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74

抑制剂 & 化合物

13

天然产物

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Cat. No. Product Name Target Signaling Pathways
T21724L Fas C-Terminal Tripeptide Acetate

Fas C-Terminal Tripeptide Acetate (189109-90-8 free base)

Others; Fatty Acid Synthase Metabolism; Others
Fas C-Terminal Tripeptide Acetate 显示出对 Fas/FAP-1 结合的抑制活性。
T11266L FAS-IN-1 Tosylate

Fatty Acid Synthase Metabolism
FAS-IN-1 Tosylate is an effective fatty acid synthase inhibitor;Has an IC50 of 10 nM.
T11266 FASN-IN-4

FAS-IN-1

Others Others
FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.
T80442 Fasciculin-II

Fas-2

Fasciculin-II (Fas-2) 是一种针对 acetylcholinesterase (AChE) 的高效抑制剂。
T82415 Fasciculin-I

FAS-I

Fasciculin-I 是从曼巴蛇的毒液中分离出的化合物。该物质通过抑制乙酰胆碱酯酶(AChE)来发挥其毒性,同时阻碍烟碱乙酰胆碱受体与α-神经毒素以及心脏毒素与细胞膜的相互作用。
T80584 Anti-Mouse Fas Ligand Antibody (MFL3)

Anti-Mouse Fas Ligand Antibody为针对小鼠Fas Ligand的IgG类抗体抑制剂,由Armenian Hamster产生。
T8616 Fasentin

N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide

transporter Metabolism
Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) 是葡萄糖摄取抑制剂,可抑制GLUT-1/GLUT-4转运蛋白,优先抑制 GLUT4,IC50为 68 μM。它是死亡受体刺激敏化剂,可敏化细胞对 FAS 诱导的细胞死亡,具有抗血管生成活性。
T39308 Boc-Asp(OMe)-fluoromethyl ketone

Boc-Asp(OMe)-fluoromethyl ketone,Boc-Asp(OMe)-FMK

Caspase Apoptosis; Proteases/Proteasome
Boc-Asp(OMe)-fluoromethyl ketone (Boc-Asp(OMe)-FMK) 是广谱的 caspase 抑制剂,可抑制 Fas 介导的吞噬作用和氧化破裂抑制,但对 IL-8 的趋化活性无影响。
T10549 Bisindolylmaleimide VIII acetate

Ro 31-7549 acetate,Bis VIII acetate

Apoptosis; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling
Bisindolylmaleimide VIII acetate (Ro 31-7549 acetate) 是一种选择性蛋白激酶 C 抑制剂。它促进 Fas 介导的细胞凋亡,并抑制 T 细胞介导的自身免疫性疾病。
T5045 GSK4112

1,1-Dimethylethyl-N-[(4-chlorophenyl)methyl]-N-[(5-nitro-2-thienyl)methyl])glycinate,SR6452

Autophagy Autophagy
GSK4112 (SR6452) 是一种 Rev-erbα 激动剂,EC50 为 0.4 μM。它也是一种用于核血红素受体 Rev-erbα 的细胞生物学的小分子化学探针。
T77135 Tafasitamab

MOR00208,XmAb5574,Tafasitamab-cxix

Apoptosis; Immunology/Inflammation related Apoptosis; Immunology/Inflammation
Tafasitamab (XmAb5574) 是一种 Fc 修饰的人源化单克隆抗体,靶向人 B 细胞表面抗原 CD19 ,可用于研究弥漫性大B细胞淋巴瘤。
T11557 FASN-IN-3

Fatty Acid Synthase Metabolism
FASN-IN-3 是脂肪酸合酶抑制剂。
T0907 Sulfasalazine

柳氮磺吡啶,NSC 667219,Azulfidine

Apoptosis; Ferroptosis; NF-κB; COX; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience; NF-κB
Sulfasalazine (Azulfidine) 是一种合成的水杨酸衍生物,对含有弹性蛋白的结缔组织具有亲和力,并配制成前药。
T4640 Parimifasor

LYC30937

Others Others
Parimifasor (LYC30937) 是免疫调节剂,具有抗炎作用。
T4276 Hydroxyfasudil Hydrochloride

