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57

抑制剂 & 化合物

3

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Cat. No. Product Name Target Signaling Pathways
T74557 α1A-AR Degrader 9c

PROTACs PROTAC
α1A-AR Degrader 9c(化合物 9c)是一种高效、选择性且可逆的α1A-AR PROTAC降解剂,DC50值为2.86 μM。它通过蛋白酶体途径诱导α1A-AR的降解,并且在抑制PC-3细胞增殖方面表现出活性,IC50为6.12 μM。此外,α1A-AR Degrader 9c展现出在前列腺癌研究中的抗肿瘤潜力。
T41231 GP 1a

Cannabinoid Receptor; PERK; Arrestin Apoptosis; GPCR/G Protein
GP 1a 是cannabinoid receptor 2(CB2)的强效激动剂(EC50=7.1),是在cAMP、GTPγS 和β-arrestin 招募试验中显示的。GP 1a 对CB2受体的选择性约为CB1受体的30倍,且在体外增加HL-60细胞的P-ERK1/2表达。GP 1a 对皮肤伤口愈合有益。GP 1a 可抑制炎症和纤维生成,同时促进上皮的重新形成。
T1132 Nicergoline

尼麦角林,Nicergolinum,Nimergoline

Adrenergic Receptor GPCR/G Protein; Neuroscience
Nicergoline (Nicergolinum) 是一种有效的,选择性的、具有口服活性的α1A-肾上腺素能受体拮抗剂,是一种溴烟碱酸的麦角林衍生物。它具有血管舒张作用,可以改善阿尔茨海默症小鼠的认知功能。
T38160 STING Agonist 1a

STING agonist 1a is an agonist of stimulator of interferon genes (STING).1It induces expression of an IRF-inducible SEAP reporter gene in a cell-based assay (EC50= 16.77 μM). STING agonist 1a (12.5-100 μM) induces expression of IFN-β, IL-6, and chemokine (C-X-C motif) ligand 10 (CXCL10) in THP-1 cells, an effect that can be reversed by STING knockout or the STING inhibitor H-151 . 1.Hou, H., Yang, R., Liu, X., et al.Discovery of triazoloquinoxaline as novel STING agonists via structure-based vir...
T76469 Esculentin 1A

Esculentin 1A 是一种青蛙皮肤来源的抗菌肽(AMP),具有强大的体外抗假单胞菌活性。
T30873 Chelator 1a

Chelator1a,Chelator-1a

Antifungal Microbiology/Virology
Chelator 1a 具有抗真菌活性,抑制曲霉菌和念珠菌,可用于研究真菌感染和癌症。
T63873 Anti-Aβ agent 1A

Anti-Aβ agent 1A 是有效的抗淀粉样蛋白-β (amyloid-β) 剂。Anti-Aβ agent 1A 可明显抑制 LPS 诱导的 IL-1β、IL-6 和 TNF-α 水平,并能够利用线粒体途径减少 H2O2诱导的 SH-SY5Y 细胞凋亡,表现出抗氧化、抗炎、抗 Aβ 毒性和神经保护活性。Anti-Aβ agent 1A 能够用于研究阿尔兹海默症。
T83857 Soluble Epoxide Hydrolase PROTAC 1a

sEH Proteolysis-targeting Chimera 1a,Soluble Epoxide Hydrolase Proteolysis-targeting Chimera 1a,sEH PROTAC 1a

Soluble epoxide hydrolase (sEH) PROTAC 1a是一种利用蛋白质降解靶向嵌合体(PROTAC)技术,通过连接区域将cereblon配体1与sEH抑制剂t-TUCB结合。该化合物通过促进sEH的降解,特异性抑制sEH的水解酶活性(IC50 = 0.8 nM),相较于其磷酸酶活性(IC50 = >10,000 nM)具有较高选择性。sEH PROTAC 1a还特定促进细胞质中而非过氧体中的sEH降解,并通过溶酶体而非蛋白酶体实现其降解。它能够降低thapsigargin诱导的HepG2与293T细胞中磷酸化的inositol-requiring enzyme 1α (IRE1α)水平和X-box结合蛋白1 (XBP1)剪接,表明能减少ER应激。
T36045 1a,1b-dihomo Prostaglandin E2

