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76

抑制剂 & 化合物

22

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T5421	KDU691	Parasite; PI4K	Microbiology/Virology; PI3K/Akt/mTOR signaling
	KDU691 是一种咪唑吡嗪类药物，对血阶段的裂殖体、配子体和肝期具有较强的抗寄生虫活性，它是 PI4K 抑制剂，选择性抑制双氢青蒿素预处理的恶性疟原虫。
T10096L	Voruciclib	CDK	Cell Cycle/Checkpoint
	Voruciclib 是一种具有口服活性和选择性 CDK 抑制剂，Ki 为 0.626 nM-9.1 nM。它在多种弥漫性大 B 细胞淋巴瘤模型中抑制 MCL-1 的表达。它有效阻断 MCL-1 的转录调节子 CDK9。
T27400L	Ganaplacide phosphate Ganaplacide phosphate (1261113-96-5 Free base)	Others	Others
	Ganaplacide phosphate 对疟原虫症状性无性血期感染具有多阶段抗疟活性，并且能够在动物模型中预防传播和阻断感染。
T14766	BPH-715	Others; Parasite	Microbiology/Virology; Others
	BPH-715 抑制恶性疟原虫的肝脏阶段生长，对 HepG2 细胞中的恶性疟原虫外红细胞的形成的 IC50 为 10 μM。
T79535	Antimalarial agent 30	Parasite	Microbiology/Virology
	Antimalarial agent 30 具有抗伯氏疟原虫肝期寄生虫活性和抗疟活性，可用于研究疟感染。
T11828	LDC7559	Pyroptosis	Apoptosis; Immunology/Inflammation
	LDC7559 通过在晚期阻断中性粒细胞胞外陷阱 (NET)来抑制gasdermin D (GSDMD)。
T9269	N-Chloroacetyl-3,5-bis(trifluoromethyl)aniline N1-[3,5-双(三氟甲基)苯基]-2-氯乙酰胺,N-(3,5-Bis(trifluoromethyl)phenyl)-2-chloroacetamide	Others	Others
	N-Chloroacetyl-3,5-bis(trifluoromethyl)aniline (KM1954) 是一种杀虫剂，对第一阶段Ae 有效。 LC50 值为 125μM 的埃及伊蚊幼虫。
T37376	PHY34	Autophagy	Autophagy
	PHY34是一种晚期自噬抑制剂，具有纳摩尔水平的抑制作用。在体内，PHY34具有抗高级别浆液性卵巢癌（HGSOC）活性。
T11244	Etimizol Ethymisol,Ethimizole,Ethymisole	Others	Others
	Etimizol (Ethimizole) 对缺氧造成的失忆症有效果。
T9246	JNJ-63576253	Androgen Receptor	Endocrinology/Hormones
	JNJ63576253 是具有口服活性的、有效的雄激素受体的完全拮抗剂，在 LNCaP 细胞中对 F877L 突变型 AR 和野生型 AR 的IC50值分别为 37 和 54 nM。它可用于研究去势抵抗性前列腺癌。
T9379	L-Threonic acid magnesium salt	Others	Others
	L-Threonic acid magnesium salt 可增加老年大鼠和晚期阿尔茨海默病 (AD) 模型小鼠的突触密度和记忆能力。
T9925	Ofatumumab	Others	Others
	Ofatumumab 是一种人源化靶向抗 CD20单克隆抗体。它作用于表达 CD20 的 B 淋巴细胞，能够诱导产生抗体依赖性细胞介导的细胞毒性和补体依赖性细胞毒性的作用。
T5181	CA-5f	Apoptosis; Autophagy	Apoptosis; Autophagy
	CA-5f 是晚期巨自噬/自噬抑制剂，通过抑制自噬体-溶酶体融合起作用。它能够增加监控自噬的标记物 LC3B-II 和 SQSTM1 蛋白水平，促进 ROS 的产生，具有抗肿瘤活性。
T29421	LY195448 4-(3-(2-Hydroxy-2-phenyl)ethylamino-3-methylbutyl)benzamide	Others	Others
	LY 195448 (4-(3-(2-Hydroxy-2-phenyl)ethylamino-3-methylbutyl)benzamide) 是存在于人血液和尿液中的一种物质，在小鼠肿瘤模型中显示出抗肿瘤活性,可在中期阻断细胞。
T3131	Fosfomycin calcium Phosphomycin calcium salt,Fosmicin,磷霉素钙	Antibacterial; Antibiotic	Microbiology/Virology
	Fosfomycin calcium (Phosphomycin calcium salt) 是一种能透过血脑屏障的广谱抗生素，不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性，包括耐多药、广泛耐药和耐全药细菌。
T3710	XMD16-5	Tyrosinase; PPAR	DNA Damage/DNA Repair; Metabolism; Proteases/Proteasome
	XMD16-5 是TNK2抑制剂，对D163E 和R806Q 突变体的IC50值分别为16和77nM。
T2180	Hexythiazox	Parasite	Microbiology/Virology
