101
18
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7872 |
Monolaurin
|
Others | Others |
Monolaurin 是椰子油中的一种表面活性剂和乳化剂。它抑制葡萄球菌、链球菌、加德纳菌、念珠菌和嗜血杆菌的生长,并减少促炎细胞因子的产生。 | |||
T3583 |
Macozinone
PBTZ169 |
Antibacterial; DprE1 | Microbiology/Virology; Others |
Macozinone (PBTZ169) 是具有杀菌作用的苯并噻嗪酮,也有抗结核作用。它也是一种 DprE1有效抑制剂,可通过与活性位点 Cys387 残基形成共价键来抑制必需的黄素蛋白 DprE1。 | |||
T1312 |
Nafcillin sodium monohydrate
CL 8491,萘夫西林钠,nafcillin sodium |
Antibacterial; Antibiotic | Microbiology/Virology |
Nafcillin sodium monohydrate (CL 8491) 是一种抗生素,是可逆的β-lactamase 抑制剂。它用于治疗由耐青霉素的葡萄球菌菌株引起的感染。 | |||
T16073 |
Micronomicin
小诺霉素,Gentamicin C2b,Antibiotic XK-62-2,Sagamicin |
Others; Antibacterial | Microbiology/Virology; Others |
Micronomicin (Gentamicin C2b) 是一种具有抗菌和杀菌能力的抗生素。 | |||
T40417 |
Ethylhydrocupreine hydrochloride
Optochin hydrochloride,乙氢去甲奎宁盐酸盐;奥普托欣盐酸盐 |
Antibacterial; Parasite | Microbiology/Virology |
Ethylhydrocupreine hydrochloride (Optochin hydrochloride) 是奎宁的一种衍生物,具有抗菌作用,可抑制肺炎链球菌的活性。Ethylhydrocupreine hydrochloride 具有抗疟活性,对 Plasmodium falciparum 的IC50为 25.75 nM。Ethylhydrocupreine hydrochloride 是Gallus gallus2 受体 (ggTas2r1,ggTas2r2和ggTas2r7) 激动剂。 | |||
T1495 |
Cefaclor monohydrate
Cefaclor,头孢克洛一水物,头孢克洛一水合物,Cefaclorum,Cefachlor |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefaclor monohydrate (Cefaclorum) 是一种抗生素,可特异性地结合青霉素结合蛋白。 | |||
T7735 |
5-Nitro-1,10-phenanthroline
5-NP,5-硝基-1,10-菲咯啉 |
Antibacterial | Microbiology/Virology |
5-Nitro-1,10-phenanthroline (5-NP) 是一种有效的杀菌剂,可抑制艰难梭菌。 | |||
T3247 |
Lysozyme from chicken egg white
鸡蛋清溶菌酶,溶菌酶,Lysozyme |
Others; Antibacterial | Microbiology/Virology; Others |
Lysozyme from chicken egg white (Lysozyme) 是一种存在于鸡蛋清中的杀菌酶,它溶解革兰氏阳性菌。 | |||
T1143 |
Carbenicillin disodium
BRL-2064,羧苄青霉素钠,Sodium carbenicillin |
Cell wall; Antibacterial; Antibiotic | Immunology/Inflammation; Microbiology/Virology |
Carbenicillin disodium (BRL-2064) 作用于细菌细胞壁合成的最后阶段,是β-内酰胺青霉素衍生物。 | |||
T0328 |
Hexetidine
NSC-17764,海克替啶 |
Antibacterial; Antifungal | Microbiology/Virology |
Hexetidine (NSC-17764) 是一种口服活性的抗菌抗真菌试剂,可用于口腔感染的相关研究。 | |||
T64346 |
DDAC
Quaternium 12 |
Antibacterial | Microbiology/Virology |
DDAC (Quaternium 12), also known as Didecyldimethylammonium chloride, is a dialkyl-quaternary ammonium compound widely utilized in various products due to its bactericidal, virucidal, and fungicidal characteristics. | |||
T3263 |
(6R,7S)-Cefminox sodium heptahydrate
Meicelin,头孢米诺钠,Cefminox Sodium,Alteporina,Tencef |
Antibiotic | Microbiology/Virology |
(6R,7S)-Cefminox sodium heptahydrate (Meicelin) 是一种 Cefminox sodium heptahydrate 的异构体。它也是一种具有广谱抗菌活性的 β-内酰胺头孢菌素抗生素。 | |||
T2211 |
Dihydrostreptomycin sulfate
Dihydrostreptomycin sesquisulfate,双氢链霉索 |
Antibacterial; Antibiotic | Microbiology/Virology |
Dihydrostreptomycin sulfate (Dihydrostreptomycin sesquisulfate) 是一种氨基糖苷类抗生素,可研究牛、猪和羊的细菌性疾病。 | |||
