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111

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TMAZ-0351 Anti-REG3A Monoclonal Antibody

TMAZ-0089B Anti-REG1A Monoclonal Antibody-Biotin

TMAZ-0089P Anti-REG1A Monoclonal Antibody-PE

TMAZ-0089 Anti-REG1A Monoclonal Antibody

TMAZ-0351P Anti-REG3A Monoclonal Antibody-PE

TMAZ-0351B Anti-REG3A Monoclonal Antibody-Biotin

TMAZ-0089A Anti-REG1A Monoclonal Antibody-APC

TMAZ-0351A Anti-REG3A Monoclonal Antibody-APC

TMAZ-0301 Anti-REG1B Monoclonal Antibody

TMAZ-0301P Anti-REG1B Monoclonal Antibody-PE

TMAZ-0301B Anti-REG1B Monoclonal Antibody-Biotin

TMAZ-0301A Anti-REG1B Monoclonal Antibody-APC

TMAZ-0351A5 Anti-REG3A Monoclonal Antibody-AF555

TMAZ-0089A6 Anti-REG1A Monoclonal Antibody-AF647

TMAZ-0089A5 Anti-REG1A Monoclonal Antibody-AF555

TMAZ-0089A4 Anti-REG1A Monoclonal Antibody-AF488

TMAZ-0351A4 Anti-REG3A Monoclonal Antibody-AF488

TMAZ-0351A6 Anti-REG3A Monoclonal Antibody-AF647

TMAZ-0301A5 Anti-REG1B Monoclonal Antibody-AF555

TMAZ-0301A6 Anti-REG1B Monoclonal Antibody-AF647

TMAZ-0301A4 Anti-REG1B Monoclonal Antibody-AF488

T1792L Regorafenib monohydrate

Raf; VEGFR; c-RET; PDGFR; c-Kit; Autophagy Angiogenesis; Apoptosis; Autophagy; MAPK; Tyrosine Kinase/Adaptors
Regorafenib monohydrate 是一种新型口服多激酶抑制剂,对VEGFR1/2/3、PDGFRβ、Kit、RET 和Raf-1的IC50分别为 13、4.2、46、22、7、1.5 和 2.5 nM。
T12218 NFAT Transcription Factor Regulator-1

IL Receptor Immunology/Inflammation
NFAT Transcription Factor Regulator-1 是 IL-2 合成 的抑制剂,IC50 值为182 nM。
TP1761L Handle region peptide, rat acetate

Handle region peptide, rat acetate(749227-53-0 free base)

Others Others
Handle region peptide, rat acetate(749227-53-0 free base) 是一种肾素原受体拮抗剂,可抑制糖尿病肾病的进展并具有抗炎作用。
T1792 Regorafenib

BAY 73-4506,瑞戈非尼,Fluoro-Sorafenib,瑞格非尼

Raf; VEGFR; c-RET; PDGFR; c-Kit; Autophagy Angiogenesis; Apoptosis; Autophagy; MAPK; Tyrosine Kinase/Adaptors
Regorafenib (BAY 73-4506) 是一种多靶点受体酪氨酸激酶抑制剂,抑制 RET、C-RAF、VEGFR2、c-Kit、VEGFR1 和 PDGFRβ (IC50=1.5/2.5/4.2/7/13/22 nM),具有口服活性。Regorafenib 具有抗肿瘤和抗血管生成活性。
T11339 Furegrelate sodium

U-63557A

PPAR DNA Damage/DNA Repair; Metabolism
Furegrelate sodium (U-63557A) 是口服有效的、血栓素合酶选择性抑制剂,抑制人血小板微粒体血栓素 A2 (TxA2) 合酶的 IC50为 15 nM。它正在开发作为抗血小板药物。
T1831 StemRegenin 1

SR1

AhR; Aryl Hydrocarbon Receptor Immunology/Inflammation; Metabolism
StemRegenin 1 (SR1) 是一种芳香烃受体拮抗剂,IC50为 127 nM。
T8402 Regorafenib Hydrochloride

