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78

抑制剂 & 化合物

55

天然产物

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Cat. No. Product Name Target Signaling Pathways
T3463 NVP-ACC789

ACC-789,ZK202650

VEGFR; PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
NVP-ACC789 (ZK202650) 是一种人VEGFR-1,VEGFR-2(鼠VEGFR-2),VEGFR-3 和 PDGFR-β 的抑制剂,它们的 IC50 值分别为 0.38,0.02 (0.23),0.18 和 1.4 μM。
T82019 JA-ACC

Jasmonyl-ACC

JA-ACC(Jasmonyl-ACC)是1-氨基环丙烷-1-羧酸(ACC)衍生物,后者是植物激素乙烯的直接前体。JA-ACC可抑制Arabidopsis根生长,此作用与茉莉酸(JA)信号通路无关。
T27286L Esprolol

ACC-9369 free base

Adrenergic Receptor GPCR/G Protein; Neuroscience
Esprolol (ACC-9369 free base) 是一种新型β肾上腺素能拮抗剂,可用于研究劳力性心绞痛。
T7066 Fosphenytoin disodium

Fosphenytoin sodium,ACC-9653,磷苯妥英钠

Sodium Channel Membrane transporter/Ion channel
Fosphenytoin disodium (ACC-9653) 是 phenytoin 的前体药物,具有抗惊厥等活性。它是电压门控钠通道阻滞剂。
T27332 Flestolol sulfate

ACC 9089,ACC-9089,ACC9089

Flestolol sulfate is an anti-adrenergic beta-receptor.
T27286 Esprolol hydrochloride

ACC9369,ACC 9369,ACC-9369

Esprolol is a β-adrenergic receptor antagonist.
T80878 Vanutide cridificar

PF 05236806,ACC-001

Vanutide cridificar (ACC-001)是一种氨基末端Aβ1-7肽的偶联物,用于阿尔茨海默病(AD)的研究。
T1768 7ACC2

Mitochondrial Metabolism; Monocarboxylate transporter Membrane transporter/Ion channel; Metabolism
7ACC2 是单羧酸盐转运蛋白抑制剂,IC50为 11 nM。它还是线粒体丙酮酸转运的有效抑制剂,可抑制乳酸涌入,通过抑制乳酸通量来发挥抗癌作用。
T3510 Olumacostat Glasaretil

Acetyl-CoA Carboxylase Metabolism
Olumacostat glasaretil 是乙酰辅酶A 羧化酶的有效抑制剂。
TQ0243 ND-646

Acetyl-CoA Carboxylase Metabolism
ND-646 是乙酰辅酶 A 羧化酶(ACC)抑制剂,对重组 hACC1 和 hACC2的IC50分别为 3.5 nM 和 4.1 nM。
T7163 PF-05175157

Acetyl-CoA Carboxylase Metabolism
PF 05175157 是一种广谱的乙酰辅酶 A 羧化酶 (ACC) 抑制剂,对 ACC1 (human),ACC2 (human), ACC1 (rat) 和 ACC2 (rat) 具有抑制作用,IC50分别为 27.0, 33.0, 23.5 和 50.4 nM。
T1889 CP-640186

CP 640186

Acetyl-CoA Carboxylase Metabolism
CP-640186 是一种有效的乙酰辅酶 A 羧化酶 (ACC)抑制剂,抑制大鼠肝脏 ACC1 和大鼠骨骼肌 ACC2 的 IC50分别为 53 nM 和 61 nM。
T14991 CMS-121

CMS121

Acetyl-CoA Carboxylase Metabolism
CMS-121 是喹诺酮衍生物,对乙酰辅酶 A 羧化酶 1 具有抑制作用,具有口服活性。CMS-121具有保护 HT22 细胞免受缺血和氧化损伤的活性,EC50分别为7 nM 和200 nM。CMS-121具有强大的抗炎,抗氧化,神经保护和肾保护作用。
T3988 TOFA

MDL14514,RMI14514

Acetyl-CoA Carboxylase Metabolism
TOFA (MDL14514) 是有效的乙酰辅酶 A 羧化酶-α (ACCA)的变构抑制剂。
T5046 Haloxyfop

Haloxyfop Acid,(±)-Haloxyfop,吡氟氯禾灵

Others; Acetyl-CoA Carboxylase Metabolism; Others
Haloxyfop (Haloxyfop Acid) 是有效的芳氯氧苯氧丙酸除草剂,广泛应用于阔叶作物的野草。对玉米幼苗叶绿体中乙酰辅酶 A 羧化酶 (EC 6.4.1.2) 具有抑制作用,IC50为 0.5 μM,而对豌豆中该酶无影响。
T7184 Firsocostat

ND-630,NDI-010976,GS-0976

Acetyl-CoA Carboxylase Metabolism
Firsocostat (GS-0976) 是有效的乙酰辅酶A 羧化酶 (ACC) 抑制剂,抑制人类 ACC1 和 ACC2 的IC50分别为2.1和6.1 nM。
T3622 CP-640186 hydrochloride