T5022 |
Ceforanide
|
Antibacterial; Antibiotic | Microbiology/Virology |
Ceforanide 是一种头孢菌素,可静脉或肌肉给药。它在体外具有一系列抗菌活性。 | |||
T72030 |
6,6'-Dimethyl-2,2'-dipyridyl
6,6'-Bi-2-picoline |
||
6,6'-Dimethyl-2,2'-dipyridyl (6,6'-Bi-2-picoline) 是一种新型的时间分辨荧光免疫分析(TRFIA)螯合物,具有较好的杀菌效果,可用于研究酒渣鼻。 | |||
T3582 |
BTZ043
|
Antibacterial; Antibiotic; DprE1 | Microbiology/Virology; Others |
BTZ043 是一种 DprE1 的抑制剂,它对结核分枝杆菌 H37Rv 和耻垢分枝杆菌具有纳摩尔杀菌活性,MIC 值分别为 2.3 nM 和 9.2 nM。 | |||
T7533 |
Taurolidine
|
Apoptosis; Others; Antibacterial; Antibiotic | Apoptosis; Microbiology/Virology; Others |
Taurolidine 是一种广谱抗菌剂,用于预防中心静脉导管相关感染。它具有抗真菌和抗肿瘤作用。 | |||
T1405 |
Cefditoren pivoxil
头孢妥仑匹酯,ME 1207,Cefditoren pivaloyloxymethyl ester,Cefditoren pivoxyl |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefditoren pivoxil (ME 1207) 是一种半合成、广谱、β-内酰胺酶耐药的第三代头孢菌素抗生素,具有杀菌活性。 | |||
T12593 |
Pyrithione
1-hydroxyl-1H-pyridine-2-thione,吡啶硫酮 |
Others | Others |
Pyrithione (1-hydroxyl-1H-pyridine-2-thione) 是一种锌离子载体,过渡金属配合物,可引起哺乳动物细胞内锌水平的升高,有杀菌和抗真菌作用。 | |||
T28229 |
Olanexidine hydrochloride
OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045 |
Antibacterial | Microbiology/Virology |
Olanexidine hydrochloride (OPB-2045 HCl) 对革兰氏阳性菌和革兰氏阴性菌具有杀菌活性。 Olanexidine hydrochloride 破坏金黄色葡萄球菌的膜完整性。 | |||
T6706 |
Ticarcillin sodium
Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Ticarcillin sodium (Aerugipen hydrate) 主要用于抗革兰氏阴性菌, 也能用于研究嗜麦芽感染。 | |||
T1005L |
Amoxicillin trihydrate
Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate |
Antibacterial; Antibiotic | Microbiology/Virology |
Amoxicillin trihydrate (Moxaline trihydrate) 是一种中谱β内酰胺抗菌素。 | |||
T1305 |
Ceftazidime
GR20263,头孢他啶 |
Antibacterial; Antibiotic | Microbiology/Virology |
Ceftazidime (GR20263) 是可静脉内或肌肉给药的第头孢菌素。它对革兰氏阳性和革兰氏阴性需氧细菌有体外活性。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。 | |||
T7191 |
Diphenyleneiodonium chloride
二苯基氯化碘盐,DPI |
NOS; Reactive Oxygen Species; NADPH; TRP/TRPV Channel | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB |
Diphenyleneiodonium chloride (DPI) 是 NADPH 氧化酶抑制剂,也是 TRPA1激活剂,EC50为 1 - 3 μM 。它选择性抑制胞内活性氧。 | |||
T0868 |
Cefepime Dihydrochloride Monohydrate
Cefepime HCl,头孢吡肟二盐酸盐一水合物 |
Antibacterial; Antibiotic; Antifection | Microbiology/Virology |
Cefepime Dihydrochloride Monohydrate (Cefepime HCl) 是一种广谱头孢菌素,对革兰氏阳性菌和革兰氏阴性菌有更高的覆盖率。 | |||
T0199 |
Cephradine
Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定 |
TOPK; Antibacterial; Antibiotic | MAPK; Microbiology/Virology |
Cephradine (Anspor) 是广谱口服活性头孢菌素。它对革兰氏阳性和革兰氏阴性病原体都有活性。它已用于泌尿生殖系统、胃肠道和呼吸道感染以及皮肤和软组织感染的研究。它通过直接抑制TOPK 抑制太阳紫外线诱导的皮肤炎症。 | |||
T0377 |
Clofazimine
NSC-141046,氯法齐明,氯苯吩嗪 |
DNA; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Clofazimine (NSC-141046) 是一种具有显著的抗炎效果的亚氨基酚嗪类染料,与其它抗分支杆菌药物联用来治疗AIDS 和克罗恩病。 | |||
TP1341L |
Polymyxin B nonapeptide acetate
Polymyxin B nonapeptide acetate(86408-36-8 free base) |