1a,1b-dihomo Prostaglandin E2

1a,1b-dihomo Prostaglandin E2 (PGE2) is a rare polyunsaturated fatty acid first identified in extracts of sheep vesicular gland microsomes, known to contain COX, incubated with adrenic acid . 1a,1b-dihomo PGE2 has also been identified in conditioned media of RAW 264.7 macrophages stimulated with endotoxin and arachidonic acid . This product is thought to be produced by elongation of AA to adrenic acid, which is then metabolized sequentially by COX and PGE synthase.
T36219 1a,1b-dihomo Prostaglandin E1

1a,1b-dihomo Prostaglandin E1

1a,1b-dihomo Prostaglandin E1 是一类前列腺素化合物。
T131451 Methyl 1a,7a,14a-triacetoxy-8,15-isopimaredien-18-oate

Methyl 1a,7a,14a-triacetoxy-8,15-isopimaredien-18-oate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131451。
T16798 RS 17053 hydrochloride

RS-17053

Others; Adrenergic Receptor GPCR/G Protein; Neuroscience; Others
RS 17053 hydrochloride 是有效的、选择性的 α1A 肾上腺素受体 (α1A adrenoceptor) 拮抗剂。RS 17053 hydrochloride 在细胞膜中测得的 pKi 值为 9.1,功能分析的 pA2 值为 9.8。
T12643 (R)-Terazosin

(R)-特拉唑嗪,盐酸特拉唑嗪

Adrenergic Receptor GPCR/G Protein; Neuroscience
(R)-Terazosin 是一种 Terazosin 的活性 R 型对映体, 是 α1-肾上腺素受体拮抗剂,对 α1a,α1b 和α1d-肾上腺素受体的Ki 分别为 6.51 nM,1.01 nM 和 1.97 nM。
T23301 (S)-(+)-Niguldipine hydrochloride

Others Others
(S)-(+)-Niguldipine hydrochloride is a L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist.
T23253 RS 100329 hydrochloride

RS-100329

Adrenergic Receptor GPCR/G Protein; Neuroscience
RS 100329 hydrochloride 是α1A 肾上腺素能受体的拮抗剂。
T9762 Upidosin

SB-216469,SB 216469,Rec 15-2739,Recordati 15/2739

Adrenergic Receptor GPCR/G Protein; Neuroscience
Upidosin (SB-216469) 是一种有效的、选择性的α1-肾上腺素受体拮抗剂,α1a 亚型Ki=0.34nM,α1b 亚型Ki=3.9nM,β1d 亚型Ki=1.5nM,γ2-肾上腺素受体Ki=33.3nM。
T13110 Tedatioxetine hydrobromide

Lu AA 24530 hydrobromide

Dopamine Receptor; 5-HT Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) 是一种血清素-去甲肾上腺素-多巴胺再摄取抑制剂 ,也是 5-HT2A、5-HT2C、5-HT3 和 α1A-肾上腺素能受体的拮抗剂,可用于治疗抑郁症和焦虑症。
T15688 L-771688

SNAP 6383

Adrenergic Receptor GPCR/G Protein; Neuroscience
L-771688(SNAP 6383) 是一种新型有效和选择性的 α1A-肾上腺素受体拮抗剂, Ki 值为 0.43±0.02 nM。L-771688 KE 用于治疗良性前列腺增生。
T9220 Naftopidil hydrochloride

1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,萘哌地尔盐酸盐,KT-611 hydrochloride,BM-15275 hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Naftopidil hydrochloride (BM-15275 hydrochloride) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力 Ki 分别为 3.7 nM、20 nM、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。
T1504 Silodosin

西洛多辛,KAD 3213,KMD 3213

Adrenergic Receptor GPCR/G Protein; Neuroscience
Silodosin (KAD 3213) 是有选择性的、强效的、口服活性的 α1A-adrenergic receptor 阻滞剂,是一种有效且耐受性良好的试剂,可用于研究 LUTS/BPH。它对 α1A-AR 表现出高度的亲和力,是 α1B-AR 和 α1D-AR 亲和力的 162 和 50 倍。
T11286 Fiduxosin

