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Targets Recommended: P450 Antibiotic Antifungal

84

抑制剂 & 化合物

20

天然产物

1

TargetMol 试剂盒

6

重组蛋白

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Cat. No. Product Name Form Specificity Of Inhibition
C0110 Magrose Beads IDA-Cobalt

His-tag 蛋白纯化磁珠 IDA-Co

TargetMol 试剂盒

His-tag 蛋白纯化磁珠 IDA-Co
Cat.No: C0110
Cat. No. Product Name Target Signaling Pathways
T2305 Isavuconazole

艾沙康唑,BAL-4815,RO-0094815

P450; Antibiotic; Antifungal Metabolism; Microbiology/Virology
Isavuconazole (RO-0094815) 是一种三唑类前药,对酵母、霉菌和二型真菌具有抗真菌活性。它抑制麦角固醇生物合成,导致真菌膜结构和功能的破坏。它是 CYP3A4抑制剂。
TQ0077 Ceftobiprole

Ro 63-9141,BAL 9141,头孢吡普

Antibacterial Microbiology/Virology
Ceftobiprole (Ro 63-9141) 是一种广谱头孢菌素,对甲氧西林耐受的金黄色葡萄球菌的MIC90值为 2 μg/mL。
T14492 BAL-30072

Others Others
BAL30072 shows MIC90 values of 4 μg/mL for MDR Acinetobacter spp. and 8 μg/mL for MDR P. aeruginosa, respectively[1][2]. BAL-30072, a siderophore sulfactam, is a monocyclic beta-lactam antibiotic, with activity against multiresistant gram-negative bacilli
T21317 Avanbulin

BAL27862,BAL-27862,BAL 27862

Avanbulin is a potent inhibitor of tubulin polymerization with antitumor activity. It elicits a unique microtubule (MT) phenotype, distinct from colchicine, paclitaxel, and vinblastine has broad in vitro anti-proliferative activity against a diverse range
T40475 Ceftobiprole medocaril

BAL5788,头孢比普酯

Antibacterial Microbiology/Virology
Ceftobiprole medocaril (BAL5788) 是 Ceftobiprole 的前药。Ceftobiprole 是一种广谱的头孢菌素,对耐甲氧西林金黄色葡萄球菌具有活性。
T11679 Isavuconazole-d4

BAL-4815 D4,RO-0094815 D4,Isavuconazole D4

Others Others
Isavuconazole D4 is a deuterium labeled Isavuconazole. Isavuconazole is a triazole prodrug with antifungal activity against yeasts, molds, and dimorphic fungi.
T3104 Globalagliatin

LY2608204

Glucokinase Metabolism
Globalagliatin (LY2608204) 是一种葡萄糖激酶 (GK) 活化剂,EC50=42 nM。
T76687 Ibalizumab

TNX-355,TMB-355

HIV Protease Microbiology/Virology; Proteases/Proteasome
Ibalizumab(TMB-355) 是一种人源化 IgG4 单克隆抗体,可作为 CD4 受体抑制, 通过与 CD4 受体结合来阻止 HIV-1进入细胞。Ibalizumab 具有抗HIV-1感染活性,可用于维持机体正常免疫功能。
T4239 1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde

1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-BENZIMIDAZOLE-5-CARBALDEHYDE

Others Others
1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde 是中间体。
TP1215L Abaloparatide acetate(247062-33-5 free base)

Others Others
Abaloparatide acetate(247062-33-5 free base) 是一种甲状旁腺激素受体 1 PTHR1 类似物,是 PTHR1 信号通路的有效和选择性激活剂。
T18595 Dasatinib carbaldehyde

PROTAC ABL binding moiety 4,BMS-354825 carbaldehyde

Others; Ligands for Target Protein for PROTAC Others; PROTAC
Dasatinib carbaldehyde (PROTAC ABL binding moiety 4) 基于 ABL 抑制剂达沙替尼,通过接头与 IAP 配体结合,形成 SNIPER [1]。
T1850 Balicatib

