecholamine neurotransmitters, melanins, and thyroid hormones.3Plasma, skeletal muscle, and...
T32206 Isodityrosine

Isodityrosine is a new cross-linking amino acid from plant cell-wall glycoprotein.
T72787 Tyrosinase-IN-8

Tyrosinase-IN-8, 作为一种酪氨酸酶抑制剂, 具有1.57 µM的IC50值,其特点是低细胞毒性地抑制细胞生长。
T125596 Nemerosin

Nemerosin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125596,CAS号为 17187-79-0。
T69173 Ambrosin

Ambrosin is a sesquiterpene lactone and a potent NF-κβ inhibitor. It is currently being studied as a potential lead drug for Alzheimer disease therapeutics.
T73598 Tyrosinase

Tyrosinase(Polyphenol oxidase) 是控制黑色素产生的限速酶,由 TYR 基因编码。Tyrosinase 主要存在于皮肤黑素细胞合成的黑素体中。
T67308 3-Fluoro-L-tyrosine

3-Fluoro-L-tyrosine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67308。
T37254 Rugulotrosin A

Rugulotrosin A is an antibiotic originally isolated from Penicillium. It is active against the Gram-positive bacteria E. faecalis, B. cereus, B. subtilis, and S. aureus with 99% lethal dose (LD99) values of 1.6, 3.1, 5.5, and 200 μg/ml, respectively. Rugulotrosin A is inactive against Gram-negative bacteria.
T35136 Woodrosin I

Woodrosin I is a glycolipid.
T61460 Tyrosinase-IN-3

Tyrosinase-IN-3 (compound 54) is a powerful tyrosinase inhibitor, an enzyme involved in the key catalytic step of melanin biosynthesis and enzymatic browning. As a copper-containing metalloenzyme, tyrosinase plays a crucial role in these processes. The compound shows promise for studying skin whitening agents and food preservatives [1].
T72720 Tyrosinase-IN-10

Tyrosinase-IN-10 是一种部分竞争性酪氨酸酶 (tyrosinase) 抑制剂,其 IC50为 1.6 μM,可抑制人黑素瘤细胞裂解物中的酪氨酸酶活性。
T74243 Tyrosinase/elastase-IN-1

Tyrosinase/elastase-IN-1,一种来源于悬钩子叶的三萜类化合物,具有抑制酪氨酸酶和弹性蛋白酶活性的功能。
T76410 Tyrosinase (206-214), human

Tyrosinase(206-214), human (AFLPWHRLF),一种由9个氨基酸组成的肽,为酪氨酸酶的表位。可被HLA-A24限制性肿瘤浸润淋巴细胞(TIL)识别的Tyrosinase(206-214), human,具有重要生物医学意义。
T65630 N-Benzoyl-L-tyrosine ethyl ester

N-Benzoyl-L-tyrosine ethyl ester 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65630,CAS号为 3483-82-7。
T77237 N,O-Didansyl-L-tyrosine cyclohexylammonium

N,O-Didansyl-L-tyrosine cyclohexylammonium 是一种有效的选择性胸苷酸合成酶 (TS) 抑制剂,作用于Escherichia coli,Lactobacillus casei 和人的 TS 的IC50值分别是 5.0,3.4 和 119 μM。
T80911 Tyrosinase (192-200), human mouse

Tyrosinase(192-200), human mouse 为九肽化合物,能被HLA-B44分子所识别的细胞溶解T细胞(CTL)所识别,常用于黑色素瘤相关癌症研究。
T29828 Alanyltyrosine

Alanyltyrosine is a dipeptide composed of alanine and tyrosine. It is an incomplete breakdown product of protein digestion or protein catabolism.