A 185980.1,ABT 980

Adrenergic Receptor GPCR/G Protein; Neuroscience
Fiduxosin 是一种具有选择性和有效性的 α1-adrenoceptor 拮抗剂,对 α1a-adrenoceptor,α1b-adrenoceptor 和 α1d-adrenoceptor 有抑制作用,Ki 值分别为 0.160 nM,24.9 nM 和 0.920 nM。Fiduxosin 可用于治疗良性前列腺增生。
T1090 Perphenazine

Perphenazin,Etaperazine,Trilafon,奋乃静

CaMK; Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Perphenazine (Trilafon) 是吩噻嗪衍生物和多巴胺拮抗剂,具有止吐和抗精神病特性。它能够抑制5-HT2A 受体,α1A 肾上腺素能受体,多巴胺D2、D3、D2L 受体,以及组胺H1受体,对应的Ki 值分别为5.6、10、0.765、0.13、3.4 和 8 nM。
T6600 Naftopidil dihydrochloride

KT-611,KT-611 2HCl,盐酸萘哌地尔,Naftopidil DiHCl

5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Naftopidil dihydrochloride (KT-611 2HCl) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力Ki 分别为 3.7 nM、20 nM、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。
T3046 BMY 7378 dihydrochloride

BMY7378 HCl

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
BMY 7378 dihydrochloride (BMY7378 HCl) 是选择性 α1D 肾上腺素受体拮抗剂,也是5-HT1A 受体部分激动剂。它同表达克隆大鼠 α1D-AR 的膜结合的亲和力 (Ki=2 nM)  是同克隆大鼠 α1A-AR (Ki=800 nM) 或仓鼠 α1B-AR (Ki=600 nM) 结合的亲和力 的100 以上。
T27401 Garomefrine HCl

PNO-49B,NS-49,ABT-232,ABT232,NS49,PNO49B

Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.
T10523 β3-AR agonist 1

Others Others
β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold).
T80505 PKCα (C2-4) inhibitor peptide

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
PKCα(C2-4) inhibitor peptide为专一性PKCα抑制剂,能够抑制α1A‐肾上腺素受体激动剂A-61603对IKr通道的影响。
T14972 Cirazoline hydrochloride

LD 3098 hydrochloride

Others Others
Cirazoline hydrochloride is a competitive full agonist of the α1A-adrenergic receptor (α1A-AR; Ki: 120 nM). It is a partial agonist at α1B-AR (Ki: 960 nM) and α1D-AR (Ki: 660 nM).
T24378 L-771688 dihydrochloride

L 771688 dihydrochloride

L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.
T82072 Indoramin hydrochloride

Indoramine hydrochloride,Wy 21901 hydrochloride

Indoramin (hydrochloride) is a novel antihypertensive agent that exhibits selectivity for the α1A-adrenergic receptor.
T23532 WB 4101 hydrochloride

Others Others
α1A-adrenergic antagonist
T23374 SNAP 5089

Others Others
α1A-adrenoceptor antagonist
T28617 RS 100329

RS100329 HCl,RS 100329 HCl,RS100329,RS-100329

RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).
T23225 (R)-(-)-Niguldipine hydrochloride

Others Others
(R)-(-)-Niguldipine hydrochloride is a L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist.
T71335 PF-3774076

PF-3774076 is a CNS penetrant, potent, selective, partial agonist at the human α1A adrenoceptor. PF-3774076 is selective over α1B and α1D adrenoceptors.
T80477 Muscarinic toxin 3

MT3

Adrenergic Receptor GPCR/G Protein; Neuroscience
Muscarinic toxin 3 (MT3) 是高效的非竞争性mAChR及adrenoceptors拮抗剂,对M1、M4、α1A、α1B、α1D、α2A、α2B、α2C受体展示出不同程度的选择性,其pIC50值分别为6.71、8.79、8.86、7.57、8.13、8.49、6.5、7.29。该化合物具有显著的肾上腺素受体抑制活性。
T12815 (S)-Terazosin

