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59

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TP1122L IGF-I 30-41 acetate(82177-09-1 free base)

Insulin-like Growth Factor I (30-41) acetate

Others Others
IGF-I 30-41 acetate(82177-09-1 free base) (Insulin-like Growth Factor I (30-41) acetate) 是胰岛素样生长因子 I (IGF-I) 的氨基酸 30 至 41 片段。
T6419 BMS-536924

HY-10262,胰岛素样生长因子-1 受体拮抗剂,BMS 536924,CS-0117

Apoptosis; FAK; MEK; IGF-1R; Src Angiogenesis; Apoptosis; Cytoskeletal Signaling; MAPK; Tyrosine Kinase/Adaptors
BMS-536924 (BMS 536924) 是一种具有口服活性,竞争性和选择性的胰岛素样生长因子受体激酶和胰岛素受体抑制剂,IC50分别为 100 nM 和 73 nM。它具有抗癌活性。
T76539 Insulin-like growth factor II

Insulin-like growth factor II (IGF-2)为人血清中主要生长激素,对神经突生长具有许可性和直接作用,同时增强交感与感觉神经元的生存能力。
TP1122 IGF-I (30-41)

Insulin-like Growth Factor I (30-41),IGF-I 30-41

IGF-I (30-41) is amino acids 30 to 41 fragment of Insulin-like Growth Factor I (IGF-I).
TP1124 IGF-I (24-41)

Insulin-like Growth Factor I (24-41),IGF-I 24-41

IGF-I (24-41) is a 24-41 amino acid fragment of Insulin-like Growth Factor I (IGF-I). IGF-I is partly responsible for systemic GH activities although it possesses a wide number of own properties (anabolic, antioxidant, anti-inflammatory and cytoprotective
T6203 Saxagliptin

BMS-477118,沙克列汀,Onglyza,沙格列汀

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Saxagliptin (BMS-477118) 是一种选择性,可逆性,竞争性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin 能够用于 2 型糖尿病的研究。
TP1121 IGF-I (30-41) TFA(82177-09-1,FREE)

Insulin-like Growth Factor I (30-41) (TFA)

IGF-I (30-41) (TFA) is amino acids 30 to 41 fragment of Insulin-like Growth Factor I (IGF-I).
TP1123 IGF-I (24-41) TFA (135861-49-3 free base)

Insulin-like Growth Factor I (24-41) (TFA),IGF-I (24-41) TFA

IGF-I is partly responsible for systemic GH activities although it possesses a wide number of own properties (anabolic, antioxidant, anti-inflammatory and cytoprotective actions).IGF-I (24-41) (TFA) is amino acids 24 to 41 fragment of Insulin-like Growth
T0178 Saxagliptin hydrate

沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Saxagliptin hydrate (Onglyza hydrate) 是一种选择性,竞争性,可逆性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin hydrate 能够用于 2 型糖尿病的研究。
T2349 BMS-754807

Trk receptor; c-Met/HGFR; IGF-1R Tyrosine Kinase/Adaptors
BMS754807 是一种可逆的IGF-1R 抑制剂 (IC50:1.8 nM,Ki<2 nM),也是一种可逆的IR 抑制剂 (IC50:7 nM,Ki<2 nM)。它也抑制 Met (IC50:6 nM),RON (IC50:44 nM),TrkA (IC50:7 nM),TrkB (IC50:4 nM),AurA (IC50:9 nM) 和 AurB (IC50:25 nM) 的活性。
T8906 NBI-31772

NBI31772,NBI 31772

IGF-1R Tyrosine Kinase/Adaptors
NBI-31772 (NBI 31772) 是胰岛素样生长因子-1 结合蛋白 (IGFBP, Ki = 47 nM) 的有效抑制剂。 NBI-31772 可用于 IGF 反应性疾病的研究。
T2189 Sodium orthovanadate

Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate

ATPase; Phosphatase Membrane transporter/Ion channel; Metabolism
Sodium orthovanadate 是一种蛋白酪氨酸磷酸酶,碱性磷酸酶和一些ATP 酶的抑制剂,有可能充当磷酸盐类似物。它具有胰岛素样作用、对心室肌的正性肌力作用和其他代谢作用。
T78097L Mazdutide acetate(2259884-03-0 free base)

Mazdutide acetate(2259884-03-0 free base),OXM-3 acetate,LY-3305677 acetate,IBI-362 acetate