化合物

Erythrosin B
Cat.No: T0578
Synonym: Iodeosin,Tetraiodofluorescein,藻红B
Target: Others
Erythrosine B
Cat.No: T0305
Synonym: Erythrosine I,Erythrosin extra bluish,Erythrosin B,赤藓红B
Target: Others
Tyrosyltyrosine acetate
Cat.No: T20556L
Synonym:
Target: Others
Racemetirosine
Cat.No: T20700
Synonym:
Target: Others
Tyrosinase-IN-2
Cat.No: T60278
Synonym:
Target: Tyrosinase
Tyrosinase-IN-16
Cat.No: T67939
Synonym:
Target:
Tyrosine kinase-IN-1
Cat.No: T5466
Synonym:
Target: VEGFR, FGFR, FLT, PDGFR
PDGFR Tyrosine Kinase Inhibitor III
Cat.No: T60108
Synonym: PDGF Receptor Tyrosine Kinase Inhibitor III
Target: PDGFR
Tyrosine kinase-IN-7
Cat.No: T77746
Synonym:
Target: EGFR, Antiviral
3-METHOXY-DL-TYROSINE
Cat.No: T9492
Synonym:
Target: Others
Tildipirosin
Cat.No: T7096
Synonym:
Target: Antibacterial, Antibiotic
Leucyltyrosine acetate
Cat.No: T20698L
Synonym:
Target: Others
Metyrosine
Cat.No: T22368
Synonym: 甲酪氨酸,α-Methyltyrosine
Target: COX
Gizzerosine HCl
Cat.No: T31931L
Synonym: Gizzerosine HCl(89238-78-8 Free base)
Target: Others
L-m-Tyrosine
Cat.No: T19922
Synonym: L(-)mTyrosine,3-羟基-L-苯基丙氨酸,L (-) m Tyrosine,LmTyrosine,3-Hydroxy-L-Phenylalanine,L-(-)-m-Tyrosine
Target: Others
Tyrosinase-IN-12
Cat.No: T78554
Synonym:
Target: Tyrosinase
Cysteinyltyrosine
Cat.No: T31162
Synonym: N-L-Cysteinyl-L-tyrosine,Cys-tyr
Target:
Pterosin A
Cat.No: T124961
Synonym:
Target:
Stearyl tyrosine
Cat.No: T34713
Synonym: Stearyl-tyrosine,Stearyltyrosine
Target:
Tyrosinase-IN-19
Cat.No: T80909
Synonym:
Target: Tyrosinase
Tyrosinase-IN-15
Cat.No: T80910
Synonym:
Target: Tyrosinase
Tyrosine kinase inhibitor
Cat.No: T17184
Synonym:
Target: c-Met/HGFR, Tyrosine Kinases
N-(α-Linolenoyl) Tyrosine
Cat.No: T38222
Synonym:
Target:
Leucyl-leucyl-tyrosine
Cat.No: T32675
Synonym: L-Leu-L-leu-L-tyr
Target:
3-Nitro-L-tyrosine ethyl ester hydrochloride
Cat.No: T124433
Synonym:
Target:
Homotyrosine, (+)-
Cat.No: T25506
Synonym: alpha-Homotyrosine, (+)-,L-Homotyrosine
Target:
Tyrosinase-IN-1
Cat.No: T60449
Synonym:
Target:
N-cis-p-Coumaroyltyrosine
Cat.No: T124236
Synonym:
Target:
[Asp371]-Tyrosinase (369-377), human
Cat.No: TP1623
Synonym:
Target:
Tyrosinase-IN-14
Cat.No: T79406
Synonym:
Target: Tyrosinase
Furosine dihydrochloride
Cat.No: T39054
Synonym:
Target:
Tyrosyltyrosine
Cat.No: T20556
Synonym: Tyr-tyr,Peptide tyrosine-tyrosine,Tyrosyl tyrosine
Target:
Tyrosinase-IN-4
Cat.No: T60484
Synonym:
Target:
DL-Tyrosine-13C9,15N
Cat.No: T36384
Synonym: L-Tyrosine-13C9,15N
Target:
Isodityrosine
Cat.No: T32206
Synonym:
Target:
Tyrosinase-IN-8
Cat.No: T72787
Synonym:
Target:
Nemerosin
Cat.No: T125596
Synonym:
Target:
Ambrosin
Cat.No: T69173
Synonym:
Target:
Tyrosinase
Cat.No: T73598
Synonym:
Target:
3-Fluoro-L-tyrosine
Cat.No: T67308
Synonym:
Target:
Rugulotrosin A
Cat.No: T37254
Synonym:
Target:
Woodrosin I
Cat.No: T35136
Synonym:
Target:
Tyrosinase-IN-3
Cat.No: T61460
Synonym:
Target:
Tyrosinase-IN-10
Cat.No: T72720
Synonym:
Target:
Tyrosinase/elastase-IN-1
Cat.No: T74243
Synonym:
Target:
Tyrosinase (206-214), human
Cat.No: T76410
Synonym:
Target:
N-Benzoyl-L-tyrosine ethyl ester
Cat.No: T65630
Synonym:
Target:
N,O-Didansyl-L-tyrosine cyclohexylammonium
Cat.No: T77237
Synonym:
Target:
Tyrosinase (192-200), human mouse
Cat.No: T80911
Synonym:
Target:
Alanyltyrosine
Cat.No: T29828
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S0398 Rosin