瑞戈非尼盐酸盐,BAY73-4506 hydrochloride

Raf; VEGFR; c-RET; PDGFR; Autophagy Angiogenesis; Apoptosis; Autophagy; MAPK; Tyrosine Kinase/Adaptors
Regorafenib Hydrochloride (BAY73-4506 hydrochloride) 是一种新型口服多激酶抑制剂,可抑制血管生成、基质和致癌受体酪氨酸激酶,具有强大的临床前抗肿瘤活性。它靶向作用于 VEGFR1/2/3、PDGFRβ、Kit、RET 和 Raf-1,IC50值分别为 13/4.2/46、22、7、1.5 和 2.5 nM。
T21818 Pregnenolone Carbonitrile

Pregnenolone 16α-carbonitrile ,5-Pregnen-3β-ol-20-one-16α-carbonitrile

P450 Metabolism
Pregnenolone Carbonitrile (5-Pregnen-3β-ol-20-one-16α-carbonitrile) 是一种啮齿动物-PXR 的激活剂,可诱导 CYP3A 的表达。
T60000 STING (WT/R232) activity regulator 126

STING Immunology/Inflammation
STING (WT/R232) activity regulator 126 是一种具有抗菌和抗病毒作用的 STING 调节剂。
T34383L 2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv

Others Others
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv在Sprague Dawley大鼠上进行测试时显示出高局部抗炎效力和高肺选择性。
T3225 16,17-Epoxy-21-acetoxypregnenolone

Others Others
16,17-Epoxy-21-acetoxypregnenolone 用作药物中间体。
T62899 Tau-aggregation and neuroinflammation-IN-1

Microtubule Associated; NO Synthase Cytoskeletal Signaling; Immunology/Inflammation
Tau-aggregation and neuroinflammation-IN-1 是一种有效的 Tau 蛋白聚集体抑制剂, 对 AcPHF6 和全长 tau 蛋白聚集体显示出显著的抑制活性。Tau-aggregation and neuroinflammation-IN-1具有抗炎活性且可减少 NO 释放。Tau-aggregation and neuroinflammation-IN-1 对 LSP 刺激的 BV2 细胞具有低细胞毒性。Tau-aggregation and neuroinflammation-IN-1 可逆转冈田酸诱导的大鼠记忆障碍。
T34280 Regrelor disodium

INS-50589,INS50589,Regrelor sodium,Regrelor,INS 50589

P2Y Receptor GPCR/G Protein; Neuroscience
Regrelor disodium (INS 50589) 是一种 p2y12 受体拮抗剂,可预防血栓形成,可有效抑制血管平滑肌细胞收缩,抑制细胞增殖,减少炎症。
T2671 Regadenoson

CVT-3146,瑞加德松,Lexiscan

Adenosine Receptor GPCR/G Protein; Neuroscience
Regadenoson (CVT-3146) 是一种腺苷衍生物和选择性 A2A 腺苷受体激动剂,具有冠状动脉舒张活性,对大鼠和猪腺苷 A2A 受体的Ki 分别为 290 和 1120 nM。它是血管扩张剂,可增加啮齿动物血脑屏障的通透性。
T3222 16,17-Epoxypregnenol

16alpha,17alpha-Epoxypregnenolone,16,17-环氧孕烯醇酮

Others Others
16,17-Epoxypregnenol 用作药物中间体。
T3219 16,17-Epoxypregnenolone acetate

16alpha,17alpha-Epoxypregnenolone acetate,16,17-环氧孕烯醇酮醋酸酯

Others Others
16,17-Epoxypregnenolone acetate (16alpha,17alpha-Epoxypregnenolone acetate) 可由洋葱伯克霍尔德菌 SE-1 生产。
T11339L Furegrelate

PPAR DNA Damage/DNA Repair; Metabolism
FUREGRELATE 是一种血栓素 A2 (TxA2) 合酶抑制剂,可减缓新生仔猪肺动脉高压的发展。
T10157 Regorafénib N-oxyde (M2)

瑞戈非尼杂质 13

Raf; VEGFR; c-RET; PDGFR; c-Kit; Drug Metabolite Angiogenesis; Apoptosis; MAPK; Metabolism; Tyrosine Kinase/Adaptors
Regorafénib N-oxyde M2 是 Regorafenib 的活性代谢物。Regorafenib 是多靶点抑制剂,包括VEGFR1/2/3,PDGFRβ,Kit,RET 和 Raf-1 , IC50分别是 13/4.2/46,22,7,1.5 和 2.5 nM。
T76851 Regdanvimab