AAE581,巴利卡替

Cysteine Protease Proteases/Proteasome
Balicatib (AAE581) 是组织蛋白酶K 抑制剂,其对组织蛋白酶K 的抑制作用是组织蛋白酶B、L 和S 的抑制性的10到100倍。
T7216 Mirogabalin

DS5565

Calcium Channel Membrane transporter/Ion channel; Metabolism
Mirogabalin (DS5565) 是一种高效的、选择性的 α2δ-1 配体,作用于电压敏感性钙通道复合体的α2δ-1亚基。
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T4615 Balsalazide sodium hydrate

巴柳氮钠水合物,Balsalazide disodium dihydrate,巴柳氮钠,Balsalazide disodium salt dihydrate,Balsalazide disodium

STAT; Interleukin Immunology/Inflammation; JAK/STAT signaling; Stem Cells
Balsalazide sodium hydrate (Balsalazide disodium) 可通过调节IL-6/STAT3通路起抑癌作用,可用于治疗炎症性肠病。
T30188L1 (Iso)-Atagabalin HCl

(Iso)-Atagabalin HCl((Iso)-223445-75-8)

Others Others
(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) 是一种可用于治疗非恢复性睡眠的α -2- δ配体。
T19245 Cobalt phthalocyanine

Cobaltous phthalocyanine,酞菁钴,Phthalocyanine cobalt complex,Cobalt(II) phthalocyanine

Others Others
Cobalt phthalocyanine (Phthalocyanine cobalt complex) 是氧化还原反应的催化剂,已经成功催化醛和酮从醛肟和酮肟中的有氧再生。
T1745 Balipodect

TAK063,TAK-063,TAK 063

PDE Metabolism
Balipodect (TAK063) 是一种高效的、口服具有活性、选择性的 PDE10A 抑制剂,IC50=0.3nM,对其他PDEs 无抑制作用。
T30188L Atagabalin HCl

PD-0200390 HCl,Atagabalin HCl(223445-75-8 Free base)

Calcium Channel Membrane transporter/Ion channel; Metabolism
Atagabalin HCl 是一种新型电压依赖性钙通道(VDCC)α2δ亚基(1 和 2)配体,会影响慢波睡眠,可用于治疗失眠。
T14495 Baloxavir

Baloxavir acid,S-033447

Influenza Virus Microbiology/Virology
Baloxavir (S-033447) 是衍生自前药 Baloxavir marboxil,是流感病毒聚合酶 PA 亚基的一流帽依赖性核酸内切酶抑制剂。它抑制病毒 RNA 的转录和复制,具有强大的抗病毒活性。
TP1215 Abaloparatide TFA

BA 058 TFA,Abaloparatide TFA (247062-33-5 free base),BIM 44058 TFA

Others Others
Abaloparatide TFA (BIM 44058 TFA) 是一种甲状旁腺激素相关蛋白 (PTHrP) 类似物药物,与相关药物特立帕肽一样用于治疗骨质疏松症。
T3104L (1S,2R)-Globalagliatin

(1S,2R)-Globalagliatin(1S,2R-1234703-40-2)

Glucokinase Metabolism
(1S,2R)-Globalagliatin 是一种高效的葡萄糖激酶 (GK) 激活剂,可用于研究 2 型糖尿病。
T13730 Hydroxocobalamin acetate

Others Others
Hydroxocobalamin acetate 是可注射的天然维生素 B12,其不良反应特征良好,可用于研究维生素 B12 缺乏症 (包括恶性贫血) 。
T6195 Baloxavir marboxil

S-033188

Influenza Virus Microbiology/Virology
Baloxavir marboxil (S-033188) 是一种新型的帽依赖性核酸内切酶抑制剂,用于治疗甲型和乙型流感病毒感染。
T14494 Balovaptan

