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183

抑制剂 & 化合物

101

天然产物

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Cat. No. Product Name Target Signaling Pathways
T28869 Streptomyces A-Factor

A-Factor (Lactone)

Streptomyces A-Factor is a microbial hormone found in Streptomyces griseus. A-factor triggers streptomycin biosynthesis and cell differentiation by binding a repressor-type receptor protein (ArpA) and dissociating it from DNA.
T26231 Acetyl-pepstatin

Streptomyces pepsin inhibitor,Ac-Pepstatin,乙酰胃泌素

Streptomyces pepsin inhibitor is used as a pepsin inhibitor.
T8814 Nikkomycin Z

尼柯霉素Z,Nikkomycin Z from Streptomyces tendae,尼柯霉素 Z

Others; Antibiotic; Antifungal Microbiology/Virology; Others
Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) 是一种选择性竞争性几丁质合成抑制剂。它是一种核苷肽,可作为几丁质合酶底物 UDP-N-乙酰氨基葡萄糖的竞争性类似物,具有抗真菌作用。
T4989 Fosfomycin Tromethamine

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin tromethamine 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T24243 Kanosamine

3-Amino-3-deoxyglucose,3-氨基-3-脱氧-D-葡萄糖

Antifungal Microbiology/Virology
Kanosamine (3-Amino-3-deoxyglucose) 是一种由链霉菌产生的抗真菌剂。
T0788L Spectinomycin dihydrochloride pentahydrate

盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride pentahydrate (Spectogard) 是一种广谱氨基环糊精抗生素,可以抑制多种革兰氏阳性和革兰氏阴性生物的生长。
T60020 5'-Fluoro-5'-deoxyadenosine

5'-Fluoro-5'-deoxy-adenosine

Others Others
5'-Fluoro-5'-deoxyadenosine (5'-Fluoro-5'-deoxy-adenosine) 常用作研究放线菌卡特链霉菌的工具。
T19724 5NAA

5-NAA,2-氨基-5-硝基苯甲酸,5 NAA

Others Others
5NAA 是一种由疥疮链霉菌分泌的分子,可合成染料和其他硝基芳族化合物的原料。
T16551 Pladienolide B

Apoptosis Apoptosis
Pladienolide B 是一种有效的剪接体抑制剂,是从钝顶链霉菌 Mer-12 中分离出的大环内酯类化合物,其作用靶向剪接体的 SF3B1 亚单位。Pladienolide B 通过抑制前 mRNA 剪接发挥抗肿瘤作用,诱导调亡。Pladienolide B 具有抗肿瘤活性,可用于研究白血病和淋巴肿瘤。
T19860 Clavulanic Acid

BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151

Antibacterial; Antifungal Microbiology/Virology
Clavulanic Acid(RX-10100) 是一种由生物体克拉维链霉菌产生的主要β-内酰胺类抗生素,是一种强效的细菌 β-内酰胺酶抑制剂,用于研究细菌引起的感染。Clavulanic Acid 具有广谱的生物活性,对多种革兰氏阳性和革兰氏阴性细菌均有活性。
T30080 Ansatrienin A3

Ansatrienin A3 is produced by Streptomyces collinus.
T25422 Flambamycin

RP21190,RP-21190,RP 21190

Flambamycin is an antibiotic isolated from Streptomyces hygroscopicus.
T25037 Aldecalmycin

Aldecalmycin is a new antimicrobial antibiotic isolated from Streptomyces.
T25504 Histargin

Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.
T26116 Rokitamycin

Rokitamycin is a macrolide antibiotic produced from strains of Streptomyces kitasatoensis.
T26420 A 53868A

Dehydrophos,A-53868A,A53868A

A 53868A is an antibiotic, it is isolated from Streptomyces luridus.
T25689 Leuseramycin

TM 531,TM531,Antibiotic TM-531,TM-531

Leuseramycin is a polyether antibiotic isolated from Streptomyces hygroscopicus TM-531.
T26476 A28695B

A 28695B,A-28695B

A28695B is a polyether antibiotic, it is isolated from Streptomyces albus.
T25987 Probestin

Probestin is an aminopeptidase M inhibitor, isolated from Streptomyces azureus MH663-2F6.
T26178 SB-217452

SB217452

SB-217452 is a potent seryl tRNA synthetase inhibitor isolated from Streptomyces.
T26416 A 33853

A-33853,A33853

A 33853 is an antibiotic isolated from culture broth of Streptomyces sp.
T26275 Thrazarine

Thrazarine is a new antitumor antibiotic agent produced by Streptomyces coerulescens MH802-fF5.
T71367 OM-4842

OM-4842 is a platelet aggregation inhibitor from Streptomyces.
T33396 Misakimycin

Misakimycin is a mammalian cell growth stimulating substance produced by Streptomyces misakiensis BP-3621.
T38500 Enduracidin