	Hexythiazox 是一种螨类生长调节剂和噻唑烷类杀螨剂，对多种螨类具有长效杀虫作用，适用于植物从萌芽到结果的任何生长阶段。
T28824	SNX0723 SNX 0723,SNX- 0723	HSP	Cytoskeletal Signaling; Metabolism
	SNX0723 是一种 Hsp90 抑制剂，具有抗疟原虫活性。SNX0723 对 HsHsp90 和 PfHsp90 具有高结合亲和力，Ki 分别为 4.4 和 47 nM。SNX0723 抑制肝期伯氏疟原虫 ANKA 寄生虫，EC50 为 3.3 μM。
T21992	Vacuolin-1	PI3K; Autophagy	Autophagy; PI3K/Akt/mTOR signaling
	Vacuolin-1 是一种细胞渗透性抑制剂，可抑制 Ca2+ 依赖性溶酶体与细胞膜的融合。它通过抑制溶酶体内容物的释放起作用。它是一种有效的选择性 PIKfyve 抑制剂，通过损害溶酶体成熟来抑制晚期自噬。
T1063	Ticarcillin disodium Ticarpen,Ticarcillin disodium salt,替卡西林二钠	Antibacterial; Antibiotic	Microbiology/Virology
	Ticarcillin disodium (Ticarpen) 主要用于抗革兰氏阴性菌, 特别是绿脓杆菌, 也是少数可研究嗜麦芽感染的抗生素。
T16500	PF-3450074 PF-74	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	PF-3450074 (PF-74)是 HIV-1 衣壳蛋白的特异性抑制剂，可广谱抑制 HIV 分离株。它在 HIV-1 感染的早期阶段起作用，通过与 CPSF6 和 NUP153 的结合直接竞争来抑制病毒复制，并阻断病毒生命周期的脱膜，组装和逆转录步骤。
T36696	DMBA
	7,12-Dimethylbenz[a]anthracene (DMBA) is a polycyclic aromatic hydrocarbon (PAH) that has been found in tobacco smoke and diesel exhaust and has carcinogenic activity.1,2It undergoes metabolic activation by numerous enzymes, including the cytochrome P450 (CYP450) isoform CYP1B1, as well as microsomal epoxide hydrolase (mEH), producing a variety of reactive metabolites that form DNA adductsin vivo, and it has been commonly used to induce tumor formation in various rodent models.2,3,1DMBA increase...
T36466	Chlorin E6 Ce6,Chlorin e6,CE6	Parasite	Microbiology/Virology
	Chlorin E6 (CE6) 是一种第二代光敏剂，在与辐照结合使用时具有抗肿瘤活性。在植入性纤维肉瘤的小鼠模型中，Chlorin E6（2.5-10 毫克/千克，静脉注射，50-200 焦耳/平方厘米的辐照）在不同程度的辐照后会导致肿瘤完全消失。在一项针对支气管源性早期浅表鳞状细胞癌患者的 I 期临床研究中，对包括 Chlorin E6 在内的制剂进行了测试，结果良好（40 毫克/平方米，静脉注射，100 焦耳/平方厘米的激光辐照）。在一项针对早期肺癌患者的二期临床试验中，同样的给药模式使 82.9% 的患者获得了完全应答。Chlorin E6 已被研究为一种纳米技术给药工具。
T24566	O-1663 O 1663
	O-1663 is an advanced stage breast cancer inhibitor that acts by targeting multiple cannabinoid anti-tumor pathways.
T27333	FLI-28 FLI28
	FLI-28 is a novel general secretion inhibitor in early stage.
T39256	MMV674850 MMV674850
	MMV674850 exhibits potency against asexual stage parasites, with IC50 values of 2.7 and 4.5 nM. Furthermore, it demonstrates a preferential affinity for early-stage gametocytes, displaying an IC50 value of 4.5 ± 3.6 nM, compared to late-stage gametocytes with an IC50 value of 28.7 ± 0.2 nM.
T1769	Pardoprunox 帕多芦诺,SLV-308,DU-126891	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Pardoprunox (SLV-308) 是多巴胺受体D2、D3部分激动剂和5-HT1A 激动剂，pEC50分别为 8、9.2 和 6.3。
T9763	MMV666810
	MMV666810 是一种类似于 MMV390048 的2-氨基吡嗪，5.94 nM 的 MMV666810 对无性寄生虫有效。与早期相比，MMV666810 对晚期配子体细胞的选择性是早期的3.3倍（早期配子体:IC50603 ± 88 nM; 晚期配子体:IC50179 ± 8 nM）。
T71841	MMV085203