RG7314

Vasopressin Receptor GPCR/G Protein
Balovaptan (RG7314) 是一种高效和选择性的脑渗透性血管加压素 1a (hV1a) 受体拮抗剂,对人类 (hV1a) 和小鼠 (mV1a) 受体的 Ki 值分别为 1 和 39 nM,可用于自闭症的研究。
TP2141L Balixafortide

POL6326

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
Balixafortide (POL6326) is a potent, selective, well-tolerated peptidic CXCR4 antagonist with an IC50 < 10 nM and it is also a potent hematopoietic stem and progenitor cell (HSPC) mobilizing agent. Anti-cancer effects[1][2]. Balixafortide blocks β-arresti
T80492 Mambalgin-2

Mamb-2

Sodium Channel Membrane transporter/Ion channel
Mambalgin-2 (Mamb-2)为非洲黑曼巴蛇毒中提取的酸敏感离子通道(ASICs)抑制剂及蛇毒肽,主要用途为镇痛及神经系统疾病研究。
T75954 Mambalgin 1 TFA

Mambalgin 1 TFA, a selective inhibitor of ASIC1a (with IC50 values of 192 nM for human ASIC1a and 72 nM for the ASIC1a/1b dimer), preferentially binds to the channel in its closed/inactive state. It demonstrates selectivity for ASIC1a over a range of other channels, including ASIC2a, ASIC3, TRPV1, P2X2, 5-HT3, Nav1.8, Cav3.2, and Kv1.2. In vivo, Mambalgin 1 TFA effectively prolongs the latency of the withdrawal response in mouse tail-flick and paw-flick tests.
T67067 2-Butyl-4-chloro-1H-imidazole-5-carbaldehyde

2-Butyl-4-chloro-1H-imidazole-5-carbaldehyde 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67067,CAS号为 83857-96-9。
T124815 Barbaloin-related compound A

Barbaloin-related compound A 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124815。
T24721 Robalzotan

NAD-299,AZD 7371,AZD7371,NAD 299,AZD-7371

Robalzotan is a selective 5-HT1A receptor antagonist.
T32143 Imagabalin

PD332334,PD 0332334,PD-0332334,PD0332334,PD-332334,PD 332334

Imagabalin 是一种有活性的化合物,可用来研究神经系统疾病。
T67330 5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrole-3-carbaldehyde

5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrole-3-carbaldehyde 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67330,CAS号为 881677-11-8。
T82924 Balugrastim

CG 10639

Balugrastim (CG 10639)为新型长效G-CSF,由重组人血清白蛋白与G-CSF遗传融合制成,适用于乳腺癌研究。
T82925 Baloramotide

Baloramotide,一种重组蛋白,包含182个氨基酸,源自NY-ESO-1。该化合物能够促进免疫系统对肿瘤的响应。
T16100 Balamapimod

MKI 833

Integrin Cytoskeletal Signaling
Balamapimod is a reversible inhibitor of Ras/Raf/MEK. It also has a potential anti-tumor activity.
T75328 Hydroxocobalamin hydrochloride

Hydroxocobalamin hydrochloride 是天然维生素B12的可注射形式,因其优良的安全性质,被用于研究维生素B12缺乏症(包括恶性贫血)相关治疗。
TP2141 Balixafortide TFA (1051366-32-5 free base)

Balixafortide TFA,POL6326 TFA

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
Balixafortide TFA (POL6326 TFA) is a selective, well-tolerated peptidic CXCR4 antagonist (IC50 < 10 nM). It shows 1000-fold selective for CXCR4 than a large panel of receptors including CXCR7. Balixafortide TFA blocks β-arrestin recruitment and calcium fl
T75999 Balixafortide TFA

Balixafortide TFA (POL6326 TFA) 是一种有效的,选择性的,耐受性好的肽类CXCR4拮抗剂,其IC50小于 10 nM。Balixafortide TFA 对CXCR4的选择性比包括CXCR7在内的许多受体高出 1000 倍。Balixafortide TFA 以 IC50< 10 nM 阻断β-arrestin 募集和钙通量。Balixafortide TFA 还是一种有效的造血干细胞和祖细胞 (HSPC) 动员剂,并具有抗癌作用。
T78623 Cobalt protoporphyrin IX

