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Cat. No.	Product Name	Target	Signaling Pathways
T7061	Duloxetine	Serotonin Transporter	Neuroscience
	Duloxetine 是一种 5 羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂，Ki=4.6 nM，可作用于广泛性焦虑症的研究。
T1409	Methocarbamol Lumirelax,美索巴莫,Metocarbamol,AHR 85,Robaxin	Sodium Channel; Carbonic Anhydrase	Membrane transporter/Ion channel; Metabolism
	Methocarbamol (AHR 85) 是口服有效的中枢肌肉松弛剂，可阻断肌肉Nav1.4通道，阻断作用具有可逆性。Methocarbamol 具有用于肌肉痉挛和疼痛综合症研究的潜力。
T1471	Duloxetine hydrochloride Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl	Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine	GPCR/G Protein; Neuroscience
	Duloxetine hydrochloride ((S)-Duloxetine hydrochloride) 是一种 5-羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂 (SNRI)，Ki=4.6 nM，可用于广泛性焦虑症的研究。
T15358	Funapide TV 45070,XEN402	Sodium Channel	Membrane transporter/Ion channel
	Funapide (TV 45070) 是一个有效的钠通 Nav1.7 抑制剂，据有潜在的抗炎活性，可用来治疗红斑性肢痛症、肌肉骨骼疼痛、膝关节炎以及疱疹后神经。
T28453L	Propiram fumarate HCl Propiram fumarate HCl(15686-91-6 Free base)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Propiram fumarate HCl是一种可口服的Opioid receptors激动剂，具有镇痛活性，可用于研究肌肉骨骼疼痛。
T24755	Salnacedin G-201,SCY,G-201,G201,SCY,G 201	Others	Others
	Salnacedin (G-201) 是一种小分子化合物，可用于治疗免疫系统疾病、皮肤和肌肉骨骼疾病，可用于研究寻常痤疮、皮炎和银屑病。
T7725	Albaconazole W 0027,UR-9825,UR9825,W-0027	P450; Antifungal	Metabolism; Microbiology/Virology
	Albaconazole (W-0027)是一种小分子真菌细胞色素P450家族成员51 (fungal CYP51A1)抑制剂。它可用于治疗真菌感染、皮肤和肌肉骨骼疾病，可用于研究外阴阴道念珠菌病、Chagas病和泌尿生殖系统疾病。
T68108L	Moxilubant HCl Moxilubant hcl(146978-48-5 Free base)	LTR	Immunology/Inflammation
	Moxilubant HCl 是一种小分子白三烯 B4 受体 1（LTB4R）拮抗剂，可用于治疗免疫系统疾病、皮肤和肌肉骨骼疾病，可用于研究银屑病和类风湿关节炎。
T27209	Droxicam Droxicamum,屈昔康	Others	Others
	Droxicam (Droxicamum) 是一种非甾体抗炎化合物，可用于缓解肌肉骨骼疾病的炎症和疼痛的研究。
T72023	JB002	Myosin	Cytoskeletal Signaling
	JB002为一种肌球蛋白 II 抑制剂，IC50值不大于10 μM。适用于研究肌肉痉挛、慢性肌肉骨骼疼痛及肥厚型心肌病。
T34385	Ronacaleret HCl SB 751689,SB 751689A,SB-751689A,SB-751689,SB751689A,SB751689	CaSR	GPCR/G Protein
	Ronacaleret HCl (SB-751689) 是一种小分子 CaSR 拮抗剂，可用于治疗内分泌与代谢疾病、皮肤和肌肉骨骼疾病。
T33876L1	Panomifene TFA Panomifene TFA(77599-17-8 Free base),EGIS5650 TFA,GYKl13504 TFA	Estrogen/progestogen Receptor	Endocrinology/Hormones
	Panomifene TFA（GYKl13504 TFA）是一种小分子 ERs 拮抗剂，具有抗癌活性，可用于研究乳腺癌和肌肉骨骼疾病。
T68126	Pemedolac Dexpemedolac	COX	Immunology/Inflammation; Neuroscience
	Pemedolac (Dexpemedolac)是一种小分子 COX 抑制剂，可作为一种新型长效非麻醉性镇痛化合物，可用于治疗神经系统疾病、皮肤和肌肉骨骼疾病。
T1610	Metaxalone Skelaxin,Methaxalonum,美他沙酮,Zorane,NSC170959,AHR438	Others	Others
	Metaxalone (Methaxalonum) 具有肌肉松弛作用。
T0858	Flufenamic acid Arlef,Nichisedan,氟灭酸,氟芬那酸,Achless	Potassium Channel; Calcium Channel; Chloride channel; COX; AMPK; Parasite	Chromatin/Epigenetic; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling
	Flufenamic acid (Arlef) 是一种非甾体类抗炎剂，是一种邻氨基苯甲酸衍生物，具有镇痛、抗炎和解热的特性。它用于肌肉骨骼和关节疾病。
T29663	ADL-5747 ADL-5747 (free base),ADL5747,ADL-5747 free base	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	ADL-5747 (ADL-5747 (free base)) (free base)是一种δ opioid 受体激动剂，可用于治疗神经系统疾病、皮肤和肌肉骨骼疾病，可用于研究疱疹后神经痛、膝关节炎和疼痛。