Glucagon Receptor GPCR/G Protein
Mazdutide acetate 是一种高效的胰高血糖素样肽 (GLP-1R) 与胰高血糖素受体 (GCGR) 的共激动剂,是一种胃泌酸调节素类似物。Mazdutide acetate可刺激小鼠胰岛的胰岛素分泌 ,可用于研究肥胖和 2 型糖尿病 (T2D) 。
T68405 KW-2450 free base

IGF-1R Tyrosine Kinase/Adaptors
KW-2450 free base 是一种 IGF-1R/IR和酪氨酸激酶多重抑制剂 具有抗肿瘤活性。KW-2450 free base 在小鼠 HT-29/GFP 结肠癌异种移植模型中显示出适度的生长抑制活性并抑制 IGF-1 诱导的信号转导。
T76810 Ganitumab

AMG 479

IGF-1R Tyrosine Kinase/Adaptors
Ganitumab (AMG 479) 是一种高效的1型胰岛素样生长因子受体 (IGF1R) 单克隆抗体。Ganitumab 在低浓度下识别与 IGF1R 结合,KD 值为0.22 nM,Ganitumab 对小鼠 IGF1R 与 IGF1 和 IGF2 的相互作用有抑制作用。Ganitumab 可用于研究癌症。
T6017 Linsitinib

OSI-906,林西替尼

IGF-1R Tyrosine Kinase/Adaptors
Linsitinib (OSI-906) 是选择性的、有效的、具有口服活性的IGF-1和胰岛素受体(IR)的双重抑制剂,IC50分别为 35 和 75 nM。
T2160 Suramin Sodium Salt

苏拉明钠,BAY-205,Suramin hexasodium salt,苏拉明钠盐,NF-060

Apoptosis; Phosphatase; SARS-CoV; Sirtuin; Reverse Transcriptase; Topoisomerase; Parasite Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Suramin Sodium Salt (BAY-205) 是可逆的竞争性蛋白酪氨酸磷酸酶抑制剂。它抑制 IP5K,是抗寄生虫,抗肿瘤和抗血管生成剂。它是sirtuins 的有效抑制剂,也是 SARS-CoV-2 RNA 依赖性 RNA 聚合酶抑制剂。
T25123 AZ12253801

AZ 12253801,AZ-12253801

AZ12253801 is a type 1 insulin-like growth factor receptor (IGF-1R) inhibitor.
T70568 H-1356

H-1356 is an insulin-like growth factor 1(IGF-I) analog that inhibits autophosphorylation of IGF-I receptor.
T24106 GSK2163632A

GSK-2163632-A,GSK 2163632 A

GSK2163632A is an insulin-like growth factor 1 receptor inhibitor that acts by binding to a novel region of the GRK active site cleft.
TP2209 Xenin-8

Others Others
neurotensin-like peptide that modulate pancreatic insulin and glucagon secretion/effects
TP1361 S961 TFA (1083433-49-1 free base)

S961 TFA

S961 TFA is A high affinity insulin receptor (IR) antagonist with IC50 for hir-a, hir-b and human insulin-like growth factor I receptor (higf-ir) at 0.048, 0.027 and 630 nM, respectively.
T25110 AS1069562

AS-1069562,AS 1069562

AS1069562 is an inhibitor of serotonin (5-HT) and norepinephrine (NE) reuptake which acts by notably restoring reduced insulin-like growth factor 1 and fibroblast growth factor 2 mRNA levels in dorsal root ganglion and spinal cord, respectively.
T16101 ML-290

RXFP receptor GPCR/G Protein
ML-290 是一个松弛素/胰岛素样肽受体 (RXFP1) 偏向变构激动剂,为抗纤维化基因激活剂,EC50为 94 nM。
T80871 Veligrotug

IGF-1R Tyrosine Kinase/Adaptors
Veligrotug为IgG1-kappa型抗IGF1R(胰岛素样生长因子1受体,CD221)嵌合单克隆抗体。
T76043L S961 acetate

S961 acetate 是一种高亲和力的胰岛素受体 (insulin receptor, IR) 拮抗剂,对 HIR-A,HIR-B 和人胰岛素样生长因子 I 受体 (HIGF-IR) 的 IC50分别为 0.048,0.027 和 630 nM。
T24620 PF-06372222