CP 640186 HCl,盐酸CP-640186

Acetyl-CoA Carboxylase Metabolism
CP-640186 hydrochloride (CP 640186 HCl) 是膜渗透性的乙酰辅酶A 羧化酶(ACC)抑制剂,抑制大鼠肝脏ACC1和大鼠骨骼肌ACC2的IC50为53 nM 和61 nM。
T61978 ACC1/2-IN-2

ACC1/2-IN-2 (compound PF-3) 是有效的 ACC1/2抑制剂,IC50分别为 22 和 48 nM。 ACC1/2-IN-2 显示出抗增殖活性,可用于癌症相关研究。
T63961 ACC1/2-IN-1

ACC1/2-IN-1 是 ACC1/2 的有效抑制剂,可作用于 ACC1 (IC50: 98.06 nM) 和 ACC2 (IC50: 29.43 nM)。ACC1/2-IN-1 可用于研究癌症。
T4330 CaCCinh-A01

Chloride channel Membrane transporter/Ion channel
CaCCinh-A01 是钙激活氯离子通道和TMEM16A 抑制剂,IC50值分别为 10 和 2.1 μM。
T0582 Fructooligosaccharides

Others Others
Fructooligosaccharides 是一种左旋单糖,是葡萄糖的异构体。
T10038 11-cis-Vaccenyl acetate

(Z)-Octadec-11-enyl acetate

Endogenous Metabolite Metabolism
11-cis-Vaccenyl acetate ((Z)-Octadec-11-enyl acetate) 激活位于触角 T1 感受器的嗅觉神经元,并介导雄性和雌性果蝇的聚集行为。
T11142 EACC

Autophagy Autophagy
EACC 是自噬的可逆抑制剂,可阻断自噬通量。它对自噬体特异性的 SNARE Stx17 易位具有选择性抑制作用,从而阻止自噬体与溶酶体的融合。
T7871 Calcium D-saccharate tetrahydrate

D-Glucaric acid calcium salt,葡萄糖二酸鈣,Calcium D-saccharate tetrahydrate,D-Saccharic acid calcium salt

Others Others
Calcium D-saccharate tetrahydrate (Calcium D-saccharate tetrahydrate) 是一种氧化的非环状己糖。它可以抑制癌细胞的癌变和增殖。
T0889 Saccharin

O-Sulfobenzimide,O-Benzoic sulfimide,Saccharimide,Benzoic sulfimide,糖精

Others; Antibacterial Microbiology/Virology; Others
Saccharin (O-Sulfobenzimide) 是一种口服有效的人造甜味剂,具有抑菌和微生物调节特性。
T10789 Chitosan oligosaccharide

COS,壳聚糖低聚乳酸酯

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Chitosan oligosaccharide (COS) 是 β-(1→4)-连接的 D-氨基葡萄糖的寡聚体,Chitosan oligosaccharide可激活 AMPK ,抑制NF-κB 和 MAPK在内的炎症信号通路。
T6974 Saccharin 1-methylimidazole

糖精-1-甲基咪唑盐,SMI,Saccharin 1-methylimidazole (SMI)

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Saccharin 1-methylimidazole (SMI) 是一种用于 DNA 和 RNA 合成的通用激活剂。
T5845 7ACC1

DEAC,香豆素D1421,Coumarin D 1421,7-(二乙胺基)-2-氧代-2-苯并吡喃-3-羧酸,7-(Diethylamino)coumarin-3-carboxylic acid,D 1421

Monocarboxylate transporter Membrane transporter/Ion channel
7ACC1 (D 142) 抑制表达MCT1和MCT4肿瘤细胞的乳酸涌入,能选择性干扰肿瘤微环境乳酸通量。
T41319 D-Saccharic acid 1,4-lactone hydrate

Others Others
D-Saccharic acid 1,4-lactone hydrate 是β-葡萄糖醛酸酶的有效抑制剂(IC50=48.4 μM),可用作标准药物。D-Saccharic acid 1,4-lactone hydrate 显示出抗癌、解毒和抗氧化的活性性。
T78899 Laccase-IN-1

Laccase-IN-1 (compound 4b) 是一种口服laccase抑制剂,其IC50为11.3 μM。该化合物能够对苹果中的B. dothidea起到保护及治疗效果。它通过增强B. dothidea细胞膜的通透性、破坏其菌丝的表面形态以及细胞的超微结构,并且减少麦角甾醇和胞外多糖的含量,来发挥作用。
T76142 Laccase

Laccase(Denilite IIS) 是一种多铜氧化酶(MCOs),广泛存在于微生物、植物和真菌中,能催化多种酚类化合物的一个电子的氧化。Laccase 可以促进单木质素的氧化偶联在木质素的形成中及生物降解中起着重要作用,也具有交联食品聚合物的潜力。
T35744 Ivermectin B1a monosaccharide