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Cobalt protoporphyrin IX 作为一种特异性的血红素加氧酶-1 (HO-1) 诱导剂,表现出对甲型流感病毒 (IAV) 的广谱抗病毒活性。
T22265 Balofloxacin Dihydrate

Neuroquinoron,巴洛沙星/1-环丙基-7-(3-甲氨基-1-哌啶基)-8-甲氧基-6-氟-1,4-二氢-4-氧代-3-喹啉羧酸

Others Others
Balofloxacin is a fluoroquinolone antibiotic with oral activity.
T66775 5-Phenyl-1H-pyrrole-3-carbaldehyde

5-Phenyl-1H-pyrrole-3-carbaldehyde 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66775,CAS号为 56448-22-7。
T126003 Subalpinoside

Subalpinoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126003,CAS号为 135531-62-3。
T29977 Amicarbalide diisethionate

Amicarbalide diisethionate is a bioactive chemical.
T18592 Imatinib carbaldehyde

CGP-57148B carbaldehyde,STI571 carbaldehyde,PROTAC ABL binding moiety 1

Others Others
Imatinib carbaldehyde (also known as CGP-57148B carbaldehyde) is a compound derived from Imatinib, an inhibitor of the ABL protein. Imatinib carbaldehyde binds to the IAP ligand with the assistance of a linker, resulting in the formation of SNIPER[1].
T34128 Pregabalin arenacarbil

Pregabalin arenacarbil is a gabamimetic.
T64484 4,4'-(Cyclopent-1-ene-1,2-diyl)bis(5-methylthiophene-2-carbaldehydE)

4,4'-(Cyclopent-1-ene-1,2-diyl)bis(5-methylthiophene-2-carbaldehydE) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64484。
T73690 Abaloparatide

Abaloparatide (BA 058) 是一种甲状旁腺激素受体 1 (PTHR1) 类似物。Abaloparatide 也是一种选择性 PTHR1激活剂。Abaloparatide 增强 Gs/cAMP 信号和β-arrestin 募集。Abaloparatide 可增强小鼠的骨形成和皮质结构。Abaloparatide 具有用于骨质疏松症研究的潜力。
TP1100 [bAla8]-Neurokinin A(4-10)

MEN 10210

[bAla8]-Neurokinin A(4-10) is a neurokinin 2 (NK2) receptor agonist.
T20786 Cobaltocene

Kobaltocen,Dicyclopentadienylcobalt

Cobaltocene is used to catalyze the preparation of pyridines from nitriles and alkynes. It is also used as an oxygen stripping agent and as a paint drier.