	MMV08520 is a novel inhibitor of Plasmodium falciparum, killing both blood- and sexual-stage P. falciparum parasites.
T27264	Endochin
	Endochin is an experimental antimalarial. Endochin and analogues thereof are causal prophylactic and potent erythrocytic stage agents in avian models.
T19837	O4 O 4,O-4
	O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.
T14780	BRD9185	Dehydrogenase	Metabolism
	BRD9185 is an inhibitor of Dihydroorotate dehydrogenase (DHODH) with an EC50 of 16 nM against multidrug-resistant blood-stage parasites in vitro.
T71808	Tisopurine
	Tisopurine is a drug used in the treatment of gout in some countries. It reduces uric acid production through inhibiting an early stage in its production.
T69249	AMXT1501
	AMXT1501 is a polyamine uptake inhibitor, also inhibiting the putrescine transport in epimastigotes (the insect stage of t. cruzi)
T31837	FOLFIRI Regimen FOLFIRI
	FOLFIRI Regimen is a chemotherapy regimen consisting of leucovorin calcium (calcium folinate), 5-fluorouracil, and irinotecan used during the treatment of advanced-stage and metastatic colorectal cancer.
T24330	L 681217 L-681,217,L-681217,L681,217,L 681,217,L681217
	L 681217 is a glycolipid-type antibiotic related to the efrotomycin class. L-681217 inhibits bacterial protein synthesis at the elongation stage. L 681217 shows broad-spectrum antibiotic activity against Gram-positive and Gram-negative bacteria.
T30612	Bulaquine
	Bulaquine is a derivative of 8-aminoquinoline and has effective activity against the liver stage of plasmodium falciparum and the dormant bodies of Plasmodium vivax and Plasmodium ovale.
T35321	Zymostenol delta(8)-Cholestenol,5a-Cholest-8-en-3b-ol,Δ8-Cholesterol	Endogenous Metabolite; ROR	Metabolism
	Zymostenol (5a-Cholest-8-en-3b-ol) 是一种 RORγ 激动剂，EC50为1 μM。Zymostenol 是胆固醇生物合成的后期前体。
T39802	Nedosiran DCR-PHXC
	Nedosiran (DCR-PHXC) is a GalNAc-dsRNA conjugate designed for RNA interference (RNAi) targeting lactate dehydrogenase (LDH). It serves as a potential therapeutic option for patients with primary hyperoxaluria (PH) and end-stage renal disease (ESRD).
T37660	5-hydroxy Thiabendazole
	5-hydroxy Thiabendazole (5-OH TBZ) is a major metabolite of the anthelmintic thiabendazole . Unlike thiabendazole, 5-OH TBZ has no effect on the growth of third-stage A. caninum larvae.
T35037	Vanilmandelic acid, L-(+)- Vanilmandelic acid L-form,(+)-Vanilmandelic acid
	Vanilmandelic acid, L-(+)- is a chemical intermediate in the synthesis of artificial vanilla flavorings and is an end-stage metabolite of the catecholamines, epinephrine, and norepinephrine. It is produced via intermediary metabolites.
T60386	LCS-1