Ivermectin B1a monosaccharide is produced by selective hydrolysis of the terminal saccharide unit of ivermectin. It can inhibit nematode larval development, but does not cause paralytic activity. This compound has been used as a probe to detect some types of ivermectin resistance.
T19977 Saccharin sodium

CCRIS 706,Saccharin, sodium

Saccharin sodium is a type of artificial or nonnutritive sweetener. Saccharin sodium is used in the production of various foods and pharmaceutical products.
T25594 Laccaic acid A

Laccaic acid A is a direct, DNA-competitive DNA methyltransferase 1 inhibitor.
T125476 Vaccaroid A

Vaccaroid A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125476,CAS号为 191543-13-2。
T37730 Saccharocarcin A

Saccharocarcin A is an antibiotic originally isolated from S. aerocolonigenes subsp. antibiotica. It is active against M. luteus, S. aureus, E. coli, P. aeruginosa, and C. albicans in a disc assay. Saccharocarcin A inhibits C. trachomatis infection by 88% without inducing cytotoxicity in McCoy cells when used at a concentration of 0.5 μg/ml.
T81964 Laccase-IN-2

Laccase-IN-2作为laccase的抑制剂,在体外及体内对Magnaporthe oryzae均展现出优异的抗真菌活性。
T81424 Polysaccharidase

Tremella polysaccharide

Polysaccharidase (Tremella polysaccharide) 是一种提升免疫功能的真菌多糖。该化合物展现出治疗化疗和放疗导致的白细胞减少症的研究潜力。
T77217 Saccharopine hydrochloride

Saccharopine hydrochloride(L-Saccharopine hydrochloride)是赖氨酸降解的中间体,兼具线粒体毒性。该化合物由赖氨酸-酮戊二酸还原酶催化赖氨酸与α-酮戊二酸生成。继而,糖精脱氢酶作用于Saccharopine hydrochloride,生成α-氨基己酸酯半醛和谷氨酸。其通过干扰线粒体的稳态平衡,对生物体的发育造成损害。
T72319 Lewis y tetrasaccharide

Lewis y

Lewis Y tetrasaccharide (Lewis Y, LeY) 是Lewis X trisaccharide 的四糖衍生物。Lewis Y tetrasaccharide 是一种与恶性卵巢癌转移和预后不良相关的抗原。
T76390 Phosphate acceptor peptide

Phosphate acceptor peptide 是一种 cAMP 依赖性蛋白激酶 (PKA) 的底物。Phosphate acceptor peptide 也是一种弱的PKC 抑制剂。
T131467 1-Hydroxylbaccatin I

1-Hydroxylbaccatin I 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131467。
T13891 SNIPER(TACC3)-1

Others Others
SNIPER(TACC3)-1 targets TACC3 protein degradation via the ubiquitin-proteasome pathway.It induces cancer cell death.
T130142 Bacchabolivic acid

Bacchabolivic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T130142。
T81142 SNIPER(TACC3)-1 hydrochloride

SNIPERs PROTAC
SNIPERTACC3-1 hydrochloride 是一种基于IAPE3连接酶的化合物,其机制是针对泛素-蛋白酶体系统,靶向性地降解TACC3蛋白,从而诱导癌细胞死亡。
T13892 SNIPER(TACC3)-2

Others Others
SNIPER(TACC3)-2 targets TACC3 protein degradation via the ubiquitin-proteasome pathway. It induces cancer cell death.
T68494 Octenidine saccharin

Octenidine saccharin is a Dental Plaque Inhibitor
T124080 Saccatoside

Saccatoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124080,CAS号为 85819-35-8。
T126470 Vaccaroside I

Vaccaroside I 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126470,CAS号为 1052721-36-4。
T72631 TACC3 inhibitor 1

TACC3 inhibitor 1为一种能透过血脑屏障的有效TACC3抑制剂,能诱导Apoptosis及使细胞周期在G2/M期停滞,同时促进细胞内ROS产生,表现出抗增殖与抗肿瘤活性。

