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Cat. No. Product Name Target Signaling Pathways
T2433 NU 7026

NU7026,DNA-PK Inhibitor II,LY293646

Apoptosis; ATM/ATR; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
NU 7026 (DNA-PK Inhibitor II) 是一种新型特异性的DNA-PK 抑制剂,IC50为 0.23 μM,也抑制PI3K,IC50为 13 μM。
T4339 YU238259

DNA-PK; Others DNA Damage/DNA Repair; Others; PI3K/Akt/mTOR signaling
YU238259 是一种新型的同源依赖性 DNA 修复 (HDR) 抑制剂,在基于细胞的 GFP 报告基因检测中不抑制非同源末端连接 (NHEJ),可研究癌症。
T15789 LTURM34

DNA-PK; PI3K; PI4K DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
LTURM34 是一种 DNA-PK 抑制剂,IC50 为 34 nM。它在广泛的肿瘤细胞系中显示出有效的抗增殖活性,对 DNA-PK 的选择性比 PI3K 高 170 倍。
T2461 PIK-90

DNA-PK; PI3K DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK90 PIK-90 是一种 DNA-PK 和 PI3K 抑制剂,抑制 p110α、p110γ和DNA-PK,IC50分别为 11、18 和 13 nM。
T6100 Torin 2

Apoptosis; ATM/ATR; DNA-PK; mTOR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Torin 2 是一种特异性 mTOR 抑制剂,IC50值为0.25 nM,并改善了药代动力学特性。它抑制 ATM/ATR/DNA-PK 的 EC50 分别为 28 nM/35 nM/118 nM。
T3541 CC-115

CC 115

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
CC-115 是一种双重 mTOR/DNA-PK 的抑制剂,IC50分别为 21 nM 和 13 nM,可阻断mTORC1和mTORC2信号通路。
T3986 SF2523

DNA-PK; Epigenetic Reader Domain; PI3K; mTOR Chromatin/Epigenetic; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
SF2523 是一种选择性PI3K 抑制剂,抑制DNA-PK、PI3Kα、PI3Kγ、BRD4 和 mTOR,IC50分别为 9 nM、34 nM、158 nM、241 nM 和 280 nM。
T4459 PK11000

DNA Alkylator/Crosslinker DNA Damage/DNA Repair
PK11000 是一种烷化剂,可通过共价半胱氨酸修饰来稳定野生型和突变型p53的 DNA 结合结构域。
T9760 IC 86621

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
IC 86621 是一种选择性和可逆的 ATP 竞争性 DNA-PK 抑制剂,IC50 为 120 nM。 IC 86621 增加 DNA 双链断裂 (DSB) 诱导的抗肿瘤活性,其 EC50 为 68 µM,用于 DNA-PK 介导的细胞 DSB 修复。
T6557 KU-0060648

KU0060648

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
KU-0060648 是一种 PI3K 和 DNA-PK 的双重抑制剂,对 PI3Kα、PI3Kβ、PI3Kδ、PI3Kγ 和 DNA-PK 的 IC50值分别为 4 nM、0.5 nM、0.1 nM、0.59 nM 和 8.6 nM。
T6143 PI-103

PI103,PI 103

Apoptosis; DNA-PK; PI3K; mTOR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PI-103 是一种 PI3K 和 mTOR 抑制剂,抑制 p110α、p110β、p110δ、p110γ、mTORC1和 mTORC2,IC50分别为 8 nM、88 nM、48 nM、150 nM、20 nM 和 83 nM。它可诱导自噬,还抑制 DNA-PK,IC50为 2 nM。
T2667 PIK-75

Apoptosis; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK75 是一种可逆的DNA-PK 和p110α-选择性的抑制剂,抑制 DNA-PK、p110α 和 p110γ,IC50分别为 2、5.8 和 76 nM。它诱导凋亡,抑制 p110α 效果比抑制 p110β 高 200 多倍,p110β的IC50为 1.3 μM。
T7122 AZD-7648