Adrenergic Receptor GPCR/G Protein; Neuroscience
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with Ki values of 3.91 nM, 0.79 nM and 1.16 nM, respectively).
T35576 Phenylephrine-3-O-Sulfate

Phenylephrine-3-O-sulfate is metabolite of the α1A-adrenergic receptor agonist phenylephrine formed via sulfation.
T36071 Silodosin Glucuronide (sodium salt)

Silodosin glucuronide is an active metabolite of the α1A-adrenergic receptor antagonist silodosin . It is formed from silodosin by the UDP-glucuronosyltransferase (UGT) isoform UGT2B7. Silodosin glucuronide is toxic to rats with an LD50 value of 0.347 mg/kg.
TP2086 AdTx1

Selective, high affinity, non-competitive α1A adrenoceptor antagonist (Ki = 0.35 nM). Exhibits no significant activity against a range of other GPCRs, including α2A, β1 and β2 adrenoceptors. Antagonizes effects of phenylephrine on isolated rabbit prostate
T63980 BODIPY FL prazosin

BODIPY FL prazosin 是荧光 α1-肾上腺素 α1-adrenergic 拮抗剂,能够作用于 α1a-AR (Ki: 14.5 nM)和 α1b-AR (Ki: 43.3 nM)。BODIPY FL prazosin 是一种荧光配体,激发和发射波长分别为 485 和 535 nm。BODIPY FL prazosin 能够用于 α1-肾上腺素受体亚型的亚细胞定位差异的研究。
T64314 OxyMetazoline

OxyMetazoline 是一种 α-肾上腺素受体 (α-adrenoceptor) 激动剂,能够作用于 α1A (IC50: 0.02 μM)、α1B (IC50: 0.25 μM)、α2A (IC50: 0.58 μM) 和 α2C (IC50: 0.13 μM)。OxyMetazoline 能够用于研究缓解鼻黏膜充血。
T80175 Conopeptide rho-TIA

Adrenergic Receptor GPCR/G Protein; Neuroscience
Conopeptide rho-TIA为从掠食性海螺Conus tulipa毒液中提炼的多肽,对人类α1B-Adrenergic Receptor呈现非竞争性抑制作用,同时对α1A-Adrenergic Receptor和α1D-Adrenergic Receptor表现出竞争性抑制。Conopeptide rho-TIA与这些亚型的结合特性可能对开发针对α1-Adrenergic Receptor亚型的选择性新药具有参考价值。
T5384 RS 504393

CCR Immunology/Inflammation; Microbiology/Virology
RS 504393 是一种高度选择性的 CCR2 趋化因子受体拮抗剂,作用于人重组 CCR2 和 CCR1 受体,IC50值分别为 89 nM 和大于 100 μM。
T69031 Cirazoline (free base)

Cirazoline (free base) is a full agonist at the α1A adrenergic receptor, a partial agonist at both the α1B and α1D adrenergic receptors, and a nonselective antagonist to the α₂ adrenergic receptor. It is believed that this combination of properties could make cirazoline an effective vasoconstricting agent.
TQ0283 RS102895

CCR Immunology/Inflammation; Microbiology/Virology
RS102895 是一种CCR2拮抗剂,IC50值为 360 nM。
T78626 LY393615

NCC1048

Calcium Channel Membrane transporter/Ion channel; Metabolism
LY393615 (NCC1048) 是新型神经元 Ca2+ 与 Na+ 通道阻断剂,具备优良的脑渗透性,并在脑缺血模型中显示神经保护效果,适用于神经性疾病研究。
T67694 ZY-19489

Parasite Microbiology/Virology
ZY-19489是一种具有抗疟作用的化合物, 是一种潜在的单剂量根治性恶性疟原虫和间日疟原虫疟疾的药物,已获得美国 FDA 的孤儿药认定。
T37794 Rec 15/2615 (hydrochloride)