Hydroxyfasudil (HA-1100) HCl,羟基法舒地尔盐酸盐,RHO-激酶抑制剂,HA 1100 hydrochloride

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
Hydroxyfasudil Hydrochloride (HA 1100 hydrochloride) 是一种ROCK 抑制剂,对ROCK1和ROCK2的IC50值分别为 0.73 和 0.72 μM。
T27307L Fasnall HCl

Fasnall HCl(929978-58-5 Free base)

Fatty Acid Synthase Metabolism
Fasnall HCl 是一种FASN 选择性抑制剂,通过其辅助因子结合位点起作用。Fasnall HCl 在HER2(+)乳腺癌MMTV-Neu 模型中也显示出强大的抗肿瘤活性,特别是与卡铂联合使用时。
T4276L Hydroxyfasudil

Hydroxy-Fasudil,HA-1100,羟基法舒地尔

ROCK; PKA Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells; Tyrosine Kinase/Adaptors
Hydroxyfasudil (Hydroxy-Fasudil) 是一种ROCK 抑制剂,对ROCK1和ROCK2的IC50分别为 0.73 和 0.72 μM。
T1606 Fasudil

HA-1077,AT877,法舒地尔

ROCK; Serine/threonin kinase; Calcium Channel; PKA; PKC; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
Fasudil (HA-1077) 是一种非特异性 RhoA/ROCK 抑制剂,也是 Ca2+通道拮抗剂和血管扩张剂。它对蛋白激酶有抑制作用,ROCK1 的 Ki 值为 0.33 μM,ROCK2 和 PKA、PKC、PKG 的 IC50值分别 0.158 μM 和 4.58 μM、12.30 μM、1.650 μM。
T3060 Fasudil hydrochloride

Fasudil (HA-1077) HCl,盐酸法舒地尔,HA-1077,Fasudil HCl,HA-1077 hydrochloride,AT-877

ROCK; Serine/threonin kinase; Calcium Channel; HIV Protease; PKA; PKC; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
Fasudil hydrochloride (HA-1077) 是一种非特异性RhoA/ROCK 抑制剂,也抑制蛋白激酶,对 ROCK1、PKA、PKC 和 MLCK 的 Ki 值分别为 0.33 μM、1.0 μM、9.3 μM 和 55 μM。
TP1029 Thymalfasin

胸腺法新,Thymosin α1,醋酸胸腺α1

Others Others
Thymalfasin (Thymosin α1) 是一种免疫调节化合物,可增强 Thl 的免疫应答。
T11267 FASN-IN-1

TVB-2460

Fatty Acid Synthase Metabolism
FASN- in -1是一种有效的、特异性的脂肪酸合成酶(FASN)抑制剂,是一种专门设计用于靶向和抑制FASN 活性的化合物,是一种参与脂肪酸合成的酶,可抑制FASN 活性可以破坏脂肪酸的产生,并可能影响各种细胞过程。
T2351 Fasiglifam

TAK875

GPR Endocrinology/Hormones; GPCR/G Protein
Fasiglifam (TAK875) 是一种可口服的选择性GPR40激动剂,EC50值为 72 nM。
T9099 Disperse Fast Yellow 4K

分散黄,Disperse Yellow

Others Others
Disperse Fast Yellow 4K (Disperse Yellow) 是一种用于染料的颜色添加剂。
T27306 Fasidotril

BP 1137,BP1137,BP-1.137,BP1.137,BP-1137,BP 1.137

Fasidotril is a NEP/ACE inhibitor. Fasidotril was an effective oral antihypertensive agent during chronic treatment in high-renin renovascular rats, normal-renin SHR, and low-renin DOCA-salt hypertensive rats and in patients with essential hypertension.
T37776 FASN-IN-4 tosylate

FASN-IN-4 tosylate 是高效的脂肪酸合酶 FASN 抑制剂,IC50值为 10 nM。FASN-IN-4 tosylate 还抑制 SARS-CoV-2,EC50为 18.6 nM。
T27307 Fasnall

Fatty Acid Synthase Metabolism
Fasnall 是一种选择性 FASN 抑制剂,通过其辅因子结合位点起作用。 Fasnall 在 HER2(+) 乳腺癌的 MMTV-Neu 模型中显示出有效的抗肿瘤活性,尤其是与卡铂联合使用时。
TP2283 parathyroid hormone (7-34) [Homo sapiens]/[Macaca fascicularis]