PF-0637222,PF0637222,PF 0637222

PF-06372222 is a small-molecule negative allosteric modulator of the glucagon receptor (GCGR). PF-06372222 is also an antagonist for glucagon-like peptide-1 receptor GLP-1R, which inhibits glucagon secretion and glucose-dependent insulin secretion.
T30538 BMS-695735

CHEMBL459729,DNC008930,BMS 695735,BMS695735,BDBM27888

BMS-695735, a benzimidazole inhibitor of insulin-like growth factor-1 receptor, has broad-spectrum antitumor activity in vivo. It was found that BMS-695735 had strong inhibition of CYP3A4, induction of CYP3A4 mediated by PXR transactivation, poor water so
TP1795 S961

S961是一种高亲和力和选择性胰岛素受体(IR)拮抗剂,接近闪烁计数法试验中对HIR-A、HIR-B 和人胰岛素样生长因子I 受体(HIGF-IR)的ic50分别为0.048、0.027和630 nM。
T76043 S961 TFA

S961 TFA为一种与胰岛素受体(insulin receptor, IR)高亲和力相结合的拮抗剂,其IC50值对HIR-A、HIR-B及人胰岛素样生长因子I受体(HIGF-IR)分别为0.048、0.027及630 nM。
T38584 ALK-IN-12

ALK-IN-12 is a highly potent and orally active inhibitor of anaplastic lymphoma kinase (ALK), demonstrating an exceptional IC50 value of 0.18 nM. Additionally, ALK-IN-12 displays inhibitory activity against insulin-like growth factor 1 receptor (IGF1R) and insulin receptor (InsR), with IC50 values of 20.3 nM and 90.6 nM, respectively. Notably, its antitumor effects have been observed, making it a promising compound for targeted cancer therapy.
T80605 Dusigitumab

MEDI 573

IGF-1R Tyrosine Kinase/Adaptors
Dusigitumab (MEDI 573)为一种人源化IgG2λ单克隆抗体,具有特异性针对IGF2和IGF1。
T38502 IGF-1R inhibitor-2

IGF-1R inhibitor-2 (example 121) is a compound that inhibits the insulin-like growth factor-1 receptor (IGF-1R). By downregulating the IGF-1R, it has the potential to reverse the transformed phenotype of tumor cells and make them more susceptible to apoptosis.
T61506 NBI-31772 hydrate

NBI-31772 hydrate is a powerful inhibitor of the interaction between insulin-like growth factor (IGF) and IGF-binding proteins (IGFBPs). It acts as a nonpeptide ligand, effectively releasing bioactive IGF-I from the IGF-I/IGFBP-3 complex (Ki values for all six human subtypes range from 1-24 nM). This compound demonstrates significant anxiolytic and antidepressant-like effects [1] [2] [3].
TP1241 Adrenocorticotropic Hormone (ACTH) (18-39), human

ACTH (18-39), human

Adrenocorticotropic Hormone (ACTH) (18-39) is known as the Corticotropin-like Intermediate Lobe Peptide. It stimulates insulin secretion as well as amylase and protein secretion in a dose-dependent manner similar to those of secretin and carbamylcholine.
T76330 Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide

Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide 是一种带有生物素标签的Glucagon-like peptide-1-(7-36),后者为一种具备提升胰岛素释放功能,从而表现出抗糖尿病活性的胃肠道肽。
T70876 KW-2450 Tosylate

KW-2450 Tosylate is an orally bioavailable inhibitor of insulin-like growth factor 1 receptor (IGF-1R) and insulin receptor (IR) tyrosine kinases with potential antineoplastic activity. IGF-1R/IR inhibitor KW-2450 Tosylate selectively binds to and inhibits the activities of IGF-1R and IR, which may result in the inhibition of tumor cell proliferation and the induction of tumor cell apoptosis. IGF-R1 and IR tyrosine kinases, overexpressed in a variety of human cancers, play significant roles in t...
T76759 Robatumumab

Robatumumab (Sch 717454) 为针对人胰岛素样生长因子 1 受体(anti-humanIGF-1R)的抗体,展现出抗肿瘤及阻止癌细胞增殖的作用,适用于骨肉瘤与尤文肉瘤的研究。
T63019 GKA50 quarterhydrate