Enramycin,恩拉霉素

Enduracidin (Enramycin) is a polypeptide antibiotic produced by Streptomyces fungicides.
T32688 Leustroducsin C

LSN C

Leustroducsin C is an inducer of colony-stimulating factors CSF extracted from Streptomyces platensis SANK 60191.
T32122 Hydroxypepstatin

Hydroxypepstatin is a new peptatin produced by Streptomyces.
T26176 Saphenamycin

Racemic ssaphenamycin

Saphenamycin is an antibiotic from a strain of Streptomyces.
T26160 Rubomycin H

Rubomycin H is an anthracycline antibiotic from Streptomyces coeruleorubidus.
T33672 Nikkomycin pseudo-J

Nikkomycin pseudo-J is a nikkomycin isolated from Streptomyces tendae.
T25027 Albocycline

TA-2407,Ingramycin

Albocycline is a Macrolide antibiotic from Streptomyces bruneogriseus nov. sp. MCRL-0129; specifically anti-staphylococcal, including antibiotic-resistant strains.
T25587 Kujimycin A

Desacetyllankamycin

Kujimycin A is a macrolide antibiotics agent from various strains of Streptomyces. It has great activity against some Gram-positive bacteria.
T25938 Pepstanone A

Pepstanone A is a potent aspartyl protease inhibitor, produced by pepstatin-producing Streptomyces.
T69996 A-75943

A-75943 is a bone resorption inhibitor from streptomyces.
T68675 Porfiromycin

Porfiromycin is a n N-methyl derivative of the antineoplastic antibiotic mitomycin C isolated from the bacterium Streptomyces ardus and other Streptomyces bacterial species. Bioreduced porfiromycin generates oxygen radicals and alkylates DNA, producing interstrand cross-links and single-strand breaks, thereby inhibiting DNA synthesis. Porfiromycin is preferentially toxic to hypoxic cells.
T28185 Nogalamycin

Nogalamycinum,U 15167,Nogalamyicn,U-15167,Nogalamycine,Nogalomycin

Nogalamycin is an anthracycline antibiotic with antitumor properties produced by soil bacteria Streptomyces nogalater.
T25762 Lucimycin

FI1163,Antibiotic 1163 F.I.,FI 1163,FI-1163,NSC 143257

Lucimycin is a macrolide antibiotic from cultures of Streptomyces lucensis.
T25270 Conagenin

Conagenin is a small molecular immunomodulator isolated by Streptomyces roseosporus.
T25871 Nikkomycin J

Nikkomycin J is used as an insecticide from Streptomyces tendae.
T32810 LL-C 10037alpha

LLC 10037alpha,LL-c10037alpha

LL-C 10037alpha is a gamma-aminoepoxysemiquinone isolated from Streptomyces.
T26088 Rimocidin

Rimocidine

Rimocidin is a macrolide antifungal compound isolated from Streptomyces rimosus.
T29419 3'-Rhamnopiericidin A(1)

SN-198-C

3'-Rhamnopiericidin A(1) is a piericidin rhamnoside from Streptomyces.
T26333 WS 9326A

WS9326A,WS-326A

WS 9326A is an antagonist of tachykinin receptor from Streptomyces violaceusniger.
T35139 WS 1279

WS1279,WS-1279

WS 1279 is an immunoactive lipopeptide that is isolated from Streptomyces.
T26411 A 269A

A269A

A 269A is an antibiotic isolated from broth of Streptomyces sp., strain.
T25973 Poststatin

Poststatin is a prolyl endopeptidase inhibitor produced by Streptomyces viridochromogenes MH534-30F3.
T24190 Jadomycin B

A jadomycin is an anacyclic natural product produced by Streptomyces venezuelae ISP5230.
T28756 Septamycin

A 28695A,A28695A,A-28695A

Septamycin is a polycyclic, polyether, monocarboxylic acid antibiotic. Septamycin is isolated from strain of Streptomyces albus.
T26406 A 204

Antibiotic A-204,Antibiotic A204,A-204,Antibiotic A 204,A204

A 204 is a polycyclic polyether monocarboxylic acid antibiotic isolated from fermentation of strain of Streptomyces albus.
T32624 Leinamycin

DC107,(+)-Leinamycin,DC 107,DC-107,Antibiotic DC 107

Leinamycin is a thiazole containing macrolide that is extracted from Streptomyces possibly used as a DNA alkylator.