松香树脂

p38 MAPK MAPK
Rosin 分离自松木或松树桩中,是一种频繁接触的过敏原,能够导致过敏性接触性皮炎。
T3090 Abietic Acid

Rosin Acid,L-Abietic acid,Sylvic acid,松香酸,Abietate

MMP; Lipoxygenase; Antibacterial; PPAR DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; Proteases/Proteasome
Abietic Acid (Sylvic acid) 是从 Pimenta racemosavar. grissea 中提取出来的一种二萜,具有抗菌、抗增殖和抗肥胖的活性。它抑制脂氧合酶活性,可研究过敏性疾病。
TN1596 DL-Tyrosine

Others Others
DL-Tyrosine 是一种由必需氨基酸苯丙氨酸合成的芳香族非必需氨基酸。它是几种重要神经递质(如肾上腺素、去甲肾上腺素、多巴胺)的前体。
T1695 DL-O-Tyrosine

Amino Acids and Derivatives Metabolism
DL-O-Tyrosine 是苯丙氨酸的代谢物,是形成儿茶酚胺的前体。它被用作β-地中海贫血中蛋白质氧化损伤的生物标志物。
T5292 N-Acetyl-L-tyrosine

N-乙酰-L-酪氨酸,N-Acetyltyrosine,Ac-Tyr-OH

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-tyrosine (Ac-Tyr-OH) 是一种来源于AA 乙酰酶作用下的酪氨酸,和芳香族氨基酸脱羧酶缺乏症以及酪氨酸血症有关,能够作为儿茶酚胺的前体,用于治疗神经递质。
TN1545 D-Tyrosine

Tyrosinase Proteases/Proteasome
D-Tyrosine,是酪氨酸的D异构体,通过抑制酪氨酸酶活性,作为黑色素合成的负向调节剂。此外,D-Tyrosine还能抑制生物膜的形成,并诱导生物膜的自我分散,同时不影响细菌的生长。
TN3866 Dihydrosinapyl alcohol

Dihydrosinapylalcohol,二氢芥子醇

Others Others
Dihydrosinapyl alcohol (Dihydrosinapylalcohol) 是一种可以通过氢化和氢解从木质纤维素获得的天然产物。
T0493 L-Tyrosine

Tyrosine,P-Tyrosine,L-酪氨酸,L-p-Tyrosine,(S)-Tyrosine,酪氨酸

Amino Acids and Derivatives; Endogenous Metabolite Metabolism
L-Tyrosine ((S)-Tyrosine) 是一种非必需氨基酸,对后部皮层中柠檬酸合成酶具有抑制活性。
T8208 androsin

Others Others
Androsin 分离于印度胡黄连中,具有抗哮喘作用。
TN1057 Veratrosine

藜芦托素,Veratramine 3-glycoside,Veratramine-beta-D-glucoside

Platelet aggregation Others
Veratrosine (Veratramine-beta-D-glucoside) 是一种从藜芦草本植物中分离出来的生物碱。 Veratrosine 对血小板聚集表现出微弱的抑制活性。
T5774 Demethylsuberosin

7-去甲基软木花椒素,7-demethylsuberosin

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
7-Demethylsuberosin (7-demethylsuberosin) 是一种分离自 Angelica gigasNakai 中的香豆素类化合物,具有抗炎作用。
T2S0886 Terrestrosin D