化合物

NVP-ACC789
Cat.No: T3463
Synonym: ACC-789,ZK202650
Target: VEGFR, PDGFR
JA-ACC
Cat.No: T82019
Synonym: Jasmonyl-ACC
Target:
Esprolol
Cat.No: T27286L
Synonym: ACC-9369 free base
Target: Adrenergic Receptor
Fosphenytoin disodium
Cat.No: T7066
Synonym: Fosphenytoin sodium,ACC-9653,磷苯妥英钠
Target: Sodium Channel
Flestolol sulfate
Cat.No: T27332
Synonym: ACC 9089,ACC-9089,ACC9089
Target:
Esprolol hydrochloride
Cat.No: T27286
Synonym: ACC9369,ACC 9369,ACC-9369
Target:
Vanutide cridificar
Cat.No: T80878
Synonym: PF 05236806,ACC-001
Target:
7ACC2
Cat.No: T1768
Synonym:
Target: Mitochondrial Metabolism, Monocarboxylate transporter
Olumacostat Glasaretil
Cat.No: T3510
Synonym:
Target: Acetyl-CoA Carboxylase
ND-646
Cat.No: TQ0243
Synonym:
Target: Acetyl-CoA Carboxylase
PF-05175157
Cat.No: T7163
Synonym:
Target: Acetyl-CoA Carboxylase
CP-640186
Cat.No: T1889
Synonym: CP 640186
Target: Acetyl-CoA Carboxylase
CMS-121
Cat.No: T14991
Synonym: CMS121
Target: Acetyl-CoA Carboxylase
TOFA
Cat.No: T3988
Synonym: MDL14514,RMI14514
Target: Acetyl-CoA Carboxylase
Haloxyfop
Cat.No: T5046
Synonym: Haloxyfop Acid,(±)-Haloxyfop,吡氟氯禾灵
Target: Others, Acetyl-CoA Carboxylase
Firsocostat
Cat.No: T7184
Synonym: ND-630,NDI-010976,GS-0976
Target: Acetyl-CoA Carboxylase
CP-640186 hydrochloride
Cat.No: T3622
Synonym: CP 640186 HCl,盐酸CP-640186
Target: Acetyl-CoA Carboxylase
ACC1/2-IN-2
Cat.No: T61978
Synonym:
Target:
ACC1/2-IN-1
Cat.No: T63961
Synonym:
Target:
CaCCinh-A01
Cat.No: T4330
Synonym:
Target: Chloride channel
Fructooligosaccharides
Cat.No: T0582
Synonym:
Target: Others
11-cis-Vaccenyl acetate
Cat.No: T10038
Synonym: (Z)-Octadec-11-enyl acetate
Target: Endogenous Metabolite
EACC
Cat.No: T11142
Synonym:
Target: Autophagy
Calcium D-saccharate tetrahydrate
Cat.No: T7871
Synonym: D-Glucaric acid calcium salt,葡萄糖二酸鈣,Calcium D-saccharate tetrahydrate,D-Saccharic acid calcium salt
Target: Others
Saccharin
Cat.No: T0889
Synonym: O-Sulfobenzimide,O-Benzoic sulfimide,Saccharimide,Benzoic sulfimide,糖精
Target: Others, Antibacterial
Chitosan oligosaccharide
Cat.No: T10789
Synonym: COS,壳聚糖低聚乳酸酯
Target: AMPK
Saccharin 1-methylimidazole
Cat.No: T6974
Synonym: 糖精-1-甲基咪唑盐,SMI,Saccharin 1-methylimidazole (SMI)
Target: DNA/RNA Synthesis
7ACC1
Cat.No: T5845
Synonym: DEAC,香豆素D1421,Coumarin D 1421,7-(二乙胺基)-2-氧代-2-苯并吡喃-3-羧酸,7-(Diethylamino)coumarin-3-carboxylic acid,D 1421
Target: Monocarboxylate transporter
D-Saccharic acid 1,4-lactone hydrate
Cat.No: T41319
Synonym:
Target: Others
Laccase-IN-1
Cat.No: T78899
Synonym:
Target:
Laccase
Cat.No: T76142
Synonym:
Target:
Ivermectin B1a monosaccharide
Cat.No: T35744
Synonym:
Target:
Saccharin sodium
Cat.No: T19977
Synonym: CCRIS 706,Saccharin, sodium
Target:
Laccaic acid A
Cat.No: T25594
Synonym:
Target:
Vaccaroid A
Cat.No: T125476
Synonym:
Target:
Saccharocarcin A
Cat.No: T37730
Synonym:
Target:
Laccase-IN-2
Cat.No: T81964
Synonym:
Target:
Polysaccharidase
Cat.No: T81424
Synonym: Tremella polysaccharide
Target:
Saccharopine hydrochloride
Cat.No: T77217
Synonym:
Target:
Lewis y tetrasaccharide
Cat.No: T72319
Synonym: Lewis y
Target:
Phosphate acceptor peptide
Cat.No: T76390
Synonym:
Target:
1-Hydroxylbaccatin I
Cat.No: T131467
Synonym:
Target:
SNIPER(TACC3)-1
Cat.No: T13891
Synonym:
Target: Others
Bacchabolivic acid
Cat.No: T130142
Synonym:
Target:
SNIPER(TACC3)-1 hydrochloride
Cat.No: T81142
Synonym:
Target: SNIPERs
SNIPER(TACC3)-2
Cat.No: T13892
Synonym:
Target: Others
Octenidine saccharin
Cat.No: T68494
Synonym:
Target:
Saccatoside
Cat.No: T124080
Synonym:
Target:
Vaccaroside I
Cat.No: T126470
Synonym:
Target:
TACC3 inhibitor 1
Cat.No: T72631
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4752 1-Aminocyclopropane-1-carboxylic acid