化合物

Streptomyces A-Factor
Cat.No: T28869
Synonym: A-Factor (Lactone)
Target:
Acetyl-pepstatin
Cat.No: T26231
Synonym: Streptomyces pepsin inhibitor,Ac-Pepstatin,乙酰胃泌素
Target:
Nikkomycin Z
Cat.No: T8814
Synonym: 尼柯霉素Z,Nikkomycin Z from Streptomyces tendae,尼柯霉素 Z
Target: Others, Antibiotic, Antifungal
Fosfomycin Tromethamine
Cat.No: T4989
Synonym:
Target: Antibacterial, Antibiotic
Kanosamine
Cat.No: T24243
Synonym: 3-Amino-3-deoxyglucose,3-氨基-3-脱氧-D-葡萄糖
Target: Antifungal
Spectinomycin dihydrochloride pentahydrate
Cat.No: T0788L
Synonym: 盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
5'-Fluoro-5'-deoxyadenosine
Cat.No: T60020
Synonym: 5'-Fluoro-5'-deoxy-adenosine
Target: Others
5NAA
Cat.No: T19724
Synonym: 5-NAA,2-氨基-5-硝基苯甲酸,5 NAA
Target: Others
Pladienolide B
Cat.No: T16551
Synonym:
Target: Apoptosis
Clavulanic Acid
Cat.No: T19860
Synonym: BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151
Target: Antibacterial, Antifungal
Ansatrienin A3
Cat.No: T30080
Synonym:
Target:
Flambamycin
Cat.No: T25422
Synonym: RP21190,RP-21190,RP 21190
Target:
Aldecalmycin
Cat.No: T25037
Synonym:
Target:
Histargin
Cat.No: T25504
Synonym:
Target:
Rokitamycin
Cat.No: T26116
Synonym:
Target:
A 53868A
Cat.No: T26420
Synonym: Dehydrophos,A-53868A,A53868A
Target:
Leuseramycin
Cat.No: T25689
Synonym: TM 531,TM531,Antibiotic TM-531,TM-531
Target:
A28695B
Cat.No: T26476
Synonym: A 28695B,A-28695B
Target:
Probestin
Cat.No: T25987
Synonym:
Target:
SB-217452
Cat.No: T26178
Synonym: SB217452
Target:
A 33853
Cat.No: T26416
Synonym: A-33853,A33853
Target:
Thrazarine
Cat.No: T26275
Synonym:
Target:
OM-4842
Cat.No: T71367
Synonym:
Target:
Misakimycin
Cat.No: T33396
Synonym:
Target:
Enduracidin
Cat.No: T38500
Synonym: Enramycin,恩拉霉素
Target:
Leustroducsin C
Cat.No: T32688
Synonym: LSN C
Target:
Hydroxypepstatin
Cat.No: T32122
Synonym:
Target:
Saphenamycin
Cat.No: T26176
Synonym: Racemic ssaphenamycin
Target:
Rubomycin H
Cat.No: T26160
Synonym:
Target:
Nikkomycin pseudo-J
Cat.No: T33672
Synonym:
Target:
Albocycline
Cat.No: T25027
Synonym: TA-2407,Ingramycin
Target:
Kujimycin A
Cat.No: T25587
Synonym: Desacetyllankamycin
Target:
Pepstanone A
Cat.No: T25938
Synonym:
Target:
A-75943
Cat.No: T69996
Synonym:
Target:
Porfiromycin
Cat.No: T68675
Synonym:
Target:
Nogalamycin
Cat.No: T28185
Synonym: Nogalamycinum,U 15167,Nogalamyicn,U-15167,Nogalamycine,Nogalomycin
Target:
Lucimycin
Cat.No: T25762
Synonym: FI1163,Antibiotic 1163 F.I.,FI 1163,FI-1163,NSC 143257
Target:
Conagenin
Cat.No: T25270
Synonym:
Target:
Nikkomycin J
Cat.No: T25871
Synonym:
Target:
LL-C 10037alpha
Cat.No: T32810
Synonym: LLC 10037alpha,LL-c10037alpha
Target:
Rimocidin
Cat.No: T26088
Synonym: Rimocidine
Target:
3'-Rhamnopiericidin A(1)
Cat.No: T29419
Synonym: SN-198-C
Target:
WS 9326A
Cat.No: T26333
Synonym: WS9326A,WS-326A
Target:
WS 1279
Cat.No: T35139
Synonym: WS1279,WS-1279
Target:
A 269A
Cat.No: T26411
Synonym: A269A
Target:
Poststatin
Cat.No: T25973
Synonym:
Target:
Jadomycin B
Cat.No: T24190
Synonym:
Target:
Septamycin
Cat.No: T28756
Synonym: A 28695A,A28695A,A-28695A
Target:
A 204
Cat.No: T26406
Synonym: Antibiotic A-204,Antibiotic A204,A-204,Antibiotic A 204,A204
Target:
Leinamycin
Cat.No: T32624
Synonym: DC107,(+)-Leinamycin,DC 107,DC-107,Antibiotic DC 107
Target:
Cat. No. Product Name Target Signaling Pathways
T15277 Fervenulin

Parasite Microbiology/Virology
Fervenulin 具有杀灭线虫活性,抑制线虫M. incognita 卵孵化和 J2 的校正死亡率,MIC 分别为 30 μg/mL 和 120 μg/mL。
T1032 Erythromycin

