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Search Results for " methanesulfonate "

64

抑制剂 & 化合物

1

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T3111	Abemaciclib methanesulfonate abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate)	CDK	Cell Cycle/Checkpoint
	Abemaciclib methanesulfonate (LY2835219) 是一种选择性的CDK4/6抑制剂，能够抑制 CDK4/CDK6 的活性，IC50分别为 2 nM 和 10 nM。
T9985	Methyl methanesulfonate	DNA Alkylation	DNA Damage/DNA Repair
	Methyl methanesulfonate 是一种DNA 烷基化剂，可以分别修饰腺嘌呤（为3-甲基腺嘌呤）和鸟嘌呤（7-甲基腺嘌呤），进而导致碱基错配和复制障碍。
T12425	PF-06424439 methanesulfonate	Acyltransferase; Transferase	Metabolism
	PF-06424439 methanesulfonate 是一种口服有效咪唑并吡啶二酰基甘油酰基转移酶 2 (DGAT2)选择性抑制剂，IC50是14 nM。PF-06424439 methanesulfonate 具有缓慢可逆，时间依赖性的特点，其相对于酰基-CoA 底物以非竞争性模式抑制 DGAT2。
T21483	Tricaine methanesulfonate 3-氨基苯甲酸乙酯甲基磺酸盐,MS-222	Others	Others
	Tricaine methanesulfonate (MS-222) 常用于固定鱼的标记和运输，并能抑制入侵过程中的感觉系统。
T38979	CYH33 methanesulfonate CYH33 methanesulfonate
	CYH33 methanesulfonate is a highly selective and orally active inhibitor of PI3Kα, with IC50 values of 5.9 nM, 598 nM, 78.7 nM, and 225 nM against the α, β, δ, and γ isoforms, respectively. This compound effectively inhibits the phosphorylation of Akt and ERK, leading to a significant G1 phase arrest in breast cancer cells and non-small cell lung cancer (NSCLC) cells. Additionally, CYH33 methanesulfonate demonstrates potent activity against solid tumors.
T9894	2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate	Others	Others
	2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate 是一种天然产物，可作为参考标准。
T13087	Tariquidar methanesulfonate, hydrate XR9576 methanesulfonate, hydrate	Others	Others
	Tariquidar methanesulfonate, hydrate is a potent and specific P-glycoprotein (P-gp) inhibitor(Kd of 5.1 nM).
T68534	FK-448 methanesulfonate
	FK-448 methanesulfonate is a chymotrypsin inhibitor that has been shown to affect intestinal absorption of insulin in rats and dogs .
T1275	Phentolamine mesylate Phentolamine methanesulfonate,甲磺酸酚妥拉明,Phentolamine mesilate	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Phentolamine mesylate (Phentolamine methanesulfonate) 是一种非选择性的、可逆的，具有口服活性的 α1 和 α2 肾上腺素能受体阻滞剂，能够扩张使血管，降低周围血管阻力。它可用于研究嗜铬细胞瘤相关的高血压，心力衰竭和勃起功能障碍。
T6643	Ro 31-8220 Mesylate Ro 31-8220 methanesulfonate,Bisindolylmaleimide IX,Bisindolylmaleimide IX mesylate	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) 是PKC 抑制剂，对 PKCα、PKCβI、PKCβII、PKCγ、PKCε 和大鼠大脑 PKC 的IC50值为 5、24、14、27、24 和 23 nM。它还抑制 MAPKAP-K1b、MSK1、S6K1 和 GSK3β，IC50为3、8、15 和 38 nM。
T69185	INO-1001 methanesulfonate
	INO-1001 methanesulfonate is an isoindolinone derivative and potent inhibitor of the nuclear enzyme poly (ADP-ribose) polymerase (PARP) with chemosensitization and radiosensitization properties.
T23148	Phenamil methanesulfonate Phenamil	Others	Others
	TRPP3 channel inhibitor
T25722	Lifarizine methanesulfonate
	Lifarizine methanesulfonate is a modulator of sodium-calcium channel that reduces ischemic brain damage.
T5133	Dabigatran Etexilate Mesylate 甲磺酸达比加群酯,BIBR 1048MS,Dabigatran etexilate methanesulfonate	Thrombin	Proteases/Proteasome
	Dabigatran Etexilate Mesylate (BIBR 1048MS) 是一种口服具有活性的 Dabigatran 前药，具有抗凝作用，能够预防心房颤动引起的静脉血栓栓塞和中风。
T71096	GCC-4401C methanesulfonate
	GCC-4401C methanesulfonate is a factor Xa inhibitor similar to rivaroxaban that is currently under development for venous thromboembolic disease (VTE).