Regdanvimab (CT-P59),一种靶向SARS-CoV-2刺突蛋白受体结合域的人单克隆抗体,通过阻断与ACE2的相互作用来防止病毒进入,适用于COVID-19研究。
T76528 Hepatitis b virus pre-s region (120-145)

Hepatitis b virus pre-s region (120-145) 是一种 preS2 肽,可抑制单链 Fv 片段 (scFv) 或IgG 与 r-HBsAg 的结合。
T76237 Utreglutide

Utreglutide 是一种有效的胰高血糖素样肽 1(GLP-1)受体激动剂。
T80555 Myoregulin TFA

MLN peptide TFA

Calcium Channel Membrane transporter/Ion channel; Metabolism
Myoregulin (MLN peptide) TFA,作为调节蛋白家族成员,通过干预细胞内钙处理机制来调控肌肉功能。该化合物直接作用于肌浆网 Ca2+-ATPase (SERCA),抑制其将Ca2+传输至肌浆网。
T28511 Reglitazar

JTT501,PNU-182716,PNU182716,PNU-716,JTT-501

PPAR DNA Damage/DNA Repair; Metabolism
Reglitazar (JTT-501) 是 PPARα和 PPARγ双重激动剂,可用于研究糖尿病。
T22865 immunoglobulin light chain variable region fragment [Homo sapiens]

Others Others
Immunoglobulin light chain variable region fragment [Homo sapiens] is a fragment (Phe-Thr-Leu-Lys-Ile-Ser-Arg) on the variable region of the human immunoglobulin light chain.
T23400 StemRegenin 1 (hydrochloride)

StemRegenin 1 (hydrochloride) (1227633-49-9 free base)

Others Others
StemRegenin 1 is an aryl hydrocarbon receptor signaling antagonist (IC50: 127 nM in CD34+ cells).
T64090 Regorafenib mesylate

Others Others
Regorafenib (BAY 73-4506) mesylate 是一种口服具有活力的多靶点受体酪氨酸激酶 (tyrosine kinase) 抑制剂,能够抑制VEGFR1/2/3 (IC50=13/4.2/46 nM),PDGFRβ (IC50: 22 nM),Kit (IC50: 7 nM),RET (IC50: 1.5 nM) 和 Raf-1 (IC50: 2.5 nM)。Regorafenib mesylate 具有强大的抗肿瘤和抗血管生成作用。
T131440 21-(acetyloxy)pregna-5,17-dien-3-yl acetate

Others Others
21-(acetyloxy)pregna-5,17-dien-3-yl acetate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131440。
T34128 Pregabalin arenacarbil

Others Others
Pregabalin arenacarbil is a gabamimetic.
T131419 3,14,20-trihydroxypregn-5-en-15-one

Others Others
3,14,20-trihydroxypregn-5-en-15-one 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131419。