红霉素,E-Mycin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Erythromycin (E-Mycin) 是由放线菌产生的大环内酯类抗生素。它结合细菌的 50S 核糖体亚基,通过阻断转肽和易位反应来抑制 RNA 依赖性蛋白的合成。
T37009 Oxychlororaphine

吩嗪-1-甲酰胺,phenazine-1-carboxamide

Antibacterial Microbiology/Virology
Oxychlororaphine (phenazine-1-carboxamide) 强烈抑制 Streptomyces sp. 411 的生长。
TN7185 7-Cyano-7-deazaguanine

7-CN-7-deazaG

Others Others
7-Cyano-7-deazaguanine (7-CN-7-deazaG) 是一种海洋来源的天然产物,存在于Streptomyces qinglanensis。
TN7147 6-Hydroxyisatin

6-Hydroxy-1H-indole-2,3-dione,ZINC14455608,6-hydroxyindoline-2,3-dione,6-羟基靛红,6-hydroxy-2,3-dihydro-1H-indole-2,3-dione

Others Others
6-Hydroxyisatin (ZINC14455608) 是一种海洋来源的天然产物,存在于 Streptomyces sp.。
T2762 Kasugamycin hydrochloride

Kasumin,盐酸春雷霉素

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Kasugamycin hydrochloride (Kasumin) 是一种能结合 30s 和 70s 核糖体,但不能结合 50s 亚基的抗生素。它模拟 mRNA 核苷酸以破坏 tRNA 结合并抑制经典翻译起始。
TN6961 Heneicosane

N-HENEICOSANE,正二十一烷,henicosane

Antifungal Microbiology/Virology
Heneicosane (henicosane) 是一种信息素,是从 Streptomyces philanthiRL-1-178 或 Serapias cordigera 中分离出来的一种香气成分,可抑制黄曲霉毒素的产生。
T1255 Tobramycin

NSC 180514,妥布霉素,Nebramycin Factor 6,Deoxykanamycin B

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Tobramycin (NSC-180514) 是一种胃肠外给药的广谱氨基糖苷类抗生素,可研究由于敏感生物引起的中度至重度细菌感染疾病。
T1003 Tylosin

Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine

Antibacterial; Antibiotic Microbiology/Virology
Tylosin (Tylosine) 是一种兽医用大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高抗菌活性。它是饲料添加剂用于促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
T11665 Ionomycin calcium

SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)

Apoptosis; Calcium Channel; Antibacterial; Antibiotic; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Ionomycin calcium (SQ23377 calcium) 是选择性钙离子载体,也是一种由 Streptomyces conglobatus 产生的抗生素。它对二价阳离子具有高度特异性,还诱导蛋白激酶 C 激活。Ionomycin 促进细胞凋亡。
T1505 Imipenem monohydrate

N-Formimidoyl thienamycin monohydrate,亚胺培南,Imipenem,亚胺培南一水物

Antibacterial; Antibiotic Microbiology/Virology
Imipenem monohydrate (Imipenem) 是从微生物 Streptomyces cattleya 分离得到的碳青霉烯类抗生素,是一种用于静脉注射的β 内酰胺类抗生素,作用于细菌细胞壁,能广泛有效抑制多种革兰氏阳性和阴性菌。
TQ0158 Azaserine

CI-337,偶氮丝胺酸,P-165,氮杂丝氨酸,O-Diazoacetyl-L-serine

Others; Antibiotic Microbiology/Virology; Others
Azaserine (CI-337) 是一种从链霉菌属中分离出来的肿瘤抑制抗生素,可作为谷氨酰胺氨基转移酶的抑制剂。
T13827 Pronase E (Activity ≥ 7000 U/g)

Pronase,Pronase E

Others Others
Pronase E 是一种蛋白水解酶混合物,从灰色链霉菌 (Streptomyces griseus) 中获得,能够将蛋白质消化成单个氨基酸。
T21430 Oxytetracycline Hydrochloride

Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin

Antiviral; Endogenous Metabolite; Antibacterial; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology
Oxytetracycline Hydrochloride (Dalimycin) 是由 Streptomyces rimosus 生产的,一种具有抗菌活性的四环素衍生物。它干扰氨酰-tRNA 与 mRNA-核糖体复合物的结合,从而阻止肽延伸并抑制蛋白质合成。
T1214 Ribostamycin sulfate

Vistamycin sulfate,硫酸核糖霉素

Antibacterial; Antibiotic Microbiology/Virology
Ribostamycin sulfate (Vistamycin sulfate) 是一种广谱抗菌剂, 在30S 和50S 核糖体亚基结合抑制细菌蛋白质合成, 还抑制蛋白二硫键异构酶分子伴侣活性, 用于药代动力学和肾毒性研究。
T0974 Novobiocin Sodium