Apoptosis; Others Apoptosis; Others
Terrestrosin D 是从刺蒺藜中提取得到一种的甾体皂苷,可诱导细胞周期阻滞和癌细胞凋亡,具有抗血管生成的活性。
T2862 Desaminotyrosine

Phloretate,3-(4-Hydroxyphenyl)propanoic acid,Hydro-p-coumaric acid,对羟基苯丙酸,3-(4-Hydroxyphenyl)propionic acid,Phloretic acid,根皮酸

Others; Influenza Virus; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
Desaminotyrosine (3-(4-Hydroxyphenyl)propionic acid) 是一种与微生物相关的代谢物,通过增强 I 型干扰素信号传导来预防流感。
TN6749 3,5-Diiodo-L-tyrosine dihydrate

Others Others
3,5-Diiodo-L-tyrosine dihydrate 是一种天然产物。
TN2252 Syrosingopine

Dopamine Receptor GPCR/G Protein; Neuroscience
Syrosingopine 是 MCT1和 MCT4双重抑制剂,对 MCT4 的效力高 60 倍,可防止乳酸和 H+ 流出。它是可口服抗高血压药物,联合二甲双胍具有研究癌症疾病的潜力。
T5280 3-Chloro-L-Tyrosine

3-氯-L-酪氨酸,3-Chlorotyrosine,Chlorotyrosine

Others; Endogenous Metabolite Metabolism; Others
3-Chloro-L-Tyrosine (Chlorotyrosine) 是一种髓过氧化物酶催化氧化的特异性标志物,在从人动脉粥样硬化内膜分离的低密度脂蛋白中显著升高。
T4890 3-Nitro-L-tyrosine

3-Nitrotyrosine,3-硝基-L-酪氨酸

Endogenous Metabolite Metabolism
3-Nitro-L-tyrosine (3-Nitrotyrosine) 在系统自免疫原性条件下,能够作无氮自由基修饰蛋白的生物标记物。
T5795 Suberosin

软木花椒素

Others; NF-κB NF-κB; Others
Suberosin 可分离自Plumbago zeylanica 中,通过调节NF-AT 和NF-κB,抑制PHA-诱导的 PBMC 细胞增殖并捕获细胞周期G1过渡到 S 期,具有抗炎和抗血凝的活性。
TN4672 Norpterosin B glucoside

Others Others
Norpterosin B glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4672,CAS号为 1226785-88-1。
T40667 L-Azatyrosine

L-Azatyrosine, an antitumor antibiotic derived from Streptomyces chibaensis, exhibits the ability to restore the normal phenotypic behavior of transformed cells that carry oncogenic Ras genes.
TN4671 Norpterosin B

Others Others
Norpterosin B is a natural product from Pteris semipinnata.
T12576 Pterosin B

Others Others
Pterosin B is an salt-inducible kinase 3 (Sik3) signaling inhibitor. Pterosin B prevents chondrocyte hypertrophy and osteoarthritis by inhibiting Sik3.
T82779 Cararosinol A

Cararosinol A是Caragana sinica根部分离得到的化合物。
TN5168 trans-Norpterosin C

Others Others
trans-Norpterosin C is a natural product from Pteris semipinnata.
TN2266 Terrestrosin K

Others Others
Terrestrosin K is a natural product
TN5192 Tuberosin

NOS; Glucokinase Immunology/Inflammation; Metabolism
Tuberosin shows anti-inflammatory and antioxidant activities.It demonstrated a significantly potent inhibition on yeast α-glucosidase in a dose dependent manner.
TN5343 Pterosin D 3-O-glucoside

Pterosin D 3-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5343,CAS号为 84299-80-9。
TN2588 11-Hydroxytephrosin

TNF; NF-κB Apoptosis; NF-κB
11-Hydroxytephrosin inhibits NF-kappaB activity.
TN3975 Epipterosin L 2'-O-glucoside

Others Others
Epipterosin L 2'-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3975,CAS号为 61117-89-3。
TN5353 Pterosin C