化合物

Anti-REG3A Monoclonal Antibody
Cat.No: TMAZ-0351
Synonym:
Target:
Anti-REG1A Monoclonal Antibody-Biotin
Cat.No: TMAZ-0089B
Synonym:
Target:
Anti-REG1A Monoclonal Antibody-PE
Cat.No: TMAZ-0089P
Synonym:
Target:
Anti-REG1A Monoclonal Antibody
Cat.No: TMAZ-0089
Synonym:
Target:
Anti-REG3A Monoclonal Antibody-PE
Cat.No: TMAZ-0351P
Synonym:
Target:
Anti-REG3A Monoclonal Antibody-Biotin
Cat.No: TMAZ-0351B
Synonym:
Target:
Anti-REG1A Monoclonal Antibody-APC
Cat.No: TMAZ-0089A
Synonym:
Target:
Anti-REG3A Monoclonal Antibody-APC
Cat.No: TMAZ-0351A
Synonym:
Target:
Anti-REG1B Monoclonal Antibody
Cat.No: TMAZ-0301
Synonym:
Target:
Anti-REG1B Monoclonal Antibody-PE
Cat.No: TMAZ-0301P
Synonym:
Target:
Anti-REG1B Monoclonal Antibody-Biotin
Cat.No: TMAZ-0301B
Synonym:
Target:
Anti-REG1B Monoclonal Antibody-APC
Cat.No: TMAZ-0301A
Synonym:
Target:
Anti-REG3A Monoclonal Antibody-AF555
Cat.No: TMAZ-0351A5
Synonym:
Target:
Anti-REG1A Monoclonal Antibody-AF647
Cat.No: TMAZ-0089A6
Synonym:
Target:
Anti-REG1A Monoclonal Antibody-AF555
Cat.No: TMAZ-0089A5
Synonym:
Target:
Anti-REG1A Monoclonal Antibody-AF488
Cat.No: TMAZ-0089A4
Synonym:
Target:
Anti-REG3A Monoclonal Antibody-AF488
Cat.No: TMAZ-0351A4
Synonym:
Target:
Anti-REG3A Monoclonal Antibody-AF647
Cat.No: TMAZ-0351A6
Synonym:
Target:
Anti-REG1B Monoclonal Antibody-AF555
Cat.No: TMAZ-0301A5
Synonym:
Target:
Anti-REG1B Monoclonal Antibody-AF647
Cat.No: TMAZ-0301A6
Synonym:
Target:
Anti-REG1B Monoclonal Antibody-AF488
Cat.No: TMAZ-0301A4
Synonym:
Target:
Regorafenib monohydrate
Cat.No: T1792L
Synonym:
Target: Raf, VEGFR, c-RET, PDGFR, c-Kit, Autophagy
NFAT Transcription Factor Regulator-1
Cat.No: T12218
Synonym:
Target: IL Receptor
Handle region peptide, rat acetate
Cat.No: TP1761L
Synonym: Handle region peptide, rat acetate(749227-53-0 free base)
Target: Others
Regorafenib
Cat.No: T1792
Synonym: BAY 73-4506,瑞戈非尼,Fluoro-Sorafenib,瑞格非尼
Target: Raf, VEGFR, c-RET, PDGFR, c-Kit, Autophagy
Furegrelate sodium
Cat.No: T11339
Synonym: U-63557A
Target: PPAR
StemRegenin 1
Cat.No: T1831
Synonym: SR1
Target: AhR, Aryl Hydrocarbon Receptor
Regorafenib Hydrochloride
Cat.No: T8402
Synonym: 瑞戈非尼盐酸盐,BAY73-4506 hydrochloride
Target: Raf, VEGFR, c-RET, PDGFR, Autophagy
Pregnenolone Carbonitrile
Cat.No: T21818
Synonym: Pregnenolone 16α-carbonitrile ,5-Pregnen-3β-ol-20-one-16α-carbonitrile
Target: P450
STING (WT/R232) activity regulator 126
Cat.No: T60000
Synonym:
Target: STING
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv
Cat.No: T34383L
Synonym:
Target: Others
16,17-Epoxy-21-acetoxypregnenolone
Cat.No: T3225
Synonym:
Target: Others
Tau-aggregation and neuroinflammation-IN-1
Cat.No: T62899
Synonym:
Target: Microtubule Associated, NO Synthase
Regrelor disodium
Cat.No: T34280
Synonym: INS-50589,INS50589,Regrelor sodium,Regrelor,INS 50589
Target: P2Y Receptor
Regadenoson
Cat.No: T2671
Synonym: CVT-3146,瑞加德松,Lexiscan
Target: Adenosine Receptor
16,17-Epoxypregnenol
Cat.No: T3222
Synonym: 16alpha,17alpha-Epoxypregnenolone,16,17-环氧孕烯醇酮
Target: Others
16,17-Epoxypregnenolone acetate
Cat.No: T3219
Synonym: 16alpha,17alpha-Epoxypregnenolone acetate,16,17-环氧孕烯醇酮醋酸酯
Target: Others
Furegrelate
Cat.No: T11339L
Synonym:
Target: PPAR
Regorafénib N-oxyde (M2)
Cat.No: T10157
Synonym: 瑞戈非尼杂质 13
Target: Raf, VEGFR, c-RET, PDGFR, c-Kit, Drug Metabolite
Regdanvimab
Cat.No: T76851
Synonym:
Target:
Hepatitis b virus pre-s region (120-145)
Cat.No: T76528
Synonym:
Target:
Utreglutide
Cat.No: T76237
Synonym:
Target:
Myoregulin TFA
Cat.No: T80555
Synonym: MLN peptide TFA
Target: Calcium Channel
Reglitazar
Cat.No: T28511
Synonym: JTT501,PNU-182716,PNU182716,PNU-716,JTT-501
Target: PPAR
immunoglobulin light chain variable region fragment [Homo sapiens]
Cat.No: T22865
Synonym:
Target: Others
StemRegenin 1 (hydrochloride)
Cat.No: T23400
Synonym: StemRegenin 1 (hydrochloride) (1227633-49-9 free base)
Target: Others
Regorafenib mesylate
Cat.No: T64090
Synonym:
Target: Others
21-(acetyloxy)pregna-5,17-dien-3-yl acetate
Cat.No: T131440
Synonym:
Target: Others
Pregabalin arenacarbil
Cat.No: T34128
Synonym:
Target: Others
3,14,20-trihydroxypregn-5-en-15-one
Cat.No: T131419
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T12536 Pregnenolone monosulfate