Albamycinsodium,新生霉素钠,Cathomycin,Albamycin

Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。 它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
T64911 Blasticidin S HCl

Antibiotic Microbiology/Virology
Blasticidin S HCl 是从 Streptomyces griseochromogenes 中分离的肽基核苷类抗生素 (antibiotic),主要通过干扰核糖体中肽键的形成从而抑制原核细胞和真核细胞蛋白的合成。
T15717 Lasalocid

Lasalocid-A,Antibiotic X-537A,Ionophore X-537A

Antibacterial Microbiology/Virology
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。
T1679 Thiostrepton

Thiactin,Bryamycin,Alaninamide,硫链丝菌素

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Thiostrepton (Alaninamide) 是一种选择性抑制FOXM1的抗生素。FOXM1会与 YAP/TEAD 复合物结合,形成YAP/TEAD/FOXM1 复合物。
T0474 Erythromycin ethylsuccinate

EES,琥乙红霉素

ribosome; HIV Protease; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Erythromycin ethylsuccinate (EES) 是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗 HIV-1病毒活性。
TJS0161 Eudesmol

β-Eudesmol,桉叶醇,Β-桉叶醇

Others Others
β-Eudesmol (β-Eudesmol) 是一种倍半萜类化合物,由Streptomyces tendae 产生。
T1033 Monensin sodium salt

莫能菌素钠盐,Sodium Monensin,Monensin A sodium salt

Sodium Channel; Antibacterial; Antibiotic Membrane transporter/Ion channel; Microbiology/Virology
Monensin sodium salt (Monensin A sodium salt) 是由肉桂链霉菌 分泌的抗生素。它是一种介导Na+/H+交换的离子载体。它引起细胞多泡体 (MVBs) 增大并调节外泌体的分泌。
T67708 Thiolutin

Acetopyrrothin

Antibacterial; Antibiotic Microbiology/Virology
Thiolutin (Acetopyrrothin) 是一种内皮细胞粘附抑制剂,由链霉菌产生。 Thiolutin 具有抗生素和抗血管生成特性。 Thiolutin 可快速诱导 Hsp27 的磷酸化。
T0788 Spectinomycin dihydrochloride

淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride (Actinospectacin) 是一种能与细菌核糖体的30S 亚基结合,干扰蛋白质合成的抗生素。
T15716 Lasalocid sodium

拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Lasalocid sodium (Lasalocid-A sodium) 是一种抗菌剂。
T8373 6-Diazo-5-oxo-L-nor-Leucine

DON,L-6-Diazo-5-oxonorleucine,6-重氮-5-氧代-L-正亮氨酸,Diazooxonorleucine

Influenza Virus; Glutaminase; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
6-Diazo-5-oxo-L-nor-Leucine (L-6-Diazo-5-oxonorleucine) 是一种谷氨酰胺拮抗剂,具有抗菌、抗病毒和抗癌作用,其Ki 值为 6 μM。它能降低肿瘤细胞的自我更新能力和转移能力 ,在体外表现出遗传毒性。
T79972 Cyclo(L-leucyl-L-valyl)

Antifungal Microbiology/Virology
Cyclo(L-leucyl-L-valyl) 是从昆明链霉菌 YIM 次级代谢产物中部分离得到的多要化合物,尚未显示出抗菌活性。
T7285 Ionomycin

Calcium Channel Membrane transporter/Ion channel; Metabolism
Ionomycin 是一种钙离子载体和一种结合钙离子(Ca2+)的抗生素。它是由联合链霉菌(Streptomyces conglobatus)产生的。它在研究中用于提高细胞内钙水平(Ca2+),并作为了解 Ca2+跨生物膜运输的研究工具。Ionomycin 可促进细胞凋亡,诱导蛋白激酶 C (PKC)活化。
T0895 Oxytetracycline

土霉素,Terramycin

ribosome; Endogenous Metabolite; Antibacterial; Antibiotic; HSV Metabolism; Microbiology/Virology
Oxytetracycline (Terramycin) 是一种四环素类抗生素。它强力抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,具有抗 HSV-1的活性。
T6758 Anisomycin

茴香霉素,Flagecidin,NSC 76712,Wuningmeisu C

Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic; JNK Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; MAPK; Microbiology/Virology
Anisomycin (NSC-76712) 是一种从各种链霉菌属中分离出来的抗生素。 它通过抑制肽基转移酶或 80S 核糖体系统来干扰蛋白质和 DNA 合成。
T16340 Nosiheptide

RP 9671,Multhiomycin,那西肽

Antibacterial; Antibiotic Microbiology/Virology
Nosiheptide (Multhiomycin) 是一种由 Streptomyces actuosus 生产的硫肽类抗生素,已被广泛用作动物生长的饲料添加剂。它抑制细菌蛋白质合成,并在特征性大环核心上带有独特的吲哚侧环系统和区域特异性羟基。
T3607 Leucomycin