T0855	(R)-Naproxen	COX	Immunology/Inflammation; Neuroscience
	(R)-Naproxen 是一种抗炎剂，具有解热和镇痛作用。酸及其钠盐都用于治疗急性痛风或痛经、肌肉骨骼疾病、类风湿性关节炎和其他风湿病。
T41303	Isoflupredone Delta-Fluorocortisone,Isoflupredona,异氟泼尼松,Isoflupredonum,9-Fluoroprednisolone	Others	Others
	Isoflupredone (Isoflupredonum) 是一种合成的皮质类固醇，通过与动物 (如马) 的糖皮质激素和矿皮质激素受体结合抑制炎症细胞和抑制炎症介质的表达在生物体内发挥作用。Isoflupredone 具有抗炎和免疫抑制作用，可应用于治疗各种肌肉骨骼、过敏性和全身炎症性疾病。
T67952	JB062	Myosin	Cytoskeletal Signaling
	JB062是一种针对非肌肉肌球蛋白(nonmusclemyosin)的抑制剂，其IC50值对骨骼肌肌球蛋白为1.6μM、心肌肌球蛋白为5.4μM，而对平滑肌肌球蛋白II大于100μM。此化合物对人类癌细胞显示出细胞毒性，对正常细胞则无此作用。JB062在肌肉痉挛、慢性肌肉骨骼疼痛及肥厚型心肌病研究中有潜在应用价值。
T67385	Neratinib maleate HKI-272 maleate	EGFR; HER	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	Neratinib maleate (HKI-272 maleate) 是一种不可逆且具有口服活性和高选择性的 HER2 和 EGFR 抑制剂，IC50 值分别为 59 nM 和 92 nM。Neratinib maleate具有抗肿瘤活性，可用于治疗消化系统疾病、呼吸系统疾病、泌尿生殖系统疾病和皮肤和肌肉骨骼疾病，可用于研究乳腺癌和前列腺癌。
T0183L	Pramiracetam Sulfate CNS-1879,CI879,CI-879,CI 879,Pramiracetam
	Thurfyl salicylate is a reddening agent for the treatment of musculoskeletal, joint, periarticular, and soft tissue pain.
T27573	Ibuproxam Ibuproxamum,G-277
	Ibuproxam, a nonsteroidal antiinflammatory drug (NSAID), is used for the treatment of musculoskeletal pain, arthritis, and soft-tissue disorders.
T27633	Isonixin Nixyn,Isonixine
	Isonixin is used for the treatment of inflammation and pain associated with musculoskeletal and joint disorders.
T34863	Thurfyl Salicylate Tetrahydrofurfuryl salicylate
	Thurfyl Salicylate (tetrahydrofurfuryl Salicylate) is a redness preparation used for the treatment of musculoskeletal, joint, periarticular, and soft tissue pain.
T28685	SB236057 SB-236057,SB 236057
	SB236057 is a potent and selective inverse agonist for the 5-HT receptor, acting especially at 5-HT autoreceptors on nerve terminals. It produces a rapid increase in 5-HT levels in the brain. SB236057 also acts as a potent teratogen, producing severe musc
T68563	Piroxicam olamine
	Piroxicam olamine is a cyclooxygenase inhibiting, non-steroidal anti-inflammatory agent (NSAID) that is well established in treating rheumatoid arthritis and osteoarthritis and used for musculoskeletal disorders, dysmenorrhea, and postoperative pain. Its long half-life enables it to be administered once daily.
T68211	Piroxicam betadex
	Piroxicam betadex is a nonsteroidal anti-inflammatory drug. The mechanism of action of piroxicam is as a cyclooxygenase Inhibitor. It is well established in treating rheumatoid arthritis and osteoarthritis and used for musculoskeletal disorders, dysmenorrhea, and postoperative pain. It is used to reduce pain, swelling, and joint stiffness from arthritis. Reducing these symptoms helps you do more of your normal daily activities.
T68108	Moxilubant	LTR	Immunology/Inflammation
	Moxilubant 是一种小分子白三烯B4受体1（LTB4R）拮抗剂，可用于治疗免疫系统疾病、皮肤和肌肉骨骼疾病，可用于研究银屑病和类风湿关节炎。
TP1853	TP508
	TP508 is a 23 amino acid synthetic peptide representing residues 508-530 of human prothrombin which is identified as a potential receptor-binding domain based on competition for high-affinity thrombin binding to fibroblasts.TP508 (Chrysalin) is an investi