化合物

Isavuconazole
Cat.No: T2305
Synonym: 艾沙康唑,BAL-4815,RO-0094815
Target: P450, Antibiotic, Antifungal
Ceftobiprole
Cat.No: TQ0077
Synonym: Ro 63-9141,BAL 9141,头孢吡普
Target: Antibacterial
BAL-30072
Cat.No: T14492
Synonym:
Target: Others
Avanbulin
Cat.No: T21317
Synonym: BAL27862,BAL-27862,BAL 27862
Target:
Ceftobiprole medocaril
Cat.No: T40475
Synonym: BAL5788,头孢比普酯
Target: Antibacterial
Isavuconazole-d4
Cat.No: T11679
Synonym: BAL-4815 D4,RO-0094815 D4,Isavuconazole D4
Target: Others
Globalagliatin
Cat.No: T3104
Synonym: LY2608204
Target: Glucokinase
Ibalizumab
Cat.No: T76687
Synonym: TNX-355,TMB-355
Target: HIV Protease
1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde
Cat.No: T4239
Synonym: 1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-BENZIMIDAZOLE-5-CARBALDEHYDE
Target: Others
Abaloparatide acetate(247062-33-5 free base)
Cat.No: TP1215L
Synonym:
Target: Others
Dasatinib carbaldehyde
Cat.No: T18595
Synonym: PROTAC ABL binding moiety 4,BMS-354825 carbaldehyde
Target: Others, Ligands for Target Protein for PROTAC
Balicatib
Cat.No: T1850
Synonym: AAE581,巴利卡替
Target: Cysteine Protease
Mirogabalin
Cat.No: T7216
Synonym: DS5565
Target: Calcium Channel
Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Balsalazide sodium hydrate
Cat.No: T4615
Synonym: 巴柳氮钠水合物,Balsalazide disodium dihydrate,巴柳氮钠,Balsalazide disodium salt dihydrate,Balsalazide disodium
Target: STAT, Interleukin
(Iso)-Atagabalin HCl
Cat.No: T30188L1
Synonym: (Iso)-Atagabalin HCl((Iso)-223445-75-8)
Target: Others
Cobalt phthalocyanine
Cat.No: T19245
Synonym: Cobaltous phthalocyanine,酞菁钴,Phthalocyanine cobalt complex,Cobalt(II) phthalocyanine
Target: Others
Balipodect
Cat.No: T1745
Synonym: TAK063,TAK-063,TAK 063
Target: PDE
Atagabalin HCl
Cat.No: T30188L
Synonym: PD-0200390 HCl,Atagabalin HCl(223445-75-8 Free base)
Target: Calcium Channel
Baloxavir
Cat.No: T14495
Synonym: Baloxavir acid,S-033447
Target: Influenza Virus
Abaloparatide TFA
Cat.No: TP1215
Synonym: BA 058 TFA,Abaloparatide TFA (247062-33-5 free base),BIM 44058 TFA
Target: Others
(1S,2R)-Globalagliatin
Cat.No: T3104L
Synonym: (1S,2R)-Globalagliatin(1S,2R-1234703-40-2)
Target: Glucokinase
Hydroxocobalamin acetate
Cat.No: T13730
Synonym:
Target: Others
Baloxavir marboxil
Cat.No: T6195
Synonym: S-033188
Target: Influenza Virus
Balovaptan
Cat.No: T14494
Synonym: RG7314
Target: Vasopressin Receptor
Balixafortide
Cat.No: TP2141L
Synonym: POL6326
Target: CXCR
Mambalgin-2
Cat.No: T80492
Synonym: Mamb-2
Target: Sodium Channel
Mambalgin 1 TFA
Cat.No: T75954
Synonym:
Target:
2-Butyl-4-chloro-1H-imidazole-5-carbaldehyde
Cat.No: T67067
Synonym:
Target:
Barbaloin-related compound A
Cat.No: T124815
Synonym:
Target:
Robalzotan
Cat.No: T24721
Synonym: NAD-299,AZD 7371,AZD7371,NAD 299,AZD-7371
Target:
Imagabalin
Cat.No: T32143
Synonym: PD332334,PD 0332334,PD-0332334,PD0332334,PD-332334,PD 332334
Target:
5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrole-3-carbaldehyde
Cat.No: T67330
Synonym:
Target:
Balugrastim
Cat.No: T82924
Synonym: CG 10639
Target:
Baloramotide
Cat.No: T82925
Synonym:
Target:
Balamapimod
Cat.No: T16100
Synonym: MKI 833
Target: Integrin
Hydroxocobalamin hydrochloride
Cat.No: T75328
Synonym:
Target:
Balixafortide TFA (1051366-32-5 free base)
Cat.No: TP2141
Synonym: Balixafortide TFA,POL6326 TFA
Target: CXCR
Balixafortide TFA
Cat.No: T75999
Synonym:
Target:
Cobalt protoporphyrin IX
Cat.No: T78623
Synonym:
Target: Reactive Oxygen Species
Balofloxacin Dihydrate
Cat.No: T22265
Synonym: Neuroquinoron,巴洛沙星/1-环丙基-7-(3-甲氨基-1-哌啶基)-8-甲氧基-6-氟-1,4-二氢-4-氧代-3-喹啉羧酸
Target: Others
5-Phenyl-1H-pyrrole-3-carbaldehyde
Cat.No: T66775
Synonym:
Target:
Subalpinoside
Cat.No: T126003
Synonym:
Target:
Amicarbalide diisethionate
Cat.No: T29977
Synonym:
Target:
Imatinib carbaldehyde
Cat.No: T18592
Synonym: CGP-57148B carbaldehyde,STI571 carbaldehyde,PROTAC ABL binding moiety 1
Target: Others
Pregabalin arenacarbil
Cat.No: T34128
Synonym:
Target:
4,4'-(Cyclopent-1-ene-1,2-diyl)bis(5-methylthiophene-2-carbaldehydE)
Cat.No: T64484
Synonym:
Target:
Abaloparatide
Cat.No: T73690
Synonym:
Target:
[bAla8]-Neurokinin A(4-10)
Cat.No: TP1100
Synonym: MEN 10210
Target:
Cobaltocene
Cat.No: T20786
Synonym: Kobaltocen,Dicyclopentadienylcobalt
Target:
Cat. No. Product Name Target Signaling Pathways
T0176 Isobarbaloin