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
AZD-7648 是一种 DNA 依赖性蛋白激酶 (DNA-PK) 抑制剂,在酶试验中 IC50 为 0.63 nM,具有抗肿瘤活性。
T25399 ETP-45658

ETP45658,ETP 45658

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
ETP-45658 (ETP45658) 是一种PI3K 抑制剂,抑制PI3Kα、PI3Kδ、PI3Kβ和PI3Kγ的IC50值分别为 22.0、39.8、129.0 和 717.3 nM。它可研究癌症,还抑制DNA-PK 和mTOR,IC50分别为70.6 和 152 nM。
T6276 KU-57788

NU7441

DNA-PK; CRISPR/Cas9 DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
KU-57788 (NU7441) 是一种 NHEJ 通路抑制剂,抑制 PI3K 和 mTOR,IC50分别为 5.0 和 1.7 μM。 它是高效的选择性DNA-PK 抑制剂,IC50为 14 nM。
T6883 Samotolisib

GTPL8918,LY3023414

DNA-PK; PI3K; mTOR; Autophagy Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Samotolisib (LY3023414) 在低纳摩尔浓度下,有效抑制mTORC1/2。它选择性地有效抑制PI3Kα、PI3Kβ、PI3Kδ、PI3Kγ、DNA-PK 和mTOR,IC50分别为 6.07 nM、77.6 nM、38 nM、23.8 nM、4.24 nM 和 165 nM。它可用于多种肿瘤和癌症的试验。
T3586 Compound 401

2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Compound 401 (2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one) 是一种可靶向 mTOR 的合成 DNA-PK 抑制剂,IC50为0.28 μM。
T13017 STL127705

Compound L,7-[[2-(3,4-Dimethoxyphenyl)ethyl]amino]-3-(3-fluorophenyl)pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione

DNA-PK; Others DNA Damage/DNA Repair; Others; PI3K/Akt/mTOR signaling
STL127705 (Compound L) 是一种有效的 Ku 70/80 异二聚体蛋白抑制剂,抑制 Ku70/80-DNA 相互作用,IC50 为 3.5 μM。 它抑制 Ku 依赖性 DNA-PKCS 激酶的激活,IC50 为 2.5 μM。
T25069 AMA-37

DNA-PK Inhibitor V,ArylMorpholine Analog 37,AMA 37

AMA-37 is a selective, reversible, and ATP-competitive DNA-PK inhibitor.
T2008 LY294002

LY 294002,NSC 697286,SF 1101

Apoptosis; DNA-PK; Casein Kinase; PI3K; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling; Stem Cells
LY294002 (SF 1101) 是一种 PI3K 的广谱抑制剂,抑制 PI3Kα、PI3Kδ 和 PI3Kβ (IC50=0.5/0.57/0.97 μM)。LY294002 也是 DNA-PK 抑制剂 (IC50=1.4 μM) 和 CK2 抑制剂 (IC50=98 nM)。LY294002 可以激活凋亡和自噬。
T61828 DNA-PK-IN-8

DNA-PK-IN-8(化合物DK1)是一种高效、选择性且口服活性的DNA依赖蛋白激酶 (DNA-PK) 抑制剂,其IC50值为0.8 nM。与Doxorubicin联合应用时,该化合物能在多种癌细胞中展现出协同的抗增殖效应,并能显著地抑制HL-60肿瘤生长。
T62034 DNA-PK-IN-7

DNA-PK-IN-7 是有效的 DNA-PK 抑制剂,IC50为 1 nM (WO2021104277A1, compound 5)。
T62191 DNA-PK-IN-5

DNA-PK-IN-5 是一种 DNA-PK 的有效抑制剂。DNA-PK-IN-5 能够抑制 DNA-PKcs 活性,明显降低肿瘤 DNA 修复,并诱导细胞凋亡。DNA-PK-IN-5 能够提高肿瘤组织对放疗的敏感性,克服耐药问题,提高对多种实体瘤和血液肿瘤的抑制效果。
T61533 DNA-PK-IN-9