3β-Hydroxy-5-pregnen-20-one monosulfate

NMDAR Neuroscience
Pregnenolone monosulfate (3β-Hydroxy-5-pregnen-20-one monosulfate) 是一种强效神经类固醇,可正向调节 NMDA 记录,可用于研究神经分裂和抑郁症。
T0851 Pregnenolone

3β-Hydroxy-5-pregnen-20-one,Arthenolone,孕烯醇酮

Cannabinoid Receptor; Endogenous Metabolite; TRP/TRPV Channel; AChR; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Pregnenolone (Arthenolone) 是一种由胆固醇合成的内源性类固醇激素,用于治疗阿尔茨海默病。它是大麻素 CB1受体的信号传导特异性抑制剂,抑制由 CB1受体介导的四氢大麻酚 的作用。它也是 TRPM3通道激活剂,也可弱激活 TRPM1通道。
TN2139 Regaloside B

鸦胆子苦醇,王百合苷 B

NOS; COX; NO Synthase Immunology/Inflammation; Neuroscience
Regaloside B 是从麝香百合中分离出来的一种苯丙烷,可抑制iNOS 和COX-2的表达,具有抗炎活性。
T5556 5a-Pregnane-3,20-dione

Endogenous Metabolite Metabolism
5a-Pregnane-3,20-dione 是内源性的孕酮代谢物。
TN6490 Regaloside C

Others Others
Regaloside C 是一种从百合属的中分离出来的甘油葡糖苷,具有抗炎作用。
TN7117 regaloside I

Others Others
Regaloside I 是百合中的单体成分,可能是保护人类皮肤成纤维细胞免受 UVA 诱导的形态变化的主要成分。
TC0019 Pregnenolone acetate

孕烯醇酮醋酸酯,3β-Hydroxy-5-pregnen-20-one acetate

Cannabinoid Receptor; Endogenous Metabolite GPCR/G Protein; Metabolism
Pregnenolone acetate 是一种强大的神经类固醇,是各种类固醇激素(包括类固醇酮)的主要前体。它作为大麻素 CB1 受体的信号特异性抑制剂,抑制由 CB1 受体介导的四氢大麻酚 (THC) 的作用。它可以保护大脑免受大麻中毒。
T1688 Pregnanediol

5Beta-Pregnane-3Alpha,20alpha-Diol,孕甾二醇,Pregnandiol,孕二醇

Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Pregnanediol (5Beta-Pregnane-3Alpha,20alpha-Diol) 是一种黄体酮的主要代谢物 (metabolite),能够通过尿液排出。它提供了一种间接测定体内孕激素水平的方法。
T13518 5α-Pregnane-3β,6α-diol-20-one

Others Others
5α-Pregnane-3β,6α-diol-20-one 是促进有丝分裂的 progesterone 代谢物,可于血清不足时雄性激素反应的前列腺素癌细胞中产生。
T7646 Alloepipregnanolone

Endogenous Metabolite Metabolism
Alloepipregnanolone 是具有促进安定和睡眠的孕酮,可干扰乙醇抗焦虑作用的快速耐受。
TN7038 Regaloside H

Others Others
Regaloside H 是一种糖异生抑制剂,是一种苯丙酸甘油糖苷。它能够抑制大鼠肝癌细胞中葡萄糖的产生。
T7931 16a,17a-Epoxy-4-Pregnen-3,20-Dione