Others Others
parathyroid hormone (7-34) [Homo sapiens] [Macaca fascicularis] is a peptide with the sequence H2N-LMHNLGKHLNSMERVEWLRKKLQDVHNF-OH, MW= 3474.03. Parathyroid hormone (PTH) is secreted by the chief cells of the parathyroid glands as a polypeptide containing
T61382 Fasudil dihydrochloride

Fasudil dihydrochloride, also known as HA-1077 and AT877, is a nonspecific inhibitor of RhoA/ROCK. It exhibits inhibitory effects on protein kinases, including ROCK1 with a Ki value of 0.33 μM, as well as ROCK2, PKA, PKC, and PKG with IC 50 values of 0.158 μM, 4.58 μM, 12.30 μM, and 1.650 μM, respectively. Additionally, Fasudil dihydrochloride demonstrates potent Ca 2+ channel blocking activity and acts as a vasodilator [1] [2] [3].
T25405 Fasciculic acid B

Fasciculic acid B is the ester of fasciculol B and 3-hydroxy-3-methylglutaric acid. Fasciculic acid B is calmodulin antagonist from mushroom Naematoloma fasciculare.
T31748 Fasobegron

Fasobegron is a agonist of β3-adrenoreceptor .
T69954 Fasoracetam monohydrate

Fasoracetam monohydrate is a small synthetic molecule and a metabotropic glutamate receptor activator, which has previously undergone extensive Phase I-III clinical trials in humans for vascular dementia.
T31749 Fast Green free acid

J247.014D

Fast Green free acid is a dye that resists acid once applied.
T68486 Fasitibant

Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.
T31747 Fasitibant chloride hydrochloride

Fasitibant chloride (HCl salt),MEN 16132,Fasitibant chloride,MEN-16132,MEN16132

Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.
T16954 Sulfasymazine

Antibacterial Microbiology/Virology
Sulfasymazine is a sulfonamide drug.
T125173 Fasciculic acid D

Fasciculic acid D 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125173,CAS号为 261638-74-8。
T64582 Fasudil hydrochloride semihydrate

Fasudil hydrochloride semihydrate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64582。
T25406 Fasciculic acid C

Fasciculic acid C is a calmodulin antagonist isolated from mushroom Naematoloma fasciculare.
T78453 Fast Blue B Salt

Fast Blue B Salt作为染色剂,能溶解黑麦提取物中的脂肪及苯酚化合物和重氮剂。该化合物能够用于黑麦中的烷基间苯二酚半定量分析,并在加入丙酮的情况下形成有色沉淀。
T7772 Fast Green FCF

C.I. 42053,固绿 FCF,Food green 3,FD&C Green No. 3

Others Others
Fast Green FCF (FD&C Green No. 3) 是海绿色三芳基甲烷食用染料,最大吸收在625nm 处,将在电泳过程中的蛋白质染色,。
T79416 FASN-IN-6

FASN-IN-6(Compound 44)作为脂肪酸生物合成(FAB)抑制剂表现出高效性。该化合物具备抗菌作用,针对金黄色葡萄球菌ATCC 25923及粪肠球菌ATCC 29212的最小抑菌浓度(MIC)分别为1 μg/mL与4 μg/mL。
T25404 Fasciculic acid A

Fasciculic acid A is a calmodulin antagonist isolated from mushroom Naematoloma fasciculare.
T60483 Fasedienol

Fasedienol 是一种犁鼻器 (VON) 的神经化学刺激剂,可缓解焦虑和经前综合症。
T61319 Onfasprodil

Onfasprodil, a negative allosteric modulator of NR2B, has been identified as a potential compound for researching Alzheimer's disease. This compound, in combination with a GABA receptor regulator.[1]
T28039 Milfasartan

LR-B081,LRB-081,LR-B-081,LRB 081,LR-B 081

Milfasartan is a potent, selective antagonist of AT1 receptor with oral activity. It markedly lowers the blood-pressure in conscious renal and spontaneously hypertensive rats.
T33889 Passitrifasciatin

Passitrifasciatin is a cyclopentanoid cyanohydrin glycoside isolated from Passiflora trifasciata.
T31746 Fasciculol A

Fasciculol A is a terpenoid.
T74332 Rifasutenizol

Rifasutenizol (TNP-2198)为一种有效的口服生物利用度高的双靶向抗菌剂,对微需氧菌和厌氧菌病原体展现出强大的活性。
T76901 Afasevikumab