Pterosin C is a natural product from Pteris semipinnata.
T20555 Glycyltyrosine

NSC 118362,Gly Tyr,NSC-118362,Gly-Tyr,NSC118362,N-Glycyl-L-tyrosine

Glycyltyrosine, a dipeptide composed of tyrosine and glycine, is an incomplete breakdown product of protein catabolism or protein digestion.
TN5340 Pterosin D

Pterosin D 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5340,CAS号为 34169-70-5。
TN5237 Virosine B

Others Others
Virosine B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5237,CAS号为 1052228-70-2。
TN5234 Vindorosine

Calcium Channel; Sodium Channel Membrane transporter/Ion channel; Metabolism
Vindorosine has blood vessel relaxation effect, possible underlying mechanisms involving the inhibition of Ca(2+) entry via L-type Ca(2+) channels in vascular smooth muscles.
T83525 (Rac)-Tephrosin

(Rac)-Tephrosin为存在于Tephrosia purpurea中的天然产物。
TN6592 Isonemerosin

Isonemerosin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6592,CAS号为 181524-79-8。
TN5341 Pterosin Z

Pterosin Z has smooth muscle relaxant activity, is approximately equipotent with that of the related fungal pterosin (EC50 of 2.9 +/- 1.6 x 10(-6) M).
TN6561 N-trans-p-Coumaroyltyrosine

N-trans-p-Coumaroyltyrosine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6561,CAS号为 77201-66-2。
T13126 Tephrosin

Deguelinol I,灰叶草素,Hydroxydeguelin

Others Others
Tephrosin induces degradation of of EGFR and ErbB2 by inducing internalization of the receptors, has potent antitumor activities.
T37444 Aranorosin

Aranorosin is a fungal metabolite originally isolated from P. roseus. It has antimicrobial activity against B. subtilis, A. niger, and C. albicans when used at a concentration of 1 mg/ml. Aranorosin also reduces viability in apoptosis-resistant HeLa/Bcl-2 cells.
TN2301 Vinleurosine

长春素

Others Others
Vinleurosine can partially inhibit the energy dependent transport of alpha-aminoisobutyric acid in Ehrlich ascites tumor cells.
TN3421 Anhydrotuberosin

Others Others
Anhydrotuberosin是一种天然产物,属于豆科葛属,其产品编号为 TN3421,CAS号为 41347-49-3。Anhydrotuberosin可用作对照参考。
T83255 7(R)-7,8-Dihydrosinomenine

7(R)-7,8-Dihydrosinomenine是从青藤中分离出的异喹啉生物碱,具备抗破骨细胞活性。
T13654 DL-m-Tyrosine

Others Others
DL-m-Tyrosine shows effects on Arabidopsis root growth.
TN3976 Epipterosin L

Others Others
Epipterosin L是一种天然产物,属于蚌壳蕨科金毛狗蕨属,其产品编号为 TN3976,CAS号为 52611-75-3。Epipterosin L可用作对照参考。
T8278 (+)-Dehydroabietic acid