GKA50 quarterhydrate 是一种有效的葡萄糖激酶激活剂,其 EC50 值为 33 nM。GKA50 quarterhydrate 是一种啮齿动物和人类胰岛中 β 细胞代谢的葡萄糖样激活剂,也是一种 Ca2+依赖性胰岛素分泌调节剂。GKA50 quarterhydrate 能够刺激小鼠胰岛分泌胰岛素,可以显著降低高脂喂养的雌性大鼠血糖。
T76746 Figitumumab

Figitumumab (CP-751871) 为一种高效对抗胰岛素样生长因子 1 受体 (IGF1R) 的全人单克隆抗体。通过阻断 IGF1 与 IGF1R 的结合,其 IC50 值达到 1.8 nM。
T75157L Cimdelirsen sodium

Cimdelirsen (sodium) 为针对肝脏的反义寡核苷酸,通过减少生长激素受体(GHr)合成,抑制生长激素(GH)的过度分泌效应,进而降低肢端肥大症患者体内循环胰岛素样生长因子-1 (IGF-1)水平。
T64252 Efpeglenatide

Efpeglenatide 是一种胰高血糖素样肽 (GLP-1) 受体的长效激动剂。Efpeglenatide 能够改善糖尿病和肥胖小鼠模型的胰岛素敏感性,并减缓其体重减轻的作用。Efpeglenatide 已经被用于 II 型糖尿病的研究。
T73702 Mecasermin

Mecasermin(Human IGF-I; FK 780),一种重组人胰岛素样生长因子I(IGF-I),主要用于研究因生长激素(GH)受体缺陷或GH抑制抗体导致的GH不敏感性而引起的生长障碍。
T64553 GLP-1(7-37) TFA salt

The truncated glucagon-like peptides GLP-1(7-37) is naturally occurring peptide product of the preproglucagon gene that are synthesized primarily in the intestine and acts as incretin that are released from the intestine into the bloodstream in response to food and stimulate insulin secretion. GLP-1(7-37) produced a dose-related enhancement of the glucose-stimulated increase in plasma insulin concentration and an increased rate of glucose infusion in Sprague-Dawley Rats at a dosing rang of 0.5, ...
T76291 Des His1, Glu8 Exendin-4

Des His1, Glu8 Exendin-4 是一种高效的GLP-1-R(胰高血糖素样肽-1 受体)拮抗剂,主要通过调控胰岛素分泌和抑制葡萄糖生成来维持葡萄糖稳态。该化合物广泛应用于2型糖尿病及胃肠道相关研究领域。
TP1148 Glucagon-like peptide 1 (1-37), human

HuGLP-1

Glucagon-like peptide 1 (1-37), human is a highly potent agonist of the GLP-1 receptor.Pancreatic hormone synthesized by post-translational processing of proglucagon. Unlike truncated forms of GLP-1, it has no effect on food intake in rats and does not en
T21691 NVP DPP 728 dihydrochloride

NVP-DPP728 是一种有效、可逆、腈依赖性二肽基肽酶 IV (DPP-IV)抑制剂,Ki 值为 11 nM。NVP-DPP728 可抑制胰高血糖素样肽-1 (GLP-1)的降解,从而增强响应于葡萄糖摄入的胰岛素释放。NVP-DPP728 可用于糖尿病研究。
T75157 Cimdelirsen

Cimdelirsen为针对肝脏的反义寡核苷酸,通过降低生长激素受体(GHr)的合成量,来减少生长激素(GH)过量分泌所导致的不良影响,进而在肢端肥大症患者中降低循环胰岛素样生长因子-1(IGF-1)的水平。
T76012 IGF-I (30-41) (TFA)

IGF-I (30-41) (TFA) 是类胰岛素生长因子I 30 至 41 的氨基酸片段。IGF-I 对生长激素的活性有着重要的作用,但是IGF-I 本身也具有一些自身的特性,如合成代谢、抗氧化、抗炎和细胞保护作用。
T76333 (Ser8)-GLP-1 (7-36) amide, human

(Ser8)-GLP-1 (7-36) amide, human 为源自胰高血糖素原的胰高血糖素样肽-1酰胺,属于 GLP-1(1-36) 酰胺肽裂解产物。作为肠促胰岛素激素,该化合物促进胰腺 β 细胞在葡萄糖依赖性条件下分泌胰岛素,并对消化道的运动与分泌功能产生影响。