1-Aminocyclopropanecarboxylic acid,1-氨基环丙烷羧酸,1-Amino-1-carboxycyclopropane,ACC

Endogenous Metabolite; NMDAR Metabolism; Neuroscience
1-Aminocyclopropane-1-carboxylic acid (ACC) 是内源性代谢产物的一种。
T2788 Baccatin III

巴卡亭 Ⅲ,浆果赤霉素III,Baccatin Ⅲ

Others Others
Baccatin III (Baccatin Ⅲ) 是一种分离自太平洋紫杉树和其近缘种中的天然产物,能够减少 MDSCs 积累并抑制其功能,延缓肿瘤发展进程。
TN2256 Taccalonolide B

根薯酮内酯B,根薯酮内酯 B

Microtubule Associated Cytoskeletal Signaling
Taccalonolide B 是从广西裂果薯中分离得到的一种微管稳定剂,具有抗肿瘤活性。它抑制 SK-OV-3 细胞的生长,IC50 为 208 nM,在体外对过表达 P-糖蛋白 (Pgp) 和多药耐药蛋白 (MRP7) 的细胞系有效。
T3387 Phytolaccagenin

Others; Antibacterial Microbiology/Virology; Others
Phytolaccagenin 是一种三萜类皂苷,是商陆的活性成分,有抗真菌活性,抗炎活性和较低的毒性。在东亚国家广泛用于治疗炎症相关疾病。
T2197 10-Deacetylbaccatin III

10-脱乙酰巴卡丁 III,10-脱乙酰基巴卡丁III

Others Others
10-Deacetylbaccatin-III 是一种紫杉醇类似物制剂的中间体,具有抗癌活性。
T41335 cis-Vaccenic acid

cis-11-Octadecenoic acid,Asclepic acid,(Z)-octadec-11-enoic acid

Antiviral Immunology/Inflammation
cis-Vaccenic acid (Asclepic acid) 是来自 Rhodopseudomonas capsulate 的抗病毒提取物,是 Rhodopseudomonas capsulate 的主要活性成分,cis-Vaccenic acid 可用作潜在的胎儿血红蛋白诱导剂。
TN2540 1-Hydroxybaccatin I

Others Others
1-Hydroxybaccatin I 对对苯醌诱导的腹部收缩具有显着的镇痛活性。
T41078 Lipopolysaccharides, Escherichiacoli

Lipopolysaccharide, E. coli O111:B4

Others Others
Lipopolysaccharides, Escherichiacoli (E. coli O111:B4)是革兰阴性菌外膜的大分子成分,由脂质a、寡糖核心和o -特异性多糖(O-antigen) 3个区域组成。
TN2254 Taccalonolide A

根薯酮内酯A,根薯酮内酯 A

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Taccalonolide A 是从水田七根茎中分离得到的一种类固醇,具有细胞毒性和抗疟活性。它在体外对过表达 p 糖蛋白、多药耐药蛋白 7 细胞系有抑制作用,抑制 SK-OV-3 细胞生长的 IC50值为 622 nM。它是微管稳定剂,能引起 G2-M 期滞留、Bcl-2 磷酸化,并引发细胞凋亡。
T5132 9-dihydro-13-acetylbaccatin III

13-乙酰基-9-羟基巴卡丁 III,13-Acetyl-9-dihydrobaccatin III,9-DHAB III

Apoptosis Apoptosis
9-dihydro-13-acetylbaccatin III (9-DHAB III) 是一种制备紫杉醇类似物的中间体。
T5791 Fructo-​oligosaccharide DP7/GF6

Fructoheptasaccharide,蔗果七糖

Others Others
Fructo-​oligosaccharide DP7/GF6 (Fructoheptasaccharide) 属于一种聚果糖,聚合度 (DP=7)。其中 Fructo-oligosaccharides (FOS) 由 6 个果糖单元通过 (2→1)-β-糖苷键连接,并在非还原性末端具有 1 个 D-葡萄糖单元。
TQ0194 trans-Vaccenic acid

TVA,(11E)-octadec-11-enoic acid,11E)-octadec-11-enoic acid

Endogenous Metabolite Metabolism
Trans-Vaccenic acid(TVA)是一种天然存在的反式脂肪酸,存在于反刍动物的脂肪和乳制品中,可通过 GPCR-CREB 通路调控 CD8+ T 细胞增殖,具有抗肿瘤活性。Trans-Vaccenic acid 可在瘤胃中合成饱和脂肪酸,在组织水平合成共轭亚油酸。
TN2376 Fructo-oligosaccharide DP8/GF7