T26260	Tetrabenazine methanesulfonate NSC169886,NSC 169886,NSC-169886
	Tetrabenazine methanesulfonate is a medicine formerly utilized as an antipsychotic and therapy for various movement disorders. Tetrabenazine methanesulfonate blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high-affin
T13567	BCX 1470 methanesulfonate	Serine Protease	Proteases/Proteasome
	BCX 1470 methanesulfonate inhibits the esterolytic activity of factor D and C1s (IC50: 96 nM and 1.6 nM), 3.4- and 200-fold better than that of trypsin, respectively.
T2226	Pergolide mesylate 甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Pergolide mesylate salt(LY127809) 是一种有效的，具有口服活性的多巴胺 D1和 D2受体激动剂，是一种 Ergoline 衍生物，可用于帕金森氏病和高泌乳素血症的研究。
T19014	Hydroxystilbamidine bis(methanesulfonate)	Others	Others
	Hydroxystilbamidine bis(methanesulfonate) is a dye capable of binding to both DNA and RNA. It also is a potent inhibitor of cellular ribonucleases.
T34224	Quinacrine methanesulfonate Mepacrine dimethanesulfonate salt
	Quinacrine methanesulfonate is a bioactive chemical.
T1072	Loxeen Pridinol methanesulfonate,Α,Α-二苯基-1-哌啶丙醇(普立地诺甲磺酸盐 )	AChR	Neuroscience
	Loxeen (Pridinol methanesulfonate) 用作抗胆碱能药物和抗帕金森病药物。
T12417	PF-04217903 methanesulfonate	c-Met/HGFR	Tyrosine Kinase/Adaptors
	PF-04217903 methanesulfonate is a potent ATP-competitive inhibitor of c-Met kinase (Ki of 4.8 nM for human c-Met).
T1336	Benztropine mesylate Benzotropine mesylate,苯扎托品,Benzatropine mesylate,Benztropine methanesulfonate,甲磺酸苯扎托品	Dopamine Receptor; AChR; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Benztropine mesylate (Benztropine methanesulfonate) 是一种可口服的中枢性抗胆碱能剂，用于帕金森氏病的研究。它是抗组胺剂，抑制多巴胺的吸收。它也是人 D2多巴胺受体的变构拮抗剂，具有抗癌症干细胞的作用。
T1620	Pazufloxacin Mesylate Pazucross,Pazufloxacin mesilate,甲磺酸帕珠沙星,T-3762,帕珠沙星甲磺酸盐,Pazufloxacin methanesulfonate	Topoisomerase; Antibacterial; Antibiotic	DNA Damage/DNA Repair; Microbiology/Virology
	Pazufloxacin Mesylate (T-3762) 是一种喹诺酮类抗生素。
T30076	Aniline, p-(5-phenylpentyloxy)-, methanesulfonate
	Aniline, p-(5-phenylpentyloxy)-, methanesulfonate is a bioactive chemical.
T6835	Fenoldopam mesylate Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526,非诺多泮甲磺酸盐	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Fenoldopam mesylate (Corlopam mesylate) 是一种多巴胺受体D1选择性激动剂。
T33201	m-Anisidine, 4-(4-phenylbutoxy)-, methanesulfonate
	m-Anisidine, 4-(4-phenylbutoxy)-, methanesulfonate is a bioactive chemical.
T33312	4-(Octyloxy)-m-toluidine methanesulfonate Methanesulfonic acid, compd. with 4-(octyloxy)-m-toluidine (7CI)
	Methanesulfonic acid, compd. with 4-(octyloxy)-m-toluidine (7CI) is a bioactive chemical.
T34041	Phthalimide, N-(2-(p-aminophenoxy)ethyl)-, methanesulfonate
	Phthalimide, N-(2-(p-aminophenoxy)ethyl)-, methanesulfonate is a bioactive chemical.
T65157	Ethyl methanesulfonate
	Ethyl methanesulfonate 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65157，CAS号为 62-50-0。
T72280	PBT434 methanesulfonate
	PBT434 methanesulfonate 为一种有效、口服活性并能穿透血脑屏障的α-synuclein aggregation抑制剂，同时担任铁螯合剂和跨细胞铁运输的调节剂。该化合物抑制铁介导的氧化还原活性及α-synuclein聚集，可有效防止SNpc神经元丢失，显示出在PD研究中的应用潜力。
T33522	m-Toluidine, 4-(octyloxy)-alpha-(phenylthio)-, methanesulfonate
	m-Toluidine, 4-(octyloxy)-alpha-(phenylthio)-, methanesulfonate is a bioactive chemical.
T69008	Paroxol methanesulfonate
	Paroxol methanesulfonate is an intermediate in the synthesis of Paroxetine, a selective serotonin reuptake inhibitor.