Rec 15/2615 is an antagonist of α1B-adrenergic receptors (α1B-ARs; Ki = 0.45 nM for the recombinant human receptor).1 It selectively inhibits α1B-ARs over α1A-, α1D-, and α1L-ARs (Kis = 7.59, 10.23, and 49 nM, respectively). Rec 15/2615 inhibits norepinephrine-induced contractions of isolated rabbit prostate and urethral strips (Kis = 100 and 316.2 nM, respectively), as well as reduces norepinephrine-induced contractions of chloroethylclonidine-precontracted isolated rabbit aortic rings (Ki = 50...
T0696 Naftopidil

KT-611,萘哌地尔,BM-15275

Adrenergic Receptor GPCR/G Protein; Neuroscience
Naftopidil (KT-611) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力Ki 分别为 3.7 nM、20 nM 、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。

化合物

α1A-AR Degrader 9c
Cat.No: T74557
Synonym:
Target: PROTACs
GP 1a
Cat.No: T41231
Synonym:
Target: Cannabinoid Receptor, PERK, Arrestin
Nicergoline
Cat.No: T1132
Synonym: 尼麦角林,Nicergolinum,Nimergoline
Target: Adrenergic Receptor
STING Agonist 1a
Cat.No: T38160
Synonym:
Target:
Esculentin 1A
Cat.No: T76469
Synonym:
Target:
Chelator 1a
Cat.No: T30873
Synonym: Chelator1a,Chelator-1a
Target: Antifungal
Anti-Aβ agent 1A
Cat.No: T63873
Synonym:
Target:
Soluble Epoxide Hydrolase PROTAC 1a
Cat.No: T83857
Synonym: sEH Proteolysis-targeting Chimera 1a,Soluble Epoxide Hydrolase Proteolysis-targeting Chimera 1a,sEH PROTAC 1a
Target:
1a,1b-dihomo Prostaglandin E2
Cat.No: T36045
Synonym: 1a,1b-dihomo Prostaglandin E2
Target:
1a,1b-dihomo Prostaglandin E1
Cat.No: T36219
Synonym: 1a,1b-dihomo Prostaglandin E1
Target:
Methyl 1a,7a,14a-triacetoxy-8,15-isopimaredien-18-oate
Cat.No: T131451
Synonym:
Target:
RS 17053 hydrochloride
Cat.No: T16798
Synonym: RS-17053
Target: Others, Adrenergic Receptor
(R)-Terazosin
Cat.No: T12643
Synonym: (R)-特拉唑嗪,盐酸特拉唑嗪
Target: Adrenergic Receptor
(S)-(+)-Niguldipine hydrochloride
Cat.No: T23301
Synonym:
Target: Others
RS 100329 hydrochloride
Cat.No: T23253
Synonym: RS-100329
Target: Adrenergic Receptor
Upidosin
Cat.No: T9762
Synonym: SB-216469,SB 216469,Rec 15-2739,Recordati 15/2739
Target: Adrenergic Receptor
Tedatioxetine hydrobromide
Cat.No: T13110
Synonym: Lu AA 24530 hydrobromide
Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine
L-771688
Cat.No: T15688
Synonym: SNAP 6383
Target: Adrenergic Receptor
Naftopidil hydrochloride
Cat.No: T9220
Synonym: 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,萘哌地尔盐酸盐,KT-611 hydrochloride,BM-15275 hydrochloride
Target: Adrenergic Receptor
Silodosin
Cat.No: T1504
Synonym: 西洛多辛,KAD 3213,KMD 3213
Target: Adrenergic Receptor
Fiduxosin
Cat.No: T11286
Synonym: A 185980.1,ABT 980
Target: Adrenergic Receptor
Perphenazine
Cat.No: T1090
Synonym: Perphenazin,Etaperazine,Trilafon,奋乃静
Target: CaMK, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Naftopidil dihydrochloride
Cat.No: T6600