化合物

IGF-I 30-41 acetate(82177-09-1 free base)
Cat.No: TP1122L
Synonym: Insulin-like Growth Factor I (30-41) acetate
Target: Others
BMS-536924
Cat.No: T6419
Synonym: HY-10262,胰岛素样生长因子-1 受体拮抗剂,BMS 536924,CS-0117
Target: Apoptosis, FAK, MEK, IGF-1R, Src
Insulin-like growth factor II
Cat.No: T76539
Synonym:
Target:
IGF-I (30-41)
Cat.No: TP1122
Synonym: Insulin-like Growth Factor I (30-41),IGF-I 30-41
Target:
IGF-I (24-41)
Cat.No: TP1124
Synonym: Insulin-like Growth Factor I (24-41),IGF-I 24-41
Target:
Saxagliptin
Cat.No: T6203
Synonym: BMS-477118,沙克列汀,Onglyza,沙格列汀
Target: Proteasome, DPP-4
IGF-I (30-41) TFA(82177-09-1,FREE)
Cat.No: TP1121
Synonym: Insulin-like Growth Factor I (30-41) (TFA)
Target:
IGF-I (24-41) TFA (135861-49-3 free base)
Cat.No: TP1123
Synonym: Insulin-like Growth Factor I (24-41) (TFA),IGF-I (24-41) TFA
Target:
Saxagliptin hydrate
Cat.No: T0178
Synonym: 沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate
Target: Proteasome, DPP-4
BMS-754807
Cat.No: T2349
Synonym:
Target: Trk receptor, c-Met/HGFR, IGF-1R
NBI-31772
Cat.No: T8906
Synonym: NBI31772,NBI 31772
Target: IGF-1R
Sodium orthovanadate
Cat.No: T2189
Synonym: Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate
Target: ATPase, Phosphatase
Mazdutide acetate(2259884-03-0 free base)
Cat.No: T78097L
Synonym: Mazdutide acetate(2259884-03-0 free base),OXM-3 acetate,LY-3305677 acetate,IBI-362 acetate
Target: Glucagon Receptor
KW-2450 free base
Cat.No: T68405
Synonym:
Target: IGF-1R
Ganitumab
Cat.No: T76810
Synonym: AMG 479
Target: IGF-1R
Linsitinib
Cat.No: T6017
Synonym: OSI-906,林西替尼
Target: IGF-1R
Suramin Sodium Salt
Cat.No: T2160
Synonym: 苏拉明钠,BAY-205,Suramin hexasodium salt,苏拉明钠盐,NF-060
Target: Apoptosis, Phosphatase, SARS-CoV, Sirtuin, Reverse Transcriptase, Topoisomerase, Parasite
AZ12253801
Cat.No: T25123
Synonym: AZ 12253801,AZ-12253801
Target:
H-1356
Cat.No: T70568
Synonym:
Target:
GSK2163632A
Cat.No: T24106
Synonym: GSK-2163632-A,GSK 2163632 A
Target:
Xenin-8
Cat.No: TP2209
Synonym:
Target: Others
S961 TFA (1083433-49-1 free base)
Cat.No: TP1361
Synonym: S961 TFA
Target:
AS1069562
Cat.No: T25110
Synonym: AS-1069562,AS 1069562
Target:
ML-290
Cat.No: T16101
Synonym:
Target: RXFP receptor
Veligrotug
Cat.No: T80871
Synonym:
Target: IGF-1R
S961 acetate
Cat.No: T76043L
Synonym:
Target:
PF-06372222
Cat.No: T24620
Synonym: PF-0637222,PF0637222,PF 0637222
Target:
BMS-695735
Cat.No: T30538
Synonym: CHEMBL459729,DNC008930,BMS 695735,BMS695735,BDBM27888
Target:
S961
Cat.No: TP1795
Synonym:
Target:
S961 TFA
Cat.No: T76043
Synonym:
Target:
ALK-IN-12
Cat.No: T38584
Synonym:
Target:
Dusigitumab
Cat.No: T80605
Synonym: MEDI 573
Target: IGF-1R
IGF-1R inhibitor-2
Cat.No: T38502
Synonym:
Target:
NBI-31772 hydrate
Cat.No: T61506
Synonym:
Target:
Adrenocorticotropic Hormone (ACTH) (18-39), human
Cat.No: TP1241
Synonym: ACTH (18-39), human
Target:
Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide
Cat.No: T76330
Synonym:
Target:
KW-2450 Tosylate
Cat.No: T70876
Synonym:
Target:
Robatumumab
Cat.No: T76759
Synonym:
Target:
GKA50 quarterhydrate
Cat.No: T63019
Synonym:
Target:
Figitumumab
Cat.No: T76746
Synonym:
Target:
Cimdelirsen sodium
Cat.No: T75157L
Synonym:
Target:
Efpeglenatide
Cat.No: T64252
Synonym:
Target:
Mecasermin
Cat.No: T73702
Synonym:
Target:
GLP-1(7-37) TFA salt
Cat.No: T64553
Synonym:
Target:
Des His1, Glu8 Exendin-4
Cat.No: T76291
Synonym:
Target:
Glucagon-like peptide 1 (1-37), human
Cat.No: TP1148
Synonym: HuGLP-1
Target:
NVP DPP 728 dihydrochloride
Cat.No: T21691
Synonym:
Target:
Cimdelirsen
Cat.No: T75157
Synonym:
Target:
IGF-I (30-41) (TFA)
Cat.No: T76012
Synonym:
Target:
(Ser8)-GLP-1 (7-36) amide, human
Cat.No: T76333
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3823 D-Pinitol