Antibacterial; Antibiotic | Microbiology/Virology |
Polymyxin B nonapeptide acetate(86408-36-8 free base) 是一种阳离子环肽。 Polyxin B 九肽是 polyxin B 经酶解产生的衍生物。与 polyxin B 相比,polyxin B 九肽毒性低,缺乏杀菌活性,仍具有破坏革兰氏阴性菌外膜的能力。 | |||
T11348 |
G907
|
Antibiotic | Microbiology/Virology |
G907 是一种具有选择性和有效性的小分子ATP 结合盒 (ABC) 转运蛋白 MsbA 的拮抗剂,具有杀菌活性,可将 MsbA 捕获在朝内的脂多糖中。 G907 对大肠杆菌 MsbA 有抑制作用, IC50 值为 18 nM。 | |||
T0953 |
Cefazolin sodium
Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Cefazolin sodium (cephazolin sodium) salt 是一种头孢类抗生素, 可研究多种细菌感染。 | |||
T41275 |
PF-04753299
|
Others | Others |
PF-04753299 是一种有效的、选择性的LpxC 抑制剂。PF-04753299 对淋球菌分离株具有杀菌作用,对大肠杆菌、铜绿假单胞菌和肺炎菌株的抑制的MIC90值分别为 2 μg/ml、4 μg/ml 和 16 μg/ml。PF-04753299 用于革兰氏阴性菌感染的研究。 | |||
T76662 |
Ac-Pro-Gly-Pro-OH
|
Apoptosis; CXCR; Antibiotic | Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology |
Ac-Pro-Gly-Pro-OH 是乙酰基修饰的三肽化合物,可用作 CXCR2 激动剂。Ac-Pro-Gly-Pro-OH 具有杀菌和抗炎活性,抑制免疫细胞凋亡,抑制促炎细胞因子的产生。Ac-Pro-Gly-Pro-OH 可用于研究脓毒症和肺部炎症。 | |||
T1213 |
Piperacillin sodium
哌拉西林钠,Sodium piperacillin,CL227193,Piperacillin sodium salt |
Antibacterial; Antibiotic | Microbiology/Virology |
Piperacillin sodium salt(CL227193) )是一种β-内酰胺类广谱抗生素。 | |||
T77574 |
ROS inducer 1
|
ROS; Antibiotic | Immunology/Inflammation; Microbiology/Virology |
ROS inducer 1 是一种具有杀菌作用的小分子化合物,对 Xanthomonas axonopodis pv. citri (Xac)、Xanthomonas oryzae pv. oryzae (Xoo)和 Pseudomonas syringae pv. actinidiae (Psa) 具有抑制作用。ROS inducer 1 诱 Xanthomonas 细胞内 ROS 的产生可用于研究农作物细菌感染。 | |||
T1005 |
Amoxicillin
Amoxycillin,阿莫西林 |
Antibacterial; Antibiotic | Microbiology/Virology |
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。 | |||
T1224 |
Cefuroxime sodium
Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefuroxime sodium (Cefuroxime sodium salt) 是一种具有口服活性的头孢菌素抗生素,增加了对 β-内酰胺酶的稳定性。 | |||
T1122 |
Cephalothin sodium
头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin |
Antibacterial; Antibiotic | Microbiology/Virology |
Cephalothin sodium (Cefalotin) 是一种头孢类抗生素, 具有广泛的抗菌活性,抑制革兰氏阳性和阴性菌。 | |||
T1063 |
Ticarcillin disodium
Ticarpen,Ticarcillin disodium salt,替卡西林二钠 |
Antibacterial; Antibiotic | Microbiology/Virology |
Ticarcillin disodium (Ticarpen) 主要用于抗革兰氏阴性菌, 特别是绿脓杆菌, 也是少数可研究嗜麦芽感染的抗生素。 | |||
T23613 | ACH-702 | ||
ACH-702 is an agent of anti-tubercular. ACH-702 is an effective, bactericidal compound with activity against many antibiotic-resistant pathogens. | |||
T22390 |
Olanexidine Hydrochloride semihydrate
OPB-2045,OPB-2045G,奥兰西丁标准品HCL |
Others | Others |
Olanexidine is a monobiguanide compound with the activity of bactericidal. | |||
T29505 |
A039
A-039,A 039 |
||
A039 is a highly active bactericidal agent against M. tuberculosis. | |||
T69488 |
CB5255829
|
||
CB5255829 is a novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro. | |||
T71846 |
CB6513745
|
||