DNA-PK-IN-9 (also known as compound YK6) is a highly potent inhibitor of DNA-dependent protein kinase (DNA-PK), displaying an IC50 value of 10.47 nM. DNA-PK-IN-9 holds significant potential in anticancer research [1].
T79165 DNA-PK-IN-10

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
DNA-PK-IN-10是一种DNA-PK抑制剂, 主要应用于乳腺癌与非小细胞肺癌的研究。
T61857 DNA-PK-IN-4

DNA-PK-IN-4 (WO2021209055A1, compound 27), an imidazolinone derivative compound, is a highly effective inhibitor of DNA-PK, specifically targeting DNA-PKcs activity. By inhibiting DNA-PKcs, the compound significantly impairs tumor DNA repair mechanisms and triggers apoptosis in cells. With its potential application in cancer research, DNA-PK-IN-4 holds promise for further investigation [1].
T61370 DNA-PK-IN-6

DNA-PK-IN-6, a robust DNA-PK inhibitor, effectively hampers the activity of DNA-PKcs, thereby significantly impairing the DNA repair mechanism in tumors and instigating apoptosis in cells. Additionally, DNA-PK-IN-6 amplifies the responsiveness of tumor tissues to radiotherapy, overcomes the challenge of drug resistance, and augments its inhibitory impact on a diverse range of solid and hematological tumors[1].
T62648 DNA-PK-IN-1

DNA-PK-IN-1 是一种 DNA-PK 的有效抑制剂。DNA 依赖性蛋白激酶 (DNA-PK) 是一种由 Ku70/Ku80 异二聚体和 DNA 依赖性蛋白激酶催化亚基 (DNA-PKcs) 组成的 DNA-PK 酶复合物。DNA-PK-IN-1 具有潜力进行癌症疾病的研究。
T61633 DNA-PK-IN-2

DNA-PK-IN-2 is a highly effective inhibitor of DNA-dependent protein kinase (DNA-PK), which is a complex enzyme composed of Ku70/Ku80 heterodimer and DNA-PK catalytic subunit (DNA-PKcs). With its potential applications in cancer research, DNA-PK-IN-2 demonstrates promise as a valuable tool for studying cancer diseases [1].
T61751 DNA-PK-IN-3

DNA-PK-IN-3 is a highly potent inhibitor of DNA-PK. This compound exerts a synergistic effect when combined with radiotherapy and chemotherapy, resulting in enhanced therapeutic outcomes and significant inhibition of tumor growth. Furthermore, DNA-PK-IN-3 demonstrates remarkable efficacy in reducing damage to normal cells, effectively minimizing adverse side effects. Due to these compelling properties, DNA-PK-IN-3 holds great potential for cancer research applications[1].
T2287 PIK-75 hydrochloride

PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75

Apoptosis; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK-75 hydrochloride (PIK-75 HCl) 是一种可逆的 DNA-PK 和 p110α-选择性抑制剂,抑制 DNA-PK,p110α和 p110γ,可诱导凋亡。
T4079 LY-294002 hydrochloride

SF 1101,LY 294002,NSC 697286

PI3K PI3K/Akt/mTOR signaling
LY-294002 hydrochloride (NSC 697286) 是一种合成的 PI3Kα/δ/β 分子抑制剂(IC50:0.5/0.57/0.97 μM,在无细胞试验中);在溶液中比 Wortmannin 更稳定,也是自噬体形成的阻断剂。
T9498 BAY-8400

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
BAY-8400是一种具有口服活性、有效和选择性 DNA 依赖蛋白激酶 (DNA-PK) 抑制剂(IC50=81 nM),与靶向α疗法联合使用显示协同疗效。BAY-8400 可用于癌症研究。
T1826 PI3K-IN-1