Aloin,Aloin-A,芦荟甙,Barbaloin-A

Tyrosinase Proteases/Proteasome
Isobarbaloin (Barbaloin-A) 是一种来自芦荟的天然蒽环类药物,是一种酪氨酸酶抑制剂。
TN7136 1,7-dimethyl-1H-indole-3-carbaldehyde

1,7-dimethylindole-3-carbaldehyde,ZINC14592128,N,7-Dimethylindole-3-carbaldehyde

Others Others
1,7-dimethyl-1H-indole-3-carbaldehyde (ZINC14592128) 是一种海洋来源的天然产物,存在于 Lyngbya majuscula。
T3136 Methylcobalamin

CH3-B12,Methyl vitamin B12,Methycobal,Brassinolide,Vancomin,Cobametin,甲钴胺

Endogenous Metabolite Metabolism
Methylcobalamin (Brassinolide) 是维生素B12的一种形式,可直接参与同型半胱氨酸代谢。
TN7184 5,6-dibromo-1H-indole-3-carbaldehyde

ZINC198368276,5,6-二溴吲哚-3-甲醛

Others Others
5,6-dibromo-1H-indole-3-carbaldehyde 是一种海洋来源的天然产物,存在于Smenospongia sp.。
T5564 Tricarballylic acid

β-Carboxyglutaric acid,1,2,3-Propanetricarboxylic acid,三碳烯丙酸,Carballylic acid,Propane-1,2,3-tricarboxylic acid,丙三酸

aconitase; Mitochondrial Metabolism Metabolism
Tricarballylic acid (Carballylic acid) 是三碳烯丙酸酯的共轭酸,是一种乌头酸水合酶的竞争性抑制剂,其 Ki= 0.52 mM。
T2808 Bilobalide

白果内酯,银杏内酯,(-)-Bilobalide

Apoptosis; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism
Bilobalide ((-)-Bilobalide) 是银杏叶中的的一种倍半萜三内酯成分,抑制 NMDA 诱导的胆碱流出,IC50值为 2.3 µM。它通过激活 SH-SY5Y 细胞中的 PI3K/Akt 通路来防止细胞凋亡。对神经元发挥保护和营养作用。
T7973 BENZOFURAN-3-CARBALDEHYDE

Others Others
BENZOFURAN-3-CARBALDEHYDE 是一种天然产物。
T14128 Adenosylcobalamin

Cobamamide,Coenzyme B12,腺苷钴胺,AdoCbl

Endogenous Metabolite Metabolism
Adenosylcobalamin (AdoCbl) 是一种 Vitamin B12的特性形式,其中 Vitamin B12 是是甲基丙二酰 CoA 突变酶的辅助因子。
T78476 Hydroxocobalamin