化合物

Cat.No: T7061

Target: Serotonin Transporter

Cat.No: T1409

Synonym: Lumirelax,美索巴莫,Metocarbamol,AHR 85,Robaxin

Target: Sodium Channel, Carbonic Anhydrase

Duloxetine hydrochloride

Cat.No: T1471

Synonym: Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl

Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine

Cat.No: T15358

Synonym: TV 45070,XEN402

Target: Sodium Channel

Propiram fumarate HCl

Cat.No: T28453L

Synonym: Propiram fumarate HCl(15686-91-6 Free base)

Target: Opioid Receptor

Cat.No: T24755

Synonym: G-201,SCY,G-201,G201,SCY,G 201

Target: Others

Cat.No: T7725

Synonym: W 0027,UR-9825,UR9825,W-0027

Target: P450, Antifungal

Cat.No: T68108L

Synonym: Moxilubant hcl(146978-48-5 Free base)

Target: LTR

Cat.No: T27209

Synonym: Droxicamum,屈昔康

Target: Others

Cat.No: T72023

Target: Myosin

Ronacaleret HCl

Cat.No: T34385

Synonym: SB 751689,SB 751689A,SB-751689A,SB-751689,SB751689A,SB751689

Target: CaSR

Cat.No: T33876L1

Synonym: Panomifene TFA(77599-17-8 Free base),EGIS5650 TFA,GYKl13504 TFA

Target: Estrogen/progestogen Receptor

Cat.No: T68126

Synonym: Dexpemedolac

Target: COX

Cat.No: T1610

Synonym: Skelaxin,Methaxalonum,美他沙酮,Zorane,NSC170959,AHR438

Target: Others

Flufenamic acid

Cat.No: T0858

Synonym: Arlef,Nichisedan,氟灭酸,氟芬那酸,Achless

Target: Potassium Channel, Calcium Channel, Chloride channel, COX, AMPK, Parasite

Cat.No: T29663

Synonym: ADL-5747 (free base),ADL5747,ADL-5747 free base

Target: Opioid Receptor

Cat.No: T0855

Target: COX

Cat.No: T41303

Synonym: Delta-Fluorocortisone,Isoflupredona,异氟泼尼松,Isoflupredonum,9-Fluoroprednisolone

Target: Others

Cat.No: T67952

Target: Myosin

Neratinib maleate

Cat.No: T67385

Synonym: HKI-272 maleate

Target: EGFR, HER

Pramiracetam Sulfate

Cat.No: T0183L

Synonym: CNS-1879,CI879,CI-879,CI 879,Pramiracetam

Cat.No: T27573

Synonym: Ibuproxamum,G-277

Cat.No: T27633

Synonym: Nixyn,Isonixine

Thurfyl Salicylate

Cat.No: T34863

Synonym: Tetrahydrofurfuryl salicylate

Cat.No: T28685

Synonym: SB-236057,SB 236057

Piroxicam olamine

Cat.No: T68563

Piroxicam betadex

Cat.No: T68211

Cat.No: T68108

Target: LTR

Cat.No: TP1853

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