Voxtalisib Analogue,Voxtalisib (SAR245409, XL765) Analogue,XL765,SAR245409

DNA-PK; PI3K DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PI3K-IN-1 (Voxtalisib Analogue) 是 PI3K 抑制剂,PI3K-IN-1(25 μM) 能够阻断 PI3K/Akt 信号通路。
T6612 NU6027

ATM/ATR; DNA-PK; CDK Cell Cycle/Checkpoint; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
NU6027 是一种有效的 ATR/CDK 抑制剂,抑制 CDK1/2、ATR 和 DNA-PK,Ki 为 2.5 μM/1.3 μM、0.4 μM 和 2.2 μM。它以 ATR 依赖性方式增强羟基脲和顺铂的细胞毒性。
T7014 Voxtalisib

XL765,SAR245409

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Voxtalisib (XL765) 是一种PI3K 抑制剂,抑制p110α,p110β,p110γ和p110δ。它抑制mTORC1和mTORC2,IC50s 分别为 160 和 910 nM。它也抑制 DNA-PK (其 IC50=150 nM) 和 mTOR (其 IC50=157 nM)。
T62083 Camonsertib

ATR inhibitor 4,RP-3500

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Camonsertib (RP-3500) 是一种选择性的、口服具有活力的 ATR 激酶抑制剂 (ATRi),在生化试验中的 IC50: 1.00 nM,表现出有效的抗肿瘤作用。RP-3500 对 ATR 的选择性是 mTOR 的 30 倍 (IC50: 120 nM),是 ATM、DNA-PK 和 PI3Kα 激酶的 2,000 倍以上。
T8637 DMNB

6-Nitroveratraldehyde,6-硝基藜芦醛

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
DMNB (6-Nitroveratraldehyde) 可用于合成no-carrier-added 6-[18F]fluoro-L-DOPA (6-FDOPA)。它可用于研究多巴胺能系统的PET。
T8651 CAL-101

(S)-2-(1-(9H-Purin-6-ylamino)ethyl)-5-fluoro-3-phenylquinazolin-4(3H)-one,GS-1101,Idelalisib

PI3K PI3K/Akt/mTOR signaling
CAL-101 (Idelalisib) 是 p110δ 的选择性抑制剂(IC50:2.5 nM;在无细胞试验中);显示对 p110δ 的选择性比 p110α/β/γ 高 40 到 300 倍,对 p110δ 的选择性比 C2β、hVPS34、DNA-PK 和 mTOR 高 400 到 4000 倍。
T2415 PP121

Apoptosis; VEGFR; Bcr-Abl; PDGFR; Src; mTOR; Hck Angiogenesis; Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
PP121是一种多靶点激酶抑制剂,抑制 PDGFR、Hck、mTOR、VEGFR2、Src、Abl、DNK-PK 的 IC50值分别为2、8、10、12、14、18、60 nM。
T11067 VX-984

M9831

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
VX-984 (M9831) 是一种可口服的、具有选择性的的、可透过血脑屏障的 DNA-PK 抑制剂。VX-984 对非同源性末端 NHEJ 的接合具有抑制作用,可作用于 DSBs 使 DNA 双链断裂。VX-984常见于对胶质母细胞瘤 (GBM) 和非小细胞肺癌 (NSC-LC) 的研究。
T6319 OSI-027

ASP4786,OSI027

DNA-PK; PI3K; mTOR; Autophagy Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
OSI-027 (ASP4786) 是一种选择性、可口服和 ATP 竞争性的mTOR 激酶活性抑制剂,IC50为 4 nM。它抑制mTORC1和mTORC2,IC50分别为 22 nM 和 65 nM。
T2685 KU-55933

ATM Kinase Inhibitor

ATM/ATR; DNA-PK; PI3K; mTOR; Autophagy Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
KU-55933 (ATM Kinase Inhibitor) 是一种 ATM 抑制剂,IC50和 Ki 值分别为 12.9 和 2.2 nM。它对 ATM 的选择性比对 PI3K/PI4K、 DNA-PK、ATR 和 mTOR 高。
T12672 (Rac)-Nedisertib