Pinitol,Inzitol,D-(+)-Pinitol,D-松醇,Methylinositol,3-O-Methyl-D-chiro-inositol

Others; Influenza Virus Microbiology/Virology; Others
D-Pinitol (Methylinositol) 是一种存在于几种植物中,如松科和豆科植物的天然产物,具有抗病毒、杀幼虫、降血糖活性和心血管系统保护作用。
T5915 D-chiro-Inositol

D-手性肌醇,D-(+)-CHIRO-INOSITOL

Endogenous Metabolite Metabolism
D-chiro-Inositol (D-(+)-CHIRO-INOSITOL) 是肌醇差向异构体,存在于某些哺乳动物糖基磷脂酰肌醇蛋白锚和具有胰岛素样生物特性的肌醇磷脂聚糖中。它能够抑制高血糖,改善胰岛素抵抗。它用于多囊卵巢综合征和糖尿病的相关研究。
TN2080 Pinoresinol

松脂酚,松脂素,(+)-Pinoresinol

Apoptosis; NF-κB; CDK; p53 Apoptosis; Cell Cycle/Checkpoint; NF-κB
Pinoresinol ((+)-Pinoresinol) 是一种植物来源的木质素,具有抗炎、保肝和杀真菌活性。它导致 CDK 抑制剂 p21(WAF1/Cip1) 在 mRNA 和蛋白质水平上调,抑制 NF-kappaB 和激活蛋白 1 。
T3S0027 Picropodophyllotoxin

AXL 1717,Picropodophyllin,苦鬼臼毒素

IGF-1R Tyrosine Kinase/Adaptors
Picropodophyllotoxin (AXL 1717) 是一种环木脂素生物碱,存在于五月树(Podophyllum peltatum) 中,是一种具有潜在抗肿瘤活性的胰岛素样生长因子 1 受体 (IGF1R) 的小分子抑制剂。它特异性抑制 IGF1R 的活性并下调细胞表达,而不干扰其他生长因子受体的活性,例如胰岛素受体、表皮生长因子、血小板衍生生长因子、成纤维细胞生长因子和肥大/干细胞生长因子 (KIT) )。该药剂在抑制肿瘤细胞增殖和诱导肿瘤细胞凋亡方面显示出有效的活性。 IGF1R 是一种在多种人类癌症中过度表达的受体酪氨酸激酶,在多种癌细胞的生长和存活中起关键作用。

天然产物

D-Pinitol
Cat.No: T3823
Synonym: Pinitol,Inzitol,D-(+)-Pinitol,D-松醇,Methylinositol,3-O-Methyl-D-chiro-inositol
Target: Others, Influenza Virus
D-chiro-Inositol
Cat.No: T5915
Synonym: D-手性肌醇,D-(+)-CHIRO-INOSITOL
Target: Endogenous Metabolite
Pinoresinol
Cat.No: TN2080
Synonym: 松脂酚,松脂素,(+)-Pinoresinol
Target: Apoptosis, NF-κB, CDK, p53
Picropodophyllotoxin
Cat.No: T3S0027
Synonym: AXL 1717,Picropodophyllin,苦鬼臼毒素
Target: IGF-1R
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