T69165	Methiothepin methanesulfonate
	Methiothepin methanesulfonate is an inhibitor of HCV infection and cell-to-cell transmission that acts by targeting the HCV E2 glycoprotein.
T65303	Phenyl methanesulfonate
	Phenyl methanesulfonate 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65303，CAS号为 16156-59-5。
T34042	Phthalimide, N-(3-(p-aminophenoxy)propyl)-, methanesulfonate
	Phthalimide, N-(3-(p-aminophenoxy)propyl)-, methanesulfonate is a bioactive chemical.
T33181	m-Anisidine, 4-((5-(benzyloxy)pentyl)oxy)-, methanesulfonate
	m-Anisidine, 4-((5-(benzyloxy)pentyl)oxy)-, methanesulfonate is a bioactive chemical.
T13108L	Pamufetinib mesylate TAS-115 mesylate,TAS-115 methanesulfonate	Others	Others
	TAS-115 mesylate is a potent inhibitor of VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase(IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively).
T71094	CD4 (81-92)
	CD4 (81-92) is a peptide that was previously found to inhibit gp120 binding, HIV-1 infectivity, and syncytium formation.
T69989	(S)-Pomalidomide
	(S)-Pomalidomide is an inhibitor of angiogenesis and growth of B-cell neoplasias, which induces complete regressions of Burkitt's lymphoma cell tumors.
T67318	1-((2-(2,4-Difluorophenyl)oxiran-2-yl)methyl)-1H-1,2,4-triazole methanesulfonate
	1-((2-(2,4-Difluorophenyl)oxiran-2-yl)methyl)-1H-1,2,4-triazole methanesulfonate 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T67318，CAS号为 86386-77-8。
T70460	HM5023507
	HM5023507, an orally active dual inhibitor of δγ isoforms in immune signaling. HM5023507 inhibited PI3Kδ and PI3Kγ isoforms with greater than 100-fold selectivity against PI3Kα and PI3Kβ in recombinant enzymatic assays and in primary human immune cells with an exquisite selectivity against other targets.
T70995	GSK-256066
	GSK-256066 is a PDE4 inhibitor.
T67219	(2R,3R)-2-(2,4-Difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butane-2,3-diol methanesulfonate
	(2R,3R)-2-(2,4-Difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butane-2,3-diol methanesulfonate 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T67219，CAS号为 1175536-50-1。
T66687	[(2-Di-cyclohexylphosphino-3,6-dimethoxy-2′,4′,6′- triisopropyl-1,1′-biphenyl)-2-(2′-amino-1,1′ -biphenyl)]palladium(II) methanesulfonate
	[(2-Di-cyclohexylphosphino-3,6-dimethoxy-2′,4′,6′- triisopropyl-1,1′-biphenyl)-2-(2′-amino-1,1′ -biphenyl)]palladium(II) methanesulfonate 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T66687，CAS号为 1470372-59-8。
T70357	CM-546
	CM-546 is the trans-isomer of CM-414, and a dual inhibitor of PDE5 and HDACs.
T13689	Ethylene dimethanesulfonate	Apoptosis	Apoptosis
	Ethylene dimethanesulfonate 是温和的烷基化乙二醇非挥发性甲烷磺酸二酯，对 LC 具有选择性的促凋亡作用。
T11553	Heptamidine dimethanesulfonate SBi4211 dimethanesulfonate	Others	Others
	Heptamidine dimethanesulfonate (SBi4211 dimethanesulfonate) 是一种与喷他脒有关的、强效的钙结合蛋白 S100B 的抑制剂 (Kd=6.9 μM)，选择性地杀死表达 S100B 的黑素瘤细胞。它是有效的强直性肌营养不良 (DM) 研究工具。
T11381	Pictilisib dimethanesulfonate GDC-0941 dimethanesulfonate,GDC-0941 2 MeSO3H salt	Apoptosis; DNA-PK; PI3K; mTOR; Autophagy	Apoptosis; Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
	Pictilisib dimethanesulfonate (GDC-0941 2 MeSO3H salt) 是一种 PI3Kα/δ抑制剂，IC50值为 3 nM。对 p110β 和 p110γ的选择性分别为11倍和25倍。
T83100	Antibacterial agent 161 trifluoromethanesulfonate
	Antibacterialagent 161 (trifluoromethanesulfonate) (Compound 6) 表现出抗菌特性，并对结肠癌和非小细胞肺癌细胞线显示出显著的抗增殖活性。