	LCS-1, a superoxide dismutase 1 (SOD1) inhibitor, effectively inhibits the enzymatic activity of SOD1 with an IC50 value of 1.07 μM. Additionally, LCS-1 triggers both early and late-stage apoptosis in multiple myeloma (MM.1S) cells [1] [2] [3].
T70577	PEN-866
	PEN-866 is a potential agent for controlling early stage tumor growth for non-small cell lung cancer (NSCLC). PEN-866 is a novel esterase-cleavable conjugate of an HSP90i and a topoisomerase I inhibitor, SN-38
T37757	Tyvelose
	Tyvelose is an unusual 3,6-dideoxyhexose terminal sugar and the immunodominant component of glycoprotein antigens in the parasitic helminth T. spiralis, which is responsible for trichinosis in humans. It is produced in high amounts by the infective larva and is immunodominant during the muscle stage of infection. Mice immunized with tyvelose-BSA produce IgG1 antibodies to tyvelose but are not resistant to infection by T. spiralis. Tyvelose-specific antibodies (2.5 mg/20 g) administered to rat pu...
T69454	Cephradine dihydrate
	Cephradine dihydrate is the hydrate form of Cephradine (free base), a semi-synthetic cephalosporin antibiotic. Cefradin inhibits the last stage of bacterial cell wall synthesis by binding to certain penicillin-binding proteins which results in cell lysis. Cell lysis is mediated by bacterial cell wall autolytic enzymes. Cefradin may interfere with autolysin inhibitors.
T70654	Ciprokiren
	Ciprokiren is a renin inhibitor discovered by Roche. Ciprokinen inhibited human renin in a buffer and human plasma with an IC50 of 0.07 and 0.65 nmol/L, respectively. In animal models, acute and chronic administration of ciprokinen lead to a reduction in arterial blood pressure. Development of ciprokinen was discontinued at a preclinical stage.
T11534L	Haemanthamine hydrochloride (466-75-1 free base) Haemanthamine hydrochloride	Others	Others
	Haemanthamine hydrochloride is an alkaloid isolated from the Amaryllidaceae plants with potent anticancer activity. It inhibits protein biosynthesis during the elongation stage of translation. It has antimalarial, pro-apoptotic, antiviral, antioxidant, an
T62600	RYL-552S
	RYL-552S 是一种可杀死恶性疟原虫 Plasmodium falciparum 的耐药菌株，其可在体外有效杀灭无性血内阶段的寄生虫。
T81306	REA
	REA为一种特定的肽，具有识别癌症早期阶段的淋巴管的能力，然而对于肿瘤淋巴管则无法识别。
T69070	Cephradine sodium
	Cephradine sodium is the salt form of Cephradine (free base), a semi-synthetic cephalosporin antibiotic. Cefradin inhibits the last stage of bacterial cell wall synthesis by binding to certain penicillin-binding proteins which results in cell lysis. Cell lysis is mediated by bacterial cell wall autolytic enzymes. Cefradin may interfere with autolysin inhibitors.