吉他霉素,Kitasamycin,Leucomycin V,Turimycin

Antibacterial; Antibiotic Microbiology/Virology
Leucomycin (Turimycin) 是一种由 Streptomyces kitasatoensis 产生的大环内酯类抗生素。
T0819 Spiramycin

Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Spiramycin (Rovamycin) 是一种由安博链霉菌产生的大环内酯类抗生素,具有抗细菌和弓形虫活性,并具有抗寄生虫作用。它由 16 个内酯环组成,其上附着 mycaminose,forosamine 和 mycarose 三种糖。
T4038 Ectoine

THP(B),L-Ectoine,四氢甲基嘧啶羧酸

Others; Antibacterial Microbiology/Virology; Others
Ectoine (L-Ectoine) 是生活在极其恶劣环境中的细菌所产生的氨基酸衍生物,是一种天然的细胞保护剂。它具有良好的安全性,可研究过敏性鼻炎。它用作渗透调节相容性溶质,可增加皮肤表面的水合作用并稳定脂质层,常用于皮肤护理。
T1235 Lincomycin hydrochloride monohydrate

洁霉素盐酸盐,林可霉素,Lincomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Lincomycin hydrochloride monohydrate (Lincomycin hydrochloride hydrate) 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。
T8118 Bekanamycin

Kanamycin B,卡那霉素,卡那霉素 B

Antibacterial; Antibiotic Microbiology/Virology
Bekanamycin (Kanamycin B) 是一种提取自 Streptomyces kanamyceticus 的氨基糖苷类抗生素,抑制一系列革兰氏阳性和阴性细菌。
T15091 Decoyinine

Decynylene,Angustmycin A

Decoyinine (Decynylene) 是一种选择性的GMP 合成酶抑制剂,是一种新型的潜在微生物杀虫剂,是一种由透明链霉菌产生的次级代谢产物。Decoyinine 诱导水稻对小棕瓢虫Laodelphax striatellus 的抗性。
T5285 3-(Methylthio)propionic acid

3-Methylthiopropionate,3-甲基硫代丙酸,4-Thiapentanoic acid,3-Methylsulfanylpropionic acid

Others; Endogenous Metabolite; Antifungal Metabolism; Microbiology/Virology; Others
3-(Methylthio)propionic acid (4-Thiapentanoic acid) 是methionine 的代谢物,是中间体。
T0912 Tetracycline hydrochloride

NCI-c55561,盐酸四环素,Tetracycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Tetracycline hydrochloride (NCI-c55561) 是一种广谱抗生素,抑制多种革兰氏阳性和革兰氏阴性细菌。
T1506 Vidarabine

Adenine Arabinoside,阿糖腺苷,9-β-D-Arabinofuranosyladenine,Vira-A,Arabinosyladenine,Ara-A

Nucleoside Antimetabolite/Analog; Tyrosine Kinases; DNA/RNA Synthesis; Antibiotic; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Tyrosine Kinase/Adaptors
Vidarabine (Adenine Arabinoside) 是从链霉菌分离的核苷类抗生素,能抗单纯性疱疹和水痘-带状疱疹病毒。它对 HSV-1 和 HSV-2 的 IC50值分别为 9.3 μg/ml 和 11.3 μg/ml。
T14329 Ascamycin

Nucleoside Antimetabolite/Analog; Others; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ascamycin 是一种由链霉菌属产生的 5'-O-磺酰胺核糖核苷抗生素,对黄单胞菌类显示出选择性的抗菌活性,对柠檬黄单胞菌、口蹄疫黄单胞菌和噬菌体具有抑制作用,MIC 值分别为0.4μg/mL、12.5μg/mL 和12.5μg/mL。
T10662L Calcimycin

Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187

Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal Apoptosis; Autophagy; Microbiology/Virology
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。
T20879 Tacrolimus monohydrate

FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506

Phosphatase; Others; Antibacterial; Antibiotic; Autophagy Autophagy; Metabolism; Microbiology/Virology; Others
Tacrolimus monohydrate (LCP-Tacro) 是大环内酯类化合物,它与 FK506 结合蛋白 (FKBP) 结合形成复合物并抑制钙调神经磷酸酶,从而抑制 T 淋巴细胞信号转导和 IL-2 转录。具有强免疫抑制特性。
T0861 Tylosin tartrate

酒石酸泰洛星,酒石酸泰乐菌素

Antibacterial; Antibiotic Microbiology/Virology
Tylosin tartrate 是一种大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高效的抗菌活性。它作为饲料添加剂可促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
T8504 Dianemycin

Nanchangmycin (free acid)

Antibacterial; Antibiotic Microbiology/Virology
Dianemycin (Nanchangmycin (free acid)) 由Streptomyces nanchangensis 产生的一种聚醚抗生素,抑制革兰氏阳性菌。它也是一种针对 Zika 病毒的广谱抗病毒药物。
T7004 Tubercidin