(Rac)-M3814

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
(Rac)-Nedisertib is a racemate of Nedisertib, a potent inhibitor of DNA-PK(IC50 of <3 nM).
T6283 Wortmannin

SL-2052,渥曼青霉素,KY-12420

ATM/ATR; DNA-PK; Serine/threonin kinase; PLK; PI3K; Antibiotic; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
Wortmannin (SL-2052) 是一种 PI3K 抑制剂 (IC50=3 nM),具有共价性和不可逆性。Wortmannin 也是一种 PlK1 和 PlK3 的抑制剂 (IC50=5.8/48 nM),可以阻断自噬。
T13444 (R)-Nedisertib

(R)-M3814

Others Others
(R)-Nedisertib is a less active R-enantiomer of Nedisertib(IC50 in the range of 7-30 nM for DNA-PK).
T68192 OK-1035

OK-1035 is a potent and selective DNA-PK inhibitor. When a synthetic peptide was used as a substrate, OK-1035 caused 50% inhibition of DNA-PK activity at 8 microM. OK-1035 inhibited the phosphorylation by DNA-PK of consensus peptide as well as that of recombinant human wild type-p53. Kinetic studies indicated that OK-1035 inhibited DNA-PK activity in an ATP-competitive manner.
T24559 NU-7163

NU 7163,NU7163

NU-7163 is a potent and selective inhibitor of ATP-competitive DNA-PK.
T68978 KU-0058684

KU-0058684 is a potent PARP and DNA-PK inhibitors.
T68691 NU-7031

NU-7031 is a potent DNA-PK inhibitor with potential anticancer activity.