Afasevikumab (RG 7624; RO 5553110; NI-1401) 是一种全人单克隆 IgG1κ 抗体,可中和 IL-17A 和 IL-17F。Afasevikumab 具有抗炎活性。
T62925 FASN-IN-5

FASN-IN-5 (example 11) 是一种 FASN 抑制剂,能够用于 TH17 或 CSF1 介导的疾病或障碍(如癌症、免疫障碍、肥胖症)的研究。

化合物

Fas C-Terminal Tripeptide Acetate
Cat.No: T21724L
Synonym: Fas C-Terminal Tripeptide Acetate (189109-90-8 free base)
Target: Others, Fatty Acid Synthase
FAS-IN-1 Tosylate
Cat.No: T11266L
Synonym:
Target: Fatty Acid Synthase
FASN-IN-4
Cat.No: T11266
Synonym: FAS-IN-1
Target: Others
Fasciculin-II
Cat.No: T80442
Synonym: Fas-2
Target:
Fasciculin-I
Cat.No: T82415
Synonym: FAS-I
Target:
Anti-Mouse Fas Ligand Antibody (MFL3)
Cat.No: T80584
Synonym:
Target:
Fasentin
Cat.No: T8616
Synonym: N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide
Target: transporter
Boc-Asp(OMe)-fluoromethyl ketone
Cat.No: T39308
Synonym: Boc-Asp(OMe)-fluoromethyl ketone,Boc-Asp(OMe)-FMK
Target: Caspase
Bisindolylmaleimide VIII acetate
Cat.No: T10549
Synonym: Ro 31-7549 acetate,Bis VIII acetate
Target: Apoptosis, PKC
GSK4112
Cat.No: T5045
Synonym: 1,1-Dimethylethyl-N-[(4-chlorophenyl)methyl]-N-[(5-nitro-2-thienyl)methyl])glycinate,SR6452
Target: Autophagy
Tafasitamab
Cat.No: T77135
Synonym: MOR00208,XmAb5574,Tafasitamab-cxix
Target: Apoptosis, Immunology/Inflammation related
FASN-IN-3
Cat.No: T11557
Synonym:
Target: Fatty Acid Synthase
Sulfasalazine
Cat.No: T0907
Synonym: 柳氮磺吡啶,NSC 667219,Azulfidine
Target: Apoptosis, Ferroptosis, NF-κB, COX, Antibacterial, Antibiotic, Autophagy
Parimifasor
Cat.No: T4640
Synonym: LYC30937
Target: Others
Hydroxyfasudil Hydrochloride
Cat.No: T4276
Synonym: Hydroxyfasudil (HA-1100) HCl,羟基法舒地尔盐酸盐,RHO-激酶抑制剂,HA 1100 hydrochloride
Target: ROCK
Fasnall HCl
Cat.No: T27307L
Synonym: Fasnall HCl(929978-58-5 Free base)
Target: Fatty Acid Synthase
Hydroxyfasudil
Cat.No: T4276L
Synonym: Hydroxy-Fasudil,HA-1100,羟基法舒地尔
Target: ROCK, PKA
Fasudil
Cat.No: T1606
Synonym: HA-1077,AT877,法舒地尔
Target: ROCK, Serine/threonin kinase, Calcium Channel, PKA, PKC, Autophagy
Fasudil hydrochloride
Cat.No: T3060
Synonym: Fasudil (HA-1077) HCl,盐酸法舒地尔,HA-1077,Fasudil HCl,HA-1077 hydrochloride,AT-877
Target: ROCK, Serine/threonin kinase, Calcium Channel, HIV Protease, PKA, PKC, Autophagy
Thymalfasin
Cat.No: TP1029
Synonym: 胸腺法新,Thymosin α1,醋酸胸腺α1
Target: Others
FASN-IN-1
Cat.No: T11267
Synonym: TVB-2460
Target: Fatty Acid Synthase
Fasiglifam
Cat.No: T2351
Synonym: TAK875
Target: GPR
Disperse Fast Yellow 4K
Cat.No: T9099
Synonym: 分散黄,Disperse Yellow
Target: Others
Fasidotril
Cat.No: T27306
Synonym: BP 1137,BP1137,BP-1.137,BP1.137,BP-1137,BP 1.137
Target:
FASN-IN-4 tosylate
Cat.No: T37776
Synonym:
Target:
Fasnall
Cat.No: T27307
Synonym:
Target: Fatty Acid Synthase
parathyroid hormone (7-34) [Homo sapiens]/[Macaca fascicularis]
Cat.No: TP2283
Synonym:
Target: Others
Fasudil dihydrochloride
Cat.No: T61382
Synonym:
Target:
Fasciculic acid B
Cat.No: T25405
Synonym:
Target:
Fasobegron
Cat.No: T31748
Synonym:
Target:
Fasoracetam monohydrate
Cat.No: T69954
Synonym:
Target:
Fast Green free acid
Cat.No: T31749
Synonym: J247.014D
Target:
Fasitibant
Cat.No: T68486
Synonym:
Target:
Fasitibant chloride hydrochloride
Cat.No: T31747
Synonym: Fasitibant chloride (HCl salt),MEN 16132,Fasitibant chloride,MEN-16132,MEN16132
Target:
Sulfasymazine
Cat.No: T16954
Synonym:
Target: Antibacterial
Fasciculic acid D
Cat.No: T125173
Synonym:
Target:
Fasudil hydrochloride semihydrate
Cat.No: T64582
Synonym:
Target:
Fasciculic acid C
Cat.No: T25406
Synonym:
Target:
Fast Blue B Salt
Cat.No: T78453
Synonym:
Target:
Fast Green FCF
Cat.No: T7772
Synonym: C.I. 42053,固绿 FCF,Food green 3,FD&C Green No. 3
Target: Others
FASN-IN-6
Cat.No: T79416
Synonym:
Target:
Fasciculic acid A
Cat.No: T25404
Synonym:
Target:
Fasedienol
Cat.No: T60483
Synonym:
Target:
Onfasprodil
Cat.No: T61319
Synonym:
Target:
Milfasartan
Cat.No: T28039
Synonym: LR-B081,LRB-081,LR-B-081,LRB 081,LR-B 081
Target:
Passitrifasciatin
Cat.No: T33889
Synonym:
Target:
Fasciculol A
Cat.No: T31746
Synonym:
Target:
Rifasutenizol
Cat.No: T74332
Synonym:
Target:
Afasevikumab
Cat.No: T76901
Synonym:
Target:
FASN-IN-5
Cat.No: T62925
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T21936 M50054