Others Others
16a,17a-Epoxy-4-Pregnen-3,20-Dione 是一种合成孕激素,是黄体酮激素的代谢产物,它通过与黄体酮受体结合发挥作用,已被用于研究孕激素对生殖器官的影响,激素对细胞生长和发育的影响,以及激素对免疫系统的影响。
T10048 17a-Hydroxypregnenolone

Endogenous Metabolite Metabolism
17a-Hydroxypregnenolone 是一种孕烷类固醇, 是形成脱氢表雄酮的激素原。17a-Hydroxypregnenolone 是一种神经调节剂。
TN6489 Regaloside A

Others Others
 Regaloside A 是一种从百合中提取出的苯丙烷,在 160 ppm 时显示出 DPPH 自由基清除活性。Regaloside A 具有抗炎活性和抗抑郁活性。
T13489 21-Hydroxypregnenolone

Others Others
21-Hydroxypregnenolone is an essential intermediate in corticosterone synthesis.
T26055 Regelin

Regelin C

Regelin is an antitumor ursene-type triterpenoid isolated from Tripterygium regelii.
TN4821 Pregomisin

PAFR GPCR/G Protein
Pregomisin shows platelet-activating factor (PAF) antagonistic activity and the IC 50 value is 4.8x10(-5) M.
T81303 Regaloside E

Regaloside E为自Lilium longiflorum Thunb. 提取的天然化合物。
TN5295 Dregeoside A11

Dregeoside A11 is a natural product from Dregea volubilis.
T16574 Pregnenolone monosulfate sodium salt

3β-Hydroxy-5-pregnen-20-one monosulfate sodium salt

Others Others
Pregnenolone monosulfate sodium salt is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium salt can protect the brain from cannabis intoxication. Pregnenolone monosulfate sodi
TN5310 Pregn-5-ene-3β,17α,20S-triol

(3β,17α,20S)-Pregn-5-ene-3,17,20-triol

Pregn-5-ene-3β,17α,20S-triol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5310,CAS号为 903-67-3。
TN4903 Regiolone

Caspase Apoptosis; Proteases/Proteasome
Regiolone demonstrates phytotoxicity. Regiolone also has anti-proliferative and apoptotic activities, it can induce apoptosis in MCF-7 cells through the caspase-3 independent pathway.
TN5715 Oregonin

Oregonin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5715,CAS号为 55303-93-0。
TN2140 Regaloside D

王百合苷,王百合苷D

Others Others
Regaloside D 是一种分离于 Lilium Longiflorum 的苯丙素。
TN3804 Dehydroformouregine

Others Others
Dehydroformouregine是一种天然产物,属于胡椒科胡椒属,其产品编号为 TN3804,CAS号为 107633-69-2。Dehydroformouregine可用作对照参考。
T81302 Regaloside K

Regaloside K (Compd 1) 是从Easter Lily (Lilium longiflorum Thunb.) 提取的天然化合物。
TN3893 Dregeoside Da1

Others Others
Dregeoside Da1 is a natural product from Dregea volubilis.
TN3892 Dregeoside Aa1

Others Others
Dregeoside Aa1 is a natural product from Dregea volubilis.
TN2141 Regelidine

Others Others
Regelidine 是一种天然产物,分离自雷公藤茎中。
TN5293 Dregeoside Ga1

Dregeoside Ga1 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5293,CAS号为 98665-66-8。
T38592 Regaloside F

Others Others
Regaloside F is a phenolic glycerol glucoside that can be found in Lily bulbs.
TN7486 8-epi-Helenalin

Others Others
8-epi-Helenalin是从旋复花根中提取的半萜内酯,具抗肿瘤活性。其对HL-60、A549、MCF7、HCT-15、SK-OV-3以及Malme-3M的(EC50)值分别是12.2 μM、53.8 μM、9.1 μM、8.7 μM、18.7 μM和8.3 μM。