结核菌素,杀结核菌素,Sparsomycin A,7-Deazaadenosine

Influenza Virus; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Tubercidin (Sparsomycin A) 是从Streptomyces tubercidicus 得到的抗生素,抑制粪链球菌生长的IC50值为 0.02 μM。它是腺苷磷酸化酶的弱抑制剂,并干扰腺苷和 AMP 的磷酸化。它有抗病毒作用。
T24729 Roseoflavin

Antibacterial Microbiology/Virology
Roseoflavin 是天然色素,起初分离自Streptomyces davawensis。Roseoflavin 是核黄素和黄素单核苷酸的抗代谢类似物,显示出抗菌活性。
T26405 A 201A

Antibiotic 201A,A201A,A-201A

A 201A is a nucleoside antibiotic, it is isolated from Streptomyces capreolus.
T25305 Demethoxyrapamycin

AY 24668,AY24668,AY-24668

Demethoxyrapamycin is a new antifungal antibiotic agent which is co-produced with rapamycin by Streptomyces hygroscopicus.
T25622 Lankacidins

Bundlin A,Lankacidin C,Antibiotic T-2636 C,NSC 145118,Lankacidin

Lankacidins is an antitumor antibiotic of the macrolide tetraenes family from Streptomyces.
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天然产物

Fervenulin
Cat.No: T15277
Synonym:
Target: Parasite
Erythromycin
Cat.No: T1032
Synonym: 红霉素,E-Mycin
Target: ribosome, Antibacterial, Antibiotic
Oxychlororaphine
Cat.No: T37009
Synonym: 吩嗪-1-甲酰胺,phenazine-1-carboxamide
Target: Antibacterial
7-Cyano-7-deazaguanine
Cat.No: TN7185
Synonym: 7-CN-7-deazaG
Target: Others
6-Hydroxyisatin
Cat.No: TN7147
Synonym: 6-Hydroxy-1H-indole-2,3-dione,ZINC14455608,6-hydroxyindoline-2,3-dione,6-羟基靛红,6-hydroxy-2,3-dihydro-1H-indole-2,3-dione
Target: Others
Kasugamycin hydrochloride
Cat.No: T2762
Synonym: Kasumin,盐酸春雷霉素
Target: Antibacterial, Antibiotic, Antifungal
Heneicosane
Cat.No: TN6961
Synonym: N-HENEICOSANE,正二十一烷,henicosane
Target: Antifungal
Tobramycin
Cat.No: T1255
Synonym: NSC 180514,妥布霉素,Nebramycin Factor 6,Deoxykanamycin B
Target: ribosome, Antibacterial, Antibiotic
Tylosin
Cat.No: T1003
Synonym: Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine
Target: Antibacterial, Antibiotic
Ionomycin calcium
Cat.No: T11665
Synonym: SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)
Target: Apoptosis, Calcium Channel, Antibacterial, Antibiotic, PKC
Imipenem monohydrate
Cat.No: T1505
Synonym: N-Formimidoyl thienamycin monohydrate,亚胺培南,Imipenem,亚胺培南一水物
Target: Antibacterial, Antibiotic
Azaserine
Cat.No: TQ0158
Synonym: CI-337,偶氮丝胺酸,P-165,氮杂丝氨酸,O-Diazoacetyl-L-serine
Target: Others, Antibiotic
Pronase E (Activity ≥ 7000 U/g)
Cat.No: T13827
Synonym: Pronase,Pronase E
Target: Others
Oxytetracycline Hydrochloride
Cat.No: T21430
Synonym: Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin
Target: Antiviral, Endogenous Metabolite, Antibacterial, HSV
Ribostamycin sulfate
Cat.No: T1214
Synonym: Vistamycin sulfate,硫酸核糖霉素
Target: Antibacterial, Antibiotic
Novobiocin Sodium
Cat.No: T0974
Synonym: Albamycinsodium,新生霉素钠,Cathomycin,Albamycin
Target: Potassium Channel, DNA gyrase, Topoisomerase, Antibacterial, Antibiotic, ABC, Autophagy
Blasticidin S HCl
Cat.No: T64911
Synonym:
Target: Antibiotic
Lasalocid
Cat.No: T15717
Synonym: Lasalocid-A,Antibiotic X-537A,Ionophore X-537A
Target: Antibacterial
Thiostrepton
Cat.No: T1679
Synonym: Thiactin,Bryamycin,Alaninamide,硫链丝菌素
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Erythromycin ethylsuccinate
Cat.No: T0474
Synonym: EES,琥乙红霉素
Target: ribosome, HIV Protease, Antibacterial, Antibiotic, Autophagy
Eudesmol
Cat.No: TJS0161
Synonym: β-Eudesmol,桉叶醇,Β-桉叶醇
Target: Others
Monensin sodium salt
Cat.No: T1033
Synonym: 莫能菌素钠盐,Sodium Monensin,Monensin A sodium salt