2,2′-亚甲基双(1,3-环己二酮)

Caspase Apoptosis; Proteases/Proteasome
M50054 是一种有效的细胞凋亡抑制剂,可用于研究抗 Fas 抗体引起的肝炎和化疗引起的脱发。它抑制 Etoposide 诱导的 U937 细胞 caspase-3 活化,IC50为 79 μg/mL。
T5S0246 Pseudoprotodioscin

山药

Others; Fatty Acid Synthase Metabolism; Others
Pseudoprotodioscin 是一种呋喃葡糖苷,抑制SREBP1/2和microRNA 33a/b 水平,降低胆固醇和甘油三酯合成相关的基因表达。
T27305 Fascaplysin chloride

NSC622398,NSC 622398,Fascaplysin,NSC-622398

Fascaplysin is a cyclin D kinase 4/ cyclin D1 inhibitor (IC50 = 0.35 μM). Fascaplysin induces caspase mediated crosstalk between autophagy and apoptosis through the inhibition of PI3K/AKT/mTOR signaling cascade in human leukemia HL-60 cells.
TJS0387 Desoxyrhaponticin

去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin

Apoptosis; Fatty Acid Synthase Apoptosis; Metabolism
Desoxyrhaponticin (Deoxyrhaponticin) 是来自西藏营养食品唐古特大黄中的一种二苯乙烯苷。它是脂肪酸合成酶抑制剂,抑制细胞内 FAS 活性,下调人乳腺癌 MCF-7细胞中 FAS 的表达。它是控制糖尿病餐后高血糖的潜在药物。
T13815 Penicillic acid

Apoptosis; Caspase; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology; Proteases/Proteasome
Penicillic acid, a polyketide mycotoxin, synthesized by various species of Aspergillus and Penicillium, acts as an inhibitor of Fas ligand-induced apoptosis by impeding self-processing of caspase-8. Additionally, in vitro studies have shown that Penicillic acid displays cytotoxic properties in rat alveolar macrophages.
TQ0260 Cerulenin