蔗果八糖,Fructo-oligosaccharide DP8 / GF7

Others Others
Fructo-oligosaccharide DP8/GF7 (Fructo-oligosaccharide DP8 / GF7) 是一种聚果糖,聚合度(DP=8)。Fructo-oligosaccharides 由 7 个果糖单元通过 (2→1)-β-糖苷键连接,并在非还原性末端具有 1 个 D-葡萄糖单元。
T11855 Lipopolysaccharides

脂多糖,LPS

Others Others
Lipopolysaccharides (LPS) 属于天然产物,是一种来源于革兰氏阴性菌外膜外叶的内毒素。Lipopolysaccharides 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
T3881 Vaccarin

Integrin; Akt; PERK; AMPK Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Vaccarin 是从王不留行中提取的一种黄酮糖苷,可显著促进伤口愈合以及伤口部位的内皮和成纤维细胞增殖。它通过激活 AMPK 信号通路改善胰岛素抵抗和脂肪变性。
T8154 Fructo-oligosaccharide DP9/GF8

Fructo-oligosaccharide DP9 / GF8,蔗果九糖

Others Others
Fructo-oligosaccharide DP9/GF8 (Fructo-oligosaccharide DP9 / GF8) 是一种低聚果糖(FOS),其聚合度DP=9。低聚果糖(FOS)由 8 个果糖单元通过 (2→1)-β-糖苷键连接,并在非还原性末端具有 1 个 D-葡萄糖单元。
TN2627 14beta-Benzoyloxy-2-deacetylbaccatin VI

Others Others
14beta-Benzoyloxy-2-deacetylbaccatin VI是一种天然产物,属于红豆杉科红豆杉属,其产品编号为 TN2627,CAS号为 705973-69-9。14beta-Benzoyloxy-2-deacetylbaccatin VI可用作对照参考。
T79980 Flaccidoside III

Glucosidase Metabolism
Flaccidoside III, 分离自黑种草(N. sativa)地上部分的一种类黄酮和三萜类化合物,具有抑制α-Glucosidase(IC50:256.7 μM)的活性,表现出潜在的抗氧化和抗糖尿病效应。
TN6260 Taccaoside E

Taccaoside E 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6260,CAS号为 1858199-00-4。
T83435 19-Hydroxy-10-deacetylbaccatin III

19-Hydroxy-10-deacetylbaccatin III (compound 13) 是紫杉烷类化合物,显示出潜在的抗肿瘤作用。在 A498 和 NCI-H226 细胞系中,此化合物表现出轻微的细胞毒性效应。研究指出,当浓度为 30 μg/mL 时,19-Hydroxy-10-deacetylbaccatin III 对 A498 细胞和 NCI-H226 细胞的抑制率为 16.6% 和 32%。
T83471 10-Deacetyl-13-oxobaccatin III

10-Deacetyl-13-oxobaccatin III是一款从Taxus sumatrana分离的紫杉烷。在30 μg/mL的浓度下,对A498、NCI-H226、A549、PC-3细胞系展现细胞毒性作用,其抑制率分别达到29.7%、49.2%、43.9%、65.3%。
T81937 Lewis a trisaccharide

Lewis a

Lewis a trisaccharide 是精子聚糖结构和 HL-60 细胞表面聚糖结构的主要组分。
TN3477 Baccatin VIII

Others Others
Baccatin VIII exhibits inhibitory effects on HL-60 and MCF-7, with IC50 values of 3.44 and 9.67 uM, respectively.
TN2662 19-Hydroxybaccatin III

Others Others
19-Hydroxybaccatin III, 10-deacetylcephalomannine, and 10-deacetyltaxol are new antitumor taxanes from Taxus wallichiana.
TN1356 Acetyl Perisesaccharide C

乙酰杠柳寡糖 C,乙酰杠柳寡糖C

Others Others
Acetyl Perisesaccharide C is a natural product
T72643 Saccharothrixin F

Saccharothrixin F 是一种高度氧化的糖丝菌,具有抗菌和抗炎活性。
TN2615 13-O-Cinnamoylbaccatin III

Others Others
13-O-Cinnamoylbaccatin III is a natural product from Taxus yunnanensis.
T82855 Blood group A pentasaccharide

A-Pentasaccharide

A-Pentasaccharide 是一种尿液中的寡糖,具有抑制抗 A 抗体与 A 型血物质结合的功能。
T81965 Laccaic acid C

Laccaic acid C,以8.1 μM的IC50有效抑制RNase H并能阻止病毒在细胞内的增殖。
T11555 Heptasaccharide Glc4Xyl3

Others Others
Heptasaccharide Glc4Xyl3 is a covalent inhibitor of endo-xyloglucanases. It used for the identification and analysis of diverse xyloglucan-active enzymes in nature.
TN3251 7-Xylosyl-10-deacetylbaccatin III