Vitamin B12a

Endogenous Metabolite Metabolism
Hydroxocobalamin(Vitamin B12a)为可注射型天然维生素B12,不良反应特性良好,适用于治疗维生素B12缺乏症(包括恶性贫血)的膳食补充。
TN1428 (+)-Balanophonin

Antioxidant; AChE Neuroscience; oxidation-reduction
(+)-Balanophonin 是一种从 Passiflora edulis 分离得到的天然酚类化合物,具有抗氧化、抗炎、抗癌和抗神经退行性活性,抑制胆碱酯酶,对 OPM2 和 RPMI-8226 细胞增殖有边际抑制作用。
TN5860 Euglobal Ia1

Euglobal Ia1 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5860,CAS号为 77844-93-0。
T67673 4-Hydroxy-1H-indole-3-carbaldehyde

4-Hydroxy-1H-indole-3-carbaldehyde 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T67673,CAS号为 81779-27-3。
T34323 Ribalinine

(S)-Ribalinine

Ribalinine is a quinolone alkaloid.
TN5345 8α-Methacryloyloxybalchanin

8α-Methacryloyloxybalchanin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5345,CAS号为 104021-39-8。
T13731 Hydroxocobalamin monohydrochloride

Vitamin B12a monohydrochloride,盐酸羟钴胺

Others Others
Hydroxocobalamin monohydrochloride is an injectable naturally occurring form of vitamin B12. It is used as a dietary supplement in the treatment of vitamin B12 deficiency including pernicious anemia.
TN4219 Homobaldrinal

Others Others
Homobaldrinal has low toxic activity. It has genotoxic activity in the Salmonella/microsome test and the SOS-chromotest.
TN5872 Phebalosin

Alosin

Phebalosin displays 50% effective concentrations (EC(50)) of 14.1 microg/mL against axenic amastigote forms of Leishmania panamensis. It also displays cytotoxicity (IC(50)) at concentrations of 20.7 microg/mL on human promonocytic U-937 cells.
T23772 Balanol

Ophiocordin,BA1,Azepinostatin,(-)-Balanol,(3R-trans)-Balanol

Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.
TN5858 Euglobal Ia2

Euglobal Ia2 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5858,CAS号为 77794-63-9。
TN1024 Baldrinal

Others Others
Baldrinal, valtrate, and acevaltrate are the quality control compounds of Valeriana jatamansi Jones.

天然产物

Isobarbaloin
Cat.No: T0176
Synonym: Aloin,Aloin-A,芦荟甙,Barbaloin-A
Target: Tyrosinase
1,7-dimethyl-1H-indole-3-carbaldehyde
Cat.No: TN7136
Synonym: 1,7-dimethylindole-3-carbaldehyde,ZINC14592128,N,7-Dimethylindole-3-carbaldehyde
Target: Others
Methylcobalamin
Cat.No: T3136
Synonym: CH3-B12,Methyl vitamin B12,Methycobal,Brassinolide,Vancomin,Cobametin,甲钴胺
Target: Endogenous Metabolite
5,6-dibromo-1H-indole-3-carbaldehyde
Cat.No: TN7184
Synonym: ZINC198368276,5,6-二溴吲哚-3-甲醛
Target: Others
Tricarballylic acid
Cat.No: T5564
Synonym: β-Carboxyglutaric acid,1,2,3-Propanetricarboxylic acid,三碳烯丙酸,Carballylic acid,Propane-1,2,3-tricarboxylic acid,丙三酸
Target: aconitase, Mitochondrial Metabolism
Bilobalide
Cat.No: T2808
Synonym: 白果内酯,银杏内酯,(-)-Bilobalide
Target: Apoptosis, Endogenous Metabolite, Autophagy
BENZOFURAN-3-CARBALDEHYDE
Cat.No: T7973
Synonym:
Target: Others
Adenosylcobalamin
Cat.No: T14128
Synonym: Cobamamide,Coenzyme B12,腺苷钴胺,AdoCbl
Target: Endogenous Metabolite
Hydroxocobalamin
Cat.No: T78476
Synonym: Vitamin B12a
Target: Endogenous Metabolite
(+)-Balanophonin
Cat.No: TN1428
Synonym:
Target: Antioxidant, AChE
Euglobal Ia1
Cat.No: TN5860
Synonym:
Target:
4-Hydroxy-1H-indole-3-carbaldehyde
Cat.No: T67673
Synonym:
Target:
Ribalinine
Cat.No: T34323
Synonym: (S)-Ribalinine
Target:
8α-Methacryloyloxybalchanin
Cat.No: TN5345
Synonym:
Target:
Hydroxocobalamin monohydrochloride
Cat.No: T13731
Synonym: Vitamin B12a monohydrochloride,盐酸羟钴胺
Target: Others
Homobaldrinal
Cat.No: TN4219
Synonym:
Target: Others
Phebalosin
Cat.No: TN5872
Synonym: Alosin
Target:
Balanol
Cat.No: T23772
Synonym: Ophiocordin,BA1,Azepinostatin,(-)-Balanol,(3R-trans)-Balanol
Target:
Euglobal Ia2
Cat.No: TN5858
Synonym:
Target:
Baldrinal
Cat.No: TN1024
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-03353 CEL Protein, Mouse, Recombinant (His)