Antibiotic; Antifungal; Fatty Acid Synthase Metabolism; Microbiology/Virology
Cerulenin 是广泛使用的天然脂肪酸合成酶抑制剂。它是由真菌Cephalosporium caeruleus 产生的。它抑制拓扑异构酶I 催化活性并增强 SN-38 诱导的细胞凋亡。它具有抗真菌和抗肿瘤活性。
T4S0290 Araloside A

Chikusetsusaponin IV,竹节参皂苷IV

RAAS; Fas/FasL Apoptosis; Endocrinology/Hormones
Araloside A (Chikusetsusaponin IV) 是竹节参中的一种成分,对肾素renin 具有低抑制活性(IC50:77.4 μM)。
T3S1775 Tectochrysin

NSC 80687,Techtochrysine,Techtochrysin,柚木柯因

NF-κB; STAT JAK/STAT signaling; NF-κB; Stem Cells
Tectochrysin (Techtochrysine) 是Alpinia oxyphylla 的主要黄酮类化合物之一,能够抑制NF-κB 活性。
T2854 Phillyrin

Forsythin,连翘苷

P450; Influenza Virus; AMPK Chromatin/Epigenetic; Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
Phillyrin (Forsythin) 是从连翘中分离出来的一种天然产物,具有抗甲型流感病毒的活性,以及抗菌和消炎作用。
TN1365 Albaspidin AP

Fatty Acid Synthase Metabolism
Albaspidin-AP, -PP, -PB inhibit Fatty acid synthase (FAS) with IC50 values ranging from 23.1+/-1.4 to 71.7+/-3.9 microM, they could be considered to be a promising class of FAS inhibitors, and FAS is emerging as a potential therapeutic target to treat can
TN4496 Marginatoxin

Caspase; Fas/FasL Apoptosis; Proteases/Proteasome
Marginatoxin may be a promising chemopreventive agent for treating hepatocellular carcinoma, it induces human hepatoma BEL-7402 cells apoptosis in vitro and in vivo via activation of Fas/FasL-mediated apoptotic pathway.
TN1532 Crenulatin

BCL; Caspase Apoptosis; Proteases/Proteasome
Crenulatin has dual- direction effects on apoptosis of cerebral microvascular endothelial cells, inhibitive effect in 25 mg/L and stimulative effect in 100 mg/L group, respectively; the mechanism is related to the alterations of Fas/Bcl-2 expression and caspase-3 activity.
TMA0918 Neochamaejasmine A

Caspase Apoptosis; Proteases/Proteasome
Neochamaejasmin A can inhibit cellular (3)H-thymidine incorporation (IC 50 12.5 microg/mL) and subsequent proliferation of human prostate cancer LNCaP cells, it blocks cell cycle progression at the G1 phase by activating the p21 protein and ultimately pro

天然产物

M50054
Cat.No: T21936
Synonym: 2,2′-亚甲基双(1,3-环己二酮)
Target: Caspase
Pseudoprotodioscin
Cat.No: T5S0246
Synonym: 山药
Target: Others, Fatty Acid Synthase
Fascaplysin chloride
Cat.No: T27305
Synonym: NSC622398,NSC 622398,Fascaplysin,NSC-622398
Target:
Desoxyrhaponticin
Cat.No: TJS0387
Synonym: 去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin
Target: Apoptosis, Fatty Acid Synthase
Penicillic acid
Cat.No: T13815
Synonym:
Target: Apoptosis, Caspase, Antibacterial, Antibiotic
Cerulenin
Cat.No: TQ0260
Synonym:
Target: Antibiotic, Antifungal, Fatty Acid Synthase
Araloside A
Cat.No: T4S0290
Synonym: Chikusetsusaponin IV,竹节参皂苷IV
Target: RAAS, Fas/FasL
Tectochrysin
Cat.No: T3S1775
Synonym: NSC 80687,Techtochrysine,Techtochrysin,柚木柯因
Target: NF-κB, STAT
Phillyrin
Cat.No: T2854
Synonym: Forsythin,连翘苷
Target: P450, Influenza Virus, AMPK
Albaspidin AP
Cat.No: TN1365
Synonym:
Target: Fatty Acid Synthase
Marginatoxin
Cat.No: TN4496
Synonym:
Target: Caspase, Fas/FasL
Crenulatin
Cat.No: TN1532
Synonym:
Target: BCL, Caspase
Neochamaejasmine A
Cat.No: TMA0918
Synonym:
Target: Caspase
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