Others Others
7-Xylosyl-10-deacetylbaccatin III is a natural product from Taxus brevifolia.
TN5785 Isooxoflaccidin

Isooxoflaccidin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5785,CAS号为 135010-50-3。
TN3474 Baccatin IV

Others Others
Baccatin IV is a natural product from Taxus chinensis.
T79983 Flaccidoside II

Apoptosis Apoptosis
Flaccidoside II 是一种源自Anemone flaccida根茎的三萜皂苷,能抑制恶性周围神经鞘瘤(MPNST)细胞系增殖并诱导细胞凋亡(apoptosis)。此外,Flaccidoside II 亦能改善由胶原蛋白引发的小鼠关节炎症状。
TN2358 Fructo-​oligosaccharide DP10/GF9

蔗果十糖,Fructo-oligosaccharide DP10/GF9

Others Others
Fructo-oligosaccharide DP10/GF9 is a compound classified as a fructooligosaccharide (FOS) with a degree of polymerization (DP) of 10. FOS consists of a chain of 9 fructose units connected by (2→1)-β-glycosidic bonds, with a lone D-glucosyl unit located at the non-reducing end.
TN6404 Vaccarin E

Vaccarin E是一种天然产物,属于石竹科王不留行属,其产品编号为 TN6404,CAS号为 2252345-81-4。Vaccarin E可用作对照参考。
TN2530 1-Dehydroxybaccatin IV

Others Others
1-Dehydroxybaccatin IV is a natural product from Taxus mairei.
TN2065 Phytolaccagenic acid

美商陆酸

Others Others
Phytolaccagenic acid is a natural product
T82370 Fructo-oligosaccharide DP13

Fructo-oligosaccharide DP13,一种Inulin型低聚果糖,可从Morinda Officinalis中分离。
TN3475 Baccatin IX

Others Others
Baccatin IX is a natural product from Taxus yunnanensis.
TN3476 Baccatin VI

Others Others
Baccatin VI 对对苯并醌诱发的腹部收缩具有显著的抗伤害活性。
T19328 Fructo-oligosaccharide DP11/GF10

Others Others
Fructo-oligosaccharide DP11/GF10 is a fructooligosaccharide (FOS) compound with a degree of polymerization (DP) equal to 11. FOS consists of 10 fructose units connected by (2→1)-β-glycosidic bonds, with a single D-glucosyl unit present at the non-reducing end.
TN6125 Flaccidinin

Flaccidinin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6125,CAS号为 121817-23-0。
T82369 Fructo-oligosaccharide DP14

Fructo-oligosaccharide DP14为从Atractylodes lancea中提取的寡糖。
TN2057 Perisesaccharide C

Others Others
Perisesaccharide C is a natural product
TN2255 Taccalonolide AJ

Others Others
Taccalonolide AJ is a microtubule stabilizer; it has excellent and highly persistent antitumor efficacy when administered directly to the tumor, suggesting that the lack of antitumor efficacy seen with systemic administration of AJ is likely due to its sh
T82277 GM1a Ganglioside oligosaccharide

GM1a Ganglioside oligosaccharide为ganglioside GM1的半合成形式,后者作为霍乱毒素的天然受体,在生长调节及激素诱导反应的耦合中具有关键功能。
T75573 Taccalonolide E

Taccalonolide E 是一种微管稳定剂,诱导癌细胞凋亡 (apoptosis)。
T19329 Fructo-oligosaccharide DP12/GF11

蔗果十二糖

Others Others
Fructo-oligosaccharide DP12/GF11 is a member of fructooligosaccharides (FOS) characterized by a degree of polymerization (DP) of 12. FOS compounds consist of 11 fructose units connected by (2→1)-β-glycosidic bonds, with a lone D-glucosyl unit located at the non-reducing end.
TN6134 Flaccidin

Flaccidin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6134,CAS号为 115531-76-5。
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天然产物