化合物

NU 7026
Cat.No: T2433
Synonym: NU7026,DNA-PK Inhibitor II,LY293646
Target: Apoptosis, ATM/ATR, DNA-PK, PI3K
YU238259
Cat.No: T4339
Synonym:
Target: DNA-PK, Others
LTURM34
Cat.No: T15789
Synonym:
Target: DNA-PK, PI3K, PI4K
PIK-90
Cat.No: T2461
Synonym:
Target: DNA-PK, PI3K
Torin 2
Cat.No: T6100
Synonym:
Target: Apoptosis, ATM/ATR, DNA-PK, mTOR, Autophagy
CC-115
Cat.No: T3541
Synonym: CC 115
Target: DNA-PK, PI3K, mTOR
SF2523
Cat.No: T3986
Synonym:
Target: DNA-PK, Epigenetic Reader Domain, PI3K, mTOR
PK11000
Cat.No: T4459
Synonym:
Target: DNA Alkylator/Crosslinker
IC 86621
Cat.No: T9760
Synonym:
Target: DNA-PK
KU-0060648
Cat.No: T6557
Synonym: KU0060648
Target: DNA-PK, PI3K, mTOR
PI-103
Cat.No: T6143
Synonym: PI103,PI 103
Target: Apoptosis, DNA-PK, PI3K, mTOR, Autophagy
PIK-75
Cat.No: T2667
Synonym:
Target: Apoptosis, DNA-PK, PI3K
AZD-7648
Cat.No: T7122
Synonym:
Target: DNA-PK
ETP-45658
Cat.No: T25399
Synonym: ETP45658,ETP 45658
Target: DNA-PK, PI3K, mTOR
KU-57788
Cat.No: T6276
Synonym: NU7441
Target: DNA-PK, CRISPR/Cas9
Samotolisib
Cat.No: T6883
Synonym: GTPL8918,LY3023414
Target: DNA-PK, PI3K, mTOR, Autophagy
Compound 401
Cat.No: T3586
Synonym: 2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one
Target: DNA-PK
STL127705
Cat.No: T13017
Synonym: Compound L,7-[[2-(3,4-Dimethoxyphenyl)ethyl]amino]-3-(3-fluorophenyl)pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione
Target: DNA-PK, Others
AMA-37
Cat.No: T25069
Synonym: DNA-PK Inhibitor V,ArylMorpholine Analog 37,AMA 37
Target:
LY294002
Cat.No: T2008
Synonym: LY 294002,NSC 697286,SF 1101
Target: Apoptosis, DNA-PK, Casein Kinase, PI3K, Autophagy
DNA-PK-IN-8
Cat.No: T61828
Synonym:
Target:
DNA-PK-IN-7
Cat.No: T62034
Synonym:
Target:
DNA-PK-IN-5
Cat.No: T62191
Synonym:
Target:
DNA-PK-IN-9
Cat.No: T61533
Synonym:
Target:
DNA-PK-IN-10
Cat.No: T79165
Synonym:
Target: DNA-PK
DNA-PK-IN-4
Cat.No: T61857
Synonym:
Target:
DNA-PK-IN-6
Cat.No: T61370
Synonym:
Target:
DNA-PK-IN-1
Cat.No: T62648
Synonym:
Target:
DNA-PK-IN-2
Cat.No: T61633
Synonym:
Target:
DNA-PK-IN-3
Cat.No: T61751
Synonym:
Target:
PIK-75 hydrochloride
Cat.No: T2287
Synonym: PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75
Target: Apoptosis, DNA-PK, PI3K
LY-294002 hydrochloride
Cat.No: T4079
Synonym: SF 1101,LY 294002,NSC 697286
Target: PI3K
BAY-8400
Cat.No: T9498
Synonym:
Target: DNA-PK
PI3K-IN-1
Cat.No: T1826
Synonym: Voxtalisib Analogue,Voxtalisib (SAR245409, XL765) Analogue,XL765,SAR245409
Target: DNA-PK, PI3K
NU6027
Cat.No: T6612
Synonym:
Target: ATM/ATR, DNA-PK, CDK
Voxtalisib
Cat.No: T7014
Synonym: XL765,SAR245409
Target: DNA-PK, PI3K, mTOR
Camonsertib
Cat.No: T62083
Synonym: ATR inhibitor 4,RP-3500
Target: ATM/ATR
DMNB
Cat.No: T8637
Synonym: 6-Nitroveratraldehyde,6-硝基藜芦醛
Target: DNA-PK
CAL-101
Cat.No: T8651
Synonym: (S)-2-(1-(9H-Purin-6-ylamino)ethyl)-5-fluoro-3-phenylquinazolin-4(3H)-one,GS-1101,Idelalisib
Target: PI3K
PP121
Cat.No: T2415
Synonym:
Target: Apoptosis, VEGFR, Bcr-Abl, PDGFR, Src, mTOR, Hck
VX-984
Cat.No: T11067
Synonym: M9831
Target: DNA-PK
OSI-027
Cat.No: T6319
Synonym: ASP4786,OSI027
Target: DNA-PK, PI3K, mTOR, Autophagy
KU-55933
Cat.No: T2685
Synonym: ATM Kinase Inhibitor
Target: ATM/ATR, DNA-PK, PI3K, mTOR, Autophagy
(Rac)-Nedisertib
Cat.No: T12672
Synonym: (Rac)-M3814
Target: DNA-PK
Wortmannin
Cat.No: T6283
Synonym: SL-2052,渥曼青霉素,KY-12420
Target: ATM/ATR, DNA-PK, Serine/threonin kinase, PLK, PI3K, Antibiotic, Autophagy
(R)-Nedisertib
Cat.No: T13444
Synonym: (R)-M3814
Target: Others
OK-1035
Cat.No: T68192
Synonym:
Target:
NU-7163
Cat.No: T24559
Synonym: NU 7163,NU7163
Target:
KU-0058684
Cat.No: T68978
Synonym:
Target:
NU-7031
Cat.No: T68691
Synonym:
Target:
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