化合物

Abemaciclib methanesulfonate

Cat.No: T3111

Synonym: abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate)

Target: CDK

Methyl methanesulfonate

Cat.No: T9985

Target: DNA Alkylation

PF-06424439 methanesulfonate

Cat.No: T12425

Target: Acyltransferase, Transferase

Tricaine methanesulfonate

Cat.No: T21483

Synonym: 3-氨基苯甲酸乙酯甲基磺酸盐,MS-222

Target: Others

CYH33 methanesulfonate

Cat.No: T38979

Synonym: CYH33 methanesulfonate

2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate

Cat.No: T9894

Target: Others

Tariquidar methanesulfonate, hydrate

Cat.No: T13087

Synonym: XR9576 methanesulfonate, hydrate

Target: Others

FK-448 methanesulfonate

Cat.No: T68534

Phentolamine mesylate

Cat.No: T1275

Synonym: Phentolamine methanesulfonate,甲磺酸酚妥拉明,Phentolamine mesilate

Target: Adrenergic Receptor

Ro 31-8220 Mesylate

Cat.No: T6643

Synonym: Ro 31-8220 methanesulfonate,Bisindolylmaleimide IX,Bisindolylmaleimide IX mesylate

Target: PKC

INO-1001 methanesulfonate

Cat.No: T69185

Phenamil methanesulfonate

Cat.No: T23148

Synonym: Phenamil

Target: Others

Lifarizine methanesulfonate

Cat.No: T25722

Dabigatran Etexilate Mesylate

Cat.No: T5133

Synonym: 甲磺酸达比加群酯,BIBR 1048MS,Dabigatran etexilate methanesulfonate

Target: Thrombin

GCC-4401C methanesulfonate

Cat.No: T71096

Tetrabenazine methanesulfonate

Cat.No: T26260

Synonym: NSC169886,NSC 169886,NSC-169886

BCX 1470 methanesulfonate

Cat.No: T13567

Target: Serine Protease

Pergolide mesylate

Cat.No: T2226

Synonym: 甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Hydroxystilbamidine bis(methanesulfonate)

Cat.No: T19014

Target: Others

Quinacrine methanesulfonate

Cat.No: T34224

Synonym: Mepacrine dimethanesulfonate salt

Cat.No: T1072

Synonym: Pridinol methanesulfonate,Α,Α-二苯基-1-哌啶丙醇(普立地诺甲磺酸盐 )