1-Aminocyclopropane-1-carboxylic acid
Cat.No: T4752
Synonym: 1-Aminocyclopropanecarboxylic acid,1-氨基环丙烷羧酸,1-Amino-1-carboxycyclopropane,ACC
Target: Endogenous Metabolite, NMDAR
Baccatin III
Cat.No: T2788
Synonym: 巴卡亭 Ⅲ,浆果赤霉素III,Baccatin Ⅲ
Target: Others
Taccalonolide B
Cat.No: TN2256
Synonym: 根薯酮内酯B,根薯酮内酯 B
Target: Microtubule Associated
Phytolaccagenin
Cat.No: T3387
Synonym:
Target: Others, Antibacterial
10-Deacetylbaccatin III
Cat.No: T2197
Synonym: 10-脱乙酰巴卡丁 III,10-脱乙酰基巴卡丁III
Target: Others
cis-Vaccenic acid
Cat.No: T41335
Synonym: cis-11-Octadecenoic acid,Asclepic acid,(Z)-octadec-11-enoic acid
Target: Antiviral
1-Hydroxybaccatin I
Cat.No: TN2540
Synonym:
Target: Others
Lipopolysaccharides, Escherichiacoli
Cat.No: T41078
Synonym: Lipopolysaccharide, E. coli O111:B4
Target: Others
Taccalonolide A
Cat.No: TN2254
Synonym: 根薯酮内酯A,根薯酮内酯 A
Target: Apoptosis, Microtubule Associated
9-dihydro-13-acetylbaccatin III
Cat.No: T5132
Synonym: 13-乙酰基-9-羟基巴卡丁 III,13-Acetyl-9-dihydrobaccatin III,9-DHAB III
Target: Apoptosis
Fructo-​oligosaccharide DP7/GF6
Cat.No: T5791
Synonym: Fructoheptasaccharide,蔗果七糖
Target: Others
trans-Vaccenic acid
Cat.No: TQ0194
Synonym: TVA,(11E)-octadec-11-enoic acid,11E)-octadec-11-enoic acid
Target: Endogenous Metabolite
Fructo-oligosaccharide DP8/GF7
Cat.No: TN2376
Synonym: 蔗果八糖,Fructo-oligosaccharide DP8 / GF7
Target: Others
Lipopolysaccharides
Cat.No: T11855
Synonym: 脂多糖,LPS
Target: Others
Vaccarin
Cat.No: T3881
Synonym:
Target: Integrin, Akt, PERK, AMPK
Fructo-oligosaccharide DP9/GF8
Cat.No: T8154
Synonym: Fructo-oligosaccharide DP9 / GF8,蔗果九糖
Target: Others
14beta-Benzoyloxy-2-deacetylbaccatin VI
Cat.No: TN2627
Synonym:
Target: Others
Flaccidoside III
Cat.No: T79980
Synonym:
Target: Glucosidase
Taccaoside E
Cat.No: TN6260
Synonym:
Target:
19-Hydroxy-10-deacetylbaccatin III
Cat.No: T83435
Synonym:
Target:
10-Deacetyl-13-oxobaccatin III
Cat.No: T83471
Synonym:
Target:
Lewis a trisaccharide
Cat.No: T81937
Synonym: Lewis a
Target:
Baccatin VIII
Cat.No: TN3477
Synonym:
Target: Others
19-Hydroxybaccatin III
Cat.No: TN2662
Synonym:
Target: Others
Acetyl Perisesaccharide C
Cat.No: TN1356
Synonym: 乙酰杠柳寡糖 C,乙酰杠柳寡糖C
Target: Others
Saccharothrixin F
Cat.No: T72643
Synonym:
Target:
13-O-Cinnamoylbaccatin III
Cat.No: TN2615
Synonym:
Target: Others
Blood group A pentasaccharide
Cat.No: T82855
Synonym: A-Pentasaccharide
Target:
Laccaic acid C
Cat.No: T81965
Synonym:
Target:
Heptasaccharide Glc4Xyl3
Cat.No: T11555
Synonym:
Target: Others
7-Xylosyl-10-deacetylbaccatin III
Cat.No: TN3251
Synonym:
Target: Others
Isooxoflaccidin
Cat.No: TN5785
Synonym:
Target:
Baccatin IV
Cat.No: TN3474
Synonym:
Target: Others
Flaccidoside II
Cat.No: T79983
Synonym:
Target: Apoptosis
Fructo-​oligosaccharide DP10/GF9
Cat.No: TN2358
Synonym: 蔗果十糖,Fructo-oligosaccharide DP10/GF9
Target: Others
Vaccarin E
Cat.No: TN6404
Synonym:
Target:
1-Dehydroxybaccatin IV
Cat.No: TN2530
Synonym:
Target: Others
Phytolaccagenic acid
Cat.No: TN2065
Synonym: 美商陆酸
Target: Others
Fructo-oligosaccharide DP13
Cat.No: T82370
Synonym:
Target:
Baccatin IX
Cat.No: TN3475
Synonym:
Target: Others
Baccatin VI
Cat.No: TN3476
Synonym:
Target: Others
Fructo-oligosaccharide DP11/GF10
Cat.No: T19328
Synonym:
Target: Others
Flaccidinin
Cat.No: TN6125
Synonym:
Target:
Fructo-oligosaccharide DP14
Cat.No: T82369
Synonym:
Target:
Perisesaccharide C
Cat.No: TN2057
Synonym:
Target: Others
Taccalonolide AJ
Cat.No: TN2255
Synonym:
Target: Others
GM1a Ganglioside oligosaccharide
Cat.No: T82277
Synonym:
Target:
Taccalonolide E
Cat.No: T75573
Synonym:
Target:
Fructo-oligosaccharide DP12/GF11
Cat.No: T19329
Synonym: 蔗果十二糖
Target: Others
Flaccidin
Cat.No: TN6134
Synonym:
Target:
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