CB6513745 is a novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro. | |||
T81848 |
Maximin 7
|
||
Maximin 7是一种从蟾蜍Bombina maxima分离得到的抗菌肽。 | |||
T62014 | (R,R)-BAY-Y 3118 | ||
(R,R)-BAY-Y 3118 是 BAY-Y 3118 的 R 对映体。(R,R)-BAY-Y 3118 显示出杀菌活性。 | |||
T13326 |
SPR719
VXc-486 |
Others | Others |
SPR719 is an inhibitor of gyrase B, has bactericidal activity. | |||
T38801 |
Fobrepodacin
SPR720,pVXc-486 |
||
Fobrepodacin (SPR720) is an orally active and potent phosphate prodrug of SPR719 (VXc-486). Fobrepodacin has potent bactericidal activities in vivo. | |||
T68809 | Trichomonacid | ||
Trichomonacid is a novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro. | |||
T80333 |
Cathepsin G(1-5)
|
||
CathepsinG(1-5)为位于组织蛋白酶G经梭菌蛋白酶消化后混合物中的一种抗菌肽。 | |||
T38913 |
Furaltadone L-tartrate
Furaltadone L-tartrate,Altafur L-tartrate |
||
Furaltadone L-tartrate (Altafur L-tartrate), a nitrofuran antimicrobial agent, is potentially useful for researching Salmonella enteritidis infections in chickens. It demonstrates both inhibitory and bactericidal properties against Staphylococci in vitro. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T20198 |
Potassium gluconate
Kalium-beta,Kalium Gluconate,Kaon elixir,Kaon,Potassium D-gluconate,HSDB 3165,K-Iao |
Endogenous Metabolite; Antifungal | Metabolism; Microbiology/Virology |
Potassium gluconate (Potassium D-gluconate) 是一种具有口服活性和螯合性质的氧化型羧酸,具有杀菌活性。 | |||
T1029 |
Aztreonam
SQ-26,776,氨曲南 |
Antibacterial; Antibiotic | Microbiology/Virology |
Aztreonam (SQ-26,776) 是单环β-内酰胺抗生素,与青霉素结合蛋白3有较高亲和力。 | |||
T0832 |
Vancomycin hydrochloride
盐酸万古霉素,Vancomycin HCl |
Cell wall; Antibacterial; Antibiotic; Autophagy | Autophagy; Immunology/Inflammation; Microbiology/Virology |
Vancomycin hydrochloride (Vancomycin HCl) 是Vancomycin 的盐酸盐,是一种支链三环糖基化肽,对大多数生物体具有杀菌活性,对肠球菌具有抑菌作用。 | |||
T8262 |
Fosfomycin sodium
Fosfomycin Disodium,磷霉素钠 |
Antibacterial; Antibiotic | Microbiology/Virology |
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。 | |||
T0814L |
Ampicillin
Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid |
Antibacterial; Antibiotic | Microbiology/Virology |
Ampicillin (Aminobenzylpenicillin) 属于 β-内酰胺类抗生素,是一种半合成的青霉素。Ampicillin 具有杀菌活性,对各种革兰氏阳性细菌和革兰氏阴性细菌均有抑制活性。 | |||
T1165 |
Ethionamide
Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide |
Dehydrogenase; CAT; Antibacterial; Antibiotic | Metabolism; Microbiology/Virology; oxidation-reduction |
Ethionamide (2-ethylthioisonicotinamide) 是一种抗结核抗生素。 | |||
T3123 |
Allicin
|
ERK; IL Receptor; Others; IκB/IKK; p38 MAPK; TNF; ROS; Caspase; Antifection | Apoptosis; Immunology/Inflammation; MAPK; Microbiology/Virology; NF-κB; Others; Proteases/Proteasome |
Allicin 具有抗氧化、杀菌、抗癌、抗炎活性,对肠上皮细胞具有抑制性免疫调节作用。 Allicin 能显着抑制胰岛素诱导的血管平滑肌细胞的增殖和迁移,这可能与抑制 ERK 信号通路的激活有关。 Allicin 有利于降低高胆固醇血症大鼠的血液胆固醇、甘油三酯水平和收缩压,它可能有益于影响动脉粥样硬化的两个危险因素——高脂血症和高血压。 | |||
T40797 | Essential oils, Melaleuca alternifolia | ||