Target: Sodium Channel, Antibacterial, Antibiotic
Thiolutin
Cat.No: T67708
Synonym: Acetopyrrothin
Target: Antibacterial, Antibiotic
Spectinomycin dihydrochloride
Cat.No: T0788
Synonym: 淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin
Target: ribosome, Antibacterial, Antibiotic
Lasalocid sodium
Cat.No: T15716
Synonym: 拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium
Target: Antibacterial, Antibiotic, Autophagy
6-Diazo-5-oxo-L-nor-Leucine
Cat.No: T8373
Synonym: DON,L-6-Diazo-5-oxonorleucine,6-重氮-5-氧代-L-正亮氨酸,Diazooxonorleucine
Target: Influenza Virus, Glutaminase, Antibacterial, Antibiotic
Cyclo(L-leucyl-L-valyl)
Cat.No: T79972
Synonym:
Target: Antifungal
Ionomycin
Cat.No: T7285
Synonym:
Target: Calcium Channel
Oxytetracycline
Cat.No: T0895
Synonym: 土霉素,Terramycin
Target: ribosome, Endogenous Metabolite, Antibacterial, Antibiotic, HSV
Anisomycin
Cat.No: T6758
Synonym: 茴香霉素,Flagecidin,NSC 76712,Wuningmeisu C
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic, JNK
Nosiheptide
Cat.No: T16340
Synonym: RP 9671,Multhiomycin,那西肽
Target: Antibacterial, Antibiotic
Leucomycin
Cat.No: T3607
Synonym: 吉他霉素,Kitasamycin,Leucomycin V,Turimycin
Target: Antibacterial, Antibiotic
Spiramycin
Cat.No: T0819
Synonym: Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine
Target: Antibacterial, Antibiotic, Parasite
Ectoine
Cat.No: T4038
Synonym: THP(B),L-Ectoine,四氢甲基嘧啶羧酸
Target: Others, Antibacterial
Lincomycin hydrochloride monohydrate
Cat.No: T1235
Synonym: 洁霉素盐酸盐,林可霉素,Lincomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
Bekanamycin
Cat.No: T8118
Synonym: Kanamycin B,卡那霉素,卡那霉素 B
Target: Antibacterial, Antibiotic
Decoyinine
Cat.No: T15091
Synonym: Decynylene,Angustmycin A
Target:
3-(Methylthio)propionic acid
Cat.No: T5285
Synonym: 3-Methylthiopropionate,3-甲基硫代丙酸,4-Thiapentanoic acid,3-Methylsulfanylpropionic acid
Target: Others, Endogenous Metabolite, Antifungal
Tetracycline hydrochloride
Cat.No: T0912
Synonym: NCI-c55561,盐酸四环素,Tetracycline HCl
Target: ribosome, Antibacterial, Antibiotic
Vidarabine
Cat.No: T1506
Synonym: Adenine Arabinoside,阿糖腺苷,9-β-D-Arabinofuranosyladenine,Vira-A,Arabinosyladenine,Ara-A
Target: Nucleoside Antimetabolite/Analog, Tyrosine Kinases, DNA/RNA Synthesis, Antibiotic, HSV
Ascamycin
Cat.No: T14329
Synonym:
Target: Nucleoside Antimetabolite/Analog, Others, Antibacterial, Antibiotic
Calcimycin
Cat.No: T10662L
Synonym: Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187
Target: Apoptosis, Antibacterial, Antibiotic, Autophagy, Antifungal
Tacrolimus monohydrate
Cat.No: T20879
Synonym: FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506
Target: Phosphatase, Others, Antibacterial, Antibiotic, Autophagy
Tylosin tartrate
Cat.No: T0861
Synonym: 酒石酸泰洛星,酒石酸泰乐菌素
Target: Antibacterial, Antibiotic
Dianemycin
Cat.No: T8504
Synonym: Nanchangmycin (free acid)
Target: Antibacterial, Antibiotic
Tubercidin
Cat.No: T7004
Synonym: 结核菌素,杀结核菌素,Sparsomycin A,7-Deazaadenosine
Target: Influenza Virus, DNA/RNA Synthesis, Antibacterial, Antibiotic
Roseoflavin
Cat.No: T24729
Synonym:
Target: Antibacterial
A 201A
Cat.No: T26405
Synonym: Antibiotic 201A,A201A,A-201A
Target:
Demethoxyrapamycin
Cat.No: T25305
Synonym: AY 24668,AY24668,AY-24668
Target:
Lankacidins
Cat.No: T25622
Synonym: Bundlin A,Lankacidin C,Antibiotic T-2636 C,NSC 145118,Lankacidin
Target:
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