天然产物

Pregnenolone monosulfate
Cat.No: T12536
Synonym: 3β-Hydroxy-5-pregnen-20-one monosulfate
Target: NMDAR
Pregnenolone
Cat.No: T0851
Synonym: 3β-Hydroxy-5-pregnen-20-one,Arthenolone,孕烯醇酮
Target: Cannabinoid Receptor, Endogenous Metabolite, TRP/TRPV Channel, AChR, Autophagy
Regaloside B
Cat.No: TN2139
Synonym: 鸦胆子苦醇,王百合苷 B
Target: NOS, COX, NO Synthase
5a-Pregnane-3,20-dione
Cat.No: T5556
Synonym:
Target: Endogenous Metabolite
Regaloside C
Cat.No: TN6490
Synonym:
Target: Others
regaloside I
Cat.No: TN7117
Synonym:
Target: Others
Pregnenolone acetate
Cat.No: TC0019
Synonym: 孕烯醇酮醋酸酯,3β-Hydroxy-5-pregnen-20-one acetate
Target: Cannabinoid Receptor, Endogenous Metabolite
Pregnanediol
Cat.No: T1688
Synonym: 5Beta-Pregnane-3Alpha,20alpha-Diol,孕甾二醇,Pregnandiol,孕二醇
Target: Estrogen/progestogen Receptor, Endogenous Metabolite
5α-Pregnane-3β,6α-diol-20-one
Cat.No: T13518
Synonym:
Target: Others
Alloepipregnanolone
Cat.No: T7646
Synonym:
Target: Endogenous Metabolite
Regaloside H
Cat.No: TN7038
Synonym:
Target: Others
16a,17a-Epoxy-4-Pregnen-3,20-Dione
Cat.No: T7931
Synonym:
Target: Others
17a-Hydroxypregnenolone
Cat.No: T10048
Synonym:
Target: Endogenous Metabolite
Regaloside A
Cat.No: TN6489
Synonym:
Target: Others
21-Hydroxypregnenolone
Cat.No: T13489
Synonym:
Target: Others
Regelin
Cat.No: T26055
Synonym: Regelin C
Target:
Pregomisin
Cat.No: TN4821
Synonym:
Target: PAFR
Regaloside E
Cat.No: T81303
Synonym:
Target:
Dregeoside A11
Cat.No: TN5295
Synonym:
Target:
Pregnenolone monosulfate sodium salt
Cat.No: T16574
Synonym: 3β-Hydroxy-5-pregnen-20-one monosulfate sodium salt
Target: Others
Pregn-5-ene-3β,17α,20S-triol
Cat.No: TN5310
Synonym: (3β,17α,20S)-Pregn-5-ene-3,17,20-triol
Target:
Regiolone
Cat.No: TN4903
Synonym:
Target: Caspase
Oregonin
Cat.No: TN5715
Synonym:
Target:
Regaloside D
Cat.No: TN2140
Synonym: 王百合苷,王百合苷D
Target: Others
Dehydroformouregine
Cat.No: TN3804
Synonym:
Target: Others
Regaloside K
Cat.No: T81302
Synonym:
Target:
Dregeoside Da1
Cat.No: TN3893
Synonym:
Target: Others
Dregeoside Aa1
Cat.No: TN3892
Synonym:
Target: Others
Regelidine
Cat.No: TN2141
Synonym:
Target: Others
Dregeoside Ga1
Cat.No: TN5293
Synonym:
Target:
Regaloside F
Cat.No: T38592
Synonym:
Target: Others
8-epi-Helenalin
Cat.No: TN7486
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T12698 Regorafenib-d3

Regorafenib D3,BAY 73-4506 D3

Others Others
Regorafenib D3 is a deuterium labeled Regorafenib. Regorafenib is a multi-targeted receptor inhibitor of tyrosine kinase.
TMIH-0083 Allopregnanolone-d4

Allopregnanolone-d4 是 Allopregnanolone 的氘代化合物。
TMIH-0082 Allopregnanolone isomer-d4

Allopregnanolone isomer-d4 是 Allopregnanolone isomer 的氘代化合物。Allopregnanolone isomer 的 CAS 号为 21788-58-9。

同位素

Regorafenib-d3
Cat.No: T12698
Synonym: Regorafenib D3,BAY 73-4506 D3
Target: Others
Allopregnanolone-d4
Cat.No: TMIH-0083
Synonym:
Target:
Allopregnanolone isomer-d4
Cat.No: TMIH-0082
Synonym:
Target:
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