Melaleuca alternifolia essential oil, derived from the leaves of Melaleuca alternifolia, exhibits bactericidal and anti-inflammatory properties. | |||
TN2760 | 2-Hydroxy-1,8-cineole | Antifection | Microbiology/Virology |
1. 2-endo-Hydroxy-1,8-cineole shows antimicrobial and bactericidal activities against against test bacteria (Staphylococcus aureus, Escherichia coli, and Pseudomonas fluorescens) .<BR/> | |||
TN1407 |
Artocarpin
桂木黄素,2',4',5-三羟基-7-甲氧基-6-(3-甲基-1-丁烯基)-3-(3-甲基-2-丁烯基)黄酮 |
IL Receptor; TNF; COX | Apoptosis; Immunology/Inflammation; Neuroscience |
Artocarpin has anti- bactericidal effect, can reduce the viability of pneumococci by a factor of >1000, without obvious harm to lung epithelial cells. | |||
TN3177 | 6-Methyl-5,6-dihydropyran-2-one | Antifection | Microbiology/Virology |
6-Methyl-5,6-dihydropyran-2-on is bactericidal,and antiprotozoal agents. | |||
TN4944 | Santamarine | Caspase | Apoptosis; Proteases/Proteasome |
Santamarine has significant anticancer activity, can inhibit L1210 cells because of its cytotoxic,cytostatic and blocking mitosis and reducing uptake of thymidine. Santamarine and reynosin show bactericidal activity against clinical strains of Mycobacterium tuberculosis. | |||
T10928 |
Cytochalasin A
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Cytochalasin A is a cell-permeable fungal toxin and is an oxidized derivative of cytochalasin B. Cytochalasin A is an inhibitor of HIV-1 protease (IC50 = 3 μM), inhibits actin polymerization and interferes with microtubule assembly by reacting with sulfhy | |||
T13970 | Xinjiachalcone A | Others | Others |
Xinjiachalcone A is a natural product isolated from Glycyrrhiza inflata Batalin. Xinjiachalcone A shows both a low MIC and a strong bactericidal activity against H. pylori(MIC : 12.5 to 50 µM, seventeen H. pylori strains). | |||
T80357 |
Bombinin H7
|
||
Bombinin H7 是一种抗菌肽,提取自铃蟾Bombina的皮肤分泌物。该化合物对Bacillus megateriumBm11显示出高效活性,其致死浓度达到25.2 μM。 | |||
T80360 |
Bombinin H4
|
||
Bombinin H4,蛾Bombina variegata皮肤中的抗菌肽,其对大肠杆菌D21和金黄色葡萄球菌Cowan 1的致死浓度分别为4.8 μM和3.3 μM。 | |||
T1104 |
Paromomycin Sulfate
Aminosidine sulfate,Paromomycin sulfate salt,硫酸巴龙霉素,巴龙霉素硫酸盐 |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Paromomycin Sulfate (Aminosidine sulfate) 是一种广谱氨基糖苷类抗生素 ,是具有杀螨杀菌作用的新霉素衍生物。它通过与细菌 30S 核糖体 A 位点的 RNA 寡核苷酸特异性结合,使 mRNA 的翻译提前终止,并抑制蛋白质合成。它可研究细菌和寄生虫感染。 | |||
TN4437 |
Licorisoflavan A
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MMP; IL Receptor; NF-κB; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; NF-κB; Proteases/Proteasome |
Licorisoflavan A shows weak scavenging activity against superoxide anion radical, it and licoricidin have potential for the development of novel host-modulating strategies for the treatment of cytokine and/or MMP-mediated disorders such as periodontitis.L |