化合物

Cat.No: T5421

Target: Parasite, PI4K

Cat.No: T10096L

Target: CDK

Ganaplacide phosphate

Cat.No: T27400L

Synonym: Ganaplacide phosphate (1261113-96-5 Free base)

Target: Others

Cat.No: T14766

Target: Others, Parasite

Antimalarial agent 30

Cat.No: T79535

Target: Parasite

Cat.No: T11828

Target: Pyroptosis

N-Chloroacetyl-3,5-bis(trifluoromethyl)aniline

Cat.No: T9269

Synonym: N1-[3,5-双(三氟甲基)苯基]-2-氯乙酰胺,N-(3,5-Bis(trifluoromethyl)phenyl)-2-chloroacetamide

Target: Others

Cat.No: T37376

Target: Autophagy

Cat.No: T11244

Synonym: Ethymisol,Ethimizole,Ethymisole

Target: Others

Cat.No: T9246

Target: Androgen Receptor

L-Threonic acid magnesium salt

Cat.No: T9379

Target: Others

Cat.No: T9925

Target: Others

Cat.No: T5181

Target: Apoptosis, Autophagy

Cat.No: T29421

Synonym: 4-(3-(2-Hydroxy-2-phenyl)ethylamino-3-methylbutyl)benzamide

Target: Others

Fosfomycin calcium

Cat.No: T3131

Synonym: Phosphomycin calcium salt,Fosmicin,磷霉素钙

Target: Antibacterial, Antibiotic

Cat.No: T3710

Target: Tyrosinase, PPAR

Cat.No: T2180

Target: Parasite

Cat.No: T28824

Synonym: SNX 0723,SNX- 0723

Target: HSP

Cat.No: T21992

Target: PI3K, Autophagy

Ticarcillin disodium

Cat.No: T1063

Synonym: Ticarpen,Ticarcillin disodium salt,替卡西林二钠

Target: Antibacterial, Antibiotic

Cat.No: T16500

Synonym: PF-74

Target: HIV Protease

Cat.No: T36696

Cat.No: T36466

Synonym: Ce6,Chlorin e6,CE6

Target: Parasite

Cat.No: T24566

Synonym: O 1663

Cat.No: T27333

Synonym: FLI28

Cat.No: T39256

Synonym: MMV674850

Cat.No: T1769

Synonym: 帕多芦诺,SLV-308,DU-126891

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Cat.No: T9763

Cat.No: T71841

Cat.No: T27264

Cat.No: T19837

Synonym: O 4,O-4

Cat.No: T14780

Target: Dehydrogenase

Cat.No: T71808

Cat.No: T69249

FOLFIRI Regimen

Cat.No: T31837

Synonym: FOLFIRI

Cat.No: T24330

Synonym: L-681,217,L-681217,L681,217,L 681,217,L681217

Cat.No: T30612

Cat.No: T35321

Synonym: delta(8)-Cholestenol,5a-Cholest-8-en-3b-ol,Δ8-Cholesterol

Target: Endogenous Metabolite, ROR

Cat.No: T39802

Synonym: DCR-PHXC

5-hydroxy Thiabendazole

Cat.No: T37660

Vanilmandelic acid, L-(+)-

Cat.No: T35037

Synonym: Vanilmandelic acid L-form,(+)-Vanilmandelic acid

Cat.No: T60386

Cat.No: T70577

Cat.No: T37757

Cephradine dihydrate

Cat.No: T69454

Cat.No: T70654

Haemanthamine hydrochloride (466-75-1 free base)