Target: AChR

PF-04217903 methanesulfonate

Cat.No: T12417

Target: c-Met/HGFR

Benztropine mesylate

Cat.No: T1336

Synonym: Benzotropine mesylate,苯扎托品,Benzatropine mesylate,Benztropine methanesulfonate,甲磺酸苯扎托品

Target: Dopamine Receptor, AChR, Histamine Receptor

Pazufloxacin Mesylate

Cat.No: T1620

Synonym: Pazucross,Pazufloxacin mesilate,甲磺酸帕珠沙星,T-3762,帕珠沙星甲磺酸盐,Pazufloxacin methanesulfonate

Target: Topoisomerase, Antibacterial, Antibiotic

Aniline, p-(5-phenylpentyloxy)-, methanesulfonate

Cat.No: T30076

Fenoldopam mesylate

Cat.No: T6835

Synonym: Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526,非诺多泮甲磺酸盐

Target: Dopamine Receptor

m-Anisidine, 4-(4-phenylbutoxy)-, methanesulfonate

Cat.No: T33201

4-(Octyloxy)-m-toluidine methanesulfonate

Cat.No: T33312

Synonym: Methanesulfonic acid, compd. with 4-(octyloxy)-m-toluidine (7CI)

Phthalimide, N-(2-(p-aminophenoxy)ethyl)-, methanesulfonate

Cat.No: T34041

Ethyl methanesulfonate

Cat.No: T65157

PBT434 methanesulfonate

Cat.No: T72280

m-Toluidine, 4-(octyloxy)-alpha-(phenylthio)-, methanesulfonate

Cat.No: T33522

Paroxol methanesulfonate

Cat.No: T69008

Methiothepin methanesulfonate

Cat.No: T69165

Phenyl methanesulfonate

Cat.No: T65303

Phthalimide, N-(3-(p-aminophenoxy)propyl)-, methanesulfonate

Cat.No: T34042

m-Anisidine, 4-((5-(benzyloxy)pentyl)oxy)-, methanesulfonate

Cat.No: T33181

Pamufetinib mesylate

Cat.No: T13108L

Synonym: TAS-115 mesylate,TAS-115 methanesulfonate

Target: Others

Cat.No: T71094

(S)-Pomalidomide

Cat.No: T69989

1-((2-(2,4-Difluorophenyl)oxiran-2-yl)methyl)-1H-1,2,4-triazole methanesulfonate

Cat.No: T67318

Cat.No: T70460

Cat.No: T70995

(2R,3R)-2-(2,4-Difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butane-2,3-diol methanesulfonate

Cat.No: T67219

[(2-Di-cyclohexylphosphino-3,6-dimethoxy-2′,4′,6′- triisopropyl-1,1′-biphenyl)-2-(2′-amino-1,1′ -biphenyl)]palladium(II) methanesulfonate

Cat.No: T66687

Cat.No: T70357

Ethylene dimethanesulfonate

Cat.No: T13689

Target: Apoptosis

Heptamidine dimethanesulfonate

Cat.No: T11553

Synonym: SBi4211 dimethanesulfonate

Target: Others

Pictilisib dimethanesulfonate

Cat.No: T11381

Synonym: GDC-0941 dimethanesulfonate,GDC-0941 2 MeSO3H salt

Target: Apoptosis, DNA-PK, PI3K, mTOR, Autophagy

Antibacterial agent 161 trifluoromethanesulfonate

Cat.No: T83100

Cat. No.	Product Name	Target	Signaling Pathways
T21518	Colistin methanesulfonate sodium salt 粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)	Cell wall; Antibacterial	Immunology/Inflammation; Microbiology/Virology
	Colistin methanesulfonate sodium salt (Colistimethate Sodium) 是一种来自 Bacillus colistinus 的环状多肽抗生素，由多粘菌素 E1 和 E2 组成。

天然产物

Colistin methanesulfonate sodium salt

Cat.No: T21518

Synonym: 粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)

Target: Cell wall, Antibacterial

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