Synonym: KT-611,KT-611 2HCl,盐酸萘哌地尔,Naftopidil DiHCl
Target: 5-HT Receptor, Adrenergic Receptor
BMY 7378 dihydrochloride
Cat.No: T3046
Synonym: BMY7378 HCl
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Garomefrine HCl
Cat.No: T27401
Synonym: PNO-49B,NS-49,ABT-232,ABT232,NS49,PNO49B
Target:
β3-AR agonist 1
Cat.No: T10523
Synonym:
Target: Others
PKCα (C2-4) inhibitor peptide
Cat.No: T80505
Synonym:
Target: PKC
Cirazoline hydrochloride
Cat.No: T14972
Synonym: LD 3098 hydrochloride
Target: Others
L-771688 dihydrochloride
Cat.No: T24378
Synonym: L 771688 dihydrochloride
Target:
Indoramin hydrochloride
Cat.No: T82072
Synonym: Indoramine hydrochloride,Wy 21901 hydrochloride
Target:
WB 4101 hydrochloride
Cat.No: T23532
Synonym:
Target: Others
SNAP 5089
Cat.No: T23374
Synonym:
Target: Others
RS 100329
Cat.No: T28617
Synonym: RS100329 HCl,RS 100329 HCl,RS100329,RS-100329
Target:
(R)-(-)-Niguldipine hydrochloride
Cat.No: T23225
Synonym:
Target: Others
PF-3774076
Cat.No: T71335
Synonym:
Target:
Muscarinic toxin 3
Cat.No: T80477
Synonym: MT3
Target: Adrenergic Receptor
(S)-Terazosin
Cat.No: T12815
Synonym:
Target: Adrenergic Receptor
Phenylephrine-3-O-Sulfate
Cat.No: T35576
Synonym:
Target:
Silodosin Glucuronide (sodium salt)
Cat.No: T36071
Synonym:
Target:
AdTx1
Cat.No: TP2086
Synonym:
Target:
BODIPY FL prazosin
Cat.No: T63980
Synonym:
Target:
OxyMetazoline
Cat.No: T64314
Synonym:
Target:
Conopeptide rho-TIA
Cat.No: T80175
Synonym:
Target: Adrenergic Receptor
RS 504393
Cat.No: T5384
Synonym:
Target: CCR
Cirazoline (free base)
Cat.No: T69031
Synonym:
Target:
RS102895
Cat.No: TQ0283
Synonym:
Target: CCR
LY393615
Cat.No: T78626
Synonym: NCC1048
Target: Calcium Channel
ZY-19489
Cat.No: T67694
Synonym:
Target: Parasite
Rec 15/2615 (hydrochloride)
Cat.No: T37794
Synonym:
Target:
Naftopidil
Cat.No: T0696
Synonym: KT-611,萘哌地尔,BM-15275
Target: Adrenergic Receptor
Cat. No. Product Name Target Signaling Pathways
TN4117 GB 1a

Antioxidant; Tyrosinase oxidation-reduction; Proteases/Proteasome
GB 1a 是一种从藤黄 Garcinia travancorica 叶中分离出来的天然产物。
T17310 Phenylephrine

去氧肾上腺素,L-Phenylephrine,去氧肾上腺素碱,(R)-(-)-Phenylephrine

Adrenergic Receptor GPCR/G Protein; Neuroscience
Phenylephrine ((R)-(-)-Phenylephrine) 是一种选择性的α1-肾上腺素受体激动剂,常用作减充血剂。
T0453 Phenylephrine hydrochloride

NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Phenylephrine hydrochloride (NCI-c55641) 是选择性的α1-肾上腺素能受体激动剂,对α1A,α1B 和α1D 受体的pKis 分为4.70,4.87和5.86。

天然产物

GB 1a
Cat.No: TN4117
Synonym:
Target: Antioxidant, Tyrosinase
Phenylephrine
Cat.No: T17310
Synonym: 去氧肾上腺素,L-Phenylephrine,去氧肾上腺素碱,(R)-(-)-Phenylephrine
Target: Adrenergic Receptor
Phenylephrine hydrochloride
Cat.No: T0453
Synonym: NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride
Target: Endogenous Metabolite, Adrenergic Receptor
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