Others Others
(+)-Dehydroabietic acid 是一种可用于合成丙烯酰胺水凝胶的二萜。

天然产物

Rosin
Cat.No: T4S0398
Synonym: 松香树脂
Target: p38 MAPK
Abietic Acid
Cat.No: T3090
Synonym: Rosin Acid,L-Abietic acid,Sylvic acid,松香酸,Abietate
Target: MMP, Lipoxygenase, Antibacterial, PPAR
DL-Tyrosine
Cat.No: TN1596
Synonym:
Target: Others
DL-O-Tyrosine
Cat.No: T1695
Synonym:
Target: Amino Acids and Derivatives
N-Acetyl-L-tyrosine
Cat.No: T5292
Synonym: N-乙酰-L-酪氨酸,N-Acetyltyrosine,Ac-Tyr-OH
Target: Others, Endogenous Metabolite
D-Tyrosine
Cat.No: TN1545
Synonym:
Target: Tyrosinase
Dihydrosinapyl alcohol
Cat.No: TN3866
Synonym: Dihydrosinapylalcohol,二氢芥子醇
Target: Others
L-Tyrosine
Cat.No: T0493
Synonym: Tyrosine,P-Tyrosine,L-酪氨酸,L-p-Tyrosine,(S)-Tyrosine,酪氨酸
Target: Amino Acids and Derivatives, Endogenous Metabolite
androsin
Cat.No: T8208
Synonym:
Target: Others
Veratrosine
Cat.No: TN1057
Synonym: 藜芦托素,Veratramine 3-glycoside,Veratramine-beta-D-glucoside
Target: Platelet aggregation
Demethylsuberosin
Cat.No: T5774
Synonym: 7-去甲基软木花椒素,7-demethylsuberosin
Target: Prostaglandin Receptor
Terrestrosin D
Cat.No: T2S0886
Synonym:
Target: Apoptosis, Others
Desaminotyrosine
Cat.No: T2862
Synonym: Phloretate,3-(4-Hydroxyphenyl)propanoic acid,Hydro-p-coumaric acid,对羟基苯丙酸,3-(4-Hydroxyphenyl)propionic acid,Phloretic acid,根皮酸
Target: Others, Influenza Virus, Endogenous Metabolite
3,5-Diiodo-L-tyrosine dihydrate
Cat.No: TN6749
Synonym:
Target: Others
Syrosingopine
Cat.No: TN2252
Synonym:
Target: Dopamine Receptor
3-Chloro-L-Tyrosine
Cat.No: T5280
Synonym: 3-氯-L-酪氨酸,3-Chlorotyrosine,Chlorotyrosine
Target: Others, Endogenous Metabolite
3-Nitro-L-tyrosine
Cat.No: T4890
Synonym: 3-Nitrotyrosine,3-硝基-L-酪氨酸
Target: Endogenous Metabolite
Suberosin
Cat.No: T5795
Synonym: 软木花椒素
Target: Others, NF-κB
Norpterosin B glucoside
Cat.No: TN4672
Synonym:
Target: Others
L-Azatyrosine
Cat.No: T40667
Synonym:
Target:
Norpterosin B
Cat.No: TN4671
Synonym:
Target: Others
Pterosin B
Cat.No: T12576
Synonym:
Target: Others
Cararosinol A
Cat.No: T82779
Synonym:
Target:
trans-Norpterosin C
Cat.No: TN5168
Synonym:
Target: Others
Terrestrosin K
Cat.No: TN2266
Synonym:
Target: Others
Tuberosin
Cat.No: TN5192
Synonym:
Target: NOS, Glucokinase
Pterosin D 3-O-glucoside
Cat.No: TN5343
Synonym:
Target:
11-Hydroxytephrosin
Cat.No: TN2588
Synonym:
Target: TNF, NF-κB
Epipterosin L 2'-O-glucoside
Cat.No: TN3975
Synonym:
Target: Others
Pterosin C
Cat.No: TN5353
Synonym:
Target:
Glycyltyrosine
Cat.No: T20555
Synonym: NSC 118362,Gly Tyr,NSC-118362,Gly-Tyr,NSC118362,N-Glycyl-L-tyrosine
Target:
Pterosin D
Cat.No: TN5340
Synonym:
Target:
Virosine B
Cat.No: TN5237
Synonym:
Target: Others
Vindorosine
Cat.No: TN5234
Synonym:
Target: Calcium Channel, Sodium Channel
(Rac)-Tephrosin
Cat.No: T83525
Synonym:
Target:
Isonemerosin
Cat.No: TN6592
Synonym:
Target:
Pterosin Z
Cat.No: TN5341
Synonym:
Target:
N-trans-p-Coumaroyltyrosine
Cat.No: TN6561
Synonym:
Target:
Tephrosin
Cat.No: T13126
Synonym: Deguelinol I,灰叶草素,Hydroxydeguelin
Target: Others
Aranorosin
Cat.No: T37444
Synonym:
Target:
Vinleurosine
Cat.No: TN2301
Synonym: 长春素
Target: Others
Anhydrotuberosin
Cat.No: TN3421
Synonym:
Target: Others
7(R)-7,8-Dihydrosinomenine
Cat.No: T83255
Synonym:
Target:
DL-m-Tyrosine
Cat.No: T13654
Synonym:
Target: Others
Epipterosin L
Cat.No: TN3976
Synonym:
Target: Others
(+)-Dehydroabietic acid
Cat.No: T8278
Synonym:
Target: Others
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