Cat.No: T11534L

Synonym: Haemanthamine hydrochloride

Target: Others

Cat.No: T62600

Cat.No: T81306

Cephradine sodium

Cat.No: T69070

Cat. No.	Product Name	Target	Signaling Pathways
T7344	SDMA NG,NG'-Dimethyl-L-arginine,Symmetric dimethylarginine,对称N,N-二甲基精氨酸	Endogenous Metabolite	Metabolism
	SDMA (Symmetric dimethylarginine) 是一氧化氮 (NO) 合酶的内源性抑制剂。
T8262	Fosfomycin sodium Fosfomycin Disodium,磷霉素钠	Antibacterial; Antibiotic	Microbiology/Virology
	Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素，不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性，包括耐多药、广泛耐药和耐全药的细菌。
TN2121	3,5,7,3′,4′-Pentamethoxyflavone 栎精-3,5,7,3',4'-五甲醚,槲皮素3,5,7,3',4'-五甲基醚,Quercetin 3,5,7,3,4-pentamethyl ether	Others	Others
	3,5,7,3′,4′-Pentamethoxyflavone (Quercetin 3,5,7,3,4-pentamethyl ether) 是一种分离自小花山奈中的多甲氧基黄酮。在分化早期，它可以调控转录因子，促进 3T3-L1 前脂肪细胞形成脂肪。
T13741	Isoviolanthin 异佛莱心苷,异佛来心苷	Others	Others
	Isoviolanthin 是一种黄酮类苷类化合物，提取自铁皮石斛叶中。它能减少 TGF-β1 处理的 HCC 细胞的迁移和入侵能力，对正常细胞没有毒性影响，对转移性肝癌晚期具有潜在的研究价值。
T3S0364	L-Arginine L-精氨酸,L-Arg,(S)-(+)-Arginine	IL Receptor; Endogenous Metabolite; NO Synthase	Immunology/Inflammation; Metabolism
	L-Arginine (L-Arg) 是内皮型一氧化氮合酶(eNOS) 的底物。L-Arginine 通过阳离子氨基酸转运体家族转运到血管平滑肌细胞，并被代谢成一氧化氮、多胺或 L-脯氨酸。
T11534	Haemanthamine	Others	Others
	Haemanthamine is an alkaloid isolated from the Amaryllidaceae plants with potent anticancer activity. It inhibits protein biosynthesis during the elongation stage of translation. It has antimalarial, pro-apoptotic, antiviral, antioxidant, and anticonvulsa
TN5681	Cypellocarpin C Camaldulenside,桉叶苷
	Cypellocarpin C shows potent in vitro antitumor-promoting activity, it also can suppress an in vivo two-stage carcinogenesis induced with nitric oxide and TPA on mouse skin.
T2S1115	Albaspidin AA	Antifection	Microbiology/Virology
	Albaspidin AA displays strong antibacterial activity against the vegetative form of P. larvae (MIC ranging from 0.168-220 uM). It may have in vitro nematocidal activity against L4 stage larvae.
TN4695	Odorine	Others	Others
	Odorine has potent anti-carcinogenic effect by inhibiting both the initiation and promotion stages of two-stage skin carcinogenesis. It was found to inhibit the growth of the vinblastine-resistant KB cells by enhancing the anticancer activity of vinblastine.
TN5852	Oleuropeic acid
	(+)-Oleuropeic acid shows potent in vitro antitumor-promoting activity, it also suppresses an in vivo two-stage carcinogenesis induced with nitric oxide and 12-O-tetradecanoyl phorbol 13-acetate (TPA) on mouse skin.
TN3392	Alpha-Toxicarol	Others	Others
	Alpha-Toxicarol exhibits a marked inhibitory effect on mouse skin tumor promotion in an in vivo two-stage carcinogenesis test.
TN4696	Odorinol	Antifection	Microbiology/Virology
	Odorine and odorinol inhibit both the initiation and promotion stages of two-stage skin carcinogenesis. (+)-Odorinol exhibits strong antiviral activity against Ranikhet disease virus (RVD) in chick embryo.
TN1649	Frangulin A	Others	Others
	Frangulin A 保护葡萄叶免受葡萄单胞菌感染，并抑制葡萄藤的生物营养菌丝发育。
TN2047	Pendulone	Antifection	Microbiology/Virology
	Pendulone could be a valuable chemopreventive agent, it shows strong inhibition on the effect of the cell cycle induced by TPA and shows potent anti-tumor-promoting activity for an in vivo two-stage carcinogenesis test.
TN4380	Karavilagenin D	Others	Others
	Karavilagenin D exhibits inhibitory effects on skin-tumor promotion in an in vivo two-stage mouse skin carcinogenesis test based on 7,12-dimethylbenz[a]anthracene (DMBA) as initiator, and with TPA as a promoter. It exhibits inhibition effect against human
TN4241	Hyptadienic acid
	Hyptadienic acid exhibits moderate cytotoxicity against HepG2 cells.It also shows a marked anti-inflammatory effect, it also exhibits strong antitumor-promoting activity in an in vivo two-stage carcinogenesis test of mouse tumor by using 7,12-dimethylbenz
TN4652	Niazimicin	NF-κB; PI3K; AChR; Antifection	Microbiology/Virology; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling
	Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in the two-stage carcinogenesis in mouse skin using 7,12-dimethylbenz(a)anthracene (DMBA) as ini
T73069	Kurzipene D
	Kurzipene D是一种有效的抗癌剂(anticanceragent)，通过诱导HepG2细胞凋亡(apoptosis)并使其在S期阻滞，显示出明显的抗肿瘤作用。通过体内斑马鱼模型，Kurzipene D展现了其抑制肿瘤增殖和迁移的特性。
T82406	FF-MAS
	FF-MAS是一种有效的meiotic maturation激动剂，能促进小鼠卵母细胞在体外成熟，促进其发展到MII阶段，并增强从2细胞阶段到囊胚阶段转变的潜力。
T73813	Haemanthamine hydrochloride
	Haemanthamine hydrochloride 是从Amaryllidaceae 植物中分离出来的一种蛇毒碱样生物碱，具有强大的抗癌活性。Haemanthamine hydrochloride 靶向核糖体以在翻译的延长阶段抑制蛋白质的生物合成。Haemanthamine hydrochloride 具有促凋亡，抗氧化剂，抗病毒，抗疟疾和抗惊厥活性。
TN2839	2alpha,19alpha-Dihydroxy-3-oxo-urs-12-en-28-oic acid	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	2alpha,19alpha-Dihydroxy-3-oxo-urs-12-en-28-oic acid has anti-HIV activity. It shows an inhibitory effect on the activation of Epstein-Barr virus early antigen (EBV-EA) induced by 12-O-tetradecanoylphorbol-13-acetate (TPA) and causes a significant delay o
TN4140	Glochidiol	Others	Others
	Glochidiol exhibits strong inhibitory effects against all three human tumor cell lines (MCF-7, NCI-H-460 and SF-268), it exerts its antiproliferative activity through the involvement of apoptosis. It exhibits a strong inhibitory effect on mouse skin tumor