1810036E18Rik,carboxyl ester lipase,BAL

Mouse Baculovirus Insect Cells
CEL-maturity onset diabetes of the young (MODY), diabetes with pancreatic lipomatosis and exocrine dysfunction, is due to dominant frameshift mutations in the acinar cell carboxyl ester lipase gene (CEL). Bile-salt activated carboxylic ester lipase (CEL) is a major triglyceride, cholesterol ester and vitamin ester hydrolytic enzyme contained within pancreatic and lactating mammary gland secretions. Carboxyl ester lipase is a digestive pancreatic enzyme encoded by the CEL gene. Mutations in CEL c...
TMPY-00316 HIV-1 (group M, subtype B, isolate BAL) gp120 Protein (His)

HIV HEK293 Cells
HIV-1 (group M, subtype B, isolate BAL) gp120 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 55.4 kDa and the accession number is Q03805.
TMPH-00314 Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI)

Bubalus bubalis E. coli
Has bactericidal activity. Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 19.8 kDa and the accession number is A3RJ36.
TMPY-04012 Influenza A H7N9 (A/Anhui/1-BALF_RG6/2013) Nucleoprotein/NP Protein (His)

NP Protein

H7N9 Baculovirus Insect Cells
Influenza A H7N9 (A/Anhui/1-BALF_RG6/2013) Nucleoprotein/NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.8 kDa and the accession number is A0A024E372.
TMPH-00551 IL-13 Protein, Equus caballus, Recombinant (His)

Horse P. pastoris (Yeast)
IL-13 Protein, Equus caballus, Recombinant (His) is expressed in Yeast.
TMPH-02281 UBALD2 Protein, Human, Recombinant (His & Myc)

Human E. coli
N/A. UBALD2 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 25.2 kDa and the accession number is Q8IYN6.

重组蛋白

CEL Protein, Mouse, Recombinant (His)
Cat.No: TMPY-03353
Species: Mouse
Expression System: Baculovirus Insect Cells
HIV-1 (group M, subtype B, isolate BAL) gp120 Protein (His)
Cat.No: TMPY-00316
Species: HIV
Expression System: HEK293 Cells
Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI)
Cat.No: TMPH-00314
Species: Bubalus bubalis
Expression System: E. coli
Influenza A H7N9 (A/Anhui/1-BALF_RG6/2013) Nucleoprotein/NP Protein (His)
Cat.No: TMPY-04012
Species: H7N9
Expression System: Baculovirus Insect Cells
IL-13 Protein, Equus caballus, Recombinant (His)
Cat.No: TMPH-00551
Species: Horse
Expression System: P. pastoris (Yeast)
UBALD2 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-02281
Species: Human
Expression System: E. coli
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