天然产物

Cat.No: T7344

Synonym: NG,NG'-Dimethyl-L-arginine,Symmetric dimethylarginine,对称N,N-二甲基精氨酸

Target: Endogenous Metabolite

Fosfomycin sodium

Cat.No: T8262

Synonym: Fosfomycin Disodium,磷霉素钠

Target: Antibacterial, Antibiotic

3,5,7,3′,4′-Pentamethoxyflavone

Cat.No: TN2121

Synonym: 栎精-3,5,7,3',4'-五甲醚,槲皮素3,5,7,3',4'-五甲基醚,Quercetin 3,5,7,3,4-pentamethyl ether

Target: Others

Cat.No: T13741

Synonym: 异佛莱心苷,异佛来心苷

Target: Others

Cat.No: T3S0364

Synonym: L-精氨酸,L-Arg,(S)-(+)-Arginine

Target: IL Receptor, Endogenous Metabolite, NO Synthase

Cat.No: T11534

Target: Others

Cypellocarpin C

Cat.No: TN5681

Synonym: Camaldulenside,桉叶苷

Cat.No: T2S1115

Target: Antifection

Cat.No: TN4695

Target: Others

Oleuropeic acid

Cat.No: TN5852

Alpha-Toxicarol

Cat.No: TN3392

Target: Others

Cat.No: TN4696

Target: Antifection

Cat.No: TN1649

Target: Others

Cat.No: TN2047

Target: Antifection

Karavilagenin D

Cat.No: TN4380

Target: Others

Hyptadienic acid

Cat.No: TN4241

Cat.No: TN4652

Target: NF-κB, PI3K, AChR, Antifection

Cat.No: T73069

Cat.No: T82406

Haemanthamine hydrochloride

Cat.No: T73813

2alpha,19alpha-Dihydroxy-3-oxo-urs-12-en-28-oic acid

Cat.No: TN2839

Target: HIV Protease

Cat.No: TN4140

Target: Others

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